Page last updated: 2024-09-04

ru 58841 and cyproterone acetate

ru 58841 has been researched along with cyproterone acetate in 3 studies

Compound Research Comparison

Studies
(ru 58841)
Trials
(ru 58841)
Recent Studies (post-2010)
(ru 58841)
Studies
(cyproterone acetate)
Trials
(cyproterone acetate)
Recent Studies (post-2010) (cyproterone acetate)
25041,845339261

Protein Interaction Comparison

ProteinTaxonomyru 58841 (IC50)cyproterone acetate (IC50)
Glucocorticoid receptorHomo sapiens (human)0.225
Glycine receptor subunit alpha-1Rattus norvegicus (Norway rat)0.225
Androgen receptorHomo sapiens (human)0.1408
Androgen receptorRattus norvegicus (Norway rat)0.339
Glycine receptor subunit betaRattus norvegicus (Norway rat)0.225
Glycine receptor subunit alpha-2Rattus norvegicus (Norway rat)0.225
Glycine receptor subunit alpha-3Rattus norvegicus (Norway rat)0.225
Adenosine receptor A1Rattus norvegicus (Norway rat)0.045
Mu-type opioid receptorHomo sapiens (human)2.183

Research

Studies (3)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's2 (66.67)18.2507
2000's1 (33.33)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Gaillard, M; Matias, JR1
Chang, C; Miyamoto, H; Wilding, G; Yeh, S1
Blaschke, T; Kleuser, B; Korting, HC; Kramer, KD; Mehnert, W; Schäfer-Korting, M; Seltmann, H; Sivaramakrishnan, R; Stecová, J; Zouboulis, CC1

Other Studies

3 other study(ies) available for ru 58841 and cyproterone acetate

ArticleYear
Local inhibition of sebaceous gland growth by topically applied RU 58841.
    Annals of the New York Academy of Sciences, 1995, Jun-12, Volume: 761

    Topics: Administration, Topical; Androgen Antagonists; Animals; Cricetinae; Cyproterone Acetate; Ear; Imidazoles; Indenes; Male; Mesocricetus; Models, Biological; Nitriles; Sebaceous Glands; Structure-Activity Relationship; Time Factors

1995
Promotion of agonist activity of antiandrogens by the androgen receptor coactivator, ARA70, in human prostate cancer DU145 cells.
    Proceedings of the National Academy of Sciences of the United States of America, 1998, Jun-23, Volume: 95, Issue:13

    Topics: Androgen Antagonists; Androgens; Anilides; Cyproterone Acetate; Drug Interactions; Flutamide; Humans; Imidazoles; Male; Mifepristone; Nitriles; Nuclear Receptor Coactivators; Oncogene Proteins; Prostatic Neoplasms; Protein Binding; Protein Conformation; Tosyl Compounds; Trans-Activators; Transcription Factors; Transcriptional Activation; Tumor Cells, Cultured

1998
Cyproterone acetate loading to lipid nanoparticles for topical acne treatment: particle characterisation and skin uptake.
    Pharmaceutical research, 2007, Volume: 24, Issue:5

    Topics: Acne Vulgaris; Administration, Cutaneous; Androgen Antagonists; Cell Proliferation; Cell Survival; Cells, Cultured; Cyproterone Acetate; Drug Compounding; Drug Stability; Drug Storage; Fibroblasts; Gene Expression; Humans; Imidazoles; In Vitro Techniques; Keratinocytes; Lipids; Microspheres; Nanoparticles; Nitriles; Particle Size; Receptors, Androgen; Reverse Transcriptase Polymerase Chain Reaction; Skin; Temperature; Time Factors

2007