Page last updated: 2024-09-05

rpr 104632 and licostinel

rpr 104632 has been researched along with licostinel in 3 studies

Compound Research Comparison

Studies
(rpr 104632)
Trials
(rpr 104632)
Recent Studies (post-2010)
(rpr 104632)
Studies
(licostinel)
Trials
(licostinel)
Recent Studies (post-2010) (licostinel)
5004910

Protein Interaction Comparison

ProteinTaxonomyrpr 104632 (IC50)licostinel (IC50)
Glutamate receptor ionotropic, NMDA 2DHomo sapiens (human)0.0059
Glutamate receptor ionotropic, NMDA 3BHomo sapiens (human)0.0059
Glutamate receptor 1Rattus norvegicus (Norway rat)0.766
Glutamate receptor 2Rattus norvegicus (Norway rat)0.766
Glutamate receptor 3Rattus norvegicus (Norway rat)0.766
Glutamate receptor 4Rattus norvegicus (Norway rat)0.766
Glutamate receptor ionotropic, NMDA 1 Rattus norvegicus (Norway rat)0.0068
Glutamate receptor ionotropic, NMDA 2A Rattus norvegicus (Norway rat)0.0068
Glutamate receptor ionotropic, NMDA 2BRattus norvegicus (Norway rat)0.0068
Glutamate receptor ionotropic, NMDA 2CRattus norvegicus (Norway rat)0.0068
Glutamate receptor ionotropic, NMDA 1Homo sapiens (human)0.0059
Glutamate receptor ionotropic, NMDA 2AHomo sapiens (human)0.0059
Glutamate receptor ionotropic, NMDA 2BHomo sapiens (human)0.0059
Glutamate receptor ionotropic, NMDA 2CHomo sapiens (human)0.0059
Glutamate receptor ionotropic, NMDA 2DRattus norvegicus (Norway rat)0.0068
Glutamate receptor ionotropic, NMDA 3AHomo sapiens (human)0.0059
Glutamate receptor ionotropic, NMDA 3BRattus norvegicus (Norway rat)0.0068
Glutamate receptor ionotropic, NMDA 3ARattus norvegicus (Norway rat)0.0068

Research

Studies (3)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's2 (66.67)18.2507
2000's1 (33.33)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Iversen, LL; Leeson, PD1
Bohme, GA; Boireau, A; Chevé, M; Damour, D; Doble, A; Genevois-Borella, A; Herman, F; Imperato, A; Jimonet, P; Le Guern, S; Manfré, F; Mignani, S; Pratt, J; Randle, JC; Ribeill, Y; Stutzmann, JM1
Erdõ, SL; Molnár, P1

Reviews

1 review(s) available for rpr 104632 and licostinel

ArticleYear
The glycine site on the NMDA receptor: structure-activity relationships and therapeutic potential.
    Journal of medicinal chemistry, 1994, Nov-25, Volume: 37, Issue:24

    Topics: Animals; Anti-Anxiety Agents; Antipsychotic Agents; Binding Sites; Cognition; Glycine; Humans; Kynurenic Acid; Neuroprotective Agents; Pyrrolidinones; Receptors, N-Methyl-D-Aspartate; Structure-Activity Relationship

1994

Other Studies

2 other study(ies) available for rpr 104632 and licostinel

ArticleYear
Indeno[1,2-b]pyrazin-2,3-diones: a new class of antagonists at the glycine site of the NMDA receptor with potent in vivo activity.
    Journal of medicinal chemistry, 2000, Jun-15, Volume: 43, Issue:12

    Topics: Animals; Anticonvulsants; Cells, Cultured; Cerebellum; Cerebral Cortex; Excitatory Amino Acid Antagonists; In Vitro Techniques; Long-Term Potentiation; Mice; Neurons; Patch-Clamp Techniques; Pyrazines; Rats; Rats, Sprague-Dawley; Receptors, Glycine; Receptors, N-Methyl-D-Aspartate; Stereoisomerism

2000
Differential effects of five glycine site antagonists on NMDA receptor desensitisation.
    European journal of pharmacology, 1996, Sep-12, Volume: 311, Issue:2-3

    Topics: Animals; Benzothiadiazines; Cells, Cultured; Cerebral Cortex; Dose-Response Relationship, Drug; Excitatory Amino Acid Antagonists; Glycine; Kynurenic Acid; N-Methylaspartate; Neurons; Patch-Clamp Techniques; Quinolones; Quinoxalines; Rats; Rats, Sprague-Dawley; Receptors, N-Methyl-D-Aspartate

1996