Page last updated: 2024-09-02

rx 821002 and benextramine

rx 821002 has been researched along with benextramine in 1 studies

Compound Research Comparison

Studies
(rx 821002)
Trials
(rx 821002)
Recent Studies (post-2010)
(rx 821002)
Studies
(benextramine)
Trials
(benextramine)
Recent Studies (post-2010) (benextramine)
3170458403

Protein Interaction Comparison

ProteinTaxonomyrx 821002 (IC50)benextramine (IC50)
CholinesteraseHomo sapiens (human)6.1659
Alpha-1B adrenergic receptorRattus norvegicus (Norway rat)4.02
Alpha-2B adrenergic receptorRattus norvegicus (Norway rat)4.02
Alpha-2C adrenergic receptorRattus norvegicus (Norway rat)4.02
AcetylcholinesteraseHomo sapiens (human)7.2429
Alpha-2A adrenergic receptorRattus norvegicus (Norway rat)4.02
Alpha-1D adrenergic receptorRattus norvegicus (Norway rat)4.02
Adenosine receptor A2aRattus norvegicus (Norway rat)4.02
Alpha-1A adrenergic receptorRattus norvegicus (Norway rat)4.02
Carboxylic ester hydrolase Rattus norvegicus (Norway rat)6.1659

Research

Studies (1)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's1 (100.00)18.2507
2000's0 (0.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Lafontan, M; Langin, D; Paris, H1

Other Studies

1 other study(ies) available for rx 821002 and benextramine

ArticleYear
Binding of [3H]idazoxan and of its methoxy derivative [3H] RX821002 in human fat cells: [3H]idazoxan but not [3H] RX821002 labels additional non-alpha 2-adrenergic binding sites.
    Molecular pharmacology, 1990, Volume: 37, Issue:6

    Topics: Adipose Tissue; Adrenergic alpha-Antagonists; Binding Sites; Brimonidine Tartrate; Cell Membrane; Cystamine; Dioxanes; Dioxins; Epinephrine; Female; Humans; Idazoxan; Magnesium Chloride; Phenoxybenzamine; Potassium Chloride; Quinoxalines; Tritium; Yohimbine

1990