Page last updated: 2024-09-02

rx 821002 and fentanyl

rx 821002 has been researched along with fentanyl in 2 studies

Compound Research Comparison

Studies
(rx 821002)
Trials
(rx 821002)
Recent Studies (post-2010)
(rx 821002)
Studies
(fentanyl)
Trials
(fentanyl)
Recent Studies (post-2010) (fentanyl)
31704515,2884,3104,483

Protein Interaction Comparison

ProteinTaxonomyrx 821002 (IC50)fentanyl (IC50)
ATP-dependent translocase ABCB1Homo sapiens (human)6.5
Delta-type opioid receptorMus musculus (house mouse)0.6342
Delta-type opioid receptorRattus norvegicus (Norway rat)0.0122
Mu-type opioid receptorRattus norvegicus (Norway rat)0.1888
Kappa-type opioid receptorRattus norvegicus (Norway rat)0.0122
Mu-type opioid receptorHomo sapiens (human)0.0058
Delta-type opioid receptorHomo sapiens (human)0.3092
Kappa-type opioid receptorCavia porcellus (domestic guinea pig)5.893
Kappa-type opioid receptorHomo sapiens (human)1.58
Mu-type opioid receptorCavia porcellus (domestic guinea pig)0.0031
Potassium voltage-gated channel subfamily H member 2Homo sapiens (human)1.8197
Sigma non-opioid intracellular receptor 1Cavia porcellus (domestic guinea pig)4.973
Sigma non-opioid intracellular receptor 1Homo sapiens (human)0.354

Research

Studies (2)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's1 (50.00)18.2507
2000's1 (50.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Clarke, RW; Houghton, AK; Ogilvie, J; Parry-Baggott, C1
Clarke, RW; Ward, RE1

Other Studies

2 other study(ies) available for rx 821002 and fentanyl

ArticleYear
The involvement of bulbospinal pathways in fentanyl-induced inhibition of spinal withdrawal reflexes in the decerebrated rabbit.
    Pain, 1998, Volume: 78, Issue:3

    Topics: Adrenergic alpha-Antagonists; Analgesics, Opioid; Animals; Decerebrate State; Dose-Response Relationship, Drug; Electric Stimulation; Female; Fentanyl; Idazoxan; Injections, Intravenous; Injections, Intraventricular; Injections, Spinal; Male; Medulla Oblongata; Neural Inhibition; Neural Pathways; Rabbits; Reflex; Spinal Cord; Sural Nerve

1998
The role of 5-HT(1A)-receptors in fentanyl-induced bulbospinal inhibition of a spinal withdrawal reflex in the rabbit.
    Pain, 2000, Volume: 85, Issue:1-2

    Topics: Adrenergic alpha-Antagonists; Analgesics, Opioid; Animals; Dose-Response Relationship, Drug; Electrocardiography; Female; Fentanyl; Idazoxan; Injections, Intravenous; Injections, Intraventricular; Male; Piperazines; Pyridines; Rabbits; Receptors, Serotonin; Receptors, Serotonin, 5-HT1; Reflex; Serotonin Antagonists; Spinal Cord

2000