Page last updated: 2024-09-04

rp 73401 and dinoprostone

rp 73401 has been researched along with dinoprostone in 4 studies

Compound Research Comparison

Studies
(rp 73401)
Trials
(rp 73401)
Recent Studies (post-2010)
(rp 73401)
Studies
(dinoprostone)
Trials
(dinoprostone)
Recent Studies (post-2010) (dinoprostone)
9202329,1051,3466,357

Protein Interaction Comparison

ProteinTaxonomyrp 73401 (IC50)dinoprostone (IC50)
Prostaglandin E2 receptor EP1 subtypeHomo sapiens (human)0.0155
Prostaglandin E2 receptor EP4 subtypeHomo sapiens (human)0.0031
Prostaglandin E2 receptor EP4 subtypeRattus norvegicus (Norway rat)0.0021
Prostaglandin E2 receptor EP3 subtypeHomo sapiens (human)0.002
Prostaglandin E2 receptor EP2 subtypeHomo sapiens (human)0.0087
Prostacyclin receptorHomo sapiens (human)0.26
Prostaglandin E2 receptor EP2 subtypeRattus norvegicus (Norway rat)0.0052

Research

Studies (4)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's3 (75.00)29.6817
2010's1 (25.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Ezeamuzie, CI1
Cabrol, D; Dallot, E; Ferré, F; Leroy, MJ; Méhats, C; Tanguy, G1
Dunkern, TR; Feurstein, D; Hatzelmann, A; Rossi, GA; Sabatini, F1
Dunkern, T; Hatzelmann, A; Selige, J; Tenor, H1

Other Studies

4 other study(ies) available for rp 73401 and dinoprostone

ArticleYear
Requirement of additional adenylate cyclase activation for the inhibition of human eosinophil degranulation by phosphodiesterase IV inhibitors.
    European journal of pharmacology, 2001, Apr-06, Volume: 417, Issue:1-2

    Topics: 3',5'-Cyclic-AMP Phosphodiesterases; Adenylyl Cyclases; Adult; Albuterol; Benzamides; Cell Degranulation; Colforsin; Cyclic AMP; Cyclic Nucleotide Phosphodiesterases, Type 4; Cyclohexanecarboxylic Acids; Dinoprostone; Dose-Response Relationship, Drug; Enzyme Activation; Eosinophil Peroxidase; Eosinophils; Histamine; Humans; Nitriles; Peroxidases; Phosphodiesterase Inhibitors; Pyridines; Rolipram; Superoxides; Theophylline

2001
Is up-regulation of phosphodiesterase 4 activity by PGE2 involved in the desensitization of beta-mimetics in late pregnancy human myometrium?
    The Journal of clinical endocrinology and metabolism, 2001, Volume: 86, Issue:11

    Topics: 3',5'-Cyclic-AMP Phosphodiesterases; Adrenergic beta-Agonists; Adult; Albuterol; Benzamides; Cells, Cultured; Cyclic AMP; Cyclic Nucleotide Phosphodiesterases, Type 3; Cyclic Nucleotide Phosphodiesterases, Type 4; Dinoprostone; Female; Humans; Immunohistochemistry; In Vitro Techniques; Isoenzymes; Muscle Contraction; Myometrium; Oxytocics; Phosphodiesterase Inhibitors; Pregnancy; Prostaglandin Antagonists; Proteins; Pyridines; Reverse Transcriptase Polymerase Chain Reaction; Up-Regulation

2001
Inhibition of TGF-beta induced lung fibroblast to myofibroblast conversion by phosphodiesterase inhibiting drugs and activators of soluble guanylyl cyclase.
    European journal of pharmacology, 2007, Oct-15, Volume: 572, Issue:1

    Topics: Actins; Benzamides; Benzoates; Blotting, Western; Cell Differentiation; Cells, Cultured; Cyclic GMP; Dinoprostone; Drug Synergism; Enzyme Activators; Fibroblasts; Fibrosis; Guanylate Cyclase; Humans; Immunohistochemistry; Isoenzymes; Lung; Myocytes, Smooth Muscle; Natriuretic Peptide, Brain; Nitric Oxide Donors; Nitroso Compounds; Oxadiazoles; Phosphodiesterase Inhibitors; Piperazines; Purines; Pyridines; Quinoxalines; Receptors, Cytoplasmic and Nuclear; Sildenafil Citrate; Soluble Guanylyl Cyclase; Sulfones; Transforming Growth Factor beta

2007
Cytokine-dependent balance of mitogenic effects in primary human lung fibroblasts related to cyclic AMP signaling and phosphodiesterase 4 inhibition.
    Journal of cellular physiology, 2010, Volume: 223, Issue:2

    Topics: Benzamides; Cell Proliferation; Cells, Cultured; Cyclic AMP; Cyclic Nucleotide Phosphodiesterases, Type 3; Cyclooxygenase 2; Cytokines; Dinoprostone; DNA Replication; Dose-Response Relationship, Drug; Drug Synergism; Enzyme Inhibitors; Fibroblast Growth Factor 2; Fibroblasts; Genes, cdc; Growth Substances; Humans; Interleukin-1beta; Lung; Phosphodiesterase 3 Inhibitors; Phosphodiesterase 4 Inhibitors; Pulmonary Fibrosis; Pyridazines; Pyridines; Signal Transduction

2010