Page last updated: 2024-09-04

rpr 100893 and piperidines

rpr 100893 has been researched along with piperidines in 5 studies

Compound Research Comparison

Studies
(rpr 100893)
Trials
(rpr 100893)
Recent Studies (post-2010)
(rpr 100893)
Studies
(piperidines)
Trials
(piperidines)
Recent Studies (post-2010) (piperidines)
131040,2355,22114,545

Research

Studies (5)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's3 (60.00)18.2507
2000's2 (40.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Bock, MD; Clot, J; Emile, L; Fardin, V; Garret, C; Habert-Ortoli, E; Le Guern, J; Loquet, I; Mercken, L; Pradier, L1
Cavero, I; Floch, A; Thiry, C1
Campbell, EA; Gentry, CT; Panesar, MS; Patel, S; Urban, L; Walpole, CS1
Coupar, IM; Kerr, KP; Mitchelson, F1
Campbell, EA; Cruwys, S; Fox, AJ; Gentry, C; Kidd, B; Patel, S; Urban, L1

Other Studies

5 other study(ies) available for rpr 100893 and piperidines

ArticleYear
Molecular determinants of the species selectivity of neurokinin type 1 receptor antagonists.
    Molecular pharmacology, 1995, Volume: 47, Issue:2

    Topics: Androstanes; Animals; Benzimidazoles; Dipeptides; Humans; Indoles; Isoindoles; Neurokinin-1 Receptor Antagonists; Piperidines; Rats; Receptors, Neurokinin-1; Species Specificity; Substance P

1995
Pharmacological evidence that NK-2 tachykinin receptors mediate hypotension in the guinea pig but not in the rat.
    Fundamental & clinical pharmacology, 1996, Volume: 10, Issue:4

    Topics: Animals; Benzamides; Blood Pressure; Guinea Pigs; Hypotension; Indoles; Isoindoles; Male; Neurokinin A; Neurokinin-1 Receptor Antagonists; Peptide Fragments; Piperidines; Pyrrolidonecarboxylic Acid; Rats; Rats, Sprague-Dawley; Receptors, Neurokinin-1; Receptors, Neurokinin-2; Substance P

1996
Selective neurokinin-1 receptor antagonists are anti-hyperalgesic in a model of neuropathic pain in the guinea-pig.
    Neuroscience, 1998, Volume: 87, Issue:3

    Topics: Administration, Oral; Animals; Disease Models, Animal; Dose-Response Relationship, Drug; Guinea Pigs; Hyperalgesia; Indoles; Injections, Spinal; Isoindoles; Naphthalenes; Nerve Fibers; Neuralgia; Neurokinin-1 Receptor Antagonists; Neurons, Afferent; Piperidines; Proline; Receptors, Neurokinin-1; Spinal Cord

1998
Tachykinins play a minor role in mediating the third phase of the contractile response to vagal nerve stimulation of the guinea-pig oesophagus.
    Neuropeptides, 2000, Volume: 34, Issue:1

    Topics: Animals; Benzamides; Electric Stimulation; Esophagus; Guinea Pigs; In Vitro Techniques; Indoles; Isoindoles; Male; Muscle Contraction; Neurokinin-1 Receptor Antagonists; Piperidines; Quinuclidines; Receptors, Neurokinin-1; Receptors, Neurokinin-2; Receptors, Neurokinin-3; Receptors, Tachykinin; Vagus Nerve

2000
Oral anti-hyperalgesic and anti-inflammatory activity of NK(1) receptor antagonists in models of inflammatory hyperalgesia of the guinea-pig.
    Pain, 2000, Volume: 87, Issue:3

    Topics: Administration, Oral; Animals; Anti-Inflammatory Agents; Carrageenan; Disease Models, Animal; Female; Freund's Adjuvant; Guinea Pigs; Humans; Hyperalgesia; Indoles; Isoindoles; Male; Naphthalenes; Neurokinin-1 Receptor Antagonists; Piperidines; Proline; Quinuclidines

2000