Page last updated: 2024-09-02

rx 821002 and pilocarpine

rx 821002 has been researched along with pilocarpine in 4 studies

Compound Research Comparison

Studies
(rx 821002)
Trials
(rx 821002)
Recent Studies (post-2010)
(rx 821002)
Studies
(pilocarpine)
Trials
(pilocarpine)
Recent Studies (post-2010) (pilocarpine)
3170457,3343401,528

Protein Interaction Comparison

ProteinTaxonomyrx 821002 (IC50)pilocarpine (IC50)
Muscarinic acetylcholine receptor M1Rattus norvegicus (Norway rat)3.0267
Muscarinic acetylcholine receptor M3Rattus norvegicus (Norway rat)3.84
Muscarinic acetylcholine receptor M4Rattus norvegicus (Norway rat)3.84
Muscarinic acetylcholine receptor M5Rattus norvegicus (Norway rat)3.84
Muscarinic acetylcholine receptor M2Rattus norvegicus (Norway rat)3.84

Research

Studies (4)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's1 (25.00)18.2507
2000's3 (75.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Asier Garro, M; GarcĂ­a-Sevilla, JA; Giralt, MT; Menargues, A; Miralles, A; Obach, R; Olmos, G; Pineda, J; Ugedo, L1
De Luca, LA; Menani, JV; Moreira, Tdos S; Renzi, A; Takakura, AC1
De Luca, LA; dos Santos Moreira, T; Menani, JV; Renzi, A; Takakura, AC1
Colombari, DS; De Luca, LA; Menani, JV; Moreira, TS; Takakura, AC1

Other Studies

4 other study(ies) available for rx 821002 and pilocarpine

ArticleYear
Acute and chronic effects of cholinesterase inhibitors and pilocarpine on the density and sensitivity of central and peripheral alpha 2-adrenoceptors.
    European journal of pharmacology, 1993, Jun-04, Volume: 236, Issue:3

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Binding Sites; Brain; Brimonidine Tartrate; Cholinesterase Inhibitors; Clonidine; Dioxanes; Idazoxan; In Vitro Techniques; Isoflurophate; Male; Neostigmine; Physostigmine; Pilocarpine; Quinoxalines; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, alpha; Tyrosine 3-Monooxygenase; Vas Deferens

1993
Inhibition of pilocarpine-induced salivation in rats by central noradrenaline.
    Archives of oral biology, 2002, Volume: 47, Issue:6

    Topics: Adrenergic alpha-1 Receptor Antagonists; Adrenergic alpha-2 Receptor Antagonists; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Analysis of Variance; Animals; Idazoxan; Injections, Intraperitoneal; Injections, Intraventricular; Male; Muscarinic Agonists; Norepinephrine; Pilocarpine; Prazosin; Rats; Rats, Sprague-Dawley; Saliva; Salivation; Statistics as Topic; Yohimbine

2002
Central alpha(2) adrenergic receptors and cholinergic-induced salivation in rats.
    Brain research bulletin, 2003, Jan-30, Volume: 59, Issue:5

    Topics: Adrenergic alpha-Antagonists; Animals; Brain; Idazoxan; Imidazoles; Injections, Intraperitoneal; Injections, Intraventricular; Male; Muscarinic Agonists; Pilocarpine; Prazosin; Rats; Receptors, Adrenergic, alpha-2; Salivation; Sympatholytics; Yohimbine

2003
Activation of alpha(2)-adrenoceptors in the lateral hypothalamus reduces pilocarpine-induced salivation in rats.
    Neuroscience letters, 2009, Feb-06, Volume: 450, Issue:3

    Topics: Adrenergic alpha-2 Receptor Agonists; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Drug Interactions; Hypothalamic Area, Lateral; Idazoxan; Imidazoles; Male; Muscarinic Agonists; Norepinephrine; Pilocarpine; Prazosin; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, alpha-2; Salivation

2009