Page last updated: 2024-09-03

ru 24926 and sk&f-38393

ru 24926 has been researched along with sk&f-38393 in 13 studies

Compound Research Comparison

Studies
(ru 24926)
Trials
(ru 24926)
Recent Studies (post-2010)
(ru 24926)
Studies
(sk&f-38393)
Trials
(sk&f-38393)
Recent Studies (post-2010) (sk&f-38393)
30002,01229242

Protein Interaction Comparison

ProteinTaxonomyru 24926 (IC50)sk&f-38393 (IC50)
Replicase polyprotein 1abSevere acute respiratory syndrome coronavirus 22.8
DRattus norvegicus (Norway rat)0.19

Research

Studies (13)

TimeframeStudies, this research(%)All Research%
pre-19906 (46.15)18.7374
1990's7 (53.85)18.2507
2000's0 (0.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Azzaro, AJ; Harrison-Shahan, Y; Johnson, EA; Lucci, J; Tsai, CE1
Bousselmame, R; Costentin, J; Suaudeau, C1
Costentin, J; Duterte-Boucher, D; Ladurelle, N1
Charpentier, S; Costentin, J; Simon, P1
Besson, MJ; Penit-Soria, J; Retaux, S2
Bousselmame, R; Costentin, J; Michael-Titus, A1
Kelly, E; Nahorski, SR1
Maurin, Y; Penit-Soria, J; Retaux, S1
Protais, P; Vasse, M1
Bergstrom, DA; Braun, AR; Carlson, JH; Chase, TN; Walters, JR1
Besson, MJ; Girault, JA; Glowinski, J; Savaki, HE; Spampinato, U1
Gibb, JW; Hanson, GR; Sonsalla, PK1

Other Studies

13 other study(ies) available for ru 24926 and sk&f-38393

ArticleYear
Dopamine D2 synthesis-modulating receptors are present in the striatum of the guinea pig.
    Neuropharmacology, 1992, Volume: 31, Issue:1

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Benzazepines; Corpus Striatum; Guinea Pigs; In Vitro Techniques; Phenethylamines; Rats; Receptors, Dopamine; Receptors, Dopamine D1; Receptors, Dopamine D2; Sulpiride; Synaptosomes; Tyrosine 3-Monooxygenase

1992
A different balance in the sensitivity of D1 and D2 dopamine receptors accounts for differences in apomorphine-induced hypothermic effects in Swiss and C3H mice.
    Neuropharmacology, 1992, Volume: 31, Issue:11

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Apomorphine; Body Temperature; Male; Mice; Mice, Inbred BALB C; Mice, Inbred C3H; Mice, Inbred C57BL; Mice, Inbred DBA; Phenethylamines; Piribedil; Receptors, Dopamine D1; Receptors, Dopamine D2; Species Specificity

1992
Stimulation of D1 and D2 dopamine receptors produces additive anorectic effects.
    Fundamental & clinical pharmacology, 1991, Volume: 5, Issue:6

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Analysis of Variance; Animals; Anorexia; Apomorphine; Dopamine Agents; Dose-Response Relationship, Drug; Drug Interactions; Feeding Behavior; Male; Mice; Phenethylamines; Receptors, Dopamine; Receptors, Dopamine D1; Receptors, Dopamine D2; Sulpiride

1991
An automated method for the assessment of spontaneous and stereotyped climbing behavior in mice. Effects of the selective D1- and D2-dopamine receptor agonists SKF-38393 and RU-24926 and their association.
    Methods and findings in experimental and clinical pharmacology, 1991, Volume: 13, Issue:2

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Apomorphine; Behavior, Animal; Male; Mice; Motor Activity; Phenethylamines; Psychology, Experimental; Receptors, Dopamine; Receptors, Dopamine D1; Receptors, Dopamine D2; Stereotyped Behavior; Videotape Recording

1991
Synergism between D1 and D2 dopamine receptors in the inhibition of the evoked release of [3H]GABA in the rat prefrontal cortex.
    Neuroscience, 1991, Volume: 43, Issue:2-3

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Benzazepines; Electric Stimulation; Frontal Lobe; GABA Antagonists; Male; Phenethylamines; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Dopamine D1; Receptors, Dopamine D2; Reserpine; Tritium

1991
[D2 dopaminergic receptor activation enhances the spontaneous release of 3H-GABA in the prefrontal cortex of rats, in vitro. The facilitating role of D1 dopaminergic receptors].
    Comptes rendus de l'Academie des sciences. Serie III, Sciences de la vie, 1990, Volume: 311, Issue:8

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Cerebral Cortex; Dopamine Agents; Drug Interactions; Ergolines; gamma-Aminobutyric Acid; In Vitro Techniques; Lisuride; Phenethylamines; Quinpirole; Rats; Stimulation, Chemical

1990
Stimulation of dopamine D2 receptors induces an analgesia involving an opioidergic but non enkephalinergic link.
    European journal of pharmacology, 1990, Oct-09, Volume: 187, Issue:2

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Analgesia; Animals; Apomorphine; Benzazepines; Endorphins; Enkephalin, Leucine; Enkephalins; Injections, Intraventricular; Male; Mice; Narcotic Antagonists; Pain Measurement; Phenethylamines; Reaction Time; Receptors, Dopamine; Receptors, Opioid; Receptors, Opioid, mu; Sulpiride

1990
Specific inhibition of dopamine D-1-mediated cyclic AMP formation by dopamine D-2, muscarinic cholinergic, and opiate receptor stimulation in rat striatal slices.
    Journal of neurochemistry, 1986, Volume: 47, Issue:5

    Topics: 1-Methyl-3-isobutylxanthine; 2-Chloroadenosine; 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Adenosine; Alprostadil; Animals; Benzazepines; Carbachol; Cholera Toxin; Corpus Striatum; Cyclic AMP; Isoproterenol; Morphine; Phenethylamines; Rats; Receptors, Cholinergic; Receptors, Dopamine; Receptors, Muscarinic; Receptors, Opioid; Vasoactive Intestinal Peptide

1986
[Effects of the stimulation of D1 and D2 dopaminergic receptors on the electrically induced release of gamma-(3H)-aminobutyric acid in the prefrontal cortex of the rat].
    Comptes rendus de l'Academie des sciences. Serie III, Sciences de la vie, 1989, Volume: 309, Issue:10

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Electric Stimulation; Frontal Lobe; gamma-Aminobutyric Acid; In Vitro Techniques; Lisuride; Phenethylamines; Rats; Receptors, Dopamine; Sulpiride

1989
Potentiation of apomorphine-induced stereotyped behaviour by acute treatment with dopamine depleting agents: a potential role for an increased stimulation of D1 dopamine receptors.
    Neuropharmacology, 1989, Volume: 28, Issue:9

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Adenylyl Cyclases; alpha-Methyltyrosine; Amisulpride; Animals; Apomorphine; Corpus Striatum; Cyclic AMP; Dopamine Antagonists; Drug Synergism; In Vitro Techniques; Male; Methyltyrosines; Metoclopramide; Mice; Phenethylamines; Rats; Rats, Inbred Strains; Receptors, Dopamine; Reserpine; Stereotyped Behavior; Sulpiride

1989
D1 dopamine receptor activation required for postsynaptic expression of D2 agonist effects.
    Science (New York, N.Y.), 1987, May-08, Volume: 236, Issue:4802

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; alpha-Methyltyrosine; Animals; Apomorphine; Basal Ganglia; Benzazepines; Dopamine; Ergolines; Methyltyrosines; Neurons; Phenethylamines; Quinpirole; Rats; Receptors, Dopamine; Receptors, Dopamine D1; Receptors, Dopamine D2; Stereotyped Behavior

1987
In vivo release of [3H]gamma-aminobutyric acid in the rat neostriatum--I. Characterization and topographical heterogeneity of the effects of dopaminergic and cholinergic agents.
    Neuroscience, 1986, Volume: 19, Issue:4

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Acetylcholine; Animals; Benzazepines; Calcium; Corpus Striatum; Dopamine; gamma-Aminobutyric Acid; Male; Phenethylamines; Potassium; Rats; Rats, Inbred Strains; Tetrodotoxin

1986
Opposite responses in the striato-nigral substance P system to D1 and D2 receptor activation.
    European journal of pharmacology, 1984, Oct-01, Volume: 105, Issue:1-2

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Apomorphine; Appetite Depressants; Benzazepines; Corpus Striatum; Male; Methamphetamine; Phenethylamines; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Dopamine D1; Receptors, Dopamine D2; Substance P; Substantia Nigra

1984