Page last updated: 2024-09-04

rp 73401 and trequinsin

rp 73401 has been researched along with trequinsin in 2 studies

Compound Research Comparison

Studies
(rp 73401)
Trials
(rp 73401)
Recent Studies (post-2010)
(rp 73401)
Studies
(trequinsin)
Trials
(trequinsin)
Recent Studies (post-2010) (trequinsin)
9202354014

Protein Interaction Comparison

ProteinTaxonomyrp 73401 (IC50)trequinsin (IC50)
cGMP-dependent 3',5'-cyclic phosphodiesteraseHomo sapiens (human)1.9502
Multidrug resistance-associated protein 4Homo sapiens (human)10
High affinity cAMP-specific and IBMX-insensitive 3',5'-cyclic phosphodiesterase 8AHomo sapiens (human)1.9502
cGMP-specific 3',5'-cyclic phosphodiesteraseHomo sapiens (human)1.9502
cAMP-specific 3',5'-cyclic phosphodiesterase 4AHomo sapiens (human)0.4
cAMP-specific 3',5'-cyclic phosphodiesterase 4BHomo sapiens (human)0.4
cAMP-specific 3',5'-cyclic phosphodiesterase 4CHomo sapiens (human)0.4
cAMP-specific 3',5'-cyclic phosphodiesterase 4DHomo sapiens (human)1.4334
cGMP-inhibited 3',5'-cyclic phosphodiesterase AHomo sapiens (human)1.9502
cGMP-specific 3',5'-cyclic phosphodiesteraseBos taurus (cattle)5

Research

Studies (2)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's1 (50.00)29.6817
2010's1 (50.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Ashton, TD; Bland, ND; Campbell, RK; Cotter, K; Fang, AP; Gangurde, R; Garceau, N; Gechijian, L; Gustafson, AE; McAllister, G; Ochiana, SO; Ondrechen, MJ; Ortenberg, R; Pollastri, MP; Tallman, C; Wang, C; Wang, Z1
Alves, AC; Barreto, EO; Cordeiro, RS; Jose, PJ; Lagente, V; Martins, MA; Pires, AL; Serra, MF; Silva, JP; Silva, PM; Teixeira, MM1

Other Studies

2 other study(ies) available for rp 73401 and trequinsin

ArticleYear
Pharmacological validation of Trypanosoma brucei phosphodiesterases B1 and B2 as druggable targets for African sleeping sickness.
    Journal of medicinal chemistry, 2011, Dec-08, Volume: 54, Issue:23

    Topics: 3',5'-Cyclic-AMP Phosphodiesterases; Benzamides; Catalytic Domain; Humans; Models, Molecular; Molecular Structure; Pyridines; Recombinant Proteins; Structure-Activity Relationship; Trypanocidal Agents; Trypanosoma brucei brucei; Trypanosomiasis, African

2011
Modulation of eotaxin formation and eosinophil migration by selective inhibitors of phosphodiesterase type 4 isoenzyme.
    British journal of pharmacology, 2001, Volume: 134, Issue:2

    Topics: 3',5'-Cyclic-AMP Phosphodiesterases; Adrenergic beta-Agonists; Albuterol; Allergens; Animals; Benzamides; Bronchoalveolar Lavage Fluid; Capillary Permeability; Cell Adhesion; Cell Degranulation; Cell Movement; Chemokine CCL11; Chemokines, CC; Chemotaxis, Leukocyte; Cyclic Nucleotide Phosphodiesterases, Type 4; Cytokines; Dose-Response Relationship, Drug; Eosinophils; Female; Guinea Pigs; Immune Sera; Isoenzymes; Isoquinolines; Male; Mast Cells; Ovalbumin; Phosphodiesterase Inhibitors; Pleurisy; Pyridines; Rats; Rats, Wistar; Rolipram; Tetrahydroisoquinolines

2001