rx 821002 has been researched along with benextramine in 1 studies
Studies (rx 821002) | Trials (rx 821002) | Recent Studies (post-2010) (rx 821002) | Studies (benextramine) | Trials (benextramine) | Recent Studies (post-2010) (benextramine) |
---|---|---|---|---|---|
317 | 0 | 45 | 84 | 0 | 3 |
Protein | Taxonomy | rx 821002 (IC50) | benextramine (IC50) |
---|---|---|---|
Cholinesterase | Homo sapiens (human) | 6.1659 | |
Alpha-1B adrenergic receptor | Rattus norvegicus (Norway rat) | 4.02 | |
Alpha-2B adrenergic receptor | Rattus norvegicus (Norway rat) | 4.02 | |
Alpha-2C adrenergic receptor | Rattus norvegicus (Norway rat) | 4.02 | |
Acetylcholinesterase | Homo sapiens (human) | 7.2429 | |
Alpha-2A adrenergic receptor | Rattus norvegicus (Norway rat) | 4.02 | |
Alpha-1D adrenergic receptor | Rattus norvegicus (Norway rat) | 4.02 | |
Adenosine receptor A2a | Rattus norvegicus (Norway rat) | 4.02 | |
Alpha-1A adrenergic receptor | Rattus norvegicus (Norway rat) | 4.02 | |
Carboxylic ester hydrolase | Rattus norvegicus (Norway rat) | 6.1659 |
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 0 (0.00) | 18.7374 |
1990's | 1 (100.00) | 18.2507 |
2000's | 0 (0.00) | 29.6817 |
2010's | 0 (0.00) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
---|---|
Lafontan, M; Langin, D; Paris, H | 1 |
1 other study(ies) available for rx 821002 and benextramine
Article | Year |
---|---|
Binding of [3H]idazoxan and of its methoxy derivative [3H] RX821002 in human fat cells: [3H]idazoxan but not [3H] RX821002 labels additional non-alpha 2-adrenergic binding sites.
Topics: Adipose Tissue; Adrenergic alpha-Antagonists; Binding Sites; Brimonidine Tartrate; Cell Membrane; Cystamine; Dioxanes; Dioxins; Epinephrine; Female; Humans; Idazoxan; Magnesium Chloride; Phenoxybenzamine; Potassium Chloride; Quinoxalines; Tritium; Yohimbine | 1990 |