Page last updated: 2024-09-04

ruboxistaurin and pd 98059

ruboxistaurin has been researched along with pd 98059 in 3 studies

Compound Research Comparison

Studies
(ruboxistaurin)
Trials
(ruboxistaurin)
Recent Studies (post-2010)
(ruboxistaurin)
Studies
(pd 98059)
Trials
(pd 98059)
Recent Studies (post-2010) (pd 98059)
20329564,93931,001

Protein Interaction Comparison

ProteinTaxonomyruboxistaurin (IC50)pd 98059 (IC50)
RAF proto-oncogene serine/threonine-protein kinaseHomo sapiens (human)2.8
Luciferin 4-monooxygenasePhotinus pyralis (common eastern firefly)6.3
Amine oxidase [flavin-containing] BRattus norvegicus (Norway rat)2.8
Prostaglandin G/H synthase 1Homo sapiens (human)1
Mitogen-activated protein kinase 1Homo sapiens (human)2.8
Dual specificity mitogen-activated protein kinase kinase 2 Rattus norvegicus (Norway rat)4.2
Dual specificity mitogen-activated protein kinase kinase 1 Rattus norvegicus (Norway rat)4.2
Dual specificity mitogen-activated protein kinase kinase 1Homo sapiens (human)2.4

Research

Studies (3)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's3 (100.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Bullock, AN; Fedorov, O; Knapp, S; Marsden, B; Müller, S; Pogacic, V; Rellos, P; Schwaller, J; Sundström, M1
Chou, E; Gabriele, A; Ha, SW; King, GL; Meier, M; Naruse, K; Park, JY; Rhodes, CJ; Suzuma, K; Takahara, N; Yamauchi, T1
Andrassy, M; Belov, D; Harja, E; Katus, HA; Leitges, M; Nawroth, PP; Schmidt, AM; Yan, SD; Yan, SF; Zou, YS1

Other Studies

3 other study(ies) available for ruboxistaurin and pd 98059

ArticleYear
A systematic interaction map of validated kinase inhibitors with Ser/Thr kinases.
    Proceedings of the National Academy of Sciences of the United States of America, 2007, Dec-18, Volume: 104, Issue:51

    Topics: Amino Acid Sequence; Binding Sites; Clinical Trials as Topic; Drug Evaluation, Preclinical; Enzyme Stability; Humans; Molecular Sequence Data; Phylogeny; Protein Array Analysis; Protein Conformation; Protein Kinase Inhibitors; Protein Serine-Threonine Kinases

2007
Induction of endothelin-1 expression by glucose: an effect of protein kinase C activation.
    Diabetes, 2000, Volume: 49, Issue:7

    Topics: Animals; Capillaries; Cattle; Cells, Cultured; Endothelin-1; Endothelium, Vascular; Enzyme Activation; Enzyme Inhibitors; Flavonoids; Gene Expression Regulation; Glucose; Indoles; Isoenzymes; Maleimides; Pericytes; Protein Kinase C; Protein Kinase C beta; Protein Kinase C-alpha; Protein Kinase C-delta; Retinal Vessels; RNA, Messenger; Transcription, Genetic

2000
Central role of PKCbeta in neointimal expansion triggered by acute arterial injury.
    Circulation research, 2005, Mar-04, Volume: 96, Issue:4

    Topics: Animals; Aorta; Blood Glucose; Cell Division; Cell Movement; Cells, Cultured; Constriction, Pathologic; DNA-Binding Proteins; Early Growth Response Protein 1; Enzyme Activation; Femoral Artery; Flavonoids; Humans; Immediate-Early Proteins; Indoles; Janus Kinase 2; JNK Mitogen-Activated Protein Kinases; Maleimides; Mesylates; Mice; Mice, Inbred C57BL; Mice, Knockout; Mitogen-Activated Protein Kinase 1; Mitogen-Activated Protein Kinase 3; Muscle, Smooth, Vascular; Myocytes, Smooth Muscle; Oxidative Stress; Peroxidase; Protein Kinase C; Protein Kinase C beta; Protein-Tyrosine Kinases; Proto-Oncogene Proteins; Pyrroles; Signal Transduction; STAT3 Transcription Factor; Tetradecanoylphorbol Acetate; Trans-Activators; Transcription Factors; Tunica Intima

2005