Page last updated: 2024-08-25

rosiglitazone and amg 221

rosiglitazone has been researched along with amg 221 in 1 studies

Research

Studies (1)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's0 (0.00)29.6817
2010's1 (100.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Adams, J; Bartberger, MD; Chen, MM; Cupples, R; Emery, MG; Fotsch, C; Gahm, K; Hague, A; Hale, C; Henriksson, MA; Hungate, RW; Johansson, L; Jona, J; Jordan, S; Joseph, S; Kim, KW; Komorowski, R; Li, V; Moniz, G; St Jean, DJ; Syed, R; Vallgårda, J; Véniant, MM; Wang, M; Williams, M; Zhang, J1

Other Studies

1 other study(ies) available for rosiglitazone and amg 221

ArticleYear
Discovery of a potent, orally active 11beta-hydroxysteroid dehydrogenase type 1 inhibitor for clinical study: identification of (S)-2-((1S,2S,4R)-bicyclo[2.2.1]heptan-2-ylamino)-5-isopropyl-5-methylthiazol-4(5H)-one (AMG 221).
    Journal of medicinal chemistry, 2010, Jun-10, Volume: 53, Issue:11

    Topics: 11-beta-Hydroxysteroid Dehydrogenase Type 1; Administration, Oral; Animals; Dogs; Drug Discovery; Enzyme Inhibitors; Humans; Male; Mice; Models, Molecular; Protein Conformation; Rats; Thiazoles

2010