Page last updated: 2024-09-03

rs 45041-190 and idazoxan

rs 45041-190 has been researched along with idazoxan in 4 studies

Compound Research Comparison

Studies
(rs 45041-190)
Trials
(rs 45041-190)
Recent Studies (post-2010)
(rs 45041-190)
Studies
(idazoxan)
Trials
(idazoxan)
Recent Studies (post-2010) (idazoxan)
8021,49940123

Protein Interaction Comparison

ProteinTaxonomyrs 45041-190 (IC50)idazoxan (IC50)
Alpha-2A adrenergic receptorHomo sapiens (human)0.0083
Alpha-1B adrenergic receptorRattus norvegicus (Norway rat)0.0195
Alpha-2B adrenergic receptorHomo sapiens (human)0.0195
Alpha-2C adrenergic receptorHomo sapiens (human)0.0537
Alpha-1D adrenergic receptorRattus norvegicus (Norway rat)0.0195
Alpha-1A adrenergic receptorHomo sapiens (human)2.884
Alpha-1A adrenergic receptorRattus norvegicus (Norway rat)0.0195

Research

Studies (4)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's2 (50.00)18.2507
2000's2 (50.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Brown, CM; MacKinnon, AC; Redfern, WS1
Houghton, AK; Westlund, KN1
Clarke, RW; Harris, J; Ogilvie, J1
Choi, DH; Choi, SH; Chun, BG; Lee, JJ; Park, MS1

Other Studies

4 other study(ies) available for rs 45041-190 and idazoxan

ArticleYear
[3H]-RS-45041-190: a selective high-affinity radioligand for I2 imidazoline receptors.
    British journal of pharmacology, 1995, Volume: 116, Issue:2

    Topics: Adrenergic alpha-Antagonists; Animals; Autoradiography; Binding, Competitive; Dioxanes; Dose-Response Relationship, Drug; Idazoxan; Imidazoles; Imidazoline Receptors; Indoles; Isoindoles; Kidney; Male; Radioligand Assay; Rats; Rats, Sprague-Dawley; Receptors, Drug; Time Factors

1995
An I2 imidazoline ligand, RS 45041, potentiates hyperalgesia in acute arthritis.
    Neuroreport, 1996, Jun-17, Volume: 7, Issue:9

    Topics: Acute Disease; Adrenergic alpha-Antagonists; Animals; Arthritis; Drug Evaluation, Preclinical; Drug Synergism; Hyperalgesia; Idazoxan; Imidazoles; Imidazoline Receptors; Indoles; Injections, Spinal; Isoindoles; Neural Inhibition; Rats; Rats, Sprague-Dawley; Reaction Time; Receptors, Drug

1996
Imidazoline I(2)-receptors and spinal reflexes in the decerebrated rabbit.
    Neuropharmacology, 2000, Jul-24, Volume: 39, Issue:10

    Topics: Adrenergic alpha-Antagonists; Animals; Blood Pressure; Clorgyline; Decerebrate State; Dose-Response Relationship, Drug; Female; Heart Rate; Idazoxan; Imidazoles; Imidazoline Receptors; Indoles; Injections, Spinal; Isoindoles; Ligands; Male; Monoamine Oxidase Inhibitors; Pargyline; Rabbits; Receptors, Drug; Reflex; Spinal Cord

2000
Imidazoline drugs stabilize lysosomes and inhibit oxidative cytotoxicity in astrocytes.
    Free radical biology & medicine, 2002, Mar-01, Volume: 32, Issue:5

    Topics: Acridine Orange; Adrenergic alpha-Antagonists; Animals; Animals, Newborn; Antineoplastic Agents; Apoptosis; Astrocytes; Cathepsin D; Cell Division; Cell Line; Cerebral Cortex; Cytochrome c Group; Fish Venoms; Guanabenz; Guanfacine; HIV Protease Inhibitors; Idazoxan; Imidazoles; Indoles; Isoindoles; L-Lactate Dehydrogenase; Ligands; Lysosomes; Membrane Potentials; Mitochondria; Naphthoquinones; Neuroglia; Oxidation-Reduction; Pepstatins; Protease Inhibitors; Rats; Rats, Sprague-Dawley; Reactive Oxygen Species; Receptors, Drug

2002