Page last updated: 2024-08-16

rolipram and diazepam

rolipram has been researched along with diazepam in 14 studies

Research

Studies (14)

TimeframeStudies, this research(%)All Research%
pre-19902 (14.29)18.7374
1990's3 (21.43)18.2507
2000's6 (42.86)29.6817
2010's2 (14.29)24.3611
2020's1 (7.14)2.80

Authors

AuthorsStudies
Creveling, CR; Daly, JW; Lewandowski, GA; McNeal, ET1
Axe, FU; Bembenek, SD; Butler, CR; Coles, F; Dunford, PJ; Edwards, JP; Fourie, AM; Grice, CA; Karlsson, L; Lundeen, K; Riley, JP; Savall, BM; Tays, KL; Wei, J; Williams, KN; Xue, X1
Carmody, LC; Dandapani, S; Donckele, E; Feng, Y; Fernandez, C; Germain, AR; Gupta, PB; Lander, ES; Morgan, B; Munoz, B; Nag, PP; Palmer, M; Perez, JR; Schreiber, SL; Verplank, L1
Barocelli, E; Bertoni, S; Brullo, C; Bruno, O; Fedele, E; Flammini, L; Massa, M; Pronzato, MA; Ricciarelli, R; Rivera, D; Villa, C1
Balliano, TL; Barbosa, G; Carvalho, VF; da Silva, BA; de Souza, ET; Lima, LM; Martins, IRR; Martins, MA; Medeiros, MM; Moraes Junior, MO; Nunes, IKDC; Silva, PMR; Silva, SWD1
Dragunow, M1
Snell, CR; Snell, PH1
Beleta, J; Collado, MC; Domènech, T; Hernández, J; Martinez, E; Miralpeix, M; Palacios, JM1
Fernández, AG; Palacios, JM; Silvestre, JS1
Cherry, JA; Pho, V; Thompson, BE1
Abella, C; Hernandez, J; Vargas, ML1
Hernández, J; Juan-Fita, MJ; Vargas, ML1
González-Cuello, A; Hernández, J; Laorden, ML; Sánchez, L; Teresa Castells, M; Victoria Milanés, M1
González-Cuello, A; Laorden, ML; Milanés, MV; Núñez, C; Sánchez, L; Vargas, ML1

Other Studies

14 other study(ies) available for rolipram and diazepam

ArticleYear
[3H]Batrachotoxinin A 20 alpha-benzoate binding to voltage-sensitive sodium channels: a rapid and quantitative assay for local anesthetic activity in a variety of drugs.
    Journal of medicinal chemistry, 1985, Volume: 28, Issue:3

    Topics: Adrenergic alpha-Antagonists; Adrenergic beta-Antagonists; Anesthetics, Local; Animals; Batrachotoxins; Calcium Channel Blockers; Cyclic AMP; Guinea Pigs; Histamine H1 Antagonists; In Vitro Techniques; Ion Channels; Neurotoxins; Sodium; Tranquilizing Agents; Tritium

1985
Identification of a potent, selective, and orally active leukotriene a4 hydrolase inhibitor with anti-inflammatory activity.
    Journal of medicinal chemistry, 2008, Jul-24, Volume: 51, Issue:14

    Topics: Administration, Oral; Animals; Anti-Inflammatory Agents; Catalysis; Dogs; Drug Evaluation, Preclinical; Enzyme Inhibitors; Epoxide Hydrolases; Humans; Magnetic Resonance Spectroscopy; Mice; Structure-Activity Relationship

2008
Cinnamides as selective small-molecule inhibitors of a cellular model of breast cancer stem cells.
    Bioorganic & medicinal chemistry letters, 2013, Mar-15, Volume: 23, Issue:6

    Topics: Amides; Breast Neoplasms; Cell Line, Tumor; Drug Screening Assays, Antitumor; Female; Humans; Neoplastic Stem Cells; Small Molecule Libraries; Structure-Activity Relationship

2013
Synthesis, biological activities and pharmacokinetic properties of new fluorinated derivatives of selective PDE4D inhibitors.
    Bioorganic & medicinal chemistry, 2015, Jul-01, Volume: 23, Issue:13

    Topics: Animals; Catechols; Cell Line, Tumor; Cell Survival; Cyclic Nucleotide Phosphodiesterases, Type 4; Diazepam; Enzyme Assays; Gene Expression; Halogenation; Humans; Isoenzymes; Male; Mice; Mice, Inbred BALB C; Motor Activity; Neurons; Nootropic Agents; Phosphodiesterase Inhibitors; Rolipram; Structure-Activity Relationship

2015
Discovery of sulfonyl hydrazone derivative as a new selective PDE4A and PDE4D inhibitor by lead-optimization approach on the prototype LASSBio-448: In vitro and in vivo preclinical studies.
    European journal of medicinal chemistry, 2020, Oct-15, Volume: 204

    Topics: Animals; Cyclic AMP; Cyclic Nucleotide Phosphodiesterases, Type 4; Drug Design; Enzyme Inhibitors; Humans; Hydrazones; Hypersensitivity; Lung; Male; Mice

2020
Adenosine receptor antagonism accounts for the seizure-prolonging effects of aminophylline.
    Pharmacology, biochemistry, and behavior, 1990, Volume: 36, Issue:4

    Topics: Adenosine; Aminophylline; Amygdala; Animals; Brain; Carbolines; Diazepam; Flumazenil; Kindling, Neurologic; Male; Picrotoxin; Pyrazoles; Pyrrolidinones; Rats; Rats, Inbred Strains; Receptors, Purinergic; Rolipram; Seizures; Theophylline; Xanthines

1990
Benzodiazepines modulate the A2 adenosine binding sites on 108CC15 neuroblastoma X glioma hybrid cells.
    British journal of pharmacology, 1984, Volume: 83, Issue:3

    Topics: Animals; Anti-Anxiety Agents; Benzodiazepines; Binding, Competitive; Cells, Cultured; Clonazepam; Cyclic AMP; Diazepam; Glioma; Hybrid Cells; Kinetics; Neuroblastoma; Phosphodiesterase Inhibitors; Pyrrolidinones; Receptors, Cell Surface; Receptors, GABA-A; Receptors, Purinergic; Rolipram

1984
Functional and biochemical evidence for diazepam as a cyclic nucleotide phosphodiesterase type 4 inhibitor.
    British journal of pharmacology, 1998, Volume: 123, Issue:6

    Topics: 3',5'-Cyclic-AMP Phosphodiesterases; Animals; Chloride Channels; Cyclic AMP; Diazepam; Drug Interactions; Eosinophils; gamma-Aminobutyric Acid; Guinea Pigs; Heart; In Vitro Techniques; Isoenzymes; Isoproterenol; Myocardial Contraction; Phosphodiesterase Inhibitors; Pyrrolidinones; Rats; Receptors, GABA-A; Rolipram; Tritium

1998
Effects of rolipram on the elevated plus-maze test in rats: a preliminary study.
    Journal of psychopharmacology (Oxford, England), 1999, Volume: 13, Issue:3

    Topics: 3',5'-Cyclic-AMP Phosphodiesterases; Animals; Anti-Anxiety Agents; Antidepressive Agents, Tricyclic; Anxiety; Diazepam; Imipramine; Male; Phosphodiesterase Inhibitors; Rats; Rats, Wistar; Rolipram

1999
Diazepam and rolipram differentially inhibit cyclic AMP-specific phosphodiesterases PDE4A1 and PDE4B3 in the mouse.
    Biochimica et biophysica acta, 2001, Mar-19, Volume: 1518, Issue:1-2

    Topics: 1-Methyl-3-isobutylxanthine; 3',5'-Cyclic-AMP Phosphodiesterases; 4-(3-Butoxy-4-methoxybenzyl)-2-imidazolidinone; Amino Acid Sequence; Animals; Base Sequence; Cell Line; Cloning, Molecular; Cyclic AMP; Cyclic Nucleotide Phosphodiesterases, Type 4; Diazepam; DNA, Complementary; Humans; Immunoblotting; Mice; Milrinone; Molecular Sequence Data; Molecular Structure; Phosphodiesterase Inhibitors; Purinones; Rats; Rolipram; Sequence Homology, Amino Acid

2001
Diazepam increases the hypothalamic-pituitary-adrenocortical (HPA) axis activity by a cyclic AMP-dependent mechanism.
    British journal of pharmacology, 2001, Volume: 133, Issue:8

    Topics: Adrenal Cortex; Adrenocorticotropic Hormone; Animals; Corticosterone; Cyclic AMP; Cyclic AMP-Dependent Protein Kinases; Diazepam; Flumazenil; Hypothalamus; Isoquinolines; Male; Phosphodiesterase Inhibitors; Pituitary Gland; Rats; Rats, Sprague-Dawley; Rolipram; Sulfonamides

2001
Comparative actions of diazepam and other phosphodiesterase inhibitors on the effects of noradrenaline in rat myocardium.
    Pharmacology & toxicology, 2003, Volume: 93, Issue:1

    Topics: Adenine; Animals; Cyclic AMP; Diazepam; Dose-Response Relationship, Drug; Drug Synergism; Female; In Vitro Techniques; Isoenzymes; Male; Milrinone; Myocardial Contraction; Norepinephrine; Phosphodiesterase Inhibitors; Rats; Rats, Sprague-Dawley; Rolipram; Xanthines

2003
Phosphodiesterase 4 inhibitors, rolipram and diazepam block the adaptive changes observed during morphine withdrawal in the heart.
    European journal of pharmacology, 2007, Sep-10, Volume: 570, Issue:1-3

    Topics: Animals; Cyclic AMP; Cyclic GMP; Diazepam; Male; Morphine Dependence; Myocardium; Norepinephrine; Normetanephrine; Phosphodiesterase 4 Inhibitors; Phosphodiesterase Inhibitors; Proto-Oncogene Proteins c-fos; Rats; Rats, Sprague-Dawley; Rolipram; Substance Withdrawal Syndrome

2007
Effects of rolipram and diazepam on the adaptive changes induced by morphine withdrawal in the hypothalamic paraventricular nucleus.
    European journal of pharmacology, 2009, Oct-12, Volume: 620, Issue:1-3

    Topics: Adaptation, Physiological; Animals; Cyclic AMP; Cyclic GMP; Diazepam; Gene Expression Regulation; Male; Morphine; Neurosecretory Systems; Norepinephrine; Paraventricular Hypothalamic Nucleus; Phosphodiesterase Inhibitors; Pituitary Gland; Proto-Oncogene Proteins c-fos; Rats; Rats, Sprague-Dawley; Rolipram; Substance Withdrawal Syndrome

2009
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