rosiglitazone has been researched along with l-165041 in 17 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 0 (0.00) | 18.7374 |
1990's | 0 (0.00) | 18.2507 |
2000's | 5 (29.41) | 29.6817 |
2010's | 10 (58.82) | 24.3611 |
2020's | 2 (11.76) | 2.80 |
Authors | Studies |
---|---|
Brown, PJ; Henke, BR; Sternbach, DD; Willson, TM | 1 |
Altieri, F; Azzariti, A; Cervoni, L; Crestani, M; Di Giovanni, C; Fracchiolla, G; Gilardi, F; Giudici, M; Guerrini, U; Laghezza, A; Lavecchia, A; Loiodice, F; Mitro, N; Montanari, R; Paradiso, A; Piemontese, L; Pochetti, G; Porcelli, L; Simone, GM; Tortorella, P | 1 |
Kim, YH; Li, W; Shim, SH; Song, SB; Zhou, W | 1 |
Ammazzalorso, A; Amoroso, R; De Filippis, B; Di Giovanni, C; Fantacuzzi, M; Giampietro, L; Laghezza, A; Lavecchia, A; Linciano, P; Loiodice, F; Maccallini, C; Tortorella, P | 1 |
Angioni, C; Blöcher, R; Boß, M; Brüggerhoff, A; Brüne, B; Diehl, O; Geisslinger, G; Göbel, T; Grundmann, M; Hartmann, M; Heering, J; Kahnt, AS; Kaiser, A; Kostenis, E; Lamers, C; Merk, D; Proschak, E; Schader, T; Schubert-Zsilavecz, M; Steinhilber, D; Weizel, L; Wittmann, SK; Wurglics, M | 1 |
Cerchia, C; Colantuoni, V; Convertini, P; Dal Piaz, F; Iacobazzi, V; Infantino, V; Laghezza, A; Lavecchia, A; Loiodice, F; Lupo, A; Piemontese, L; Sblano, S; Tortorella, P; Ziccardi, P | 1 |
Ammazzalorso, A; Amoroso, R; Brunetti, L; Bruno, I; Cama, A; Capone, F; Cerchia, C; De Filippis, B; Fantacuzzi, M; Ferrante, C; Florio, R; Giampietro, L; Laghezza, A; Lavecchia, A; Loiodice, F; Maccallini, C; Recinella, L; Tortorella, P; Verginelli, F | 1 |
Brunetti, L; Cerchia, C; Genovese, M; Gilardi, F; Laghezza, A; Lavecchia, A; Leuci, R; Loiodice, F; Paoli, P; Piemontese, L; Santi, A; Sblano, S; Thomas, A; Tortorella, P | 1 |
Jacobsson, A; Jörgensen, JA; Zadravec, D | 1 |
Cheng, WT; Ding, ST; Mersmann, HJ; Wu, SC; Yu, YH | 1 |
Aleshin, S; Grabeklis, S; Hanck, T; Reiser, G; Sergeeva, M | 1 |
Chopra, B; Georgopoulos, NT; Hinley, J; Nicholl, A; Oleksiewicz, MB; Southgate, J | 1 |
Bernd, A; Kaufmann, R; Kippenberger, S; Müller, J; Ochsendorf, F; Schuster, M; Thaçi, D; Zouboulis, CC | 1 |
Bogacka, I; Bogacki, M; Gaglewska, M; Kurzynska, A; Wasielak, M | 1 |
Bogacka, I; Bogacki, M; Chojnowska, K; Kurzyńska, A | 2 |
Blitek, A; Szymanska, M | 1 |
1 review(s) available for rosiglitazone and l-165041
Article | Year |
---|---|
The PPARs: from orphan receptors to drug discovery.
Topics: Animals; Diabetes Mellitus; Drug Design; Humans; Hyperlipidemias; Hypertension; Inflammation; Ligands; Models, Molecular; Neoplasms; Nuclear Proteins; Obesity; Receptors, Cytoplasmic and Nuclear; Transcription Factors | 2000 |
16 other study(ies) available for rosiglitazone and l-165041
Article | Year |
---|---|
Synthesis, characterization and biological evaluation of ureidofibrate-like derivatives endowed with peroxisome proliferator-activated receptor activity.
Topics: Adipocytes; Animals; Antineoplastic Agents; Benzoxazoles; Body Weight; Calorimetry; Cell Differentiation; Cell Line; Cell Line, Tumor; Cell Proliferation; Crystallography, X-Ray; Drug Partial Agonism; Drug Screening Assays, Antitumor; Fibric Acids; Fibroblasts; Gene Expression Profiling; Humans; Insulin Resistance; Intra-Abdominal Fat; Liver; Mice; Mice, Inbred C57BL; Models, Molecular; PPAR alpha; PPAR gamma; Propionates; Stereoisomerism; Structure-Activity Relationship; Urea | 2012 |
Sterol fatty acid esters from the mushroom Hericium erinaceum and their PPAR transactivational effects.
Topics: Agaricales; Cells, Cultured; Dose-Response Relationship, Drug; Ergosterol; Esters; Fatty Acids, Unsaturated; Fruiting Bodies, Fungal; Luciferases; Molecular Structure; Nuclear Magnetic Resonance, Biomolecular; Peroxisome Proliferator-Activated Receptors; PPAR alpha; Republic of Korea; Sterols; Trans-Activators | 2014 |
Structural development studies of PPARs ligands based on tyrosine scaffold.
Topics: Dose-Response Relationship, Drug; Humans; Ligands; Molecular Docking Simulation; Molecular Structure; Peroxisome Proliferator-Activated Receptors; Structure-Activity Relationship; Tyrosine | 2015 |
N-Benzylbenzamides: A Novel Merged Scaffold for Orally Available Dual Soluble Epoxide Hydrolase/Peroxisome Proliferator-Activated Receptor γ Modulators.
Topics: 3T3 Cells; Administration, Oral; Animals; Benzamides; Chlorocebus aethiops; COS Cells; Diabetes Mellitus, Type 2; Drug Design; Drug Screening Assays, Antitumor; Enzyme Inhibitors; Epoxide Hydrolases; Humans; Hypertension; In Vitro Techniques; Metabolic Syndrome; Mice; Microsomes, Liver; PPAR gamma; Rats; Structure-Activity Relationship | 2016 |
New diphenylmethane derivatives as peroxisome proliferator-activated receptor alpha/gamma dual agonists endowed with anti-proliferative effects and mitochondrial activity.
Topics: Antineoplastic Agents; Benzhydryl Compounds; beta Catenin; Carnitine; Cell Proliferation; Drug Evaluation, Preclinical; Hep G2 Cells; HT29 Cells; Humans; Insulin Resistance; Mitochondria; Molecular Docking Simulation; PPAR alpha; PPAR gamma; Protein Conformation; Signal Transduction | 2017 |
Novel Phenyldiazenyl Fibrate Analogues as PPAR α/γ/δ Pan-Agonists for the Amelioration of Metabolic Syndrome.
Topics: | 2019 |
A chemoinformatics search for peroxisome proliferator-activated receptors ligands revealed a new pan-agonist able to reduce lipid accumulation and improve insulin sensitivity.
Topics: Cheminformatics; Diabetes Mellitus, Type 2; Humans; Hypoglycemic Agents; Insulin Resistance; Ligands; Lipids; Peroxisome Proliferator-Activated Receptors; PPAR gamma | 2022 |
Norepinephrine and rosiglitazone synergistically induce Elovl3 expression in brown adipocytes.
Topics: Acetyltransferases; Adipocytes; Adipose Tissue, Brown; Animals; Cell Proliferation; Cycloheximide; Dactinomycin; Drug Synergism; Fatty Acid Elongases; Gene Expression Regulation; Male; Membrane Proteins; Mice; Norepinephrine; Peroxisome Proliferators; Phenoxyacetates; PPAR gamma; Protein Synthesis Inhibitors; Pyrimidines; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Rosiglitazone; Thiazolidinediones; Transcription, Genetic | 2007 |
Ectopic expression of porcine peroxisome proliferator-activated receptor delta regulates adipogenesis in mouse myoblasts.
Topics: Adipocytes; Adipogenesis; Animals; Cell Differentiation; Cell Line; Dimethyl Sulfoxide; Gene Expression Regulation; Mice; Myoblasts; Phenoxyacetates; PPAR delta; PPAR gamma; Rosiglitazone; Swine; Thiazolidinediones | 2008 |
Peroxisome proliferator-activated receptor (PPAR)-gamma positively controls and PPARalpha negatively controls cyclooxygenase-2 expression in rat brain astrocytes through a convergence on PPARbeta/delta via mutual control of PPAR expression levels.
Topics: Animals; Animals, Newborn; Astrocytes; Biomarkers; Brain; Butyrates; Cells, Cultured; Cyclooxygenase 2; Drug Combinations; Gene Expression Regulation, Enzymologic; Glial Fibrillary Acidic Protein; Lipopolysaccharides; Peroxisome Proliferator-Activated Receptors; Phenoxyacetates; Phenylurea Compounds; PPAR alpha; PPAR delta; PPAR gamma; PPAR-beta; Protein Isoforms; Rats; Rosiglitazone; Thiazolidinediones; Time Factors | 2009 |
Structurally diverse peroxisome proliferator-activated receptor agonists induce apoptosis in human uro-epithelial cells by a receptor-independent mechanism involving store-operated calcium channels.
Topics: Apoptosis; Calcium; Calcium Channels; Caspase 3; Caspase 9; Cell Division; Cells, Cultured; Chromans; Epithelial Cells; Extracellular Signal-Regulated MAP Kinases; Fenofibrate; Humans; Hypoglycemic Agents; Hypolipidemic Agents; Membrane Potential, Mitochondrial; Oxazines; p38 Mitogen-Activated Protein Kinases; Peroxisome Proliferator-Activated Receptors; Phenoxyacetates; Phenylpropionates; Rosiglitazone; Thiazolidinediones; Troglitazone; Urothelium | 2009 |
Peroxisome proliferator-activated receptor activators protect sebocytes from apoptosis: a new treatment modality for acne?
Topics: Acne Vulgaris; Apoptosis; Blotting, Western; Bromodeoxyuridine; Cell Line; Enzyme Inhibitors; Humans; L-Lactate Dehydrogenase; Peroxisome Proliferator-Activated Receptors; Phenoxyacetates; PPAR alpha; PPAR delta; PPAR gamma; Pyrimidines; Rosiglitazone; Sebaceous Glands; Staurosporine; Thiazolidinediones | 2011 |
In vitro effect of peroxisome proliferator activated receptor (PPAR) ligands on prostaglandin E2 synthesis and secretion by porcine endometrium during the estrous cycle and early pregnancy.
Topics: Animals; Dinoprostone; Endometrium; Estrous Cycle; Female; Indoles; Intramolecular Oxidoreductases; Ligands; Peroxisome Proliferator-Activated Receptors; Phenoxyacetates; Pregnancy; Prostaglandin-E Synthases; Pyrimidines; RNA, Messenger; Rosiglitazone; Swine; Thiazolidinediones | 2013 |
The involvement of peroxisome proliferator activated receptors (PPARs) in prostaglandin F2α production by porcine endometrium.
Topics: Analysis of Variance; Anilides; Animals; Benzamides; Culture Media; Dinoprost; DNA Primers; Endometrium; Estrous Cycle; Female; Indoles; Peroxisome Proliferator-Activated Receptors; Phenoxyacetates; Pregnancy; Prostaglandin D2; Pyridines; Pyrimidines; Radioimmunoassay; Real-Time Polymerase Chain Reaction; Reverse Transcriptase Polymerase Chain Reaction; Rosiglitazone; Swine; Thiazolidinediones | 2013 |
Peroxisome proliferator activated receptor ligands affect progesterone and 17β-estradiol secretion by porcine corpus luteum during early pregnancy.
Topics: 3-Hydroxysteroid Dehydrogenases; Anilides; Animals; Benzamides; Corpus Luteum; Estradiol; Estrous Cycle; Female; Gene Expression; Indoles; Ligands; Peroxisome Proliferator-Activated Receptors; Phenoxyacetates; Pregnancy; Progesterone; Prostaglandin D2; Pyridines; Pyrimidines; RNA, Messenger; Rosiglitazone; Swine; Thiazolidinediones | 2014 |
Peroxisome proliferator-activated receptor β/δ and γ agonists differentially affect prostaglandin E2 and cytokine synthesis and nutrient transporter expression in porcine trophoblast cells during implantation.
Topics: Anilides; Animals; Benzamides; Butadienes; Carrier Proteins; Cells, Cultured; Cytokines; Dinoprostone; Female; Gene Expression Regulation; Nitriles; Phenoxyacetates; PPAR delta; PPAR gamma; PPAR-beta; Pregnancy; Rosiglitazone; Sulfones; Swine; Trophoblasts | 2020 |