Page last updated: 2024-09-05

roxifiban acetate and isoxazoles

roxifiban acetate has been researched along with isoxazoles in 8 studies

Compound Research Comparison

Studies
(roxifiban acetate)
Trials
(roxifiban acetate)
Recent Studies (post-2010)
(roxifiban acetate)
Studies
(isoxazoles)
Trials
(isoxazoles)
Recent Studies (post-2010) (isoxazoles)
8008,6339003,337

Research

Studies (8)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's6 (75.00)18.2507
2000's2 (25.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Bozarth, J; DeGrado, W; Forsythe, M; Hussain, M; Kapil, R; Lorelli, W; Mousa, SA; Olson, RE; Reilly, TM; Sielecki, TM; Thoolen, MJ; Wexler, R; Wityak, J; Xue, CB1
Bozarth, J; Forsythe, M; Mousa, SA; Mu, DX; Wityak, J1
Bozarth, J; Levine, B; Mousa, SA; Youssef, A1
Badawy, SI; Gilbert, DL; Williams, RC2
Barrett, JS; Bozarth, JM; Brown, F; Corjay, MH; Ebling, WF; Kapil, R; Mousa, SA; Padovani, P; Pieniaszek, HJ; Reilly, TM; Yu, J1
Badawy, SI1
Hausner, EA; Liu, J; Mousa, SA; Olson, RE; Racanelli, AL; Sielecki, TM; Wexler, RR1

Other Studies

8 other study(ies) available for roxifiban acetate and isoxazoles

ArticleYear
Novel nonpeptide antiplatelet glycoprotein IIb/IIIa receptor antagonist, DMP754: receptor binding affinity and specificity.
    Coronary artery disease, 1996, Volume: 7, Issue:10

    Topics: Amino Acids; Animals; Cell Adhesion; Dogs; Fibrinogen; Guinea Pigs; Humans; Integrins; Isoxazoles; Mice; Platelet Aggregation; Platelet Aggregation Inhibitors; Platelet Glycoprotein GPIIb-IIIa Complex; Rabbits; Rats; Sensitivity and Specificity; Species Specificity

1996
Intravenous and oral antiplatelet/antithrombotic efficacy and specificity of XR300, a novel nonpeptide platelet GPIIb/IIIa antagonist.
    Journal of cardiovascular pharmacology, 1998, Volume: 31, Issue:3

    Topics: Administration, Oral; Amino Acids; Animals; Antithrombins; Carotid Arteries; Disease Models, Animal; Dogs; Female; Humans; Hydrolysis; Infusions, Intravenous; Isoxazoles; Kinetics; Male; Platelet Aggregation Inhibitors; Platelet Glycoprotein GPIIb-IIIa Complex; Thrombosis

1998
Oral antiplatelet efficacy of the platelet GPIIb/IIIa antagonist, DMP754 in non-human primates.
    Thrombosis research, 1998, Mar-01, Volume: 89, Issue:5

    Topics: Administration, Oral; Amino Acids; Animals; Blood Platelets; Dogs; Drug Evaluation, Preclinical; Humans; Isoxazoles; Kinetics; Papio; Platelet Aggregation; Platelet Aggregation Inhibitors; Platelet Count; Platelet Glycoprotein GPIIb-IIIa Complex

1998
Chemical stability of an ester prodrug of a glycoprotein IIb/IIIa receptor antagonist in solid dosage forms.
    Journal of pharmaceutical sciences, 1999, Volume: 88, Issue:4

    Topics: Amino Acids; Capsules; Chromatography, High Pressure Liquid; Citrates; Drug Compounding; Drug Stability; Electron Probe Microanalysis; Excipients; Humidity; Hydrogen-Ion Concentration; Isoxazoles; Lactose; Platelet Glycoprotein GPIIb-IIIa Complex; Prodrugs; Sodium Citrate; Spectrophotometry, Ultraviolet; Tablets

1999
Effect of different acids on solid-state stability of an ester prodrug of a IIb/IIIa glycoprotein receptor antagonist.
    Pharmaceutical development and technology, 1999, Volume: 4, Issue:3

    Topics: Amino Acids; Chemistry, Pharmaceutical; Chromatography, High Pressure Liquid; Esters; Hydrogen-Ion Concentration; Hydrolysis; Isoxazoles; Lactose; Platelet Glycoprotein GPIIb-IIIa Complex; Prodrugs; Spectrophotometry, Ultraviolet

1999
Disposition and exposure of the fibrinogen receptor antagonist XV459 on alphaIIBbeta3 binding sites in the guinea pig.
    Biopharmaceutics & drug disposition, 1999, Volume: 20, Issue:6

    Topics: Amino Acids; Animals; Area Under Curve; Binding Sites; Binding, Competitive; Guinea Pigs; Humans; Infusions, Intravenous; Isoxazoles; Male; Metabolic Clearance Rate; Platelet Aggregation Inhibitors; Platelet Glycoprotein GPIIb-IIIa Complex; Species Specificity; Structure-Activity Relationship

1999
Effect of salt form on chemical stability of an ester prodrug of a glycoprotein IIb/IIIa receptor antagonist in solid dosage forms.
    International journal of pharmaceutics, 2001, Jul-31, Volume: 223, Issue:1-2

    Topics: Amino Acids; Drug Stability; Hydrogen-Ion Concentration; Isoxazoles; Platelet Aggregation Inhibitors; Platelet Glycoprotein GPIIb-IIIa Complex; Prodrugs

2001
Synthesis and pharmacology of modified amidine isoxazoline glycoprotein IIb/IIIa receptor antagonists.
    Bioorganic & medicinal chemistry letters, 2001, Aug-20, Volume: 11, Issue:16

    Topics: Amino Acids; Isoxazoles; Platelet Aggregation Inhibitors; Platelet Glycoprotein GPIIb-IIIa Complex; Structure-Activity Relationship; Sulfonamides

2001