ro 5-4864 and flunitrazepam

ro 5-4864 has been researched along with flunitrazepam in 70 studies

Research

Studies (70)

TimeframeStudies, this research(%)All Research%
pre-199047 (67.14)18.7374
1990's17 (24.29)18.2507
2000's2 (2.86)29.6817
2010's4 (5.71)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Blair, T; Webb, GA1
Bendinelli, S; Castellano, S; Cosconati, S; Costa, B; Da Pozzo, E; Da Settimo, F; Greco, G; Martini, C; Milite, C; Novellino, E; Pugliesi, I; Rizzetto, E; Sbardella, G; Stefancich, G; Taliani, S1
Kokka, N; Olsen, RW; Sapp, DW; Witte, U1
Adojaan, A; Harro, J; Kiivet, RA; Rägo, L1
Camilla, C; Courtiere, A; Drouet, J; Jadot, G; Lobert, P; Reybaud, J1
Machen, VL; Swaiman, KF3
Adojaan, A; Allikmets, L; Harro, J; Kiivet, RA; Rägo, L1
Calandra, RS; Calvo, DJ; Medina, JH; Ritta, MN1
Gavish, M; Katz, Y1
De Robertis, E; Levi de Stein, M; Medina, JH1
Harro, J; Kiivet, RA; Pŏld, M; Rägo, L1
Cooper, SJ; Deckert, J; Estall, LB; Marangos, PJ1
Armando, I; Barontini, M; Levin, G1
Cano, JP; Ciesielski, L; Hariton, C; Mandel, P1
Berg, DK; McEachern, AE1
Ciliax, BJ; Mancini, WR; Olson, JM; Young, AB1
Backus, KH; Kettenmann, H; Schachner, M1
Clow, A; Glover, V; Sandler, M1
Boespflug, O; Swaiman, KF1
Bachy, A; Biziere, K; Keane, PE; Morre, M1
Haumont, J; Lenfant, M; Potier, P; Zavala, F1
Barrett, JE; Basile, AS; Bolger, GT; Lueddens, H; Mantione, CR; Paul, SM; Skolnick, P; Weissman, BA; Witkin, JM1
Hornykiewicz, O; Kish, SJ; Perry, TL; Sweeney, VP1
Abraham, CJ; De Blas, AL; Haney, SA; Park, D; Rayner, CA; Sangameswaran, L1
Machen, VL; Neale, EA; Sher, PK1
Fioretti, P; Galbani, P; Gambacciani, M; Melis, GB; Ronca-Testoni, S1
Hrelia, S; Lucacchini, A; Martini, C; Rossi, CA1
Insel, T; Marangos, PJ; Tamborska, E1
Cecchi, L; Filacchioni, G; Lucacchini, A; Martini, C; Melani, F; Palazzino, G; Pennacchi, E1
Lafaille, F; Lal, S; Nair, NP; Quirion, R; Suranyi-Cadotte, B1
Calvo, D; De Robertis, E; Medina, JH; Novas, ML1
Machen, VL; Sher, PK1
Junck, L; Mancini, WR; Olson, JM; Penney, JB; Young, AB1
Borden, LA; Farb, DH; Gibbs, TT1
Villiger, JW2
Bolger, GT; Cott, J; Mezey, E; Paul, SM; Skolnick, P; Weissman, BA1
Bender, AS; Hertz, L1
Burnham, WM; Kish, SJ; Niznik, HB1
Beaumont, K; Fanestil, DD; Healy, DP1
Fioretti, P; Galbani, P; Gambacciani, M; Melis, G; Ronca-Testoni, S1
Anderson, RA; Mitchell, R1
Bylund, DB; Feller, DJ; Schroeder, F1
Keane, P; Morre, M1
Dudai, Y; Sherman-Gold, R1
Deshmukh, P; Morelli, M; Schoemaker, H; Yamamura, HI1
Sher, PK1
Burnham, WM; Kish, SJ; Niznik, HB; Okazaki, MM1
Bolger, GT; Isaac, L; Paul, SM; Skolnick, P; Weissman, BA1
Garattini, S; Mennini, T1
Hirsch, JD1
Crow, TJ; Mashal, RD; Owen, F; Poulter, M; Waddington, JL1
Cott, J; Hommer, D; Paul, S; Quirion, R; Skolnick, P; Weissman, BA1
Cazin, L; Louiset, E; Vaudry, H1
Alenfall, J; Batra, S1
Giannaccini, G; Lucacchini, A; Martini, C; Piccolino, M; Strettoi, E1
Barton, JM; Olson, MS; Svetlov, SI1
Courtiere, A; Molard, F; Reybaud, J1
Nakamoto, Y; Shiotani, T; Watabe, S; Yoshii, M1
Friend, JM; Gee, KW; Xue, BG1
Biggio, G; Cagetti, E; Franco, M; Genchi, G; Latrofa, A; Liso, G; Ricciardi, L; Sanna, E; Trapani, G; Tuveri, F1
Chaki, S; Nagamine, M; Nakazato, A; Ogawa, S; Okubo, T; Okuyama, S; Suzuki, Y; Tomisawa, K; Yoshikawa, R1
Bono, F; Herbert, JM; Lamarche, I; Le Fur, G; Prabonnaud, V1
Kitazumi, K; Mori, M; Noguchi, H; Shiba, T1
Lopes, DV; Mendonça-Silva, DL; Noël, F; Thibaut, JP1
Elbim, C; Fasseu, M; Issop, L; Lacapere, JJ; Ostuni, MA; Papadopoulos, V; Péranzi, G; Walker, F1
Haenisch, B; Huber, M; Molderings, GJ; Steffens, M; Wilhelm, T1
Novozheeva, TP; Shushpanova, TV; Solonskii, AV; Udut, VV1

Reviews

1 review(s) available for ro 5-4864 and flunitrazepam

ArticleYear
[Is the benzodiazepine binding site a receptor?].
    L'Encephale, 1983, Volume: 9, Issue:4 Suppl 2

    Topics: Animals; Anti-Anxiety Agents; Benzodiazepinones; Binding Sites; Binding, Competitive; Brain; Brain Chemistry; Carbolines; Cats; Flunitrazepam; Pyridazines; Rats; Receptors, Cell Surface; Receptors, GABA-A; Receptors, Neurotransmitter; Structure-Activity Relationship

1983

Other Studies

69 other study(ies) available for ro 5-4864 and flunitrazepam

ArticleYear
Electronic factors in the structure-activity relationship of some 1,4-benzodiazepin-2-ones.
    Journal of medicinal chemistry, 1977, Volume: 20, Issue:9

    Topics: Benzodiazepinones; Electrochemistry; Structure-Activity Relationship

1977
Synthesis and biological evaluation of 4-phenylquinazoline-2-carboxamides designed as a novel class of potent ligands of the translocator protein.
    Journal of medicinal chemistry, 2012, May-10, Volume: 55, Issue:9

    Topics: Animals; Binding, Competitive; Carrier Proteins; Cell Line, Tumor; Cell Survival; Inhibitory Concentration 50; Molecular Structure; Quinazolines; Rats; Receptors, GABA-A; Structure-Activity Relationship

2012
Sex differences in sensitivity to pentylenetetrazol but not in GABAA receptor binding.
    Pharmacology, biochemistry, and behavior, 1992, Volume: 43, Issue:2

    Topics: Anesthetics; Animals; Anticonvulsants; Autoradiography; Benzodiazepinones; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Convulsants; Diazepam; Electroshock; Ethanol; Female; Flunitrazepam; Male; Muscimol; Orchiectomy; Ovariectomy; Pentylenetetrazole; Pregnanediones; Rats; Rats, Sprague-Dawley; Receptors, GABA-A; Seizures; Sex Characteristics

1992
Correlation between exploratory activity in an elevated plus-maze and number of central and peripheral benzodiazepine binding sites.
    Naunyn-Schmiedeberg's archives of pharmacology, 1991, Volume: 343, Issue:3

    Topics: Adrenal Glands; Animals; Behavior, Animal; Benzodiazepinones; Blood Platelets; Brain; Convulsants; Flunitrazepam; Kidney; Lymphocytes; Male; Myocardium; Rats; Receptors, GABA-A; Tritium

1991
Oxygen-induced modifications of benzodiazepine receptors and D2 dopamine receptors in the rat under hyperoxia.
    Free radical research communications, 1991, Volume: 15, Issue:1

    Topics: Animals; Benzodiazepinones; Cerebral Cortex; Corpus Striatum; Down-Regulation; Flunitrazepam; Hyperbaric Oxygenation; Kidney; Liver; Mitochondria; Oxygen; Rats; Receptors, Dopamine; Receptors, GABA-A; Spiperone

1991
Effects of phenobarbital and phenytoin on cortical glial cells in culture.
    Brain & development, 1991, Volume: 13, Issue:4

    Topics: Animals; Animals, Newborn; Benzodiazepinones; Cells, Cultured; Cerebral Cortex; Flunitrazepam; Mice; Neuroglia; Phenobarbital; Phenytoin; Radioligand Assay

1991
Stress-protection action of beta-phenyl(GABA): involvement of central and peripheral type benzodiazepine binding sites.
    Pharmacology & toxicology, 1990, Volume: 66, Issue:1

    Topics: Animals; Behavior, Animal; Benzodiazepinones; Blood Proteins; Carbolines; Drug Combinations; Female; Flunitrazepam; gamma-Aminobutyric Acid; Male; Premedication; Rats; Rats, Inbred Strains; Receptors, GABA-A; Stress, Physiological; Time Factors

1990
Peripheral-type benzodiazepine receptors are highly concentrated in mitochondrial membranes of rat testicular interstitial cells.
    Neuroendocrinology, 1990, Volume: 52, Issue:4

    Topics: Animals; Benzodiazepinones; Binding, Competitive; Diazepam; Flunitrazepam; Intracellular Membranes; Isoquinolines; Kinetics; Leydig Cells; Male; Mitochondria; Rats; Rats, Inbred Strains; Receptors, GABA-A

1990
Effect of ferric nitrilotriacetate on predominantly cortical glial cell cultures.
    Neurochemical research, 1990, Volume: 15, Issue:5

    Topics: Acetates; Animals; Animals, Newborn; Benzodiazepinones; Cells, Cultured; Cerebral Cortex; Ferric Compounds; Flunitrazepam; Mice; Neuroglia; Nitrilotriacetic Acid; Proteins; Time Factors

1990
Laudanosine does not displace receptor-specific ligands from the benzodiazepinergic or muscarinic receptors.
    Anesthesiology, 1989, Volume: 70, Issue:1

    Topics: Animals; Benzodiazepinones; Cerebral Cortex; Flunitrazepam; Isoquinolines; Kidney; Quinuclidinyl Benzilate; Rats; Rats, Inbred Strains; Receptors, GABA-A; Receptors, Muscarinic; Seizures

1989
In vivo and in vitro modulation of central type benzodiazepine receptors by phosphatidylserine.
    Brain research. Molecular brain research, 1989, Volume: 5, Issue:1

    Topics: Animals; Benzodiazepinones; Brain; Cattle; Cell Membrane; Cerebellum; Cerebral Cortex; Convulsants; Flunitrazepam; Hippocampus; Kinetics; Liposomes; Phosphatidylserines; Rats; Rats, Inbred Strains; Receptors, GABA-A; Reference Values

1989
Central- and peripheral-type benzodiazepine receptors: similar regulation by stress and GABA receptor agonists.
    Pharmacology, biochemistry, and behavior, 1989, Volume: 32, Issue:4

    Topics: Animals; Anxiety; Baclofen; Behavior, Animal; Benzodiazepinones; Binding Sites; Brain; Flunitrazepam; gamma-Aminobutyric Acid; Kidney; Male; Mice; Muscimol; Myocardium; Rats; Receptors, GABA-A; Stress, Physiological

1989
Effect of ferric nitrilotriacetate on predominantly cortical neuronal cell cultures.
    Neurochemical research, 1989, Volume: 14, Issue:7

    Topics: Acetates; Animals; Benzodiazepinones; Binding, Competitive; Cerebral Cortex; Choline O-Acetyltransferase; Clonazepam; Ferric Compounds; Flunitrazepam; gamma-Aminobutyric Acid; Mice; Neurons; Nitrilotriacetic Acid; Proteins

1989
CGS 8216 treatment decreases central-type benzodiazepine receptors in rat brain.
    European journal of pharmacology, 1987, Oct-27, Volume: 142, Issue:3

    Topics: Animals; Benzodiazepines; Benzodiazepinones; Brain; Carbolines; Convulsants; Flunitrazepam; Male; Pyrazoles; Rats; Receptors, GABA-A

1987
Stress increases endogenous benzodiazepine receptor ligand-monoamine oxidase inhibitory activity (tribulin) in rat tissues.
    Journal of neural transmission, 1988, Volume: 71, Issue:1

    Topics: Animals; Benzodiazepinones; Catecholamines; Flunitrazepam; Isatin; Kidney; Male; Monoamine Oxidase; Monoamine Oxidase Inhibitors; Myocardium; Rats; Rats, Inbred Strains; Receptors, GABA-A; Restraint, Physical; Stress, Physiological

1988
Studies on benzodiazepine receptor subtypes in a model of chronic spontaneous petit mal-like seizures.
    Neuroscience letters, 1988, Jan-11, Volume: 84, Issue:1

    Topics: Animals; Benzodiazepinones; Cerebellum; Cerebral Cortex; Chronic Disease; Epilepsy, Absence; Flunitrazepam; Hippocampus; Rats; Rats, Inbred Strains; Receptors, GABA-A; Reference Values

1988
Benzodiazepine interactions with GABAA receptors on chick ciliary ganglion neurons.
    Molecular pharmacology, 1988, Volume: 34, Issue:2

    Topics: Animals; Benzodiazepines; Benzodiazepinones; Cell Membrane; Cells, Cultured; Chick Embryo; Flumazenil; Flunitrazepam; Ganglia, Parasympathetic; Membrane Potentials; Receptors, GABA-A; Spinal Cord

1988
Presence of peripheral-type benzodiazepine binding sites on human erythrocyte membranes.
    European journal of pharmacology, 1988, Jul-26, Volume: 152, Issue:1-2

    Topics: Benzodiazepinones; Clonazepam; Convulsants; Erythrocyte Membrane; Flunitrazepam; Humans; In Vitro Techniques; Isoquinolines; Kinetics; Monoamine Oxidase; Receptors, GABA-A

1988
Effect of benzodiazepines and pentobarbital on the GABA-induced depolarization in cultured astrocytes.
    Glia, 1988, Volume: 1, Issue:2

    Topics: Animals; Astrocytes; Benzodiazepines; Benzodiazepinones; Brain; Cells, Cultured; Flunitrazepam; gamma-Aminobutyric Acid; Membrane Potentials; Pentobarbital; Rats; Rats, Inbred Strains; Receptors, GABA-A

1988
Triazolam, an anomalous benzodiazepine receptor ligand: in vitro characterization of alprazolam and triazolam binding.
    Journal of neurochemistry, 1985, Volume: 45, Issue:2

    Topics: Alprazolam; Animals; Anti-Anxiety Agents; Benzodiazepines; Benzodiazepinones; Carbolines; Clonazepam; Flunitrazepam; gamma-Aminobutyric Acid; Humans; Kinetics; Male; Rats; Rats, Inbred Strains; Receptors, GABA-A; Triazolam

1985
Neurotransmitter changes during development of cortical neuronal cultures.
    Developmental neuroscience, 1986, Volume: 8, Issue:2

    Topics: Animals; Benzodiazepinones; Cells, Cultured; Cerebral Cortex; Choline O-Acetyltransferase; Clonazepam; Diazepam; Fetus; Flunitrazepam; gamma-Aminobutyric Acid; Glutamate Decarboxylase; Mice; Neurotransmitter Agents

1986
Tetrazepam: a benzodiazepine which dissociates sedation from other benzodiazepine activities. II. In vitro and in vivo interactions with benzodiazepine binding sites.
    The Journal of pharmacology and experimental therapeutics, 1988, Volume: 245, Issue:2

    Topics: Animals; Anti-Anxiety Agents; Autoradiography; Benzodiazepines; Benzodiazepinones; Binding, Competitive; Brain; Cell Membrane; Convulsants; Flunitrazepam; Kidney; Kinetics; Male; Mice; Rats; Receptors, GABA-A; Tritium

1988
[Presence of a peripheral type benzodiazepine binding site on the macrophage; its possible role in immunomodulation].
    Comptes rendus de l'Academie des sciences. Serie III, Sciences de la vie, 1985, Volume: 300, Issue:8

    Topics: Animals; Antibody Formation; Benzodiazepines; Benzodiazepinones; Clonazepam; Erythrocytes; Ethanol; Female; Flunitrazepam; Macrophages; Mice; Receptors, GABA-A; Sheep

1985
Late evolutionary appearance of 'peripheral-type' binding sites for benzodiazepines.
    Brain research, 1985, Jul-15, Volume: 338, Issue:2

    Topics: Animals; Benzodiazepinones; Biological Evolution; Brain Chemistry; Columbidae; Flunitrazepam; Lizards; Male; Organ Specificity; Radioligand Assay; Rana catesbeiana; Rats; Rats, Inbred Strains; Receptors, GABA-A; Trout; Vertebrates

1985
Brain gamma-aminobutyric acid and benzodiazepine receptor binding in dialysis encephalopathy.
    Neuroscience letters, 1985, Jul-31, Volume: 58, Issue:2

    Topics: Benzodiazepinones; Brain Diseases; Flunitrazepam; Frontal Lobe; gamma-Aminobutyric Acid; Humans; Middle Aged; Receptors, GABA-A; Renal Dialysis

1985
Monoclonal antibodies to benzodiazepines.
    Journal of neurochemistry, 1985, Volume: 45, Issue:6

    Topics: Animals; Anti-Anxiety Agents; Antibodies, Monoclonal; Benzodiazepines; Benzodiazepinones; Diazepam; Flumazenil; Flunitrazepam; Flurazepam; Mice; Mice, Inbred BALB C; Receptors, GABA-A; Structure-Activity Relationship

1985
Autoradiographic localization of benzodiazepine receptor binding in dissociated cultures of fetal mouse cerebral cortex.
    Journal of neurochemistry, 1986, Volume: 46, Issue:3

    Topics: Affinity Labels; Animals; Autoradiography; Benzodiazepinones; Binding, Competitive; Cells, Cultured; Cerebral Cortex; Clonazepam; Embryo, Mammalian; Flunitrazepam; Mice; Neurons; Photochemistry; Receptors, GABA-A

1986
Evidence of specific benzodiazepine binding to myometrial membrane preparations from human pregnant uterus.
    Acta obstetricia et gynecologica Scandinavica, 1986, Volume: 65, Issue:4

    Topics: Adult; Benzodiazepines; Benzodiazepinones; Cell Membrane; Chlordiazepoxide; Diazepam; Female; Flunitrazepam; Humans; Lorazepam; Myometrium; Pregnancy; Receptors, Cell Surface

1986
Central- and peripheral-type benzodiazepine receptors.
    Advances in biochemical psychopharmacology, 1986, Volume: 41

    Topics: Animals; Benzodiazepinones; Binding, Competitive; Brain; Clonazepam; Convulsants; Flunitrazepam; Kidney; Kinetics; Membranes; Muscimol; Rats; Receptors, GABA-A; Subcellular Fractions; Tissue Distribution

1986
'Peripheral' and 'central' type benzodiazepine receptors in Maudsley rats.
    European journal of pharmacology, 1986, Jul-31, Volume: 126, Issue:3

    Topics: Animals; Behavior, Animal; Benzodiazepinones; Brain; Carbolines; Female; Flunitrazepam; Kinetics; Male; Rats; Rats, Mutant Strains; Receptors, GABA-A; Tissue Distribution

1986
Pyrazolo[4,5-c]quinolines. 3. Synthesis, receptor binding, and 13C NMR study.
    Journal of pharmaceutical sciences, 1986, Volume: 75, Issue:12

    Topics: Animals; Benzodiazepinones; Binding, Competitive; Brain; Cattle; Chemical Phenomena; Chemistry; Clonazepam; Flunitrazepam; In Vitro Techniques; Magnetic Resonance Spectroscopy; Pyrazoles; Quinolines; Receptors, GABA-A

1986
Coexistence of central and peripheral benzodiazepine binding sites in the human pineal gland.
    Life sciences, 1987, Apr-13, Volume: 40, Issue:15

    Topics: Aged; Benzodiazepinones; Binding, Competitive; Cell Membrane; Clonazepam; Female; Flumazenil; Flunitrazepam; Humans; Isoquinolines; Male; Middle Aged; Pineal Gland; Receptors, GABA-A

1987
Increase of peripheral type benzodiazepine binding sites in kidney and olfactory bulb in acutely stressed rats.
    European journal of pharmacology, 1987, Mar-17, Volume: 135, Issue:2

    Topics: Animals; Benzodiazepinones; Cerebral Cortex; Convulsants; Female; Flunitrazepam; Kidney; Kinetics; Male; Olfactory Bulb; Rats; Rats, Inbred Strains; Receptors, GABA-A; Stress, Psychological

1987
Benzodiazepine receptor affinity alterations at physiologic temperature after chronic clonazepam exposure.
    Brain & development, 1987, Volume: 9, Issue:1

    Topics: Animals; Benzodiazepinones; Body Temperature; Cells, Cultured; Cerebral Cortex; Clonazepam; Convulsants; Flunitrazepam; Kinetics; Mice; Receptors, GABA-A; Time Factors

1987
Isoquinoline and peripheral-type benzodiazepine binding in gliomas: implications for diagnostic imaging.
    Cancer research, 1988, Oct-15, Volume: 48, Issue:20

    Topics: Benzodiazepines; Benzodiazepinones; Brain Neoplasms; Cells, Cultured; Flunitrazepam; Glioma; Humans; Isoquinolines; Kinetics; Tomography, Emission-Computed

1988
Identification, characterization, and developmental regulation of embryonic benzodiazepine binding sites.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 1987, Volume: 7, Issue:6

    Topics: Affinity Labels; Animals; Benzodiazepines; Benzodiazepinones; Binding Sites; Brain; Chick Embryo; Flunitrazepam; Kinetics; Membranes; Time Factors; Tritium

1987
Characterization of peripheral-type benzodiazepine recognition sites in the rat spinal cord.
    Neuropharmacology, 1985, Volume: 24, Issue:2

    Topics: Animals; Benzodiazepines; Benzodiazepinones; Binding Sites; Brain; Diazepam; Flunitrazepam; Kinetics; Male; Rats; Rats, Inbred Strains; Spinal Cord

1985
Differential regulation of 'central' and 'peripheral' benzodiazepine binding sites in the rat olfactory bulb.
    European journal of pharmacology, 1984, Oct-01, Volume: 105, Issue:1-2

    Topics: Animals; Benzodiazepines; Benzodiazepinones; Cerebellum; Convulsants; Flunitrazepam; Kinetics; Male; Olfactory Bulb; Pentylenetetrazole; Rats; Rats, Inbred Strains; Receptors, GABA-A

1984
Flunitrazepam binding to intact and homogenized astrocytes and neurons in primary cultures.
    Journal of neurochemistry, 1984, Volume: 43, Issue:5

    Topics: Animals; Astrocytes; Benzodiazepinones; Cells, Cultured; Clonazepam; Diazepam; Flunitrazepam; Kinetics; Mice; Neurons; Receptors, GABA-A; Temperature

1984
Benzodiazepine receptor binding following amygdala-kindled convulsions: differing results in washed and unwashed brain membranes.
    Journal of neurochemistry, 1984, Volume: 43, Issue:6

    Topics: Amygdala; Animals; Benzodiazepinones; Brain; Buffers; Cell Membrane; Cerebral Cortex; Flunitrazepam; gamma-Aminobutyric Acid; Hypothalamus; Kindling, Neurologic; Male; Rats; Receptors, GABA-A; Seizures; Specimen Handling

1984
Autoradiographic localization of benzodiazepine receptors in the rat kidney.
    The American journal of physiology, 1984, Volume: 247, Issue:5 Pt 2

    Topics: Animals; Autoradiography; Benzodiazepinones; Clonazepam; Diazepam; Flunitrazepam; Kidney; Kidney Tubules, Distal; Loop of Henle; Male; Mucoproteins; Rats; Rats, Inbred Strains; Receptors, GABA-A; Tritium; Uromodulin

1984
Benzodiazepine binding sites in human myometrium.
    International journal of tissue reactions, 1984, Volume: 6, Issue:5

    Topics: Adult; Benzodiazepinones; Binding Sites; Cell Membrane; Clonazepam; Diazepam; Female; Flunitrazepam; Humans; In Vitro Techniques; Lorazepam; Middle Aged; Myometrium; Receptors, GABA-A

1984
Analysis of benzodiazepine binding sites in rat pituitary gland.
    Brain research, 1984, Dec-10, Volume: 323, Issue:2

    Topics: Animals; Benzodiazepinones; Binding, Competitive; Clonazepam; Diazepam; Flunitrazepam; gamma-Aminobutyric Acid; In Vitro Techniques; Male; Pituitary Gland; Rats; Rats, Inbred Strains; Receptors, GABA-A

1984
Binding of [3H]flunitrazepam to the LM cell, a transformed murine fibroblast.
    Biochemical pharmacology, 1983, Jul-15, Volume: 32, Issue:14

    Topics: Animals; Anti-Anxiety Agents; Benzodiazepinones; Binding Sites; Cell Line; Cell Membrane; Choline; Clonazepam; Culture Media; Cyclic AMP; Flunitrazepam; Kinetics; Mice; Neoplasms, Experimental; Phospholipids

1983
Involvement of tyrosyl residues in the binding of benzodiazepines to their brain receptors.
    FEBS letters, 1981, Aug-31, Volume: 131, Issue:2

    Topics: Animals; Benzodiazepines; Benzodiazepinones; Brain; Cattle; Diazepam; Flunitrazepam; gamma-Aminobutyric Acid; Imidazoles; Nitrazepam; Receptors, Drug; Receptors, GABA-A; Receptors, Neurotransmitter; Tetranitromethane; Tyrosine

1981
[3H]Ro5-4864 benzodiazepine binding in the kainate lesioned striatum and Huntington's diseased basal ganglia.
    Brain research, 1982, Sep-30, Volume: 248, Issue:2

    Topics: Aged; Animals; Benzodiazepinones; Binding Sites; Corpus Striatum; Flunitrazepam; Humans; Huntington Disease; Kainic Acid; Male; Middle Aged; Neuroglia; Pyrrolidines; Rats; Rats, Inbred Strains; Receptors, Drug; Receptors, GABA-A

1982
Development and differentiation of the benzodiazepine receptor in cultures of fetal mouse spinal cord.
    Brain research, 1983, Volume: 283, Issue:2-3

    Topics: Animals; Benzodiazepinones; Cell Differentiation; Clonazepam; Diazepam; Fetus; Flunitrazepam; Kinetics; Mice; Neurons; Receptors, Cell Surface; Receptors, GABA-A; Spinal Cord

1983
Binding of [3H]flunitrazepam and [3H]Ro5-4864 to crude homogenates of amygdala-kindled rat brain: two months post-seizure.
    Brain research, 1983, Nov-21, Volume: 279, Issue:1-2

    Topics: Amygdala; Animals; Benzodiazepinones; Brain; Flunitrazepam; Kindling, Neurologic; Kinetics; Male; Muridae; Receptors, Cell Surface; Receptors, GABA-A; Seizures

1983
Characterization of the binding of [3H]Ro 5-4864, a convulsant benzodiazepine, to guinea pig brain.
    Journal of neurochemistry, 1984, Volume: 42, Issue:4

    Topics: Animals; Benzodiazepinones; Binding Sites; Brain; Cats; Convulsants; Diazepam; Flunitrazepam; Guinea Pigs; Kinetics; Male; Mice; Rats; Receptors, Cell Surface; Receptors, GABA-A; Species Specificity; Tissue Distribution

1984
Benzodiazepines receptor binding in vivo: pharmacokinetic and pharmacological significance.
    Advances in biochemical psychopharmacology, 1983, Volume: 38

    Topics: Adrenal Glands; Animals; Benzodiazepinones; Brain; Carbolines; Corticosterone; Diazepam; Flumazenil; Flunitrazepam; Kinetics; Rats; Receptors, Cell Surface; Receptors, GABA-A

1983
Specific [3H]Ro 5-4864 binding to rat spinal cord membranes: evidence for peripheral type benzodiazepine recognition sites.
    Neuroscience letters, 1984, May-18, Volume: 46, Issue:3

    Topics: Animals; Benzodiazepines; Benzodiazepinones; Binding, Competitive; Cell Membrane; Flunitrazepam; Kinetics; Male; Rats; Rats, Inbred Strains; Receptors, Cell Surface; Receptors, GABA-A; Spinal Cord

1984
Peripheral and central-type benzodiazepine binding sites in mammalian ocular tissues.
    Experimental eye research, 1984, Volume: 38, Issue:1

    Topics: Animals; Benzodiazepines; Benzodiazepinones; Binding Sites; Eye; Female; Flumazenil; Flunitrazepam; Macaca mulatta; Male; Rabbits; Rats; Rats, Inbred Strains

1984
[3H]R05-4864 and [3H]flunitrazepam binding in kainate-lesioned rat striatum and in temporal cortex of brains from patients with senile dementia of the Alzheimer type.
    Brain research, 1983, Nov-14, Volume: 278, Issue:1-2

    Topics: Aged; Alzheimer Disease; Animals; Benzodiazepinones; Binding Sites; Corpus Striatum; Female; Flunitrazepam; Glutamate Decarboxylase; Humans; Kainic Acid; Male; Pyrrolidines; Rats; Temporal Lobe; Tritium

1983
Pharmacological, electrophysiological, and neurochemical actions of the convulsant benzodiazepine Ro 5-4864 (4'-chlordiazepam).
    Advances in biochemical psychopharmacology, 1983, Volume: 38

    Topics: Animals; Autoradiography; Benzodiazepinones; Brain Chemistry; Cats; Convulsants; Electrophysiology; Flunitrazepam; Guinea Pigs; Male; Mice; Neurons; Rats; Rats, Inbred Strains; Subcellular Fractions

1983
Allosteric modulation of the GABA-induced chloride current in frog melanotrophs.
    Annals of the New York Academy of Sciences, 1993, May-31, Volume: 680

    Topics: Action Potentials; Allosteric Regulation; Animals; Anti-Anxiety Agents; Azepines; Benzodiazepinones; Chloride Channels; Convulsants; Diazepam; Flunitrazepam; gamma-Aminobutyric Acid; Ion Channels; Melanocyte-Stimulating Hormones; Membrane Proteins; Pituitary Gland; Ranidae; Receptors, GABA-A

1993
Characterization of peripheral benzodiazepine receptors in rat prostatic adenocarcinoma.
    The Prostate, 1994, Volume: 24, Issue:5

    Topics: Adenocarcinoma; Animals; Benzodiazepinones; Binding, Competitive; Diazepam; Flunitrazepam; Isoquinolines; Male; Mesoporphyrins; Microsomes; Mitochondria; Neoplasm Transplantation; Prostatic Neoplasms; Rats; Receptors, GABA-A

1994
The peripheral-type benzodiazepine receptor ligands [3H]Ro 5-4864 and [3H]PK 11195 bind to the retina of rabbit, but not of turtle.
    Journal of neurochemistry, 1993, Volume: 61, Issue:4

    Topics: Animals; Benzodiazepinones; Flunitrazepam; Isoquinolines; Ligands; Rabbits; Receptors, GABA-A; Retina; Tritium; Turtles

1993
The specific binding of the platelet-activating factor (PAF) receptor antagonist WEB 2086 and the benzodiazepine flunitrazepam to rat hepatocytes.
    Life sciences, 1996, Volume: 58, Issue:5

    Topics: Animals; Anti-Anxiety Agents; Anticonvulsants; Azepines; Benzodiazepinones; Bicuculline; Cells, Cultured; Clonazepam; Convulsants; Flunitrazepam; Kinetics; Liver; Male; Platelet Aggregation Inhibitors; Platelet Membrane Glycoproteins; Rats; Rats, Sprague-Dawley; Receptors, Cell Surface; Receptors, G-Protein-Coupled; Triazoles; Tritium

1996
Differential effects of in vitro peroxidation on peripheral- and central-type benzodiazepine receptors. Protection by diverse antioxidants.
    Biochemical pharmacology, 1995, Nov-27, Volume: 50, Issue:11

    Topics: Animals; Antioxidants; Ascorbic Acid; Benzodiazepinones; Brain; Cell Membrane; Chromans; Deferoxamine; Edetic Acid; Ferrous Compounds; Flunitrazepam; Hypolipidemic Agents; Lipid Peroxidation; Liver; Malondialdehyde; Receptors, GABA-A; Rutin; Vitamin E

1995
Peripheral-type benzodiazepine receptors in association with epileptic seizures in EL mice.
    Brain research, 1996, Apr-22, Volume: 717, Issue:1-2

    Topics: Animals; Anti-Anxiety Agents; Benzodiazepinones; Binding Sites; Cell Fractionation; Convulsants; Epilepsy; Flunitrazepam; GABA-A Receptor Agonists; Isoquinolines; Membrane Proteins; Mice; Mice, Mutant Strains; Mitochondria; Pentylenetetrazole; Prosencephalon; Receptors, GABA-A; Tritium

1996
Loreclezole modulates [35S]t-butylbicyclophosphorothionate and [3H]flunitrazepam binding via a distinct site on the GABAA receptor complex.
    European journal of pharmacology, 1996, Apr-04, Volume: 300, Issue:1-2

    Topics: Animals; Anticonvulsants; Benzodiazepinones; Binding Sites; Brain; Bridged Bicyclo Compounds, Heterocyclic; Convulsants; Drug Interactions; Flunitrazepam; Male; Rats; Rats, Sprague-Dawley; Receptors, GABA; Triazoles

1996
Synthesis and binding affinity of 2-phenylimidazo[1,2-alpha]pyridine derivatives for both central and peripheral benzodiazepine receptors. A new series of high-affinity and selective ligands for the peripheral type.
    Journal of medicinal chemistry, 1997, Sep-12, Volume: 40, Issue:19

    Topics: Animals; Benzodiazepinones; Binding, Competitive; Brain; Female; Flunitrazepam; Humans; Hypnotics and Sedatives; Imidazoles; Kidney; Kinetics; Male; Mitochondria; Molecular Structure; Oocytes; Pyridines; Radioligand Assay; Rats; Rats, Wistar; Receptors, GABA-A; Recombinant Proteins; Structure-Activity Relationship; Xenopus laevis; Zolpidem

1997
Neuropharmacological profile of peripheral benzodiazepine receptor agonists, DAA1097 and DAA1106.
    Life sciences, 1999, Volume: 64, Issue:16

    Topics: Acetamides; Anesthesia; Animals; Anti-Anxiety Agents; Benzodiazepinones; Brain; Buspirone; Cell Membrane; Diazepam; Exploratory Behavior; Flunitrazepam; GABA Modulators; GABA-A Receptor Agonists; Hexobarbital; Isoquinolines; Male; Mice; Mice, Inbred ICR; Mitochondria; Motor Activity; Phenyl Ethers

1999
Peripheral benzodiazepine receptor agonists exhibit potent antiapoptotic activities.
    Biochemical and biophysical research communications, 1999, Nov-19, Volume: 265, Issue:2

    Topics: Apoptosis; Benzodiazepinones; Clonazepam; Diazepam; Flunitrazepam; GABA-A Receptor Agonists; GABA-A Receptor Antagonists; Humans; Isoquinolines; Jurkat Cells; Kinetics; Ligands; Receptors, GABA-A; Transfection; Tumor Necrosis Factor-alpha; U937 Cells

1999
Binding and neuropharmacological profile of zaleplon, a novel nonbenzodiazepine sedative/hypnotic.
    European journal of pharmacology, 2002, Jan-02, Volume: 434, Issue:1-2

    Topics: Acetamides; Animals; Benzodiazepinones; Electroencephalography; Flunitrazepam; gamma-Aminobutyric Acid; Hypnotics and Sedatives; Male; Muscimol; Pyrimidines; Rabbits; Rats; Rats, Sprague-Dawley; Sleep

2002
Characterization of two classes of benzodiazepine binding sites in Schistosoma mansoni.
    Parasitology, 2007, Volume: 134, Issue:Pt 7

    Topics: Animals; Benzodiazepines; Benzodiazepinones; Binding Sites; Clonazepam; Diazepam; Flunitrazepam; GABA Agonists; GABA Modulators; Inhibitory Concentration 50; Isoquinolines; Ligands; Male; Pyridines; Rats; Rats, Wistar; Receptors, GABA-A; Schistosoma mansoni; Synaptosomes; Temperature; Time Factors; Tritium; Zolpidem

2007
Overexpression of translocator protein in inflammatory bowel disease: potential diagnostic and treatment value.
    Inflammatory bowel diseases, 2010, Volume: 16, Issue:9

    Topics: Animals; Antineoplastic Agents; Benzodiazepinones; Carrier Proteins; Case-Control Studies; Colitis; Colon; Colonic Neoplasms; Cytokines; Dextran Sulfate; Enterocytes; Flunitrazepam; GABA Modulators; Humans; Hypolipidemic Agents; Immunoenzyme Techniques; Inflammatory Bowel Diseases; Isoquinolines; Male; Mitochondria; Rats; Rats, Wistar; Receptors, GABA; Receptors, GABA-A; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger

2010
Investigation into mechanisms mediating the inhibitory effect of 1,4-benzodiazepines on mast cells by gene expression profiling.
    Life sciences, 2013, Mar-14, Volume: 92, Issue:6-7

    Topics: Adult; Aged; Benzodiazepinones; Clonazepam; Female; Flunitrazepam; Gene Expression; Gene Expression Profiling; HL-60 Cells; Humans; Male; Mast Cells; Mastocytosis; Microarray Analysis; Middle Aged; Polymerase Chain Reaction

2013
Effect of meta-chlorobenzhydryl urea (m-ClBHU) on benzodiazepine receptor system in rat brain during experimental alcoholism.
    Bulletin of experimental biology and medicine, 2014, Volume: 156, Issue:6

    Topics: Alcoholism; Animals; Anticonvulsants; Benzodiazepinones; Brain; Flunitrazepam; gamma-Aminobutyric Acid; Genetic Predisposition to Disease; Hydrocarbons, Chlorinated; Male; Phenylurea Compounds; Rats; Rats, Wistar; Receptors, GABA-A; Synaptic Transmission; Tritium

2014