Page last updated: 2024-09-02

rx 821002 and guanfacine

rx 821002 has been researched along with guanfacine in 6 studies

Compound Research Comparison

Studies
(rx 821002)
Trials
(rx 821002)
Recent Studies (post-2010)
(rx 821002)
Studies
(guanfacine)
Trials
(guanfacine)
Recent Studies (post-2010) (guanfacine)
317045784180273

Protein Interaction Comparison

ProteinTaxonomyrx 821002 (IC50)guanfacine (IC50)
5-hydroxytryptamine receptor 4Cavia porcellus (domestic guinea pig)1.453
Alpha-2A adrenergic receptorHomo sapiens (human)0.134
Alpha-2B adrenergic receptorHomo sapiens (human)0.249
Alpha-2C adrenergic receptorHomo sapiens (human)6.447
5-hydroxytryptamine receptor 2AHomo sapiens (human)3.014
5-hydroxytryptamine receptor 2CHomo sapiens (human)1.453
5-hydroxytryptamine receptor 2BHomo sapiens (human)2.098

Research

Studies (6)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's3 (50.00)18.2507
2000's3 (50.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Uhlén, S; Wikberg, JE1
Intengan, HD; Smyth, DD1
Audinot, V; Chaput, C; Gavaudan, S; Millan, MJ; Newman-Tancredi, A; Nicolas, JP; Richard, N; Touzard, M; Verrièle, L1
Bisgard, GE; Herman, JK; O'Halloran, KD1
Dausse, JP; Giudicelli, Y; Ilhami, N; Khalid, M1
Angst, MJ; Fresquet, N; Gobaille, S; Sandner, G; Schleef, C1

Other Studies

6 other study(ies) available for rx 821002 and guanfacine

ArticleYear
Delineation of rat kidney alpha 2A- and alpha 2B-adrenoceptors with [3H]RX821002 radioligand binding: computer modelling reveals that guanfacine is an alpha 2A-selective compound.
    European journal of pharmacology, 1991, Sep-17, Volume: 202, Issue:2

    Topics: Animals; Computer Simulation; Dioxanes; Guanfacine; Idazoxan; In Vitro Techniques; Isoquinolines; Kidney; Male; Monte Carlo Method; Piperazines; Radioligand Assay; Rats; Rats, Inbred Strains; Receptors, Adrenergic, alpha

1991
Alpha-2a/d adrenoceptor subtype stimulation by guanfacine increases osmolar clearance.
    The Journal of pharmacology and experimental therapeutics, 1997, Volume: 281, Issue:1

    Topics: Adrenergic alpha-Agonists; Animals; Body Water; Brimonidine Tartrate; Guanfacine; Idazoxan; Kidney; Male; Naltrexone; Prazosin; Quinoxalines; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, alpha-2

1997
Actions of alpha2 adrenoceptor ligands at alpha2A and 5-HT1A receptors: the antagonist, atipamezole, and the agonist, dexmedetomidine, are highly selective for alpha2A adrenoceptors.
    Naunyn-Schmiedeberg's archives of pharmacology, 1998, Volume: 358, Issue:2

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Binding, Competitive; Brimonidine Tartrate; CHO Cells; Cricetinae; Guanfacine; Humans; Idazoxan; Imidazoles; Ligands; Medetomidine; Quinoxalines; Radioligand Assay; Rats; Receptors, Adrenergic, alpha-2; Receptors, Serotonin; Receptors, Serotonin, 5-HT1; Yohimbine

1998
Alpha2A-adrenoceptor mediated tachypnea in awake goats.
    Respiration physiology, 2001, Volume: 125, Issue:3

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Blood Pressure; Clonidine; Dose-Response Relationship, Drug; Female; Goats; Guanfacine; Heart Rate; Idazoxan; Periodicity; Receptors, Adrenergic, alpha-2; Respiratory Mechanics

2001
Testosterone dependence of salt-induced hypertension in Sabra rats and role of renal alpha(2)-adrenoceptor subtypes.
    The Journal of pharmacology and experimental therapeutics, 2002, Volume: 300, Issue:1

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Blood Pressure; Gene Expression Regulation; Guanfacine; Hypertension; Idazoxan; Kidney; Male; Orchiectomy; Prazosin; Rats; Receptors, Adrenergic, alpha-2; RNA, Messenger; Sodium Chloride; Testosterone

2002
Adrenergic drugs modify the level of noradrenaline in the insular cortex and alter extinction of conditioned taste aversion in rats.
    Behavioural brain research, 2007, Mar-12, Volume: 178, Issue:1

    Topics: Adrenergic Agents; Analysis of Variance; Animals; Avoidance Learning; Blood Glucose; Cerebral Cortex; Conditioning, Classical; Drinking Behavior; Extinction, Psychological; Guanfacine; Idazoxan; Male; Microdialysis; Norepinephrine; Rats; Rats, Long-Evans; Receptors, Adrenergic, alpha-2; Taste

2007