ro 5-4864 has been researched along with clonazepam in 98 studies
Timeframe | Studies, this research(%) | All Research% |
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pre-1990 | 54 (55.10) | 18.7374 |
1990's | 33 (33.67) | 18.2507 |
2000's | 8 (8.16) | 29.6817 |
2010's | 1 (1.02) | 24.3611 |
2020's | 2 (2.04) | 2.80 |
Authors | Studies |
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Blair, T; Webb, GA | 1 |
Campiani, G; Ciani, SM; De Filippis, MP; Fiorini, I; Garofalo, A; Greco, G; Manzoni, C; Mennini, T; Mihai, C; Nacci, V; Novellino, E; Williams, DC; Woods, MJ; Zisterer, DM | 1 |
Cleary, J; Glick, GD; Johnson, KM; Opipari, AW | 1 |
Baglini, E; Barresi, E; Robello, M; Salerno, S; Settimo, FD; Taliani, S | 1 |
Advenier, C; Candenas, ML; Devillier, P; Naline, E | 1 |
Järvinen, A; Männistö, PT; Rägo, L | 1 |
Berdeu, D; Loubatières-Mariani, MM; Manteghetti, M; Petit, P; Ribes, G | 1 |
Diana, G; Massotti, M | 1 |
Järvinen, A; Männistö, PT; Paakkari, I | 1 |
Becker, DP; Black, KL; Ikezaki, K; Shiraishi, T | 1 |
Abraham, S; Bolger, GT; Oz, N; Weissman, BA | 1 |
Bravo, C; Chiang, PK; Gutiérrez, J; Moreno-Sánchez, R; Newman, AH | 1 |
Lichtensteiger, W; Parmar, R; Ramseier, HR; Schlumpf, M | 1 |
Izquierdo, I; Medina, JH; Pereira, ME | 1 |
Elgoyhen, AB; Kazanietz, MG | 1 |
O'Beirne, GB; Williams, DC; Woods, MJ | 1 |
De Luca, C; Massotti, M; Mele, L | 1 |
Sher, PK | 3 |
Griffith, JA; Woolley, DE | 1 |
Adler-Graschinsky, E; Elgoyhen, B | 1 |
Daval, JL; Marangos, PJ; Post, RM | 1 |
Gorman, AM; O'Beirne, GB; Regan, CM; Williams, DC | 1 |
Duerson, KC; Gerrish, KE; Laird, HE; Putnam, CW; Russell, DH | 1 |
Calandra, RS; Ritta, MN | 1 |
Machen, VL; Swaiman, KF | 1 |
Sher, PK; Talwar, D | 1 |
Brinton, RE; Gee, KW; McEwen, BS | 1 |
Salmona, M; Tacconi, MT | 1 |
Ciliax, BJ; Mancini, WR; Olson, JM; Young, AB | 1 |
Basile, AS; Crawley, JN; Drugan, RC; Paul, SM; Skolnick, P | 1 |
Randall, JI; Rodgers, RJ | 1 |
Clow, A; Glover, V; Sandler, M | 1 |
Boespflug, O; Swaiman, KF | 1 |
Falk, JL; Plaessmann, WR; Tang, M | 1 |
Anholt, RR; De Souza, EB; Kuhar, MJ; Murphy, KM; Snyder, SH | 1 |
Haumont, J; Lenfant, M; Potier, P; Zavala, F | 1 |
Cooper, SJ; Gilbert, DB | 1 |
Paul, SM; Pert, CB; Ruff, MR; Wahl, LM; Wahl, SM; Weber, RJ | 1 |
Cole, R; De Vellis, J; Noble, EP; Syapin, PJ | 1 |
Fares, F; Gavish, M | 1 |
Belin, C; Carriot, T; Dubroeucq, MC; Guérémy, C; Le Fur, G; Mestre, M; Renault, C; Uzan, A | 2 |
Machen, VL; Neale, EA; Sher, PK | 1 |
Bryere, P; Naquet, R; Valin, A | 1 |
Deckert, J; Marangos, PJ | 1 |
Hrelia, S; Lucacchini, A; Martini, C; Rossi, CA | 1 |
Cecchi, L; Filacchioni, G; Lucacchini, A; Martini, C; Melani, F; Palazzino, G; Pennacchi, E | 1 |
Lafaille, F; Lal, S; Nair, NP; Quirion, R; Suranyi-Cadotte, B | 1 |
Machen, VL; Sher, PK | 2 |
Lenfant, M; Zavala, F | 1 |
Teo, WL; Wong, PT | 1 |
Kunert-Radek, J; Pawlikowski, M; Radek, A; Stepien, H | 1 |
Brown, T; Fogel, R; Gaginella, T; Marshall, D; Michelson, G; Senler, T | 1 |
French, JF; Grupp, IL; Matlib, MA | 1 |
Brown, C; Martin, IL | 1 |
Bender, AS; Hertz, L | 1 |
Beaumont, K; Fanestil, DD; Healy, DP | 1 |
Fioretti, P; Galbani, P; Gambacciani, M; Melis, G; Ronca-Testoni, S | 1 |
Anderson, RA; Mitchell, R | 1 |
Bylund, DB; Feller, DJ; Schroeder, F | 1 |
Spector, S; Taniguchi, T; Wang, JK | 1 |
Benavides, J; Dubroeucq, MC; Flamier, A; Guérémy, C; Imbault, F; Le Fur, G; Perrier, ML; Renault, C; Uzan, A; Vaucher, N | 1 |
Benavides, J; Dubroeucq, MC; Guérémy, C; Guilloux, F; Le Fur, G; Renault, C; Rufat, P; Uzan, A | 1 |
Benavides, J; Dubroeucq, MC; Flamier, A; Guérémy, C; Le Fur, G; Perrier, ML; Renault, C; Uzan, A; Vaucher, N | 1 |
Butlen, D | 1 |
Lichtensteiger, W; Möhler, H; Richards, JG; Schlumpf, M | 1 |
Khalansky, AS; Kondakova, LI; Zlobina, GP | 1 |
Ebel, C; Mallorga, P; Roth-Schechter, BF | 1 |
Elías, MM; Monasterolo, LA; Ochoa, JE; Trumper, L | 1 |
Antonenko, YN; Kinnally, KW; McEnery, MW; Snyder, SH; Tedeschi, H; Zorov, DB | 1 |
Chen, JS; Gee, KW; Johnson, D; Lan, NC | 1 |
Matthews, EK; Ratcliffe, SL | 1 |
Koga, K; Matsumoto, T; Ogata, M; Shigematsu, A | 1 |
Lichtensteiger, W; Ramseier, H; Schlumpf, M | 1 |
Barton, JM; Olson, MS; Svetlov, SI | 1 |
Cespuglio, R; Miachon, S | 1 |
Boujrad, N; Kotoula, M; Kozikowski, AP; Ma, D; Papadopoulos, V; Tückmantel, W | 1 |
Gavish, M; Kelly-Hershkovitz, E; Lahav, M; Leschiner, S; Spanier, I; Weisinger, G; Weizman, R | 1 |
Butterworth, RF; Rao, VL | 1 |
Caldiroli, E; Cattaneo, S; Cosentino, M; Di Grazia, L; Frigo, G; Lecchini, S; Marino, F | 1 |
Beery, E; Brenner, S; Gavish, M; Landau, M; Landau, O; Nordenberg, J; Wasseman, L; Weizman, A; Zoref-Shani, E | 1 |
Kawaguchi, M; Okubo, M | 1 |
Bender, AS; Norenberg, MD | 1 |
Kizaki, H; Onishi, Y; Sato, Y; Tanimoto, Y | 1 |
Fornai, F; Gesi, M; Lenzi, P; Natale, G; Paparelli, A; Pellegrini, A; Riva, A; Soldani, P | 1 |
Bono, F; Herbert, JM; Lamarche, I; Le Fur, G; Prabonnaud, V | 1 |
Bruni, F; Ciciani, G; Costa, B; Costagli, C; Costanzo, A; Guerrini, G; Martini, C; Selleri, S | 1 |
Gekker, G; Hegg, CC; Hu, S; Lokensgard, JR; Peterson, PK; Thayer, SA | 1 |
Kohjitani, A; Maeda, S; Miyawaki, T; Shimada, M; Sogawa, N | 1 |
Jayakumar, AR; Norenberg, MD; Panickar, KS | 1 |
Dagli, ML; Fonseca, ES; Leite, KR; Massoco, CO; Matsuzaki, P; Oloris, SC; Otake, AH; Palermo-Neto, J; Sakai, M | 1 |
Lopes, DV; Mendonça-Silva, DL; Noël, F; Thibaut, JP | 1 |
Buckingham, SD; Higashino, Y; Sattelle, DB | 1 |
Haenisch, B; Huber, M; Molderings, GJ; Steffens, M; Wilhelm, T | 1 |
Hughes, DA | 1 |
1 review(s) available for ro 5-4864 and clonazepam
Article | Year |
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The Alpha Keto Amide Moiety as a Privileged Motif in Medicinal Chemistry: Current Insights and Emerging Opportunities.
Topics: Amides; Animals; Cell Line, Tumor; Chemistry, Pharmaceutical; Humans; Ketones | 2021 |
97 other study(ies) available for ro 5-4864 and clonazepam
Article | Year |
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Electronic factors in the structure-activity relationship of some 1,4-benzodiazepin-2-ones.
Topics: Benzodiazepinones; Electrochemistry; Structure-Activity Relationship | 1977 |
Synthesis, biological activity, and SARs of pyrrolobenzoxazepine derivatives, a new class of specific "peripheral-type" benzodiazepine receptor ligands.
Topics: Animals; Benzodiazepinones; Binding Sites; Cerebral Cortex; Isoquinolines; Ligands; Mice; Rats; Rats, Wistar; Receptors, GABA-A; Structure-Activity Relationship | 1996 |
Inhibition of the mitochondrial F1F0-ATPase by ligands of the peripheral benzodiazepine receptor.
Topics: Adenosine Triphosphate; Antineoplastic Agents; Apoptosis; Benzodiazepines; Cell Line, Tumor; Cell Proliferation; GABA-A Receptor Antagonists; Humans; Hydrolysis; Isoquinolines; Kinetics; Ligands; Mitochondria; Proton-Translocating ATPases; Structure-Activity Relationship | 2007 |
Contractile effect of alpha,beta-methylene ATP on the guinea-pig isolated trachea.
Topics: 2-Chloroadenosine; Adenosine Triphosphate; Animals; Benzodiazepinones; Clonazepam; Diazepam; Drug Synergism; GABA-A Receptor Antagonists; Guinea Pigs; Male; Muscle Contraction; Muscle, Smooth; Phenylisopropyladenosine; Trachea | 1992 |
Effects of central and peripheral type benzodiazepine ligands on thyrotropin and prolactin secretion.
Topics: Animals; Benzodiazepinones; Carbolines; Clonazepam; Cold Temperature; Diazepam; Flumazenil; Hypothalamo-Hypophyseal System; Isoquinolines; Male; Pituitary Gland, Anterior; Prolactin; Rats; Rats, Inbred Strains; Receptors, GABA-A; Secretory Rate; Thyrotropin; Thyrotropin-Releasing Hormone | 1992 |
Effects of a peripheral-type benzodiazepine on glucose-induced insulin secretion.
Topics: Animals; Benzodiazepinones; Clonazepam; Glucose; In Vitro Techniques; Insulin; Insulin Secretion; Islets of Langerhans; Isoquinolines; Male; Perfusion; Rats; Rats, Wistar | 1992 |
Repeated administration of diazepam reduces [3H]Ro 5-4864 binding in cerebral cortex of rats.
Topics: Animals; Benzodiazepinones; Cerebral Cortex; Clonazepam; Diazepam; Down-Regulation; Electroencephalography; In Vitro Techniques; Male; Mitochondria; Rats; Rats, Inbred Strains | 1992 |
Central and peripheral type benzodiazepine ligands displace [3H][3-ME-HIS2]TRH from its binding sites in the brain and the anterior pituitary and antagonize the effect of TRH in the rat duodenum.
Topics: Animals; Benzodiazepinones; Binding Sites; Brain; Brain Stem; Carbolines; Clonazepam; Diazepam; Duodenum; Hypothalamus; Isoquinolines; Male; Muscle, Smooth; Pituitary Gland, Anterior; Pyrrolidonecarboxylic Acid; Rats; Rats, Inbred Strains; Receptors, GABA-A; Receptors, Neurotransmitter; Receptors, Thyrotropin-Releasing Hormone; Thyrotropin-Releasing Hormone | 1991 |
Peripheral benzodiazepine induces morphological changes and proliferation of mitochondria in glioma cells.
Topics: Animals; Benzodiazepinones; Cell Line; Clonazepam; Culture Media, Serum-Free; Fluorescent Dyes; Glioma; Isoquinolines; Microscopy, Electron; Microscopy, Fluorescence; Mitochondria; Rats; Receptors, GABA-A; Rhodamine 123; Rhodamines | 1991 |
Interactions between peripheral-type benzodiazepine receptor ligands and an activator of voltage-operated calcium channels.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Benzodiazepinones; Blood Pressure; Calcium Channels; Clonazepam; Coronary Disease; Electrocardiography; Guinea Pigs; In Vitro Techniques; Isoquinolines; Male; Myocardial Contraction; Receptors, GABA-A | 1990 |
Release of Ca2+ from heart and kidney mitochondria by peripheral-type benzodiazepine receptor ligands.
Topics: Animals; Benzodiazepines; Benzodiazepinones; Calcium; Clonazepam; Kidney; Magnesium; Mitochondria; Mitochondria, Heart; Rats; Rats, Inbred Strains; Receptors, GABA-A; Strontium | 1991 |
Prenatal benzodiazepine immunosuppression: possible involvement of peripheral benzodiazepine site.
Topics: Animals; Autoradiography; Benzodiazepinones; Binding Sites; Cell Division; Clonazepam; Convulsants; Diazepam; Female; Immune Tolerance; Immunity, Cellular; Lymphocytes; Male; Maternal-Fetal Exchange; Pregnancy; Prenatal Exposure Delayed Effects; Rats; Receptors, GABA-A | 1990 |
Benzodiazepine receptor ligand influences on acquisition: suggestion of an endogenous modulatory mechanism mediated by benzodiazepine receptors.
Topics: Animals; Anti-Anxiety Agents; Arousal; Avoidance Learning; Benzodiazepinones; Brain; Carbolines; Clonazepam; Diazepam; Dose-Response Relationship, Drug; Exploratory Behavior; Female; Flumazenil; Habituation, Psychophysiologic; Memory; Mental Recall; Rats; Rats, Inbred Strains; Reaction Time; Receptors, GABA-A; Retention, Psychology | 1990 |
Relaxant effect of benzodiazepines on uterine rings isolated from estrogen-treated rats.
Topics: Animals; Anti-Anxiety Agents; Benzodiazepinones; Bicuculline; Clonazepam; Convulsants; Diazepam; Estradiol; Estrogens; Female; Flumazenil; In Vitro Techniques; Isoquinolines; Muscle, Smooth; Potassium Chloride; Propranolol; Rats; Rats, Inbred Strains; Uterine Contraction | 1990 |
Two subcellular locations for peripheral-type benzodiazepine acceptors in rat liver.
Topics: Affinity Labels; Animals; Benzodiazepinones; Catalase; Centrifugation, Density Gradient; Clonazepam; Electrophoresis, Polyacrylamide Gel; Glutamate Dehydrogenase; Intracellular Membranes; Isoquinolines; Liver; Mitochondria, Liver; Polyethyleneimine; Rats; Receptors, GABA-A; Sonication; Subcellular Fractions; Succinate Dehydrogenase | 1990 |
Involvement of the "peripheral" benzodiazepine receptor type (omega 3) in the tolerance to the electroencephalographic effects of benzodiazepines in rats: comparison of diazepam and clonazepam.
Topics: Animals; Benzodiazepinones; Clonazepam; Diazepam; Drug Tolerance; Electroencephalography; Isoquinolines; Male; Rats; Rats, Inbred Strains; Receptors, GABA-A | 1990 |
The effects of acidosis on chronically hypoxic neurons in culture.
Topics: Acidosis; Animals; Benzodiazepines; Benzodiazepinones; Binding, Competitive; Cells, Cultured; Chronic Disease; Clonazepam; Culture Media; Hypoxia; Neurons; Reference Values; Time Factors | 1990 |
"Central" and "peripheral" benzodiazepines and kinetics of lindane-induced toxicity.
Topics: Animals; Anti-Anxiety Agents; Benzodiazepinones; Body Temperature; Clonazepam; Diazepam; Drug Interactions; Female; Hexachlorocyclohexane; Male; Phenytoin; Rats; Rats, Inbred Strains | 1989 |
Diminution by benzodiazepines of the chronotropic responses to noradrenaline in rat isolated atria.
Topics: 1-Methyl-3-isobutylxanthine; 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Anti-Anxiety Agents; Benzodiazepinones; Clonazepam; Colforsin; Cyclic AMP; Diazepam; Female; Flumazenil; Heart; Heart Rate; In Vitro Techniques; Isoquinolines; Male; Myocardium; Norepinephrine; Rats; Rats, Inbred Strains | 1989 |
Pyruvate dehydrogenase interactions with peripheral-type benzodiazepine receptors.
Topics: Animals; Benzodiazepinones; Brain; Clonazepam; Isoquinolines; Ketoglutarate Dehydrogenase Complex; Male; Pyruvate Dehydrogenase Complex; Rats; Rats, Inbred Strains; Receptors, GABA-A; Solubility | 1989 |
Antiproliferative action of benzodiazepines in cultured brain cells is not mediated through the peripheral-type benzodiazepine acceptor.
Topics: Animals; Benzodiazepines; Benzodiazepinones; Blood; Cell Division; Clonazepam; Diazepam; DNA; Glioma; Isoquinolines; Mice; Neuroblastoma; Rats; Receptors, GABA-A; Tumor Cells, Cultured | 1989 |
Peripheral benzodiazepine binding sites in Nb 2 node lymphoma cells: effects on prolactin-stimulated proliferation and ornithine decarboxylase activity.
Topics: Benzodiazepinones; Cell Division; Clonazepam; Humans; Isoquinolines; Kinetics; Lymph Nodes; Lymphoma; Ornithine Decarboxylase; Prolactin; Receptors, GABA-A; Thymidine; Tumor Cells, Cultured | 1989 |
Testicular interstitial cells as targets for peripheral benzodiazepines.
Topics: Animals; Benzodiazepinones; Clonazepam; Diazepam; In Vitro Techniques; Isoquinolines; Leydig Cells; Male; Rats; Rats, Inbred Strains; Testosterone | 1989 |
Effect of ferric nitrilotriacetate on predominantly cortical neuronal cell cultures.
Topics: Acetates; Animals; Benzodiazepinones; Binding, Competitive; Cerebral Cortex; Choline O-Acetyltransferase; Clonazepam; Ferric Compounds; Flunitrazepam; gamma-Aminobutyric Acid; Mice; Neurons; Nitrilotriacetic Acid; Proteins | 1989 |
Benzodiazepine receptor development in murine glial cultures.
Topics: Animals; Animals, Newborn; Benzodiazepinones; Binding, Competitive; Cells, Cultured; Clonazepam; Diazepam; Mice; Neuroglia; Receptors, GABA-A | 1987 |
Regional distribution of a Ro5 4864 binding site that is functionally coupled to the gamma-aminobutyric acid/benzodiazepine receptor complex in rat brain.
Topics: Affinity Labels; Animals; Autoradiography; Azides; Benzodiazepines; Benzodiazepinones; Brain; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Clonazepam; Male; Photochemistry; Rats; Rats, Inbred Strains; Receptors, GABA-A | 1988 |
Differential effects of benzodiazepines on phospholipid methylation in hippocampus and cerebellum of rats.
Topics: Animals; Benzodiazepines; Benzodiazepinones; Cell Membrane; Cerebellum; Clonazepam; Hippocampus; Isoquinolines; Male; Methylation; Methyltransferases; Neurons; Phosphatidylcholines; Phosphatidylethanolamine N-Methyltransferase; Phosphatidylethanolamines; Phospholipids; Rats; Receptors, GABA-A; Synaptosomes | 1988 |
Presence of peripheral-type benzodiazepine binding sites on human erythrocyte membranes.
Topics: Benzodiazepinones; Clonazepam; Convulsants; Erythrocyte Membrane; Flunitrazepam; Humans; In Vitro Techniques; Isoquinolines; Kinetics; Monoamine Oxidase; Receptors, GABA-A | 1988 |
Characterization of stress-induced alterations in [3H] Ro5-4864 binding to peripheral benzodiazepine receptors in rat heart and kidney.
Topics: Adrenalectomy; Animals; Benzodiazepinones; Clonazepam; Convulsants; Electroshock; Hypophysectomy; Kidney; Male; Myocardium; Rats; Rats, Inbred Strains; Receptors, GABA-A; Reference Values; Stress, Psychological | 1988 |
Blockade of non-opioid analgesia in intruder mice by selective neuronal and non-neuronal benzodiazepine recognition site ligands.
Topics: Aggression; Analgesia; Animals; Benzodiazepinones; Clonazepam; Convulsants; Isoquinolines; Ligands; Male; Mice; Mice, Inbred DBA; Neurons; Nociceptors; Reaction Time; Receptors, GABA-A | 1988 |
Triazolam, an anomalous benzodiazepine receptor ligand: in vitro characterization of alprazolam and triazolam binding.
Topics: Alprazolam; Animals; Anti-Anxiety Agents; Benzodiazepines; Benzodiazepinones; Carbolines; Clonazepam; Flunitrazepam; gamma-Aminobutyric Acid; Humans; Kinetics; Male; Rats; Rats, Inbred Strains; Receptors, GABA-A; Triazolam | 1985 |
Neurotransmitter changes during development of cortical neuronal cultures.
Topics: Animals; Benzodiazepinones; Cells, Cultured; Cerebral Cortex; Choline O-Acetyltransferase; Clonazepam; Diazepam; Fetus; Flunitrazepam; gamma-Aminobutyric Acid; Glutamate Decarboxylase; Mice; Neurotransmitter Agents | 1986 |
The role of central- and peripheral-type benzodiazepine receptors in anxiolytic-agent augmentation of NaCl solution intake: effects of clonazepam and Ro 5-4864.
Topics: Animals; Anti-Anxiety Agents; Benzodiazepinones; Clonazepam; Dose-Response Relationship, Drug; Drinking Behavior; Drug Interactions; Male; Rats; Receptors, GABA-A; Reference Values; Saline Solution, Hypertonic; Water Deprivation | 1988 |
Peripheral-type benzodiazepine receptors in endocrine organs: autoradiographic localization in rat pituitary, adrenal, and testis.
Topics: Adrenal Glands; Animals; Autoradiography; Benzodiazepinones; Binding, Competitive; Clonazepam; Isoquinolines; Male; Pituitary Gland; Rats; Rats, Inbred Strains; Receptors, GABA-A; Testis; Tissue Distribution | 1985 |
[Presence of a peripheral type benzodiazepine binding site on the macrophage; its possible role in immunomodulation].
Topics: Animals; Antibody Formation; Benzodiazepines; Benzodiazepinones; Clonazepam; Erythrocytes; Ethanol; Female; Flunitrazepam; Macrophages; Mice; Receptors, GABA-A; Sheep | 1985 |
Clonazepam-induced hyperphagia in nondeprived rats: tests of pharmacological specificity with Ro5-4864, Ro5-3663, Ro15-1788 and CGS 9896.
Topics: Animals; Benzodiazepinones; Clonazepam; Drug Interactions; Feeding Behavior; Flumazenil; Humans; Hyperphagia; Male; Pyrazoles; Rats; Receptors, GABA-A | 1985 |
Characteristics of benzodiazepine receptor binding in living cultures of mouse cerebral cortex at physiologic temperature.
Topics: Animals; Benzodiazepinones; Cerebral Cortex; Clonazepam; Culture Techniques; Kinetics; Mice; Receptors, GABA-A; Temperature | 1985 |
Benzodiazepine receptor-mediated chemotaxis of human monocytes.
Topics: Benzodiazepinones; Binding, Competitive; Chemotaxis, Leukocyte; Clonazepam; Humans; Isoquinolines; Monocytes; Receptors, GABA-A | 1985 |
Benzodiazepine binding characteristics of embryonic rat brain neurons grown in culture.
Topics: Animals; Benzodiazepines; Benzodiazepinones; Brain; Carbolines; Cells, Cultured; Clonazepam; Diazepam; Dose-Response Relationship, Drug; Flumazenil; gamma-Aminobutyric Acid; Neurons; Pyridazines; Rats; Receptors, GABA-A | 1985 |
Solubilization of peripheral benzodiazepine-binding sites from rat kidney.
Topics: Animals; Benzodiazepinones; Binding, Competitive; Carbolines; Chlordiazepoxide; Clonazepam; Diazepam; Digitonin; Flumazenil; Flurazepam; Guanidine; Guanidines; Hot Temperature; Isoquinolines; Kidney; Kinetics; Male; Rats; Rats, Inbred Strains; Receptors, GABA-A; Solubility; Time Factors; Urea | 1985 |
Pharmacology of peripheral type benzodiazepine receptors in the heart.
Topics: Action Potentials; Animals; Benzodiazepinones; Clonazepam; Convulsants; Diazepam; Electric Stimulation; Guinea Pigs; Heart; Heart Ventricles; Isoquinolines; Kinetics; Myocardial Contraction; Myocardium; Receptors, GABA-A; Ventricular Function | 1985 |
Autoradiographic localization of benzodiazepine receptor binding in dissociated cultures of fetal mouse cerebral cortex.
Topics: Affinity Labels; Animals; Autoradiography; Benzodiazepinones; Binding, Competitive; Cells, Cultured; Cerebral Cortex; Clonazepam; Embryo, Mammalian; Flunitrazepam; Mice; Neurons; Photochemistry; Receptors, GABA-A | 1986 |
Convulsant effect of Ro 5-4864, a peripheral type benzodiazepine, on the baboon (Papio papio).
Topics: Animals; Benzodiazepines; Benzodiazepinones; Clonazepam; Diazepam; Dose-Response Relationship, Drug; Flumazenil; Isoquinolines; Papio; Receptors, GABA-A; Seizures | 1986 |
Hormonal interactions with benzodiazepine binding sites in vitro.
Topics: Adrenal Cortex Hormones; Animals; Benzodiazepinones; Binding, Competitive; Clonazepam; Hormones; In Vitro Techniques; Male; Prostaglandins; Radioligand Assay; Rats; Rats, Inbred Strains; Receptors, GABA-A; Thyroxine | 1986 |
Central- and peripheral-type benzodiazepine receptors.
Topics: Animals; Benzodiazepinones; Binding, Competitive; Brain; Clonazepam; Convulsants; Flunitrazepam; Kidney; Kinetics; Membranes; Muscimol; Rats; Receptors, GABA-A; Subcellular Fractions; Tissue Distribution | 1986 |
Pyrazolo[4,5-c]quinolines. 3. Synthesis, receptor binding, and 13C NMR study.
Topics: Animals; Benzodiazepinones; Binding, Competitive; Brain; Cattle; Chemical Phenomena; Chemistry; Clonazepam; Flunitrazepam; In Vitro Techniques; Magnetic Resonance Spectroscopy; Pyrazoles; Quinolines; Receptors, GABA-A | 1986 |
Coexistence of central and peripheral benzodiazepine binding sites in the human pineal gland.
Topics: Aged; Benzodiazepinones; Binding, Competitive; Cell Membrane; Clonazepam; Female; Flumazenil; Flunitrazepam; Humans; Isoquinolines; Male; Middle Aged; Pineal Gland; Receptors, GABA-A | 1987 |
Benzodiazepine receptor affinity alterations at physiologic temperature after chronic clonazepam exposure.
Topics: Animals; Benzodiazepinones; Body Temperature; Cells, Cultured; Cerebral Cortex; Clonazepam; Convulsants; Flunitrazepam; Kinetics; Mice; Receptors, GABA-A; Time Factors | 1987 |
Peripheral benzodiazepines enhance the respiratory burst of macrophage-like P388D1 cells stimulated by arachidonic acid.
Topics: Animals; Arachidonic Acid; Arachidonic Acids; Benzodiazepinones; Cell Line; Clonazepam; Diazepam; Isoquinolines; Kinetics; Macrophages; Receptors, GABA-A; Superoxides | 1987 |
Diazepam-sensitive specific binding of phenytoin in rat brain.
Topics: Animals; Benzodiazepinones; Binding Sites; Cell Membrane; Cerebral Cortex; Clonazepam; Diazepam; Flumazenil; Male; Phenytoin; Rats; Rats, Inbred Strains | 1986 |
Inhibition of cell proliferation of human gliomas by benzodiazepines in vitro.
Topics: Astrocytoma; Benzodiazepines; Benzodiazepinones; Cell Division; Clonazepam; Diazepam; Female; Flumazenil; Glioma; Humans; Male; Middle Aged; Thymidine; Tumor Cells, Cultured | 1988 |
Central administration of benzodiazepines alters water absorption by the rat ileum in vivo.
Topics: Animals; Benzodiazepines; Benzodiazepinones; Clonazepam; Diazepam; Ileum; Injections, Intraventricular; Intestinal Absorption; Lorazepam; Male; Nifedipine; Nitrendipine; Rats; Rats, Inbred Strains; Water | 1987 |
Benzodiazepine Ro 5-4864 increases coronary flow.
Topics: Animals; Benzodiazepinones; Clonazepam; Convulsants; Coronary Circulation; Heart Rate; In Vitro Techniques; Isoquinolines; Male; Muscle Contraction; Rats; Rats, Inbred Strains | 1987 |
Electrophysiological and pharmacological characterization of peripheral benzodiazepine receptors in a guinea pig heart preparation.
Topics: Action Potentials; Animals; Benzodiazepinones; Clonazepam; Convulsants; Diazepam; Dose-Response Relationship, Drug; Electric Stimulation; Flumazenil; Guinea Pigs; Heart; In Vitro Techniques; Isoquinolines; Myocardial Contraction; Myocardium; Receptors, Cell Surface; Receptors, GABA-A | 1984 |
Autoradiographic localisation of benzodiazepine receptors in the rat pituitary gland.
Topics: Animals; Autoradiography; Benzodiazepinones; Clonazepam; Flumazenil; gamma-Aminobutyric Acid; In Vitro Techniques; Male; Pituitary Gland; Rats; Rats, Inbred Strains; Receptors, GABA-A | 1984 |
Flunitrazepam binding to intact and homogenized astrocytes and neurons in primary cultures.
Topics: Animals; Astrocytes; Benzodiazepinones; Cells, Cultured; Clonazepam; Diazepam; Flunitrazepam; Kinetics; Mice; Neurons; Receptors, GABA-A; Temperature | 1984 |
Autoradiographic localization of benzodiazepine receptors in the rat kidney.
Topics: Animals; Autoradiography; Benzodiazepinones; Clonazepam; Diazepam; Flunitrazepam; Kidney; Kidney Tubules, Distal; Loop of Henle; Male; Mucoproteins; Rats; Rats, Inbred Strains; Receptors, GABA-A; Tritium; Uromodulin | 1984 |
Benzodiazepine binding sites in human myometrium.
Topics: Adult; Benzodiazepinones; Binding Sites; Cell Membrane; Clonazepam; Diazepam; Female; Flunitrazepam; Humans; In Vitro Techniques; Lorazepam; Middle Aged; Myometrium; Receptors, GABA-A | 1984 |
Analysis of benzodiazepine binding sites in rat pituitary gland.
Topics: Animals; Benzodiazepinones; Binding, Competitive; Clonazepam; Diazepam; Flunitrazepam; gamma-Aminobutyric Acid; In Vitro Techniques; Male; Pituitary Gland; Rats; Rats, Inbred Strains; Receptors, GABA-A | 1984 |
Binding of [3H]flunitrazepam to the LM cell, a transformed murine fibroblast.
Topics: Animals; Anti-Anxiety Agents; Benzodiazepinones; Binding Sites; Cell Line; Cell Membrane; Choline; Clonazepam; Culture Media; Cyclic AMP; Flunitrazepam; Kinetics; Mice; Neoplasms, Experimental; Phospholipids | 1983 |
Properties of [3H]diazepam binding sites on rat blood platelets.
Topics: Animals; Benzodiazepinones; Blood Platelets; Clonazepam; Diazepam; Hydrogen-Ion Concentration; Kinetics; Male; Rats; Receptors, Drug; Receptors, GABA-A; Temperature | 1980 |
Peripheral benzodiazepine binding sites: effect of PK 11195, 1-(2-chlorophenyl)-N-methyl-N-(1-methylpropyl)-3-isoquinolinecarboxamide. I. In vitro studies.
Topics: Adrenal Glands; Animals; Benzodiazepinones; Blood Platelets; Brain; Clonazepam; Diazepam; In Vitro Techniques; Isoquinolines; Kidney; Male; Myocardium; Rats; Rats, Inbred Strains; Receptors, Cell Surface; Receptors, GABA-A; Tissue Distribution | 1983 |
Peripheral benzodiazepine binding sites: effect of PK 11195, 1-(2-chlorophenyl)-N-methyl-(1-methylpropyl)-3 isoquinolinecarboxamide. II. In vivo studies.
Topics: Animals; Benzodiazepinones; Brain; Clonazepam; Diazepam; Isoquinolines; Kidney; Kinetics; Male; Mice; Myocardium; Receptors, Cell Surface; Receptors, GABA-A | 1983 |
Development and differentiation of the benzodiazepine receptor in cultures of fetal mouse spinal cord.
Topics: Animals; Benzodiazepinones; Cell Differentiation; Clonazepam; Diazepam; Fetus; Flunitrazepam; Kinetics; Mice; Neurons; Receptors, Cell Surface; Receptors, GABA-A; Spinal Cord | 1983 |
Differentiation between two ligands for peripheral benzodiazepine binding sites, [3H]RO5-4864 and [3H]PK 11195, by thermodynamic studies.
Topics: Animals; Benzodiazepinones; Clonazepam; Diazepam; Dipyridamole; Isoquinolines; Ligands; Male; Membranes; Myocardium; Rats; Receptors, Cell Surface; Receptors, GABA-A; Thermodynamics | 1983 |
Benzodiazepine receptors along the nephron: [3H]PK 11195 binding in rat tubules.
Topics: Animals; Benzodiazepinones; Clonazepam; Dose-Response Relationship, Drug; Isoquinolines; Kidney Tubules; Male; Nephrons; Rats; Rats, Inbred Strains; Receptors, Cell Surface; Receptors, GABA-A; Tissue Distribution | 1984 |
Receptors for psychoactive drugs: autoradiographic visualization of benzodiazepine binding sites.
Topics: Animals; Autoradiography; Benzodiazepinones; Binding Sites; Brain; Brain Chemistry; Clonazepam; Convulsants; Rats; Receptors, Cell Surface; Receptors, GABA-A | 1984 |
Specific binding of [3H]diazepam in mouse glioblastoma: the influence of clonazepam and Ro 5-4864 on [3H]diazepam binding.
Topics: Animals; Benzodiazepinones; Binding Sites; Cell Line; Clonazepam; Diazepam; Glioma; Mice; Neuroglia | 1984 |
[3H]diazepam binding sites on chick neurons in primary culture.
Topics: Animals; Benzodiazepinones; Binding Sites; Binding, Competitive; Cells, Cultured; Chick Embryo; Clonazepam; Diazepam; gamma-Aminobutyric Acid; Neurons; Pentobarbital; Telencephalon | 1983 |
Properties of [3H]diazepam binding sites on cultured murine glia and neurons.
Topics: Animals; Animals, Newborn; Benzodiazepinones; Binding Sites; Cells, Cultured; Cerebral Cortex; Clonazepam; Diazepam; Kinetics; Mice; Neuroglia; Neurons | 1984 |
Vascular and tubular actions of diazepam in isolated and perfused rat kidney.
Topics: Animals; Benzodiazepinones; Biological Transport, Active; Blood Vessels; Clonazepam; Convulsants; Diazepam; Diuresis; In Vitro Techniques; Kidney Function Tests; Kidney Tubules; Male; Muscle Contraction; Muscle Relaxation; Muscle, Smooth, Vascular; Natriuresis; Norepinephrine; Potassium Chloride; Rats; Rats, Wistar; Renal Circulation | 1995 |
Mitochondrial benzodiazepine receptor linked to inner membrane ion channels by nanomolar actions of ligands.
Topics: Animals; Benzodiazepinones; Clonazepam; Convulsants; Flumazenil; Intracellular Membranes; Ion Channels; Isoquinolines; Male; Membrane Potentials; Mitochondria, Heart; Protoporphyrins; Rats; Rats, Sprague-Dawley; Receptors, GABA-A; Submitochondrial Particles | 1993 |
Differential effects of 4'-chlorodiazepam on expressed human GABAA receptors.
Topics: Benzodiazepinones; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cell Line; Clonazepam; Flumazenil; Humans; Quinolines; Receptors, GABA; Transfection | 1995 |
Modification of the photodynamic action of delta-aminolaevulinic acid (ALA) on rat pancreatoma cells by mitochondrial benzodiazepine receptor ligands.
Topics: Aminolevulinic Acid; Animals; Benzodiazepines; Benzodiazepinones; Cell Division; Cell Survival; Clonazepam; Flumazenil; Isoquinolines; Ligands; Mitochondria; Oxygen; Pancreatic Neoplasms; Photochemotherapy; Protoporphyrins; Radiation-Protective Agents; Radiation-Sensitizing Agents; Rats; Receptors, GABA-A; Singlet Oxygen; Tumor Cells, Cultured | 1995 |
Effect of peripheral benzodiazepine receptor ligands on lipopolysaccharide-induced tumor necrosis factor activity in thioglycolate-treated mice.
Topics: Animals; Benzodiazepinones; Clonazepam; GABA-A Receptor Antagonists; Isoquinolines; Ligands; Lipopolysaccharides; Macrophages, Peritoneal; Male; Mice; Mice, Inbred C3H; Midazolam; Receptors, GABA-A; Thioglycolates; Tumor Necrosis Factor-alpha | 1994 |
In vitro inhibition of cellular immune responses by benzodiazepines and PK 11195. Effects on mitogen- and alloantigen-driven lymphocyte proliferation and on IL-1, IL-2 synthesis and IL-2 receptor expression.
Topics: Animals; B-Lymphocytes; Benzodiazepines; Benzodiazepinones; Clonazepam; Diazepam; Female; Flumazenil; Immunity, Cellular; In Vitro Techniques; Interleukin-1; Interleukin-2; Isoquinolines; Lymphocyte Activation; Male; Mice; Mice, Inbred A; Mice, Inbred C57BL; Neuroimmunomodulation; Receptors, GABA-A; T-Lymphocytes | 1993 |
The specific binding of the platelet-activating factor (PAF) receptor antagonist WEB 2086 and the benzodiazepine flunitrazepam to rat hepatocytes.
Topics: Animals; Anti-Anxiety Agents; Anticonvulsants; Azepines; Benzodiazepinones; Bicuculline; Cells, Cultured; Clonazepam; Convulsants; Flunitrazepam; Kinetics; Liver; Male; Platelet Aggregation Inhibitors; Platelet Membrane Glycoproteins; Rats; Rats, Sprague-Dawley; Receptors, Cell Surface; Receptors, G-Protein-Coupled; Triazoles; Tritium | 1996 |
Prevention of ACTH- and adrenalectomy-induced muricidal behavior: by benzodiazepinic ligands.
Topics: Adrenalectomy; Adrenocorticotropic Hormone; Aggression; Animals; Benzodiazepinones; Clonazepam; Flumazenil; GABA Modulators; Isoquinolines; Male; Mice; Muscimol; Rats; Rats, Wistar; Receptors, GABA-A; Time Factors | 1997 |
Synthesis and biology of a 7-nitro-2,1,3-benzoxadiazol-4-yl derivative of 2-phenylindole-3-acetamide: a fluorescent probe for the peripheral-type benzodiazepine receptor.
Topics: 4-Chloro-7-nitrobenzofurazan; Animals; Benzodiazepinones; Biological Transport; Cholesterol; Clonazepam; Fluorescent Dyes; Hypolipidemic Agents; Indoleacetic Acids; Isoquinolines; Ligands; Male; Mice; Microscopy, Fluorescence; Mitochondria; Rats; Receptors, GABA-A; Tumor Cells, Cultured | 1997 |
Effects of peripheral-type benzodiazepine receptor antisense knockout on MA-10 Leydig cell proliferation and steroidogenesis.
Topics: Algestone; Androstenedione; Animals; Benzodiazepinones; Cell Division; Clonazepam; Cyclic AMP; DNA, Antisense; GABA-A Receptor Antagonists; Isoquinolines; Leydig Cells; Male; Mice; Plasmids; Progesterone; Protein Binding; Receptors, GABA-A; RNA, Messenger; Transfection; Tumor Cells, Cultured | 1998 |
Characterization of binding sites for the omega3 receptor ligands [3H]PK11195 and [3H]RO5-4864 in human brain.
Topics: Allosteric Regulation; Benzodiazepines; Benzodiazepinones; Binding Sites; Binding, Competitive; Clonazepam; Convulsants; Detergents; Diazepam; Dithiothreitol; Female; Histidine; Humans; Isoquinolines; Ligands; Male; Occipital Lobe; Receptors, GABA-A; Sulfhydryl Reagents; Tritium | 1997 |
Modulation of intracellular calcium in human neutrophils by peripheral benzodiazepine receptor ligands.
Topics: Anti-Anxiety Agents; Benzodiazepinones; Calcium; Clonazepam; Cytosol; Diazepam; Drug Antagonism; GABA Modulators; Humans; Isoquinolines; Neutrophils; Receptors, GABA-A | 1998 |
Antiproliferative and differentiating effects of benzodiazepine receptor ligands on B16 melanoma cells.
Topics: Animals; Antineoplastic Agents; Benzodiazepinones; Cell Cycle; Cell Differentiation; Cell Division; Clonazepam; Diazepam; GABA Agents; gamma-Glutamyltransferase; Isoquinolines; Melanoma, Experimental; Mice; Nucleotides; Phenotype; Tumor Cells, Cultured | 1998 |
Inhibitory regulation of amylase release in rat parotid acinar cells by benzodiazepine receptors.
Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Amylases; Animals; Atropine; Benzodiazepinones; Carbachol; Clonazepam; Diazepam; Dose-Response Relationship, Drug; Flumazenil; GABA Modulators; GABA-A Receptor Agonists; GABA-A Receptor Antagonists; Isoproterenol; Male; Muscarinic Agonists; Muscarinic Antagonists; Parotid Gland; Propranolol; Rats; Rats, Wistar; Receptors, GABA-A | 1998 |
Effect of benzodiazepines and neurosteroids on ammonia-induced swelling in cultured astrocytes.
Topics: Ammonia; Astrocytes; Atrial Natriuretic Factor; Benzodiazepines; Benzodiazepinones; Brain Edema; Cell Size; Clonazepam; Dehydroepiandrosterone Sulfate; Desoxycorticosterone; Diazepam; Diazepam Binding Inhibitor; Flumazenil; GABA-A Receptor Agonists; GABA-A Receptor Antagonists; Isoquinolines; Nerve Tissue Proteins; Neuropeptides; Peptide Fragments; Pregnanolone; Pregnenolone; Protoporphyrins; Receptors, GABA-A; Steroids; Up-Regulation | 1998 |
Benzodiazepine receptor agonists modulate thymocyte apoptosis through reduction of the mitochondrial transmembrane potential.
Topics: Animals; Apoptosis; Benzodiazepines; Benzodiazepinones; Binding Sites; Caspase Inhibitors; Cells, Cultured; Clonazepam; Dexamethasone; Diazepam; Drug Interactions; Drug Synergism; Etoposide; GABA-A Receptor Agonists; Male; Membrane Potentials; Mice; Mice, Inbred BALB C; Mitochondria; Protease Inhibitors; Protein Biosynthesis; Proteins; RNA, Messenger; Thymus Gland | 1999 |
Central and peripheral benzodiazepine ligands prevent mitochondrial damage induced by noise exposure in the rat myocardium: an ultrastructural study.
Topics: Animals; Benzodiazepines; Benzodiazepinones; Clonazepam; Diazepam; GABA Modulators; Isoquinolines; Male; Microscopy, Electron; Microscopy, Electron, Scanning; Mitochondria, Heart; Myocardium; Noise; Rats; Rats, Wistar; Time Factors | 1999 |
Peripheral benzodiazepine receptor agonists exhibit potent antiapoptotic activities.
Topics: Apoptosis; Benzodiazepinones; Clonazepam; Diazepam; Flunitrazepam; GABA-A Receptor Agonists; GABA-A Receptor Antagonists; Humans; Isoquinolines; Jurkat Cells; Kinetics; Ligands; Receptors, GABA-A; Transfection; Tumor Necrosis Factor-alpha; U937 Cells | 1999 |
2-Arylpyrazolo[1,5-a]pyrimidin-3-yl acetamides. New potent and selective peripheral benzodiazepine receptor ligands.
Topics: Acetamides; Animals; Benzodiazepinones; Binding Sites; Cerebral Cortex; Clonazepam; Flumazenil; Glioma; Intracellular Membranes; Isoquinolines; Kidney; Ligands; Magnetic Resonance Spectroscopy; Molecular Structure; Pyrazoles; Pyrimidines; Rats; Receptors, GABA-A; Structure-Activity Relationship; Thermodynamics; Tumor Cells, Cultured | 2001 |
Diazepam inhibits HIV-1 Tat-induced migration of human microglia.
Topics: Adjuvants, Immunologic; Benzodiazepinones; Calcium Signaling; Chemotaxis; Clonazepam; Diazepam; Gene Products, tat; HIV-1; Humans; Microglia; Nerve Tissue Proteins; Receptors, CCR5; Receptors, GABA-A; tat Gene Products, Human Immunodeficiency Virus; Up-Regulation | 2001 |
Effect of midazolam on interleukin-6 mRNA expression in human peripheral blood mononuclear cells in the absence of lipopolysaccharide.
Topics: Anti-Anxiety Agents; Anticonvulsants; Benzodiazepinones; Binding, Competitive; Cell Survival; Cells, Cultured; Clonazepam; Convulsants; DNA, Complementary; Dose-Response Relationship, Drug; GABA-A Receptor Agonists; Humans; Interleukin-6; Leukocytes, Mononuclear; Ligands; Lipopolysaccharides; Midazolam; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Time Factors | 2001 |
Effects on free radical generation by ligands of the peripheral benzodiazepine receptor in cultured neural cells.
Topics: Animals; Antioxidants; Astrocytes; Benzodiazepinones; Binding, Competitive; Cells, Cultured; Clonazepam; Cyclosporine; Dose-Response Relationship, Drug; Free Radicals; Isoquinolines; Ligands; Microglia; Mitochondria; Neurons; Protoporphyrins; Rats; Receptors, GABA-A | 2002 |
Effects of peripheral-type benzodiazepine receptor ligands on Ehrlich tumor cell proliferation.
Topics: Animals; Benzodiazepinones; Carcinoma, Ehrlich Tumor; Cell Cycle; Cell Division; Cell Proliferation; Clonazepam; Flow Cytometry; GABA Modulators; Immunohistochemistry; Isoquinolines; Ligands; Mice; Receptors, GABA-A | 2006 |
Characterization of two classes of benzodiazepine binding sites in Schistosoma mansoni.
Topics: Animals; Benzodiazepines; Benzodiazepinones; Binding Sites; Clonazepam; Diazepam; Flunitrazepam; GABA Agonists; GABA Modulators; Inhibitory Concentration 50; Isoquinolines; Ligands; Male; Pyridines; Rats; Rats, Wistar; Receptors, GABA-A; Schistosoma mansoni; Synaptosomes; Temperature; Time Factors; Tritium; Zolpidem | 2007 |
Allosteric modulation by benzodiazepines of GABA-gated chloride channels of an identified insect motor neurone.
Topics: Animals; Benzodiazepines; Benzodiazepinones; Chloride Channels; Clonazepam; Diazepam; Dose-Response Relationship, Drug; Evoked Potentials; GABA Modulators; gamma-Aminobutyric Acid; Glutamic Acid; In Vitro Techniques; Insect Proteins; Male; Membrane Potentials; Microelectrodes; Motor Neurons; Periplaneta | 2009 |
Investigation into mechanisms mediating the inhibitory effect of 1,4-benzodiazepines on mast cells by gene expression profiling.
Topics: Adult; Aged; Benzodiazepinones; Clonazepam; Female; Flunitrazepam; Gene Expression; Gene Expression Profiling; HL-60 Cells; Humans; Male; Mast Cells; Mastocytosis; Microarray Analysis; Middle Aged; Polymerase Chain Reaction | 2013 |
Acute chloroquine poisoning: A comprehensive experimental toxicology assessment of the role of diazepam.
Topics: Animals; Arrhythmias, Cardiac; Benzodiazepinones; Cardiotoxicity; Chloroquine; Clonazepam; Coronavirus Infections; COVID-19; Diazepam; Dose-Response Relationship, Drug; Drug Overdose; Electrocardiography; Female; Hypokalemia; Male; Pandemics; Pneumonia, Viral; Rabbits; Random Allocation; Rats; Rats, Wistar | 2020 |