Page last updated: 2024-09-05

rpr 104632 and kynurenic acid

rpr 104632 has been researched along with kynurenic acid in 3 studies

Compound Research Comparison

Studies
(rpr 104632)
Trials
(rpr 104632)
Recent Studies (post-2010)
(rpr 104632)
Studies
(kynurenic acid)
Trials
(kynurenic acid)
Recent Studies (post-2010) (kynurenic acid)
5002,61128750

Protein Interaction Comparison

ProteinTaxonomyrpr 104632 (IC50)kynurenic acid (IC50)
Neuronal acetylcholine receptor subunit alpha-7Homo sapiens (human)7

Research

Studies (3)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's3 (100.00)18.2507
2000's0 (0.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Iversen, LL; Leeson, PD1
Blanchard, JC; Boireau, A; Bordier, F; Burgevin, MC; Chevet, T; Daniel, M; Doble, A; Durand, G; Jimonet, P; Malgouris, C; Meunier, M; Mignani, S; Miquet, JM; Pény, C1
Erdõ, SL; Molnár, P1

Reviews

1 review(s) available for rpr 104632 and kynurenic acid

ArticleYear
The glycine site on the NMDA receptor: structure-activity relationships and therapeutic potential.
    Journal of medicinal chemistry, 1994, Nov-25, Volume: 37, Issue:24

    Topics: Animals; Anti-Anxiety Agents; Antipsychotic Agents; Binding Sites; Cognition; Glycine; Humans; Kynurenic Acid; Neuroprotective Agents; Pyrrolidinones; Receptors, N-Methyl-D-Aspartate; Structure-Activity Relationship

1994

Other Studies

2 other study(ies) available for rpr 104632 and kynurenic acid

ArticleYear
Neuroprotective effects of RPR 104632, a novel antagonist at the glycine site of the NMDA receptor, in vitro.
    European journal of pharmacology, 1996, Apr-11, Volume: 300, Issue:3

    Topics: Aminoquinolines; Animals; Benzothiadiazines; Binding, Competitive; Cerebral Cortex; Cyclic GMP; Excitatory Amino Acid Antagonists; Hippocampus; In Vitro Techniques; Kynurenic Acid; Nerve Degeneration; Phencyclidine; Rats; Rats, Sprague-Dawley; Receptors, N-Methyl-D-Aspartate

1996
Differential effects of five glycine site antagonists on NMDA receptor desensitisation.
    European journal of pharmacology, 1996, Sep-12, Volume: 311, Issue:2-3

    Topics: Animals; Benzothiadiazines; Cells, Cultured; Cerebral Cortex; Dose-Response Relationship, Drug; Excitatory Amino Acid Antagonists; Glycine; Kynurenic Acid; N-Methylaspartate; Neurons; Patch-Clamp Techniques; Quinolones; Quinoxalines; Rats; Rats, Sprague-Dawley; Receptors, N-Methyl-D-Aspartate

1996