Page last updated: 2024-09-02

rx 821002 and clorgyline

rx 821002 has been researched along with clorgyline in 4 studies

Compound Research Comparison

Studies
(rx 821002)
Trials
(rx 821002)
Recent Studies (post-2010)
(rx 821002)
Studies
(clorgyline)
Trials
(clorgyline)
Recent Studies (post-2010) (clorgyline)
3170451,07523170

Protein Interaction Comparison

ProteinTaxonomyrx 821002 (IC50)clorgyline (IC50)
Amine oxidase [flavin-containing] BRattus norvegicus (Norway rat)0.8602
Amine oxidase [flavin-containing] A Rattus norvegicus (Norway rat)0.5688
Amine oxidase [flavin-containing] AHomo sapiens (human)0.2574
Amine oxidase [flavin-containing] A Bos taurus (cattle)0.0032
Amine oxidase [flavin-containing] BHomo sapiens (human)3.6869

Research

Studies (4)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's2 (50.00)18.2507
2000's1 (25.00)29.6817
2010's1 (25.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
García-Sevilla, JA; Miralles, A; Ribas, C1
Callado, LF; Gabilondo, AM; Meana, JJ1
Clarke, RW; Harris, J; Ogilvie, J1
García-Fuster, MJ; García-Sevilla, JA1

Other Studies

4 other study(ies) available for rx 821002 and clorgyline

ArticleYear
Acceleration by chronic treatment with clorgyline of the turnover of brain alpha 2-adrenoceptors in normotensive but not in spontaneously hypertensive rats.
    British journal of pharmacology, 1993, Volume: 110, Issue:1

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Brain Chemistry; Brimonidine Tartrate; Cerebral Cortex; Clorgyline; Dioxanes; Down-Regulation; Hypertension; Idazoxan; In Vitro Techniques; Kinetics; Male; Membranes; Quinolines; Quinoxalines; Rats; Rats, Inbred SHR; Rats, Inbred WKY; Rats, Sprague-Dawley; Receptors, Adrenergic, alpha-2; Species Specificity

1993
Differential modulation of alpha2-adrenoceptor subtypes in rat kidney by chronic desipramine treatment.
    Life sciences, 1999, Volume: 64, Issue:25

    Topics: Adrenergic alpha-Antagonists; Adrenergic Uptake Inhibitors; Animals; Binding, Competitive; Clorgyline; Desipramine; Epinephrine; Idazoxan; Imidazoles; In Vitro Techniques; Indoles; Isoindoles; Isoquinolines; Kidney; Kinetics; Male; Monoamine Oxidase Inhibitors; Piperazines; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, alpha-2

1999
Imidazoline I(2)-receptors and spinal reflexes in the decerebrated rabbit.
    Neuropharmacology, 2000, Jul-24, Volume: 39, Issue:10

    Topics: Adrenergic alpha-Antagonists; Animals; Blood Pressure; Clorgyline; Decerebrate State; Dose-Response Relationship, Drug; Female; Heart Rate; Idazoxan; Imidazoles; Imidazoline Receptors; Indoles; Injections, Spinal; Isoindoles; Ligands; Male; Monoamine Oxidase Inhibitors; Pargyline; Rabbits; Receptors, Drug; Reflex; Spinal Cord

2000
Effects of anti-depressant treatments on FADD and p-FADD protein in rat brain cortex: enhanced anti-apoptotic p-FADD/FADD ratio after chronic desipramine and fluoxetine administration.
    Psychopharmacology, 2016, Volume: 233, Issue:15-16

    Topics: Adrenergic alpha-Antagonists; Animals; Antidepressive Agents; Apoptosis; Autoreceptors; Blotting, Western; Brain; CASP8 and FADD-Like Apoptosis Regulating Protein; Cerebral Cortex; Clorgyline; Desipramine; Electroshock; Excitatory Amino Acid Antagonists; Fas-Associated Death Domain Protein; Fluoxetine; Idazoxan; Indans; Ketamine; Male; Mianserin; Mirtazapine; Monoamine Oxidase Inhibitors; Norepinephrine Plasma Membrane Transport Proteins; Phenelzine; Phosphoproteins; Phosphorylation; Rats; RNA-Binding Proteins; Thiazoles

2016