Page last updated: 2024-09-02

rx 821002 and dextroamphetamine

rx 821002 has been researched along with dextroamphetamine in 3 studies

Compound Research Comparison

Studies
(rx 821002)
Trials
(rx 821002)
Recent Studies (post-2010)
(rx 821002)
Studies
(dextroamphetamine)
Trials
(dextroamphetamine)
Recent Studies (post-2010) (dextroamphetamine)
3170457,044697660

Protein Interaction Comparison

ProteinTaxonomyrx 821002 (IC50)dextroamphetamine (IC50)
Sodium-dependent noradrenaline transporter Homo sapiens (human)0.631
Sodium-dependent dopamine transporter Homo sapiens (human)0.2884

Research

Studies (3)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's1 (33.33)18.2507
2000's2 (66.67)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Heal, DJ; Hughes, ZA; Stanford, SC; Wortley, KE1
Hudson, AL; Hume, SP; Lalies, MD; Nutt, DJ; Robinson, ES; Tyacke, RJ1
Schmidt, WJ; Srinivasan, J1

Other Studies

3 other study(ies) available for rx 821002 and dextroamphetamine

ArticleYear
Comparison of changes in the extracellular concentration of noradrenaline in rat frontal cortex induced by sibutramine or d-amphetamine: modulation by alpha2-adrenoceptors.
    British journal of pharmacology, 1999, Volume: 127, Issue:8

    Topics: Adrenergic alpha-Antagonists; Animals; Appetite Depressants; Cerebral Cortex; Cyclobutanes; Dextroamphetamine; Idazoxan; Male; Norepinephrine; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, alpha-2

1999
Estimation of endogenous noradrenaline release in rat brain in vivo using [3H]RX 821002.
    Synapse (New York, N.Y.), 2005, Volume: 55, Issue:2

    Topics: Adrenergic alpha-Antagonists; Adrenergic Uptake Inhibitors; Animals; Binding, Competitive; Brain; Dextroamphetamine; Idazoxan; Imidazoles; Male; Microdialysis; Monoamine Oxidase Inhibitors; Norepinephrine; Radioligand Assay; Rats; Rats, Wistar; Selegiline; Time Factors; Tissue Distribution; Tritium

2005
Serotonergic influence on the potentiation of D-amphetamine and apomorphine-induced rotational behavior by the alpha2-adrenoceptor antagonist 2-methoxy idazoxan in hemiparkinsonian rats.
    Journal of neural transmission (Vienna, Austria : 1996), 2005, Volume: 112, Issue:9

    Topics: Adrenergic Agents; Adrenergic alpha-2 Receptor Antagonists; Adrenergic alpha-Antagonists; Animals; Antiparkinson Agents; Apomorphine; Behavior, Animal; Dextroamphetamine; Drug Synergism; Idazoxan; Male; Motor Activity; Oxidopamine; Parkinsonian Disorders; Rats; Rats, Sprague-Dawley; Serotonin; Sympatholytics

2005