Page last updated: 2024-09-05

rs 67333 and prucalopride

rs 67333 has been researched along with prucalopride in 8 studies

Compound Research Comparison

Studies
(rs 67333)
Trials
(rs 67333)
Recent Studies (post-2010)
(rs 67333)
Studies
(prucalopride)
Trials
(prucalopride)
Recent Studies (post-2010) (prucalopride)
6303423857167

Research

Studies (8)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's3 (37.50)29.6817
2010's5 (62.50)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Fischmeister, R; Langlois, M1
Benade, V; Bhyrapuneni, G; Bogaraju, N; Gagginapalli, SR; Goyal, VK; Jayarajan, P; Kota, L; Mohammed, AR; Muddana, NR; Nirogi, R; Palacharla, RC; Ravella, SR; Shinde, AK; Subramanian, R1
Benade, V; Birangal, SR; Bogaraju, N; Gagginapally, SR; Jayarajan, P; Kancharla, DM; Middekadi, VR; Mohammed, AR; Muddana, N; Nirogi, R; Palacharla, RC; Ravella, SR; Shinde, AK; Singh, P; Subramanian, R1
Barrot, M; Bockaert, J; Charnay, Y; Compan, V; Debonnel, G; Lucas, G; Nestler, EJ; Neve, RL1
Belzung, C; Cachard-Chastel, M; Devers, S; Gardier, AM; Langlois, M; Lezoualc'h, F; Sicsic, S1
Debonnel, G; Du, J; Haddjeri, N; Lucas, G; Mnie-Filali, O; PiƱeyro, G; Romeas, T1
Chinkwo, KA; Coupar, IM; Grabbe, C; Irving, HR; Li, JG; Pouton, CW; Shapiro, M; Tochon-Danguy, N1
Ajjala, DR; Aleti, RR; Bhyrapuneni, G; Kandikere, V; Nirogi, R; Rasheed, MA; Saralaya, R1

Reviews

1 review(s) available for rs 67333 and prucalopride

ArticleYear
5-HT4 receptor ligands: applications and new prospects.
    Journal of medicinal chemistry, 2003, Jan-30, Volume: 46, Issue:3

    Topics: Animals; Benzamides; Benzimidazoles; Benzoates; Binding Sites; Cardiovascular Physiological Phenomena; Central Nervous System; Digestive System Physiological Phenomena; Humans; Indoles; Ketones; Ligands; Receptors, Serotonin; Receptors, Serotonin, 5-HT4; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists

2003

Other Studies

7 other study(ies) available for rs 67333 and prucalopride

ArticleYear
Synthesis and SAR of Imidazo[1,5-a]pyridine derivatives as 5-HT4 receptor partial agonists for the treatment of cognitive disorders associated with Alzheimer's disease.
    European journal of medicinal chemistry, 2015, Oct-20, Volume: 103

    Topics: Alzheimer Disease; Animals; Cognition Disorders; Dogs; Dose-Response Relationship, Drug; Drug Design; Drug Partial Agonism; Humans; Molecular Structure; Pyridines; Rats; Receptors, Serotonin, 5-HT4; Structure-Activity Relationship

2015
Synthesis, Structure-Activity Relationships, and Preclinical Evaluation of Heteroaromatic Amides and 1,3,4-Oxadiazole Derivatives as 5-HT
    Journal of medicinal chemistry, 2018, 06-14, Volume: 61, Issue:11

    Topics: Amides; Animals; Chemistry Techniques, Synthetic; Drug Evaluation, Preclinical; Humans; Male; Oxadiazoles; Rats; Rats, Wistar; Receptors, Serotonin, 5-HT4; Serotonin 5-HT4 Receptor Agonists; Structure-Activity Relationship

2018
Frontocortical 5-HT4 receptors exert positive feedback on serotonergic activity: viral transfections, subacute and chronic treatments with 5-HT4 agonists.
    Biological psychiatry, 2005, Apr-15, Volume: 57, Issue:8

    Topics: Aniline Compounds; Animals; Benzofurans; Electrophysiology; Extracellular Space; Feedback; Frontal Lobe; Gene Transfer Techniques; Genetic Vectors; Herpesvirus 1, Human; In Situ Hybridization; Indoles; Iontophoresis; Male; Neurons; Piperidines; Pyramidal Cells; Raphe Nuclei; Rats; Rats, Sprague-Dawley; Receptors, Serotonin, 5-HT4; RNA Probes; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Sulfonamides

2005
Prucalopride and donepezil act synergistically to reverse scopolamine-induced memory deficit in C57Bl/6j mice.
    Behavioural brain research, 2008, Mar-05, Volume: 187, Issue:2

    Topics: Amyloid beta-Protein Precursor; Analysis of Variance; Aniline Compounds; Animals; Benzofurans; Cerebral Cortex; Cholinesterase Inhibitors; Donepezil; Drug Synergism; Hippocampus; Indans; Male; Maze Learning; Memory Disorders; Mice; Mice, Inbred C57BL; Motor Activity; Nootropic Agents; Piperidines; Scopolamine; Serotonin 5-HT4 Receptor Agonists; Statistics, Nonparametric

2008
Selective serotonin reuptake inhibitors potentiate the rapid antidepressant-like effects of serotonin4 receptor agonists in the rat.
    PloS one, 2010, Feb-16, Volume: 5, Issue:2

    Topics: Action Potentials; Aniline Compounds; Animals; Antidepressive Agents; Benzofurans; CA3 Region, Hippocampal; Citalopram; Cyclic AMP Response Element-Binding Protein; Drug Synergism; Fluvoxamine; Male; Motor Activity; Neurons; Phosphorylation; Piperazines; Piperidines; Pyridines; Raphe Nuclei; Rats; Rats, Sprague-Dawley; Selective Serotonin Reuptake Inhibitors; Serotonin; Serotonin 5-HT1 Receptor Antagonists; Serotonin 5-HT4 Receptor Agonists; Serotonin Antagonists; Serotonin Receptor Agonists

2010
Investigations into the binding affinities of different human 5-HT4 receptor splice variants.
    Pharmacology, 2010, Volume: 85, Issue:4

    Topics: Aniline Compounds; Animals; Benzamides; Benzimidazoles; Benzofurans; Binding Sites; Binding, Competitive; Bridged Bicyclo Compounds, Heterocyclic; Chlorocebus aethiops; COS Cells; Cyclic AMP; Dose-Response Relationship, Drug; Humans; Indoles; Kinetics; Ligands; Piperidines; Protein Isoforms; Receptors, Serotonin, 5-HT4; Serotonin 5-HT4 Receptor Agonists; Serotonin Antagonists

2010
In-vivo rat striatal 5-HT4 receptor occupancy using non-radiolabelled SB207145.
    The Journal of pharmacy and pharmacology, 2013, Volume: 65, Issue:5

    Topics: Aniline Compounds; Animals; Benzofurans; Binding, Competitive; Brain; Drug Discovery; Indoles; Ligands; Male; Oxazines; Piperidines; Rats; Rats, Sprague-Dawley; Receptors, Serotonin, 5-HT4; Serotonin Receptor Agonists; Sulfonamides; Tandem Mass Spectrometry; Tissue Distribution

2013