rx 821002 has been researched along with rauwolscine in 3 studies
| Studies (rx 821002) | Trials (rx 821002) | Recent Studies (post-2010) (rx 821002) | Studies (rauwolscine) | Trials (rauwolscine) | Recent Studies (post-2010) (rauwolscine) |
|---|---|---|---|---|---|
| 317 | 0 | 45 | 47 | 0 | 14 |
| Protein | Taxonomy | rx 821002 (IC50) | rauwolscine (IC50) |
|---|---|---|---|
| Alpha-2C adrenergic receptor | Homo sapiens (human) | 0.016 | |
| Alpha-2B adrenergic receptor | Rattus norvegicus (Norway rat) | 0.165 | |
| Alpha-2C adrenergic receptor | Rattus norvegicus (Norway rat) | 0.165 | |
| Alpha-2A adrenergic receptor | Rattus norvegicus (Norway rat) | 0.165 |
| Timeframe | Studies, this research(%) | All Research% |
|---|---|---|
| pre-1990 | 0 (0.00) | 18.7374 |
| 1990's | 2 (66.67) | 18.2507 |
| 2000's | 1 (33.33) | 29.6817 |
| 2010's | 0 (0.00) | 24.3611 |
| 2020's | 0 (0.00) | 2.80 |
| Authors | Studies |
|---|---|
| Neubig, RR; Porter, AC; Uhlén, S | 1 |
| Bylund, DB; Cerutis, DR; Deupree, JD; Hinton, KA | 1 |
| Harms, GS; Lohse, MJ; Steinmeyer, R; Vilardaga, JP | 1 |
3 other study(ies) available for rx 821002 and rauwolscine
| Article | Year |
|---|---|
The novel alpha-2 adrenergic radioligand [3H]-MK912 is alpha-2C selective among human alpha-2A, alpha-2B and alpha-2C adrenoceptors.
Topics: Adrenergic alpha-Antagonists; Animals; Binding, Competitive; CHO Cells; Cricetinae; Dibenzazepines; Humans; Imidazoles; Indoles; Isoindoles; Quinolizines; Radioligand Assay; Receptors, Adrenergic, alpha-2 | 1994 |
Buffers differentially alter the binding of [3H]rauwolscine and [3H]RX821002 to the alpha-2 adrenergic receptor subtypes.
Topics: Animals; Buffers; CHO Cells; Cricetinae; Humans; Idazoxan; Kinetics; Opossums; Oxymetazoline; Prazosin; Radioligand Assay; Rats; Receptors, Adrenergic, alpha-2; Recombinant Proteins; Species Specificity; Yohimbine | 1996 |
Molecular basis of inverse agonism in a G protein-coupled receptor.
Topics: Adrenergic alpha-2 Receptor Agonists; Cell Line; Fluorescence Resonance Energy Transfer; Humans; Ligands; Protein Binding; Receptors, Adrenergic, alpha-2; Receptors, G-Protein-Coupled; Signal Transduction | 2005 |