Page last updated: 2024-09-03

ru 24926 and sulpiride

ru 24926 has been researched along with sulpiride in 10 studies

Compound Research Comparison

Studies
(ru 24926)
Trials
(ru 24926)
Recent Studies (post-2010)
(ru 24926)
Studies
(sulpiride)
Trials
(sulpiride)
Recent Studies (post-2010) (sulpiride)
30004,152427635

Protein Interaction Comparison

ProteinTaxonomyru 24926 (IC50)sulpiride (IC50)
Carbonic anhydrase 1Homo sapiens (human)1.2
Carbonic anhydrase 2Homo sapiens (human)0.04
Alpha-2A adrenergic receptorHomo sapiens (human)2.019
D(2) dopamine receptorHomo sapiens (human)0.0858
D(3) dopamine receptorHomo sapiens (human)0.2651
D(2) dopamine receptorRattus norvegicus (Norway rat)0.2215
Carbonic anhydrase 4Bos taurus (cattle)0.62
D(2) dopamine receptorCanis lupus familiaris (dog)0.2

Research

Studies (10)

TimeframeStudies, this research(%)All Research%
pre-19905 (50.00)18.7374
1990's5 (50.00)18.2507
2000's0 (0.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Azzaro, AJ; Harrison-Shahan, Y; Johnson, EA; Lucci, J; Tsai, CE1
Besson, MJ; Penit-Soria, J; Rétaux, S1
Costentin, J; Duterte-Boucher, D; Ladurelle, N1
Costentin, J; Duterte-Boucher, D; Michael-Titus, A; Panissaud, C1
Bousselmame, R; Costentin, J; Michael-Titus, A1
Maurin, Y; Penit-Soria, J; Retaux, S1
Martres, MP; Riou, JF; Schwartz, JC; Sokoloff, P1
Protais, P; Vasse, M1
Conzelmann, U; Holland, A; Meyer, DK1
Bockaert, J; Enjalbert, A1

Other Studies

10 other study(ies) available for ru 24926 and sulpiride

ArticleYear
Dopamine D2 synthesis-modulating receptors are present in the striatum of the guinea pig.
    Neuropharmacology, 1992, Volume: 31, Issue:1

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Benzazepines; Corpus Striatum; Guinea Pigs; In Vitro Techniques; Phenethylamines; Rats; Receptors, Dopamine; Receptors, Dopamine D1; Receptors, Dopamine D2; Sulpiride; Synaptosomes; Tyrosine 3-Monooxygenase

1992
Opposing effects of dopamine D2 receptor stimulation on the spontaneous and the electrically evoked release of [3H]GABA on rat prefrontal cortex slices.
    Neuroscience, 1991, Volume: 42, Issue:1

    Topics: Amphetamine; Animals; Calcium; Cerebral Cortex; Dopamine Agents; Electric Stimulation; Ergolines; Frontal Lobe; gamma-Aminobutyric Acid; In Vitro Techniques; Interneurons; Lisuride; Male; Phenethylamines; Quinpirole; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Dopamine D2; Sulpiride

1991
Stimulation of D1 and D2 dopamine receptors produces additive anorectic effects.
    Fundamental & clinical pharmacology, 1991, Volume: 5, Issue:6

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Analysis of Variance; Animals; Anorexia; Apomorphine; Dopamine Agents; Dose-Response Relationship, Drug; Drug Interactions; Feeding Behavior; Male; Mice; Phenethylamines; Receptors, Dopamine; Receptors, Dopamine D1; Receptors, Dopamine D2; Sulpiride

1991
Dopamine D1 and D2 receptors mediate opposite effects of apomorphine on the body temperature of reserpinized mice.
    Neuropharmacology, 1990, Volume: 29, Issue:1

    Topics: Animals; Apomorphine; Benzazepines; Body Temperature; Dopamine Agents; Dose-Response Relationship, Drug; Male; Mice; Phenethylamines; Receptors, Dopamine; Reserpine; Sulpiride

1990
Stimulation of dopamine D2 receptors induces an analgesia involving an opioidergic but non enkephalinergic link.
    European journal of pharmacology, 1990, Oct-09, Volume: 187, Issue:2

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Analgesia; Animals; Apomorphine; Benzazepines; Endorphins; Enkephalin, Leucine; Enkephalins; Injections, Intraventricular; Male; Mice; Narcotic Antagonists; Pain Measurement; Phenethylamines; Reaction Time; Receptors, Dopamine; Receptors, Opioid; Receptors, Opioid, mu; Sulpiride

1990
[Effects of the stimulation of D1 and D2 dopaminergic receptors on the electrically induced release of gamma-(3H)-aminobutyric acid in the prefrontal cortex of the rat].
    Comptes rendus de l'Academie des sciences. Serie III, Sciences de la vie, 1989, Volume: 309, Issue:10

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Electric Stimulation; Frontal Lobe; gamma-Aminobutyric Acid; In Vitro Techniques; Lisuride; Phenethylamines; Rats; Receptors, Dopamine; Sulpiride

1989
Presence of dopamine D-2 receptors in human tumoral cell lines.
    Biochemical and biophysical research communications, 1989, Jul-31, Volume: 162, Issue:2

    Topics: Apomorphine; Breast Neoplasms; Cell Membrane; Digestive System Neoplasms; Dopamine; Humans; Iodine Radioisotopes; Leukemia; Lung Neoplasms; Neoplasms; Neuroblastoma; Phenethylamines; Receptors, Dopamine; Receptors, Dopamine D2; Sulpiride; Tumor Cells, Cultured

1989
Potentiation of apomorphine-induced stereotyped behaviour by acute treatment with dopamine depleting agents: a potential role for an increased stimulation of D1 dopamine receptors.
    Neuropharmacology, 1989, Volume: 28, Issue:9

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Adenylyl Cyclases; alpha-Methyltyrosine; Amisulpride; Animals; Apomorphine; Corpus Striatum; Cyclic AMP; Dopamine Antagonists; Drug Synergism; In Vitro Techniques; Male; Methyltyrosines; Metoclopramide; Mice; Phenethylamines; Rats; Rats, Inbred Strains; Receptors, Dopamine; Reserpine; Stereotyped Behavior; Sulpiride

1989
Effects of selective dopamine D2-receptor agonists on the release of cholecystokinin-like immunoreactivity from rat neostriatum.
    European journal of pharmacology, 1984, May-18, Volume: 101, Issue:1-2

    Topics: Animals; Caudate Nucleus; Cholecystokinin; Domperidone; Ergolines; Female; In Vitro Techniques; Phenethylamines; Potassium; Putamen; Quinpirole; Radioimmunoassay; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Dopamine D2; Sulpiride

1984
Pharmacological characterization of the D2 dopamine receptor negatively coupled with adenylate cyclase in rat anterior pituitary.
    Molecular pharmacology, 1983, Volume: 23, Issue:3

    Topics: Adenylyl Cyclases; Animals; Binding, Competitive; Cyclic AMP; Dopamine; Female; Kinetics; Male; Phenethylamines; Pituitary Gland, Anterior; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Dopamine D2; Sulpiride; Vasoactive Intestinal Peptide

1983