Page last updated: 2024-09-02

rx 821002 and prazosin

rx 821002 has been researched along with prazosin in 44 studies

Compound Research Comparison

Studies
(rx 821002)
Trials
(rx 821002)
Recent Studies (post-2010)
(rx 821002)
Studies
(prazosin)
Trials
(prazosin)
Recent Studies (post-2010) (prazosin)
3170457,914713682

Protein Interaction Comparison

ProteinTaxonomyrx 821002 (IC50)prazosin (IC50)
Solute carrier family 22 member 1 Homo sapiens (human)5.87
Interstitial collagenaseHomo sapiens (human)4.036
Alpha-2A adrenergic receptorHomo sapiens (human)2.638
Matrix metalloproteinase-9Homo sapiens (human)6.963
Alpha-1B adrenergic receptorRattus norvegicus (Norway rat)0.0008
Ribosyldihydronicotinamide dehydrogenase [quinone]Homo sapiens (human)0.0078
Alpha-2B adrenergic receptorHomo sapiens (human)0.29
Alpha-2C adrenergic receptorHomo sapiens (human)0.647
Alpha-1D adrenergic receptorRattus norvegicus (Norway rat)0.0008
Alpha-1D adrenergic receptorHomo sapiens (human)0.0007
Bromodomain-containing protein 2Homo sapiens (human)0.0009
Alpha-1A adrenergic receptorHomo sapiens (human)0.0006
Alpha-1B adrenergic receptorHomo sapiens (human)0.0006
5-hydroxytryptamine receptor 2BHomo sapiens (human)4.118
Alpha-1A adrenergic receptorRattus norvegicus (Norway rat)0.0008
5-hydroxytryptamine receptor 7Cavia porcellus (domestic guinea pig)9.9
Potassium voltage-gated channel subfamily H member 2Homo sapiens (human)1.5849
Multidrug and toxin extrusion protein 1Homo sapiens (human)1.6

Research

Studies (44)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's22 (50.00)18.2507
2000's15 (34.09)29.6817
2010's7 (15.91)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Denis-Pouxviel, C; Devedjian, JC; Esclapez, F; Paris, H1
Neubig, RR; Porter, AC; Uhlén, S1
De Backer, JP; De Keyser, J; De Vos, H; Van Liefde, I; Vauquelin, G1
Berlan, M; Galitzky, J; Lafontan, M; Montastruc, JL; Senard, JM; Stillings, M1
Berlan, M; Estan, L; Montastruc, JL; Senard, JM; Tran, MA1
Advenier, C; Biyah, K1
Hussain, JF; Kendall, DA; Pinthong, D; Wilson, VG1
Blaylock, NA; Kendall, DA; Wilson, VG; Wright, IK1
Atrens, DM; Fleischhauer, AE; Kuhlman, SJ; Siviy, SM1
Ala-Uotila, S; Kurose, H; Marjamäki, A; Oker-Blom, C; Pohjanoksa, K; Scheinin, M; Sizmann, D1
Blandizzi, C; Carignani, D; Colucci, R; Crema, F; Del Tacca, M; Lazzeri, G; Natale, G1
Bylund, DB; Cerutis, DR; Deupree, JD; Hinton, KA1
Herman, CA; Luczy, G; Uhlén, S; Wikberg, JE1
Intengan, HD; Smyth, DD1
Elliott, J1
Bearham, MC; Heal, DJ; Hutchins, LJ; Jackson, HC; Mazurkiewicz, SE; Needham, AM1
Guyenet, PG; Huangfu, D1
Butterworth, RF; Buu, PN; Michalak, A; Rose, C1
Audinot, V; Cistarelli, L; Gobert, A; Millan, MJ; Newman-Tancredi, A; Rivet, JM1
Caramona, MM; Figueiredo, IV; Guimarães, S; Moura, D; Paiva, MQ1
Aicher, SA; Drake, CT1
Goepel, M; Krege, S; Michel, MC; Michelotti, GA; Price, DT; Schwinn, DA1
Benamour, K; Chang-Fong, J; Cussac, M; Morand, JM; Szymonski, B; Thomasson, F1
Dausse, JP; Giudicelli, Y; Ilhami, N; Khalid, M1
Corrêa, FM; Peres-Polon, VL; Tavares, RF1
De Luca, LA; Menani, JV; Moreira, Tdos S; Renzi, A; Takakura, AC1
Goldstein, I; Huang, YH; Kim, NN; Min, K; Traish, AM1
De Luca, LA; dos Santos Moreira, T; Menani, JV; Renzi, A; Takakura, AC1
Kindlundh, A; Lindblom, J; Mugisha, P; Nyberg, F; Uhlén, S1
Fagerholm, V; Hein, L; Philipp, M; Scheinin, M1
Blum, JW; Hammon, HM; Ontsouka, EC; Zbinden, Y1
Greenup, JL; Leverenz, JB; Peskind, ER; Raskind, MA; Szot, P; White, SS2
Ahsan, MR; Lehmann, ML; Quartermain, D; Stone, EA; Yan, L; Yeretsian, J1
Bylund, DB; Happe, HK; Murrin, LC; Sanders, JD; Szot, P; Weinshenker, D1
Colombari, DS; De Luca, LA; Menani, JV; Moreira, TS; Takakura, AC1
Chang, ST; Chuang, CH; Kao, YC; Lin, YL; Liu, YP; Tung, CS1
Acheson, AG; Dashwood, MR; Eames, T; Gruss, H; Henry, Y; Rayment, SJ; Scholefield, JH; Simpson, JA; Wilson, VG1
Bennett, DJ; D'Amico, J; Gorassini, MA; Murray, KC; Rank, MM; Stephens, MJ1
Aono, Y; Cools, AR; Koshikawa, N; Saigusa, T; Takada, K; Uchida, T; Verheij, MM1
Hackett, D; Heal, DJ; Hutson, PH; Murray, F; Vickers, SP1
Essali, N; Sanders, J1
Dobrzański, G; Kwiatkowska, K; Pradel, K; Przewłocki, R; Solecki, WB; Szklarczyk, K1
Hartzler, LK; Santin, JM; Vallejo, M1

Other Studies

44 other study(ies) available for rx 821002 and prazosin

ArticleYear
Further characterization of human alpha 2-adrenoceptor subtypes: [3H]RX821002 binding and definition of additional selective drugs.
    European journal of pharmacology, 1994, Jan-24, Volume: 252, Issue:1

    Topics: Adrenergic alpha-Antagonists; Animals; Binding, Competitive; Cell Line; Dioxanes; Humans; Idazoxan; Plasmids; Radioligand Assay; Receptors, Adrenergic, alpha; Transfection

1994
The novel alpha-2 adrenergic radioligand [3H]-MK912 is alpha-2C selective among human alpha-2A, alpha-2B and alpha-2C adrenoceptors.
    The Journal of pharmacology and experimental therapeutics, 1994, Volume: 271, Issue:3

    Topics: Adrenergic alpha-Antagonists; Animals; Binding, Competitive; CHO Cells; Cricetinae; Dibenzazepines; Humans; Imidazoles; Indoles; Isoindoles; Quinolizines; Radioligand Assay; Receptors, Adrenergic, alpha-2

1994
Regional distribution of alpha 2A- and alpha 2B-adrenoceptor subtypes in postmortem human brain.
    Journal of neurochemistry, 1992, Volume: 58, Issue:4

    Topics: Adrenergic alpha-Antagonists; Aged; Binding, Competitive; Brain; Cadaver; Dioxanes; Humans; Idazoxan; Middle Aged; Oxymetazoline; Prazosin; Receptors, Adrenergic, alpha; Receptors, Adrenergic, beta; Tissue Distribution

1992
Identification of human platelet alpha 2-adrenoceptors with a new antagonist [3H]-RX821002, a 2-methoxy derivative of idazoxan.
    British journal of pharmacology, 1990, Volume: 100, Issue:4

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Adult; Blood Platelets; Brimonidine Tartrate; Dioxanes; Epinephrine; Humans; Idazoxan; In Vitro Techniques; Kinetics; Male; Membranes; Oxymetazoline; Prazosin; Quinoxalines; Radioligand Assay; Receptors, Adrenergic, alpha; Yohimbine

1990
Reserpine induces vascular alpha 2-adrenergic supersensitivity and platelet alpha 2-adrenoceptor up-regulation in dog.
    British journal of pharmacology, 1990, Volume: 101, Issue:2

    Topics: Adipose Tissue; Animals; Blood Platelets; Blood Pressure; Cardiovascular System; Catecholamines; Cell Membrane; Clonidine; Dioxanes; Dogs; Heart Rate; Idazoxan; Male; Norepinephrine; Posture; Prazosin; Receptors, Adrenergic, alpha; Reserpine; Up-Regulation; Yohimbine

1990
Effects of three alpha 2-adrenoceptor agonists, rilmenidine, UK 14304 and clonidine on bradykinin- and substance P-induced airway microvascular leakage in guinea-pigs.
    Neuropeptides, 1995, Volume: 28, Issue:4

    Topics: Acetylcholine; Adrenergic alpha-1 Receptor Antagonists; Adrenergic alpha-2 Receptor Agonists; Adrenergic alpha-2 Receptor Antagonists; Adrenergic alpha-Agonists; Animals; Bradykinin; Brimonidine Tartrate; Capillaries; Capillary Permeability; Clonidine; Dioxanes; Extravascular Lung Water; Guinea Pigs; Idazoxan; Oxazoles; Prazosin; Quinoxalines; Rilmenidine; Substance P; Trachea

1995
Comparison of the interaction of agmatine and crude methanolic extracts of bovine lung and brain with alpha 2-adrenoceptor binding sites.
    British journal of pharmacology, 1995, Volume: 115, Issue:4

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Agmatine; Animals; Binding, Competitive; Brimonidine Tartrate; Cattle; Cerebral Cortex; Clonidine; Dioxanes; Idazoxan; Imidazoles; Lung; Methanol; Prazosin; Quinoxalines; Receptors, Adrenergic, alpha-2; Yohimbine

1995
The relationship between density of alpha-adrenoceptor binding sites and contractile responses in several porcine isolated blood vessels.
    British journal of pharmacology, 1995, Volume: 114, Issue:3

    Topics: 5'-Nucleotidase; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Aorta, Thoracic; Binding, Competitive; Cell Membrane; Dioxanes; Dose-Response Relationship, Drug; Drug Interactions; Ear, External; Idazoxan; Male; Microscopy, Electron; Muscle Contraction; Muscle, Smooth, Vascular; Prazosin; Radioligand Assay; Receptors, Adrenergic, alpha; Splenic Artery; Structure-Activity Relationship; Swine; Veins; Yohimbine

1995
Effects of alpha-2 adrenoceptor antagonists on rough-and-tumble play in juvenile rats: evidence for a site of action independent of non-adrenoceptor imidazoline binding sites.
    Psychopharmacology, 1994, Volume: 113, Issue:3-4

    Topics: Adrenergic alpha-2 Receptor Antagonists; Adrenergic alpha-Agonists; Agonistic Behavior; Animals; Clonidine; Dioxanes; Female; Idazoxan; Imidazoline Receptors; Interpersonal Relations; Male; Prazosin; Rats; Rats, Sprague-Dawley; Rats, Wistar; Receptors, Drug

1994
Similar ligand binding in recombinant human alpha 2 C2-adrenoceptors produced in mammalian, insect and yeast cells.
    European journal of pharmacology, 1994, Mar-15, Volume: 267, Issue:1

    Topics: Adrenergic alpha-Antagonists; Amino Acid Sequence; Animals; Cells, Cultured; Chlorpromazine; Dioxanes; Humans; Idazoxan; Immunoblotting; Mammary Neoplasms, Experimental; Mice; Molecular Sequence Data; Moths; Oxymetazoline; Prazosin; Receptors, Adrenergic, alpha; Recombinant Proteins; Saccharomyces cerevisiae; Transfection; Tumor Cells, Cultured; Yohimbine

1994
Determination on functional basis of presynaptic alpha 2-adrenoceptor subtypes in guinea-pig duodenum.
    Neuroscience letters, 1996, May-24, Volume: 210, Issue:1

    Topics: Adrenergic alpha-2 Receptor Agonists; Adrenergic alpha-2 Receptor Antagonists; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Cholinergic Fibers; Duodenum; Electric Stimulation; Gastrointestinal Motility; Guinea Pigs; Idazoxan; Imidazoles; Indoles; Isoindoles; Isoquinolines; Male; Medetomidine; Muscle Contraction; Nordefrin; Norepinephrine; Oxymetazoline; Piperazines; Prazosin; Receptors, Adrenergic, alpha-2; Synaptic Membranes; Vasoconstrictor Agents; Xylazine; Yohimbine

1996
Buffers differentially alter the binding of [3H]rauwolscine and [3H]RX821002 to the alpha-2 adrenergic receptor subtypes.
    The Journal of pharmacology and experimental therapeutics, 1996, Volume: 278, Issue:3

    Topics: Animals; Buffers; CHO Cells; Cricetinae; Humans; Idazoxan; Kinetics; Opossums; Oxymetazoline; Prazosin; Radioligand Assay; Rats; Receptors, Adrenergic, alpha-2; Recombinant Proteins; Species Specificity; Yohimbine

1996
Characterization of adrenoceptor types and subtypes in American bullfrogs acclimated to warm or cold temperature.
    General and comparative endocrinology, 1996, Volume: 104, Issue:2

    Topics: Acclimatization; Adrenergic alpha-Antagonists; Adrenergic beta-Antagonists; Animals; Binding, Competitive; Dose-Response Relationship, Drug; Humans; Idazoxan; Kidney; Membrane Proteins; Myocardium; Pindolol; Prazosin; Radioligand Assay; Rana catesbeiana; Receptors, Adrenergic; Receptors, Adrenergic, alpha-1; Receptors, Adrenergic, alpha-2; Receptors, Adrenergic, beta; Spinal Cord; Temperature

1996
Alpha-2a/d adrenoceptor subtype stimulation by guanfacine increases osmolar clearance.
    The Journal of pharmacology and experimental therapeutics, 1997, Volume: 281, Issue:1

    Topics: Adrenergic alpha-Agonists; Animals; Body Water; Brimonidine Tartrate; Guanfacine; Idazoxan; Kidney; Male; Naltrexone; Prazosin; Quinoxalines; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, alpha-2

1997
Alpha-adrenoceptors in equine digital veins: evidence for the presence of both alpha1 and alpha2-receptors mediating vasoconstriction.
    Journal of veterinary pharmacology and therapeutics, 1997, Volume: 20, Issue:4

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Azepines; Binding, Competitive; Brimonidine Tartrate; Dopamine; Horses; Idazoxan; In Vitro Techniques; Isometric Contraction; Methoxamine; Muscle, Smooth, Vascular; Norepinephrine; Phenylephrine; Prazosin; Quinoxalines; Receptors, Adrenergic, alpha-1; Receptors, Adrenergic, alpha-2; Vasoconstriction; Veins; Yohimbine

1997
Investigation of the mechanisms underlying the hypophagic effects of the 5-HT and noradrenaline reuptake inhibitor, sibutramine, in the rat.
    British journal of pharmacology, 1997, Volume: 121, Issue:8

    Topics: Adrenergic Uptake Inhibitors; Animals; Cyclobutanes; Eating; Idazoxan; Male; Metoprolol; Prazosin; Propanolamines; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, beta; Receptors, Serotonin; Selective Serotonin Reuptake Inhibitors

1997
Alpha 2-adrenergic autoreceptors in A5 and A6 neurons of neonate rats.
    The American journal of physiology, 1997, Volume: 273, Issue:5

    Topics: Adrenergic alpha-Antagonists; Animals; Animals, Newborn; Brain; Idazoxan; In Vitro Techniques; Locus Coeruleus; Meglumine; Membrane Potentials; Neurons; Norepinephrine; Potassium; Potassium Channels; Prazosin; Rats; Receptors, Adrenergic, alpha-2; Sodium; Tetrodotoxin

1997
Evidence for altered central noradrenergic function in experimental acute liver failure in the rat.
    Hepatology (Baltimore, Md.), 1998, Volume: 27, Issue:2

    Topics: Adrenergic alpha-Antagonists; Adrenergic beta-Antagonists; Animals; Autoradiography; Cerebral Cortex; Chromatography, High Pressure Liquid; Coma; Dopamine; Frontal Lobe; Hippocampus; Hypothalamus; Idazoxan; Liver Failure, Acute; Microdialysis; Norepinephrine; Pindolol; Prazosin; Propanolamines; Putamen; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic; Serotonin; Thalamus

1998
Simultaneous quantification of serotonin, dopamine and noradrenaline levels in single frontal cortex dialysates of freely-moving rats reveals a complex pattern of reciprocal auto- and heteroreceptor-mediated control of release.
    Neuroscience, 1998, Volume: 84, Issue:2

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Benzopyrans; Dopamine; Dopamine Agonists; Frontal Lobe; Guanabenz; Guinea Pigs; Homeostasis; Idazoxan; Imidazoles; Indoles; Isoindoles; Male; Medetomidine; Models, Neurological; Motor Activity; Norepinephrine; Oxadiazoles; Piperazines; Prazosin; Raclopride; Rats; Rats, Wistar; Receptors, Adrenergic; Receptors, Dopamine; Receptors, Serotonin; Salicylamides; Serotonin

1998
Prejunctional alpha2A-autoreceptors in the human gastric and ileocolic arteries.
    Naunyn-Schmiedeberg's archives of pharmacology, 1998, Volume: 358, Issue:2

    Topics: Adrenergic alpha-Antagonists; Aged; Arteries; Autoreceptors; Colon; Dioxanes; Dopamine Antagonists; Dose-Response Relationship, Drug; Electric Stimulation; Female; Gastric Mucosa; Humans; Idazoxan; Ileum; In Vitro Techniques; Male; Middle Aged; Neuromuscular Junction; Norepinephrine; Phentolamine; Prazosin; Receptors, Adrenergic, alpha-2; Spiro Compounds; Stomach; Tritium; Yohimbine

1998
Clonidine evokes vasodepressor responses via alpha2-adrenergic receptors in gigantocellular reticular formation.
    The Journal of pharmacology and experimental therapeutics, 1999, Volume: 289, Issue:2

    Topics: Adrenergic alpha-2 Receptor Agonists; Adrenergic alpha-2 Receptor Antagonists; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Blood Pressure; Clonidine; Depression, Chemical; Dose-Response Relationship, Drug; Heart Rate; Hemodynamics; Idazoxan; Male; Medulla Oblongata; Microinjections; Neurons; Prazosin; Rats; Rats, Sprague-Dawley; Reticular Formation

1999
Characterization of alpha-adrenoceptor subtypes in the corpus cavernosum of patients undergoing sex change surgery.
    The Journal of urology, 1999, Volume: 162, Issue:5

    Topics: Adrenergic alpha-Antagonists; Binding, Competitive; Disorders of Sex Development; Dose-Response Relationship, Drug; Humans; Idazoxan; Male; Penis; Prazosin; Receptors, Adrenergic, alpha; Sulfonamides; Tamsulosin

1999
Synthesis and alpha-adrenergic binding ligand affinities of 2-iminoimidazolidine derivatives.
    Chemical & pharmaceutical bulletin, 2000, Volume: 48, Issue:5

    Topics: Adrenergic alpha-2 Receptor Agonists; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Binding, Competitive; Clonidine; Idazoxan; Imidazoles; In Vitro Techniques; Ligands; Magnetic Resonance Spectroscopy; Prazosin; Rats; Receptors, Adrenergic, alpha-2; Spectrophotometry, Infrared; Yohimbine

2000
Testosterone dependence of salt-induced hypertension in Sabra rats and role of renal alpha(2)-adrenoceptor subtypes.
    The Journal of pharmacology and experimental therapeutics, 2002, Volume: 300, Issue:1

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Blood Pressure; Gene Expression Regulation; Guanfacine; Hypertension; Idazoxan; Kidney; Male; Orchiectomy; Prazosin; Rats; Receptors, Adrenergic, alpha-2; RNA, Messenger; Sodium Chloride; Testosterone

2002
Mechanisms involved in the water intake-related pressor response in the rat.
    Journal of hypertension, 2002, Volume: 20, Issue:2

    Topics: Animals; Antihypertensive Agents; Arteries; Blood Pressure; Brazil; Diazepam; Dose-Response Relationship, Drug; Drinking; Heart Rate; Idazoxan; Lidocaine; Losartan; Male; Mecamylamine; Models, Animal; Muscle Relaxants, Central; Prazosin; Quinine; Rats; Rats, Wistar; Sodium Chloride; Tropanes; Water

2002
Inhibition of pilocarpine-induced salivation in rats by central noradrenaline.
    Archives of oral biology, 2002, Volume: 47, Issue:6

    Topics: Adrenergic alpha-1 Receptor Antagonists; Adrenergic alpha-2 Receptor Antagonists; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Analysis of Variance; Animals; Idazoxan; Injections, Intraperitoneal; Injections, Intraventricular; Male; Muscarinic Agonists; Norepinephrine; Pilocarpine; Prazosin; Rats; Rats, Sprague-Dawley; Saliva; Salivation; Statistics as Topic; Yohimbine

2002
Biochemical and functional characterization of alpha-adrenergic receptors in the rabbit vagina.
    Life sciences, 2002, Nov-01, Volume: 71, Issue:24

    Topics: Administration, Intravaginal; Adrenergic alpha-Antagonists; Animals; Behavior, Animal; Drug Therapy, Combination; Female; Idazoxan; In Vitro Techniques; Isometric Contraction; Ligands; Muscle, Smooth, Vascular; Oxyhemoglobins; Prazosin; Rabbits; Radioligand Assay; Receptors, Adrenergic, alpha; Sexual Behavior; Vagina; Vasodilator Agents

2002
Central alpha(2) adrenergic receptors and cholinergic-induced salivation in rats.
    Brain research bulletin, 2003, Jan-30, Volume: 59, Issue:5

    Topics: Adrenergic alpha-Antagonists; Animals; Brain; Idazoxan; Imidazoles; Injections, Intraperitoneal; Injections, Intraventricular; Male; Muscarinic Agonists; Pilocarpine; Prazosin; Rats; Receptors, Adrenergic, alpha-2; Salivation; Sympatholytics; Yohimbine

2003
Nandrolone treatment decreases the level of rat kidney alpha(1B)-adrenoceptors.
    Naunyn-Schmiedeberg's archives of pharmacology, 2003, Volume: 368, Issue:2

    Topics: Adrenergic alpha-1 Receptor Antagonists; Adrenergic alpha-2 Receptor Antagonists; Adrenergic alpha-Antagonists; Anabolic Agents; Animals; Idazoxan; Injections, Intramuscular; Kidney; Ligands; Male; Nandrolone; Prazosin; Radioligand Assay; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, alpha-1; Receptors, Adrenergic, alpha-2; Spleen

2003
[Ethyl-3H]RS-79948-197 alpha2-adrenoceptor autoradiography validation in alpha2-adrenoceptor knockout mice.
    European journal of pharmacology, 2004, Aug-30, Volume: 497, Issue:3

    Topics: Adrenergic alpha-2 Receptor Antagonists; Adrenergic alpha-Agonists; Animals; Autoradiography; Binding Sites; Binding, Competitive; Cerebral Cortex; Idazoxan; In Vitro Techniques; Isoquinolines; Ligands; Mice; Mice, Knockout; Naphthyridines; Oxymetazoline; Phentolamine; Prazosin; Putamen; Radioligand Assay; Receptors, Adrenergic, alpha-2; Tritium; Yohimbine

2004
Ontogenesis of mRNA levels and binding sites of hepatic alpha-adrenoceptors in young cattle.
    Domestic animal endocrinology, 2006, Volume: 30, Issue:3

    Topics: Adrenergic alpha-Antagonists; Animals; Animals, Newborn; Binding, Competitive; Blood Glucose; Cattle; Female; Glycogen; Idazoxan; Liver; Phosphoenolpyruvate; Prazosin; Pregnancy; Pyruvate Carboxylase; Receptors, Adrenergic, alpha; Receptors, Adrenergic, beta; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger

2006
Compensatory changes in the noradrenergic nervous system in the locus ceruleus and hippocampus of postmortem subjects with Alzheimer's disease and dementia with Lewy bodies.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 2006, Jan-11, Volume: 26, Issue:2

    Topics: Adrenergic alpha-Antagonists; Adult; Aged; Aged, 80 and over; Alzheimer Disease; Dendrites; Female; Fluoxetine; Hippocampus; Humans; Idazoxan; In Situ Hybridization; Lewy Body Disease; Locus Coeruleus; Male; Middle Aged; Nerve Tissue Proteins; Norepinephrine; Norepinephrine Plasma Membrane Transport Proteins; Prazosin; Receptors, Adrenergic, alpha-1; Receptors, Adrenergic, alpha-2; RNA, Messenger; Tetralones; Tyrosine 3-Monooxygenase

2006
Role of CNS alpha1-adrenoceptor activity in central fos responses to novelty.
    Synapse (New York, N.Y.), 2006, Volume: 59, Issue:5

    Topics: Adrenergic alpha-Antagonists; Animals; Behavior, Animal; Brain Chemistry; Central Nervous System; Dialysis; Exploratory Behavior; Idazoxan; Immunohistochemistry; Male; Oncogene Proteins v-fos; Phenylephrine; Prazosin; Protein Binding; Rats; Rats, Wistar; Receptors, Adrenergic, alpha-1

2006
Analysis of brain adrenergic receptors in dopamine-beta-hydroxylase knockout mice.
    Brain research, 2006, Sep-13, Volume: 1109, Issue:1

    Topics: Analysis of Variance; Animals; Animals, Newborn; Autoradiography; Brain; Dopamine beta-Hydroxylase; Gene Expression Regulation, Developmental; Guanosine 5'-O-(3-Thiotriphosphate); Idazoxan; Isotopes; Mice; Mice, Inbred C57BL; Mice, Knockout; Pindolol; Prazosin; Receptors, Adrenergic, alpha-1; Receptors, Adrenergic, alpha-2

2006
Changes in adrenoreceptors in the prefrontal cortex of subjects with dementia: evidence of compensatory changes.
    Neuroscience, 2007, Apr-25, Volume: 146, Issue:1

    Topics: Adrenergic alpha-Antagonists; Adult; Aged; Aged, 80 and over; Dementia; Female; Gene Expression Regulation; Humans; Idazoxan; Male; Middle Aged; Postmortem Changes; Prazosin; Prefrontal Cortex; Receptors, Adrenergic; RNA, Messenger

2007
Activation of alpha(2)-adrenoceptors in the lateral hypothalamus reduces pilocarpine-induced salivation in rats.
    Neuroscience letters, 2009, Feb-06, Volume: 450, Issue:3

    Topics: Adrenergic alpha-2 Receptor Agonists; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Drug Interactions; Hypothalamic Area, Lateral; Idazoxan; Imidazoles; Male; Muscarinic Agonists; Norepinephrine; Pilocarpine; Prazosin; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, alpha-2; Salivation

2009
Alpha adrenergic modulation on effects of norepinephrine transporter inhibitor reboxetine in five-choice serial reaction time task.
    Journal of biomedical science, 2009, Aug-14, Volume: 16

    Topics: Adrenergic alpha-1 Receptor Antagonists; Adrenergic alpha-2 Receptor Antagonists; Adrenergic alpha-Antagonists; Adrenergic Uptake Inhibitors; Animals; Attention; Discrimination, Psychological; Drug Evaluation, Preclinical; Drug Interactions; Feeding Behavior; Idazoxan; Impulsive Behavior; Male; Morpholines; Norepinephrine Plasma Membrane Transport Proteins; Prazosin; Rats; Rats, Sprague-Dawley; Reaction Time; Reboxetine; Receptors, Adrenergic, alpha-1; Receptors, Adrenergic, alpha-2; Spatial Behavior; Time Perception

2009
Investigation of the distribution and function of alpha-adrenoceptors in the sheep isolated internal anal sphincter.
    British journal of pharmacology, 2010, Volume: 160, Issue:7

    Topics: Adrenergic alpha-1 Receptor Antagonists; Adrenergic alpha-2 Receptor Antagonists; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Anal Canal; Animals; Antibodies, Monoclonal; Autoradiography; Binding, Competitive; Dose-Response Relationship, Drug; Fecal Incontinence; Humans; Idazoxan; Immunohistochemistry; In Vitro Techniques; Muscle Contraction; Prazosin; Protein Binding; Radioligand Assay; Receptors, Adrenergic, alpha-1; Receptors, Adrenergic, alpha-2; Sheep

2010
Adrenergic receptors modulate motoneuron excitability, sensory synaptic transmission and muscle spasms after chronic spinal cord injury.
    Journal of neurophysiology, 2011, Volume: 105, Issue:1

    Topics: Adrenergic Agonists; Adrenergic Antagonists; Animals; Chromones; Clonidine; Excitatory Postsynaptic Potentials; Female; Idazoxan; Models, Animal; Motor Neurons; Norepinephrine; Prazosin; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic; Sensory Receptor Cells; Spasm; Spinal Cord Injuries; Synaptic Transmission

2011
The α₁-, but not α₂-, adrenoceptor in the nucleus accumbens plays an inhibitory role upon the accumbal noradrenaline and dopamine efflux of freely moving rats.
    European journal of pharmacology, 2012, Aug-05, Volume: 688, Issue:1-3

    Topics: Adrenergic alpha-2 Receptor Agonists; Adrenergic alpha-2 Receptor Antagonists; Animals; Brimonidine Tartrate; Clonidine; Dopamine; Dose-Response Relationship, Drug; Extracellular Space; Idazoxan; Male; Methoxamine; Movement; Neurons; Norepinephrine; Nucleus Accumbens; Prazosin; Quinoxalines; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, alpha-1; Receptors, Adrenergic, alpha-2

2012
Effects of lisdexamfetamine in a rat model of binge-eating.
    Journal of psychopharmacology (Oxford, England), 2015, Volume: 29, Issue:12

    Topics: Animals; Baclofen; Behavior, Animal; Benzazepines; Benzodiazepines; Body Weight; Bulimia; Disease Models, Animal; Eating; Feeding Behavior; Female; Idazoxan; Lisdexamfetamine Dimesylate; Naltrexone; Olanzapine; Prazosin; Prodrugs; Raclopride; Rats; Rats, Wistar; Rolipram

2015
Interdependent adrenergic receptor regulation of Arc and Zif268 mRNA in cerebral cortex.
    Neuroscience letters, 2016, Jan-26, Volume: 612

    Topics: Adrenergic Antagonists; Animals; Cerebral Cortex; Cytoskeletal Proteins; Early Growth Response Protein 1; Idazoxan; Nerve Tissue Proteins; Prazosin; Propranolol; Rats, Sprague-Dawley; Receptors, Adrenergic; Receptors, Adrenergic, alpha-1; Receptors, Adrenergic, alpha-2; Receptors, Adrenergic, beta; RNA, Messenger

2016
Noradrenergic signaling in the VTA modulates cocaine craving.
    Addiction biology, 2018, Volume: 23, Issue:2

    Topics: Adrenergic alpha-1 Receptor Agonists; Adrenergic alpha-1 Receptor Antagonists; Adrenergic alpha-2 Receptor Antagonists; Adrenergic beta-Antagonists; Animals; Behavior, Animal; Cocaine; Conditioning, Operant; Craving; Dopamine Uptake Inhibitors; Drug-Seeking Behavior; Idazoxan; Male; Phenylephrine; Prazosin; Propranolol; Rats; Rats, Sprague-Dawley; Self Administration; Ventral Tegmental Area

2018
Noradrenergic modulation determines respiratory network activity during temperature changes in the in vitro brainstem of bullfrogs.
    Respiratory physiology & neurobiology, 2018, Volume: 258

    Topics: Action Potentials; Adrenergic alpha-Antagonists; Analysis of Variance; Animals; Brain Stem; Female; Idazoxan; In Vitro Techniques; Motor Neurons; Norepinephrine; Prazosin; Rana catesbeiana; Respiration; Spinal Cord; Temperature

2018