Page last updated: 2024-09-02

rx 821002 and nisoxetine

rx 821002 has been researched along with nisoxetine in 3 studies

Compound Research Comparison

Studies
(rx 821002)
Trials
(rx 821002)
Recent Studies (post-2010)
(rx 821002)
Studies
(nisoxetine)
Trials
(nisoxetine)
Recent Studies (post-2010) (nisoxetine)
317045316262

Protein Interaction Comparison

ProteinTaxonomyrx 821002 (IC50)nisoxetine (IC50)
Cytochrome P450 1A1Homo sapiens (human)0.0079
Cytochrome P450 1A2Homo sapiens (human)0.0079
Prostaglandin G/H synthase 1Homo sapiens (human)2.4
Sodium-dependent noradrenaline transporter Homo sapiens (human)0.0131
Sodium-dependent dopamine transporterRattus norvegicus (Norway rat)0.0083
Sodium-dependent serotonin transporterHomo sapiens (human)0.8628
Sodium-dependent dopamine transporter Homo sapiens (human)1.65

Research

Studies (3)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's1 (33.33)29.6817
2010's2 (66.67)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Greenup, JL; Leverenz, JB; Peskind, ER; Raskind, MA; Szot, P; White, SS1
Beveridge, TJ; Nader, MA; Porrino, LJ; Smith, HR1
García-Fuster, MJ; García-Sevilla, JA1

Other Studies

3 other study(ies) available for rx 821002 and nisoxetine

ArticleYear
Compensatory changes in the noradrenergic nervous system in the locus ceruleus and hippocampus of postmortem subjects with Alzheimer's disease and dementia with Lewy bodies.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 2006, Jan-11, Volume: 26, Issue:2

    Topics: Adrenergic alpha-Antagonists; Adult; Aged; Aged, 80 and over; Alzheimer Disease; Dendrites; Female; Fluoxetine; Hippocampus; Humans; Idazoxan; In Situ Hybridization; Lewy Body Disease; Locus Coeruleus; Male; Middle Aged; Nerve Tissue Proteins; Norepinephrine; Norepinephrine Plasma Membrane Transport Proteins; Prazosin; Receptors, Adrenergic, alpha-1; Receptors, Adrenergic, alpha-2; RNA, Messenger; Tetralones; Tyrosine 3-Monooxygenase

2006
Effects of abstinence from chronic cocaine self-administration on nonhuman primate dorsal and ventral noradrenergic bundle terminal field structures.
    Brain structure & function, 2016, Volume: 221, Issue:5

    Topics: Adrenergic alpha-2 Receptor Antagonists; Animals; Autoradiography; Brain; Cocaine; Cocaine-Related Disorders; Fluoxetine; Idazoxan; Macaca mulatta; Male; Neural Pathways; Norepinephrine Plasma Membrane Transport Proteins; Receptors, Adrenergic, alpha-2; Reinforcement Schedule; Self Administration

2016
Effects of anti-depressant treatments on FADD and p-FADD protein in rat brain cortex: enhanced anti-apoptotic p-FADD/FADD ratio after chronic desipramine and fluoxetine administration.
    Psychopharmacology, 2016, Volume: 233, Issue:15-16

    Topics: Adrenergic alpha-Antagonists; Animals; Antidepressive Agents; Apoptosis; Autoreceptors; Blotting, Western; Brain; CASP8 and FADD-Like Apoptosis Regulating Protein; Cerebral Cortex; Clorgyline; Desipramine; Electroshock; Excitatory Amino Acid Antagonists; Fas-Associated Death Domain Protein; Fluoxetine; Idazoxan; Indans; Ketamine; Male; Mianserin; Mirtazapine; Monoamine Oxidase Inhibitors; Norepinephrine Plasma Membrane Transport Proteins; Phenelzine; Phosphoproteins; Phosphorylation; Rats; RNA-Binding Proteins; Thiazoles

2016