Page last updated: 2024-08-25

rosiglitazone and int 131

rosiglitazone has been researched along with int 131 in 4 studies

Research

Studies (4)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's1 (25.00)29.6817
2010's3 (75.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Aramaki, H; Beckmann, H; Biermann, D; Chen, JL; Cushing, TD; Flygare, J; Frankmoelle, W; Furukawa, N; Hagiwara, A; Houze, JB; Iida, T; Jaen, J; Kearney, P; Kitao, Y; Learned, MR; Li, Y; Lindstrom, M; Liu, J; McGee, LR; Miao, S; Motani, A; Nakamura, M; Nishiu, J; Rubenstein, SM; Shinkai, H; Taygerly, JP; Thoolen, M; Timmermans, PB; Walker, N; Wang, Z; Weiszmann, J; Ye, G1
Hashimoto, Y; Ishikawa, M; Makishima, M; Noguchi-Yachide, T; Okazaki, S; Shioi, R; Yamaguchi, T1
Biermann, DH; Chen, JL; Fang, Z; Fuentes, H; Jaen, J; Learned, RM; Lee, G; Li, Y; Lindstrom, M; Liu, J; Liu, Q; McGee, LR; Motani, A; Staunton, J; Walker, NP; Wang, Z; Weiszmann, J1
Depaoli, AM; Higgins, LS1

Reviews

1 review(s) available for rosiglitazone and int 131

ArticleYear
Selective peroxisome proliferator-activated receptor gamma (PPARgamma) modulation as a strategy for safer therapeutic PPARgamma activation.
    The American journal of clinical nutrition, 2010, Volume: 91, Issue:1

    Topics: Diabetes Mellitus, Type 2; Dipeptidyl-Peptidase IV Inhibitors; Gluconeogenesis; Humans; Hypoglycemia; Hypoglycemic Agents; Incretins; Insulin Resistance; Pioglitazone; PPAR gamma; Quinolines; Retinoid X Receptors; Rosiglitazone; Sulfonamides; Thiazolidinediones

2010

Other Studies

3 other study(ies) available for rosiglitazone and int 131

ArticleYear
Discovery of INT131: a selective PPARγ modulator that enhances insulin sensitivity.
    Bioorganic & medicinal chemistry, 2013, Feb-15, Volume: 21, Issue:4

    Topics: Administration, Oral; Animals; Binding Sites; Crystallography, X-Ray; Cytochrome P-450 CYP3A; Cytochrome P-450 Enzyme Inhibitors; Cytochrome P-450 Enzyme System; Diabetes Mellitus, Experimental; Half-Life; Insulin Resistance; Male; Mice; PPAR gamma; Protein Structure, Tertiary; Quinolines; Rats; Rats, Sprague-Dawley; Rats, Zucker; Structure-Activity Relationship; Sulfonamides

2013
Structure-activity relationship studies of non-carboxylic acid peroxisome proliferator-activated receptor α/δ (PPARα/δ) dual agonists.
    Bioorganic & medicinal chemistry, 2016, 11-01, Volume: 24, Issue:21

    Topics: Acetamides; Dose-Response Relationship, Drug; HEK293 Cells; Humans; Molecular Structure; PPAR alpha; PPAR delta; Structure-Activity Relationship

2016
INT131: a selective modulator of PPAR gamma.
    Journal of molecular biology, 2009, Mar-13, Volume: 386, Issue:5

    Topics: Adipocytes; Amino Acid Sequence; Animals; Blood Glucose; Cell Differentiation; Cells, Cultured; Crystallography, X-Ray; Drug Partial Agonism; Hydrophobic and Hydrophilic Interactions; Hypoglycemic Agents; Insulin; Mice; Molecular Sequence Data; PPAR gamma; Protein Binding; Quinolines; Rats; Rats, Zucker; Rosiglitazone; Sulfonamides; Thiazolidinediones

2009