Page last updated: 2024-09-02

rx 821002 and apraclonidine

rx 821002 has been researched along with apraclonidine in 3 studies

Compound Research Comparison

Studies
(rx 821002)
Trials
(rx 821002)
Recent Studies (post-2010)
(rx 821002)
Studies
(apraclonidine)
Trials
(apraclonidine)
Recent Studies (post-2010) (apraclonidine)
3170454279856

Protein Interaction Comparison

ProteinTaxonomyrx 821002 (IC50)apraclonidine (IC50)
Alpha-2A adrenergic receptorHomo sapiens (human)0.004
Alpha-2B adrenergic receptorHomo sapiens (human)0.004
Alpha-2C adrenergic receptorHomo sapiens (human)0.004

Research

Studies (3)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's3 (100.00)18.2507
2000's0 (0.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Evans, RG; Haynes, JM1
Escribá, PV; García-Sevilla, JA; Regunathan, S; Reis, DJ; Sastre, M; Wang, H1
Fukazawa, H; Ishida, H; Koda, H; Kuriyama, K; Matsumoto, N; Nukaya, H; Suwa, Y; Tsuji, K; Yokoo, Y1

Other Studies

3 other study(ies) available for rx 821002 and apraclonidine

ArticleYear
Characterization of binding sites for [3H]-idazoxan, [3H]-P-aminoclonidine and [3H]-rauwolscine in the kidney of the dog.
    Clinical and experimental pharmacology & physiology, 1994, Volume: 21, Issue:8

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Binding Sites; Binding, Competitive; Clonidine; Dioxanes; Dogs; GTP-Binding Proteins; Idazoxan; Imidazoline Receptors; Kidney; Male; Radioligand Assay; Receptors, Drug; Yohimbine

1994
Immunodetection of putative imidazoline receptor proteins in the human and rat brain and other tissues.
    Neuroscience letters, 1994, Aug-29, Volume: 178, Issue:1

    Topics: Adrenal Medulla; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Autoradiography; Brain Chemistry; Chromatography, Affinity; Clonidine; Dioxanes; Electrophoresis, Polyacrylamide Gel; Humans; Idazoxan; Imidazoline Receptors; Immunoblotting; Liver; Male; Medulla Oblongata; Rats; Rats, Sprague-Dawley; Receptors, Drug; Tritium

1994
Antagonistic effect of N-methyltyramine on alpha2-adrenoceptor in mice.
    Japanese journal of pharmacology, 1999, Volume: 81, Issue:3

    Topics: Adrenergic alpha-2 Receptor Antagonists; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Clonidine; Idazoxan; Male; Mice; Radioligand Assay; Receptors, Adrenergic, alpha-2; Scopolamine; Tyramine

1999