rp 73401 has been researched along with albuterol in 5 studies
Studies (rp 73401) | Trials (rp 73401) | Recent Studies (post-2010) (rp 73401) | Studies (albuterol) | Trials (albuterol) | Recent Studies (post-2010) (albuterol) |
---|---|---|---|---|---|
92 | 0 | 23 | 10,108 | 3,059 | 2,058 |
Protein | Taxonomy | rp 73401 (IC50) | albuterol (IC50) |
---|---|---|---|
Beta-2 adrenergic receptor | Homo sapiens (human) | 1.2618 |
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 0 (0.00) | 18.7374 |
1990's | 2 (40.00) | 18.2507 |
2000's | 3 (60.00) | 29.6817 |
2010's | 0 (0.00) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
---|---|
Battram, CH; Jordan, R; Lewis, SA; Raeburn, D; Sharma, S; Souness, JE; Tomkinson, A; Underwood, SL; Webber, SE; Woodman, VR | 1 |
Au, BT; Collins, PD; Teixeira, MM; Williams, TJ | 1 |
Ezeamuzie, CI | 1 |
Alves, AC; Barreto, EO; Cordeiro, RS; Jose, PJ; Lagente, V; Martins, MA; Pires, AL; Serra, MF; Silva, JP; Silva, PM; Teixeira, MM | 1 |
Cabrol, D; Dallot, E; Ferré, F; Leroy, MJ; Méhats, C; Tanguy, G | 1 |
5 other study(ies) available for rp 73401 and albuterol
Article | Year |
---|---|
Anti-inflammatory and bronchodilator properties of RP 73401, a novel and selective phosphodiesterase type IV inhibitor.
Topics: Albuterol; Animals; Anti-Inflammatory Agents, Non-Steroidal; Benzamides; Bronchial Hyperreactivity; Bronchial Spasm; Bronchodilator Agents; Capillary Permeability; Guinea Pigs; Hemodynamics; Histamine; Inflammation; Male; Muscle Contraction; Muscle, Smooth; Phosphodiesterase Inhibitors; Platelet Activating Factor; Pyridines; Pyrrolidinones; Rats; Rats, Sprague-Dawley; Rolipram | 1994 |
Effect of PDE4 inhibitors on zymosan-induced IL-8 release from human neutrophils: synergism with prostanoids and salbutamol.
Topics: 3',5'-Cyclic-AMP Phosphodiesterases; Adult; Albuterol; Benzamides; Cyclic Nucleotide Phosphodiesterases, Type 4; Cyclohexanecarboxylic Acids; Drug Synergism; Humans; Interleukin-8; Neutrophils; Nitriles; Phosphodiesterase Inhibitors; Prostaglandins; Pyridines; Pyrrolidinones; Rolipram; Zymosan | 1998 |
Requirement of additional adenylate cyclase activation for the inhibition of human eosinophil degranulation by phosphodiesterase IV inhibitors.
Topics: 3',5'-Cyclic-AMP Phosphodiesterases; Adenylyl Cyclases; Adult; Albuterol; Benzamides; Cell Degranulation; Colforsin; Cyclic AMP; Cyclic Nucleotide Phosphodiesterases, Type 4; Cyclohexanecarboxylic Acids; Dinoprostone; Dose-Response Relationship, Drug; Enzyme Activation; Eosinophil Peroxidase; Eosinophils; Histamine; Humans; Nitriles; Peroxidases; Phosphodiesterase Inhibitors; Pyridines; Rolipram; Superoxides; Theophylline | 2001 |
Modulation of eotaxin formation and eosinophil migration by selective inhibitors of phosphodiesterase type 4 isoenzyme.
Topics: 3',5'-Cyclic-AMP Phosphodiesterases; Adrenergic beta-Agonists; Albuterol; Allergens; Animals; Benzamides; Bronchoalveolar Lavage Fluid; Capillary Permeability; Cell Adhesion; Cell Degranulation; Cell Movement; Chemokine CCL11; Chemokines, CC; Chemotaxis, Leukocyte; Cyclic Nucleotide Phosphodiesterases, Type 4; Cytokines; Dose-Response Relationship, Drug; Eosinophils; Female; Guinea Pigs; Immune Sera; Isoenzymes; Isoquinolines; Male; Mast Cells; Ovalbumin; Phosphodiesterase Inhibitors; Pleurisy; Pyridines; Rats; Rats, Wistar; Rolipram; Tetrahydroisoquinolines | 2001 |
Is up-regulation of phosphodiesterase 4 activity by PGE2 involved in the desensitization of beta-mimetics in late pregnancy human myometrium?
Topics: 3',5'-Cyclic-AMP Phosphodiesterases; Adrenergic beta-Agonists; Adult; Albuterol; Benzamides; Cells, Cultured; Cyclic AMP; Cyclic Nucleotide Phosphodiesterases, Type 3; Cyclic Nucleotide Phosphodiesterases, Type 4; Dinoprostone; Female; Humans; Immunohistochemistry; In Vitro Techniques; Isoenzymes; Muscle Contraction; Myometrium; Oxytocics; Phosphodiesterase Inhibitors; Pregnancy; Prostaglandin Antagonists; Proteins; Pyridines; Reverse Transcriptase Polymerase Chain Reaction; Up-Regulation | 2001 |