Page last updated: 2024-09-02

rx 821002 and selegiline

rx 821002 has been researched along with selegiline in 1 studies

Compound Research Comparison

Studies
(rx 821002)
Trials
(rx 821002)
Recent Studies (post-2010)
(rx 821002)
Studies
(selegiline)
Trials
(selegiline)
Recent Studies (post-2010) (selegiline)
3170452,575319394

Protein Interaction Comparison

ProteinTaxonomyrx 821002 (IC50)selegiline (IC50)
CholinesteraseHomo sapiens (human)0.0055
Cytochrome P450 3A4Homo sapiens (human)0.0039
Alpha-2A adrenergic receptorHomo sapiens (human)1.798
Alpha-2B adrenergic receptorHomo sapiens (human)0.376
Amine oxidase [flavin-containing] BRattus norvegicus (Norway rat)0.2127
Amine oxidase [flavin-containing] A Rattus norvegicus (Norway rat)0.9046
Amine oxidase [flavin-containing] AHomo sapiens (human)1.4408
Adenosine receptor A1Rattus norvegicus (Norway rat)0.0067
Amine oxidase [flavin-containing] BHomo sapiens (human)0.1001
Type-1 angiotensin II receptorSus scrofa (pig)0.048
Alpha-synucleinHomo sapiens (human)0.27
Amine oxidase [flavin-containing] BBos taurus (cattle)1
Sigma intracellular receptor 2Rattus norvegicus (Norway rat)0.017

Research

Studies (1)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's1 (100.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Hudson, AL; Hume, SP; Lalies, MD; Nutt, DJ; Robinson, ES; Tyacke, RJ1

Other Studies

1 other study(ies) available for rx 821002 and selegiline

ArticleYear
Estimation of endogenous noradrenaline release in rat brain in vivo using [3H]RX 821002.
    Synapse (New York, N.Y.), 2005, Volume: 55, Issue:2

    Topics: Adrenergic alpha-Antagonists; Adrenergic Uptake Inhibitors; Animals; Binding, Competitive; Brain; Dextroamphetamine; Idazoxan; Imidazoles; Male; Microdialysis; Monoamine Oxidase Inhibitors; Norepinephrine; Radioligand Assay; Rats; Rats, Wistar; Selegiline; Time Factors; Tissue Distribution; Tritium

2005