Page last updated: 2024-09-04

rs 42358-197 and granisetron

rs 42358-197 has been researched along with granisetron in 1 studies

*Granisetron: A serotonin receptor (5HT-3 selective) antagonist that has been used as an antiemetic for cancer chemotherapy patients. [MeSH]

*Granisetron: A serotonin receptor (5HT-3 selective) antagonist that has been used as an antiemetic for cancer chemotherapy patients. [MeSH]

Compound Research Comparison

Studies
(rs 42358-197)
Trials
(rs 42358-197)
Recent Studies (post-2010)
(rs 42358-197)
Studies
(granisetron)
Trials
(granisetron)
Recent Studies (post-2010) (granisetron)
60059016

Protein Interaction Comparison

ProteinTaxonomyrs 42358-197 (IC50)granisetron (IC50)
Solute carrier family 22 member 2Homo sapiens (human)4.3
DRattus norvegicus (Norway rat)3.8019
Alpha-2B adrenergic receptorRattus norvegicus (Norway rat)3.8019
Alpha-2C adrenergic receptorRattus norvegicus (Norway rat)3.8019
Alpha-2A adrenergic receptorRattus norvegicus (Norway rat)3.8019
Sodium-dependent dopamine transporterRattus norvegicus (Norway rat)3.8019
5-hydroxytryptamine receptor 3ARattus norvegicus (Norway rat)1.76
Potassium voltage-gated channel subfamily H member 2Homo sapiens (human)3.7702
Multidrug and toxin extrusion protein 1Homo sapiens (human)5
5-hydroxytryptamine receptor 3BRattus norvegicus (Norway rat)1.76

Research

Studies (1)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's1 (100.00)18.2507
2000's0 (0.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Berger, J; Bonhaus, DW; Clark, RD; Eglen, RM; Kowalczyk, BA; Lee, CH; Michel, AD; Miller, AB; Repke, DB; Weinhardt, KK1

Other Studies

1 other study(ies) available for rs 42358-197 and granisetron

ArticleYear
2-(Quinuclidin-3-yl)pyrido[4,3-b]indol-1-ones and isoquinolin-1-ones. Potent conformationally restricted 5-HT3 receptor antagonists.
    Journal of medicinal chemistry, 1993, Sep-03, Volume: 36, Issue:18

    Topics: Animals; Cisplatin; Computer Simulation; Dogs; Ferrets; Isoquinolines; Male; Models, Molecular; Molecular Structure; Palonosetron; Pyridones; Quinuclidines; Rats; Rats, Sprague-Dawley; Receptors, Serotonin; Serotonin Antagonists; Stereoisomerism; Structure-Activity Relationship; Vomiting

1993