Page last updated: 2024-09-02

rx 821002 and physostigmine

rx 821002 has been researched along with physostigmine in 1 studies

Compound Research Comparison

Studies
(rx 821002)
Trials
(rx 821002)
Recent Studies (post-2010)
(rx 821002)
Studies
(physostigmine)
Trials
(physostigmine)
Recent Studies (post-2010) (physostigmine)
3170456,230252331

Protein Interaction Comparison

ProteinTaxonomyrx 821002 (IC50)physostigmine (IC50)
AcetylcholinesteraseElectrophorus electricus (electric eel)0.1666
AcetylcholinesteraseTetronarce californica (Pacific electric ray)0.3023
CholinesteraseHomo sapiens (human)0.3055
Cytochrome P450 2D6Homo sapiens (human)0.2
Alpha-1B adrenergic receptorRattus norvegicus (Norway rat)0.857
AcetylcholinesteraseMus musculus (house mouse)0.0269
AcetylcholinesteraseHomo sapiens (human)0.0853
Acetylcholinesterase Bos taurus (cattle)0.7197
Alpha-1D adrenergic receptorRattus norvegicus (Norway rat)0.857
Delta-type opioid receptorMus musculus (house mouse)1.1821
AcetylcholinesteraseGallus gallus (chicken)0.02
AcetylcholinesteraseRattus norvegicus (Norway rat)0.0416
Alpha-1A adrenergic receptorRattus norvegicus (Norway rat)0.857
CholinesteraseEquus caballus (horse)0.4081
CholinesteraseMus musculus (house mouse)0.28
Acyl-CoA:cholesterol acyltransferase Oryctolagus cuniculus (rabbit)0.0189
Carboxylic ester hydrolase Rattus norvegicus (Norway rat)0.018
Carboxylic ester hydrolase Equus caballus (horse)1.263

Research

Studies (1)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's1 (100.00)18.2507
2000's0 (0.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Asier Garro, M; GarcĂ­a-Sevilla, JA; Giralt, MT; Menargues, A; Miralles, A; Obach, R; Olmos, G; Pineda, J; Ugedo, L1

Other Studies

1 other study(ies) available for rx 821002 and physostigmine

ArticleYear
Acute and chronic effects of cholinesterase inhibitors and pilocarpine on the density and sensitivity of central and peripheral alpha 2-adrenoceptors.
    European journal of pharmacology, 1993, Jun-04, Volume: 236, Issue:3

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Binding Sites; Brain; Brimonidine Tartrate; Cholinesterase Inhibitors; Clonidine; Dioxanes; Idazoxan; In Vitro Techniques; Isoflurophate; Male; Neostigmine; Physostigmine; Pilocarpine; Quinoxalines; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, alpha; Tyrosine 3-Monooxygenase; Vas Deferens

1993