ro 5-4864 and clonazepam

ro 5-4864 has been researched along with clonazepam in 98 studies

Research

Studies (98)

TimeframeStudies, this research(%)All Research%
pre-199054 (55.10)18.7374
1990's33 (33.67)18.2507
2000's8 (8.16)29.6817
2010's1 (1.02)24.3611
2020's2 (2.04)2.80

Authors

AuthorsStudies
Blair, T; Webb, GA1
Campiani, G; Ciani, SM; De Filippis, MP; Fiorini, I; Garofalo, A; Greco, G; Manzoni, C; Mennini, T; Mihai, C; Nacci, V; Novellino, E; Williams, DC; Woods, MJ; Zisterer, DM1
Cleary, J; Glick, GD; Johnson, KM; Opipari, AW1
Baglini, E; Barresi, E; Robello, M; Salerno, S; Settimo, FD; Taliani, S1
Advenier, C; Candenas, ML; Devillier, P; Naline, E1
Järvinen, A; Männistö, PT; Rägo, L1
Berdeu, D; Loubatières-Mariani, MM; Manteghetti, M; Petit, P; Ribes, G1
Diana, G; Massotti, M1
Järvinen, A; Männistö, PT; Paakkari, I1
Becker, DP; Black, KL; Ikezaki, K; Shiraishi, T1
Abraham, S; Bolger, GT; Oz, N; Weissman, BA1
Bravo, C; Chiang, PK; Gutiérrez, J; Moreno-Sánchez, R; Newman, AH1
Lichtensteiger, W; Parmar, R; Ramseier, HR; Schlumpf, M1
Izquierdo, I; Medina, JH; Pereira, ME1
Elgoyhen, AB; Kazanietz, MG1
O'Beirne, GB; Williams, DC; Woods, MJ1
De Luca, C; Massotti, M; Mele, L1
Sher, PK3
Griffith, JA; Woolley, DE1
Adler-Graschinsky, E; Elgoyhen, B1
Daval, JL; Marangos, PJ; Post, RM1
Gorman, AM; O'Beirne, GB; Regan, CM; Williams, DC1
Duerson, KC; Gerrish, KE; Laird, HE; Putnam, CW; Russell, DH1
Calandra, RS; Ritta, MN1
Machen, VL; Swaiman, KF1
Sher, PK; Talwar, D1
Brinton, RE; Gee, KW; McEwen, BS1
Salmona, M; Tacconi, MT1
Ciliax, BJ; Mancini, WR; Olson, JM; Young, AB1
Basile, AS; Crawley, JN; Drugan, RC; Paul, SM; Skolnick, P1
Randall, JI; Rodgers, RJ1
Clow, A; Glover, V; Sandler, M1
Boespflug, O; Swaiman, KF1
Falk, JL; Plaessmann, WR; Tang, M1
Anholt, RR; De Souza, EB; Kuhar, MJ; Murphy, KM; Snyder, SH1
Haumont, J; Lenfant, M; Potier, P; Zavala, F1
Cooper, SJ; Gilbert, DB1
Paul, SM; Pert, CB; Ruff, MR; Wahl, LM; Wahl, SM; Weber, RJ1
Cole, R; De Vellis, J; Noble, EP; Syapin, PJ1
Fares, F; Gavish, M1
Belin, C; Carriot, T; Dubroeucq, MC; Guérémy, C; Le Fur, G; Mestre, M; Renault, C; Uzan, A2
Machen, VL; Neale, EA; Sher, PK1
Bryere, P; Naquet, R; Valin, A1
Deckert, J; Marangos, PJ1
Hrelia, S; Lucacchini, A; Martini, C; Rossi, CA1
Cecchi, L; Filacchioni, G; Lucacchini, A; Martini, C; Melani, F; Palazzino, G; Pennacchi, E1
Lafaille, F; Lal, S; Nair, NP; Quirion, R; Suranyi-Cadotte, B1
Machen, VL; Sher, PK2
Lenfant, M; Zavala, F1
Teo, WL; Wong, PT1
Kunert-Radek, J; Pawlikowski, M; Radek, A; Stepien, H1
Brown, T; Fogel, R; Gaginella, T; Marshall, D; Michelson, G; Senler, T1
French, JF; Grupp, IL; Matlib, MA1
Brown, C; Martin, IL1
Bender, AS; Hertz, L1
Beaumont, K; Fanestil, DD; Healy, DP1
Fioretti, P; Galbani, P; Gambacciani, M; Melis, G; Ronca-Testoni, S1
Anderson, RA; Mitchell, R1
Bylund, DB; Feller, DJ; Schroeder, F1
Spector, S; Taniguchi, T; Wang, JK1
Benavides, J; Dubroeucq, MC; Flamier, A; Guérémy, C; Imbault, F; Le Fur, G; Perrier, ML; Renault, C; Uzan, A; Vaucher, N1
Benavides, J; Dubroeucq, MC; Guérémy, C; Guilloux, F; Le Fur, G; Renault, C; Rufat, P; Uzan, A1
Benavides, J; Dubroeucq, MC; Flamier, A; Guérémy, C; Le Fur, G; Perrier, ML; Renault, C; Uzan, A; Vaucher, N1
Butlen, D1
Lichtensteiger, W; Möhler, H; Richards, JG; Schlumpf, M1
Khalansky, AS; Kondakova, LI; Zlobina, GP1
Ebel, C; Mallorga, P; Roth-Schechter, BF1
Elías, MM; Monasterolo, LA; Ochoa, JE; Trumper, L1
Antonenko, YN; Kinnally, KW; McEnery, MW; Snyder, SH; Tedeschi, H; Zorov, DB1
Chen, JS; Gee, KW; Johnson, D; Lan, NC1
Matthews, EK; Ratcliffe, SL1
Koga, K; Matsumoto, T; Ogata, M; Shigematsu, A1
Lichtensteiger, W; Ramseier, H; Schlumpf, M1
Barton, JM; Olson, MS; Svetlov, SI1
Cespuglio, R; Miachon, S1
Boujrad, N; Kotoula, M; Kozikowski, AP; Ma, D; Papadopoulos, V; Tückmantel, W1
Gavish, M; Kelly-Hershkovitz, E; Lahav, M; Leschiner, S; Spanier, I; Weisinger, G; Weizman, R1
Butterworth, RF; Rao, VL1
Caldiroli, E; Cattaneo, S; Cosentino, M; Di Grazia, L; Frigo, G; Lecchini, S; Marino, F1
Beery, E; Brenner, S; Gavish, M; Landau, M; Landau, O; Nordenberg, J; Wasseman, L; Weizman, A; Zoref-Shani, E1
Kawaguchi, M; Okubo, M1
Bender, AS; Norenberg, MD1
Kizaki, H; Onishi, Y; Sato, Y; Tanimoto, Y1
Fornai, F; Gesi, M; Lenzi, P; Natale, G; Paparelli, A; Pellegrini, A; Riva, A; Soldani, P1
Bono, F; Herbert, JM; Lamarche, I; Le Fur, G; Prabonnaud, V1
Bruni, F; Ciciani, G; Costa, B; Costagli, C; Costanzo, A; Guerrini, G; Martini, C; Selleri, S1
Gekker, G; Hegg, CC; Hu, S; Lokensgard, JR; Peterson, PK; Thayer, SA1
Kohjitani, A; Maeda, S; Miyawaki, T; Shimada, M; Sogawa, N1
Jayakumar, AR; Norenberg, MD; Panickar, KS1
Dagli, ML; Fonseca, ES; Leite, KR; Massoco, CO; Matsuzaki, P; Oloris, SC; Otake, AH; Palermo-Neto, J; Sakai, M1
Lopes, DV; Mendonça-Silva, DL; Noël, F; Thibaut, JP1
Buckingham, SD; Higashino, Y; Sattelle, DB1
Haenisch, B; Huber, M; Molderings, GJ; Steffens, M; Wilhelm, T1
Hughes, DA1

Reviews

1 review(s) available for ro 5-4864 and clonazepam

ArticleYear
The Alpha Keto Amide Moiety as a Privileged Motif in Medicinal Chemistry: Current Insights and Emerging Opportunities.
    Journal of medicinal chemistry, 2021, 04-08, Volume: 64, Issue:7

    Topics: Amides; Animals; Cell Line, Tumor; Chemistry, Pharmaceutical; Humans; Ketones

2021

Other Studies

97 other study(ies) available for ro 5-4864 and clonazepam

ArticleYear
Electronic factors in the structure-activity relationship of some 1,4-benzodiazepin-2-ones.
    Journal of medicinal chemistry, 1977, Volume: 20, Issue:9

    Topics: Benzodiazepinones; Electrochemistry; Structure-Activity Relationship

1977
Synthesis, biological activity, and SARs of pyrrolobenzoxazepine derivatives, a new class of specific "peripheral-type" benzodiazepine receptor ligands.
    Journal of medicinal chemistry, 1996, Aug-30, Volume: 39, Issue:18

    Topics: Animals; Benzodiazepinones; Binding Sites; Cerebral Cortex; Isoquinolines; Ligands; Mice; Rats; Rats, Wistar; Receptors, GABA-A; Structure-Activity Relationship

1996
Inhibition of the mitochondrial F1F0-ATPase by ligands of the peripheral benzodiazepine receptor.
    Bioorganic & medicinal chemistry letters, 2007, Mar-15, Volume: 17, Issue:6

    Topics: Adenosine Triphosphate; Antineoplastic Agents; Apoptosis; Benzodiazepines; Cell Line, Tumor; Cell Proliferation; GABA-A Receptor Antagonists; Humans; Hydrolysis; Isoquinolines; Kinetics; Ligands; Mitochondria; Proton-Translocating ATPases; Structure-Activity Relationship

2007
Contractile effect of alpha,beta-methylene ATP on the guinea-pig isolated trachea.
    Fundamental & clinical pharmacology, 1992, Volume: 6, Issue:3

    Topics: 2-Chloroadenosine; Adenosine Triphosphate; Animals; Benzodiazepinones; Clonazepam; Diazepam; Drug Synergism; GABA-A Receptor Antagonists; Guinea Pigs; Male; Muscle Contraction; Muscle, Smooth; Phenylisopropyladenosine; Trachea

1992
Effects of central and peripheral type benzodiazepine ligands on thyrotropin and prolactin secretion.
    Neuropeptides, 1992, Volume: 21, Issue:3

    Topics: Animals; Benzodiazepinones; Carbolines; Clonazepam; Cold Temperature; Diazepam; Flumazenil; Hypothalamo-Hypophyseal System; Isoquinolines; Male; Pituitary Gland, Anterior; Prolactin; Rats; Rats, Inbred Strains; Receptors, GABA-A; Secretory Rate; Thyrotropin; Thyrotropin-Releasing Hormone

1992
Effects of a peripheral-type benzodiazepine on glucose-induced insulin secretion.
    European journal of pharmacology, 1992, Oct-20, Volume: 221, Issue:2-3

    Topics: Animals; Benzodiazepinones; Clonazepam; Glucose; In Vitro Techniques; Insulin; Insulin Secretion; Islets of Langerhans; Isoquinolines; Male; Perfusion; Rats; Rats, Wistar

1992
Repeated administration of diazepam reduces [3H]Ro 5-4864 binding in cerebral cortex of rats.
    Pharmacology, biochemistry, and behavior, 1992, Volume: 42, Issue:2

    Topics: Animals; Benzodiazepinones; Cerebral Cortex; Clonazepam; Diazepam; Down-Regulation; Electroencephalography; In Vitro Techniques; Male; Mitochondria; Rats; Rats, Inbred Strains

1992
Central and peripheral type benzodiazepine ligands displace [3H][3-ME-HIS2]TRH from its binding sites in the brain and the anterior pituitary and antagonize the effect of TRH in the rat duodenum.
    Neuropeptides, 1991, Volume: 19, Issue:3

    Topics: Animals; Benzodiazepinones; Binding Sites; Brain; Brain Stem; Carbolines; Clonazepam; Diazepam; Duodenum; Hypothalamus; Isoquinolines; Male; Muscle, Smooth; Pituitary Gland, Anterior; Pyrrolidonecarboxylic Acid; Rats; Rats, Inbred Strains; Receptors, GABA-A; Receptors, Neurotransmitter; Receptors, Thyrotropin-Releasing Hormone; Thyrotropin-Releasing Hormone

1991
Peripheral benzodiazepine induces morphological changes and proliferation of mitochondria in glioma cells.
    Journal of neuroscience research, 1991, Volume: 30, Issue:3

    Topics: Animals; Benzodiazepinones; Cell Line; Clonazepam; Culture Media, Serum-Free; Fluorescent Dyes; Glioma; Isoquinolines; Microscopy, Electron; Microscopy, Fluorescence; Mitochondria; Rats; Receptors, GABA-A; Rhodamine 123; Rhodamines

1991
Interactions between peripheral-type benzodiazepine receptor ligands and an activator of voltage-operated calcium channels.
    Canadian journal of physiology and pharmacology, 1990, Volume: 68, Issue:1

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Benzodiazepinones; Blood Pressure; Calcium Channels; Clonazepam; Coronary Disease; Electrocardiography; Guinea Pigs; In Vitro Techniques; Isoquinolines; Male; Myocardial Contraction; Receptors, GABA-A

1990
Release of Ca2+ from heart and kidney mitochondria by peripheral-type benzodiazepine receptor ligands.
    The International journal of biochemistry, 1991, Volume: 23, Issue:2

    Topics: Animals; Benzodiazepines; Benzodiazepinones; Calcium; Clonazepam; Kidney; Magnesium; Mitochondria; Mitochondria, Heart; Rats; Rats, Inbred Strains; Receptors, GABA-A; Strontium

1991
Prenatal benzodiazepine immunosuppression: possible involvement of peripheral benzodiazepine site.
    Developmental pharmacology and therapeutics, 1990, Volume: 15, Issue:3-4

    Topics: Animals; Autoradiography; Benzodiazepinones; Binding Sites; Cell Division; Clonazepam; Convulsants; Diazepam; Female; Immune Tolerance; Immunity, Cellular; Lymphocytes; Male; Maternal-Fetal Exchange; Pregnancy; Prenatal Exposure Delayed Effects; Rats; Receptors, GABA-A

1990
Benzodiazepine receptor ligand influences on acquisition: suggestion of an endogenous modulatory mechanism mediated by benzodiazepine receptors.
    Behavioral and neural biology, 1990, Volume: 54, Issue:1

    Topics: Animals; Anti-Anxiety Agents; Arousal; Avoidance Learning; Benzodiazepinones; Brain; Carbolines; Clonazepam; Diazepam; Dose-Response Relationship, Drug; Exploratory Behavior; Female; Flumazenil; Habituation, Psychophysiologic; Memory; Mental Recall; Rats; Rats, Inbred Strains; Reaction Time; Receptors, GABA-A; Retention, Psychology

1990
Relaxant effect of benzodiazepines on uterine rings isolated from estrogen-treated rats.
    European journal of pharmacology, 1990, Aug-28, Volume: 185, Issue:2-3

    Topics: Animals; Anti-Anxiety Agents; Benzodiazepinones; Bicuculline; Clonazepam; Convulsants; Diazepam; Estradiol; Estrogens; Female; Flumazenil; In Vitro Techniques; Isoquinolines; Muscle, Smooth; Potassium Chloride; Propranolol; Rats; Rats, Inbred Strains; Uterine Contraction

1990
Two subcellular locations for peripheral-type benzodiazepine acceptors in rat liver.
    European journal of biochemistry, 1990, Feb-22, Volume: 188, Issue:1

    Topics: Affinity Labels; Animals; Benzodiazepinones; Catalase; Centrifugation, Density Gradient; Clonazepam; Electrophoresis, Polyacrylamide Gel; Glutamate Dehydrogenase; Intracellular Membranes; Isoquinolines; Liver; Mitochondria, Liver; Polyethyleneimine; Rats; Receptors, GABA-A; Sonication; Subcellular Fractions; Succinate Dehydrogenase

1990
Involvement of the "peripheral" benzodiazepine receptor type (omega 3) in the tolerance to the electroencephalographic effects of benzodiazepines in rats: comparison of diazepam and clonazepam.
    Pharmacology, biochemistry, and behavior, 1990, Volume: 35, Issue:4

    Topics: Animals; Benzodiazepinones; Clonazepam; Diazepam; Drug Tolerance; Electroencephalography; Isoquinolines; Male; Rats; Rats, Inbred Strains; Receptors, GABA-A

1990
The effects of acidosis on chronically hypoxic neurons in culture.
    Experimental neurology, 1990, Volume: 107, Issue:3

    Topics: Acidosis; Animals; Benzodiazepines; Benzodiazepinones; Binding, Competitive; Cells, Cultured; Chronic Disease; Clonazepam; Culture Media; Hypoxia; Neurons; Reference Values; Time Factors

1990
"Central" and "peripheral" benzodiazepines and kinetics of lindane-induced toxicity.
    Pharmacology, biochemistry, and behavior, 1989, Volume: 32, Issue:2

    Topics: Animals; Anti-Anxiety Agents; Benzodiazepinones; Body Temperature; Clonazepam; Diazepam; Drug Interactions; Female; Hexachlorocyclohexane; Male; Phenytoin; Rats; Rats, Inbred Strains

1989
Diminution by benzodiazepines of the chronotropic responses to noradrenaline in rat isolated atria.
    European journal of pharmacology, 1989, May-30, Volume: 164, Issue:3

    Topics: 1-Methyl-3-isobutylxanthine; 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Anti-Anxiety Agents; Benzodiazepinones; Clonazepam; Colforsin; Cyclic AMP; Diazepam; Female; Flumazenil; Heart; Heart Rate; In Vitro Techniques; Isoquinolines; Male; Myocardium; Norepinephrine; Rats; Rats, Inbred Strains

1989
Pyruvate dehydrogenase interactions with peripheral-type benzodiazepine receptors.
    Journal of neurochemistry, 1989, Volume: 52, Issue:1

    Topics: Animals; Benzodiazepinones; Brain; Clonazepam; Isoquinolines; Ketoglutarate Dehydrogenase Complex; Male; Pyruvate Dehydrogenase Complex; Rats; Rats, Inbred Strains; Receptors, GABA-A; Solubility

1989
Antiproliferative action of benzodiazepines in cultured brain cells is not mediated through the peripheral-type benzodiazepine acceptor.
    Journal of neurochemistry, 1989, Volume: 53, Issue:3

    Topics: Animals; Benzodiazepines; Benzodiazepinones; Blood; Cell Division; Clonazepam; Diazepam; DNA; Glioma; Isoquinolines; Mice; Neuroblastoma; Rats; Receptors, GABA-A; Tumor Cells, Cultured

1989
Peripheral benzodiazepine binding sites in Nb 2 node lymphoma cells: effects on prolactin-stimulated proliferation and ornithine decarboxylase activity.
    European journal of pharmacology, 1989, Nov-14, Volume: 171, Issue:1

    Topics: Benzodiazepinones; Cell Division; Clonazepam; Humans; Isoquinolines; Kinetics; Lymph Nodes; Lymphoma; Ornithine Decarboxylase; Prolactin; Receptors, GABA-A; Thymidine; Tumor Cells, Cultured

1989
Testicular interstitial cells as targets for peripheral benzodiazepines.
    Neuroendocrinology, 1989, Volume: 49, Issue:3

    Topics: Animals; Benzodiazepinones; Clonazepam; Diazepam; In Vitro Techniques; Isoquinolines; Leydig Cells; Male; Rats; Rats, Inbred Strains; Testosterone

1989
Effect of ferric nitrilotriacetate on predominantly cortical neuronal cell cultures.
    Neurochemical research, 1989, Volume: 14, Issue:7

    Topics: Acetates; Animals; Benzodiazepinones; Binding, Competitive; Cerebral Cortex; Choline O-Acetyltransferase; Clonazepam; Ferric Compounds; Flunitrazepam; gamma-Aminobutyric Acid; Mice; Neurons; Nitrilotriacetic Acid; Proteins

1989
Benzodiazepine receptor development in murine glial cultures.
    Developmental neuroscience, 1987, Volume: 9, Issue:3

    Topics: Animals; Animals, Newborn; Benzodiazepinones; Binding, Competitive; Cells, Cultured; Clonazepam; Diazepam; Mice; Neuroglia; Receptors, GABA-A

1987
Regional distribution of a Ro5 4864 binding site that is functionally coupled to the gamma-aminobutyric acid/benzodiazepine receptor complex in rat brain.
    The Journal of pharmacology and experimental therapeutics, 1988, Volume: 244, Issue:1

    Topics: Affinity Labels; Animals; Autoradiography; Azides; Benzodiazepines; Benzodiazepinones; Brain; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Clonazepam; Male; Photochemistry; Rats; Rats, Inbred Strains; Receptors, GABA-A

1988
Differential effects of benzodiazepines on phospholipid methylation in hippocampus and cerebellum of rats.
    Life sciences, 1988, Volume: 42, Issue:5

    Topics: Animals; Benzodiazepines; Benzodiazepinones; Cell Membrane; Cerebellum; Clonazepam; Hippocampus; Isoquinolines; Male; Methylation; Methyltransferases; Neurons; Phosphatidylcholines; Phosphatidylethanolamine N-Methyltransferase; Phosphatidylethanolamines; Phospholipids; Rats; Receptors, GABA-A; Synaptosomes

1988
Presence of peripheral-type benzodiazepine binding sites on human erythrocyte membranes.
    European journal of pharmacology, 1988, Jul-26, Volume: 152, Issue:1-2

    Topics: Benzodiazepinones; Clonazepam; Convulsants; Erythrocyte Membrane; Flunitrazepam; Humans; In Vitro Techniques; Isoquinolines; Kinetics; Monoamine Oxidase; Receptors, GABA-A

1988
Characterization of stress-induced alterations in [3H] Ro5-4864 binding to peripheral benzodiazepine receptors in rat heart and kidney.
    Pharmacology, biochemistry, and behavior, 1988, Volume: 30, Issue:4

    Topics: Adrenalectomy; Animals; Benzodiazepinones; Clonazepam; Convulsants; Electroshock; Hypophysectomy; Kidney; Male; Myocardium; Rats; Rats, Inbred Strains; Receptors, GABA-A; Reference Values; Stress, Psychological

1988
Blockade of non-opioid analgesia in intruder mice by selective neuronal and non-neuronal benzodiazepine recognition site ligands.
    Psychopharmacology, 1988, Volume: 96, Issue:1

    Topics: Aggression; Analgesia; Animals; Benzodiazepinones; Clonazepam; Convulsants; Isoquinolines; Ligands; Male; Mice; Mice, Inbred DBA; Neurons; Nociceptors; Reaction Time; Receptors, GABA-A

1988
Triazolam, an anomalous benzodiazepine receptor ligand: in vitro characterization of alprazolam and triazolam binding.
    Journal of neurochemistry, 1985, Volume: 45, Issue:2

    Topics: Alprazolam; Animals; Anti-Anxiety Agents; Benzodiazepines; Benzodiazepinones; Carbolines; Clonazepam; Flunitrazepam; gamma-Aminobutyric Acid; Humans; Kinetics; Male; Rats; Rats, Inbred Strains; Receptors, GABA-A; Triazolam

1985
Neurotransmitter changes during development of cortical neuronal cultures.
    Developmental neuroscience, 1986, Volume: 8, Issue:2

    Topics: Animals; Benzodiazepinones; Cells, Cultured; Cerebral Cortex; Choline O-Acetyltransferase; Clonazepam; Diazepam; Fetus; Flunitrazepam; gamma-Aminobutyric Acid; Glutamate Decarboxylase; Mice; Neurotransmitter Agents

1986
The role of central- and peripheral-type benzodiazepine receptors in anxiolytic-agent augmentation of NaCl solution intake: effects of clonazepam and Ro 5-4864.
    Pharmacology, biochemistry, and behavior, 1988, Volume: 30, Issue:3

    Topics: Animals; Anti-Anxiety Agents; Benzodiazepinones; Clonazepam; Dose-Response Relationship, Drug; Drinking Behavior; Drug Interactions; Male; Rats; Receptors, GABA-A; Reference Values; Saline Solution, Hypertonic; Water Deprivation

1988
Peripheral-type benzodiazepine receptors in endocrine organs: autoradiographic localization in rat pituitary, adrenal, and testis.
    Endocrinology, 1985, Volume: 116, Issue:2

    Topics: Adrenal Glands; Animals; Autoradiography; Benzodiazepinones; Binding, Competitive; Clonazepam; Isoquinolines; Male; Pituitary Gland; Rats; Rats, Inbred Strains; Receptors, GABA-A; Testis; Tissue Distribution

1985
[Presence of a peripheral type benzodiazepine binding site on the macrophage; its possible role in immunomodulation].
    Comptes rendus de l'Academie des sciences. Serie III, Sciences de la vie, 1985, Volume: 300, Issue:8

    Topics: Animals; Antibody Formation; Benzodiazepines; Benzodiazepinones; Clonazepam; Erythrocytes; Ethanol; Female; Flunitrazepam; Macrophages; Mice; Receptors, GABA-A; Sheep

1985
Clonazepam-induced hyperphagia in nondeprived rats: tests of pharmacological specificity with Ro5-4864, Ro5-3663, Ro15-1788 and CGS 9896.
    Pharmacology, biochemistry, and behavior, 1985, Volume: 22, Issue:5

    Topics: Animals; Benzodiazepinones; Clonazepam; Drug Interactions; Feeding Behavior; Flumazenil; Humans; Hyperphagia; Male; Pyrazoles; Rats; Receptors, GABA-A

1985
Characteristics of benzodiazepine receptor binding in living cultures of mouse cerebral cortex at physiologic temperature.
    Brain research, 1985, Volume: 353, Issue:1

    Topics: Animals; Benzodiazepinones; Cerebral Cortex; Clonazepam; Culture Techniques; Kinetics; Mice; Receptors, GABA-A; Temperature

1985
Benzodiazepine receptor-mediated chemotaxis of human monocytes.
    Science (New York, N.Y.), 1985, Sep-20, Volume: 229, Issue:4719

    Topics: Benzodiazepinones; Binding, Competitive; Chemotaxis, Leukocyte; Clonazepam; Humans; Isoquinolines; Monocytes; Receptors, GABA-A

1985
Benzodiazepine binding characteristics of embryonic rat brain neurons grown in culture.
    Journal of neurochemistry, 1985, Volume: 45, Issue:6

    Topics: Animals; Benzodiazepines; Benzodiazepinones; Brain; Carbolines; Cells, Cultured; Clonazepam; Diazepam; Dose-Response Relationship, Drug; Flumazenil; gamma-Aminobutyric Acid; Neurons; Pyridazines; Rats; Receptors, GABA-A

1985
Solubilization of peripheral benzodiazepine-binding sites from rat kidney.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 1985, Volume: 5, Issue:11

    Topics: Animals; Benzodiazepinones; Binding, Competitive; Carbolines; Chlordiazepoxide; Clonazepam; Diazepam; Digitonin; Flumazenil; Flurazepam; Guanidine; Guanidines; Hot Temperature; Isoquinolines; Kidney; Kinetics; Male; Rats; Rats, Inbred Strains; Receptors, GABA-A; Solubility; Time Factors; Urea

1985
Pharmacology of peripheral type benzodiazepine receptors in the heart.
    Progress in clinical and biological research, 1985, Volume: 192

    Topics: Action Potentials; Animals; Benzodiazepinones; Clonazepam; Convulsants; Diazepam; Electric Stimulation; Guinea Pigs; Heart; Heart Ventricles; Isoquinolines; Kinetics; Myocardial Contraction; Myocardium; Receptors, GABA-A; Ventricular Function

1985
Autoradiographic localization of benzodiazepine receptor binding in dissociated cultures of fetal mouse cerebral cortex.
    Journal of neurochemistry, 1986, Volume: 46, Issue:3

    Topics: Affinity Labels; Animals; Autoradiography; Benzodiazepinones; Binding, Competitive; Cells, Cultured; Cerebral Cortex; Clonazepam; Embryo, Mammalian; Flunitrazepam; Mice; Neurons; Photochemistry; Receptors, GABA-A

1986
Convulsant effect of Ro 5-4864, a peripheral type benzodiazepine, on the baboon (Papio papio).
    Neuroscience letters, 1986, May-15, Volume: 66, Issue:2

    Topics: Animals; Benzodiazepines; Benzodiazepinones; Clonazepam; Diazepam; Dose-Response Relationship, Drug; Flumazenil; Isoquinolines; Papio; Receptors, GABA-A; Seizures

1986
Hormonal interactions with benzodiazepine binding sites in vitro.
    Life sciences, 1986, Aug-25, Volume: 39, Issue:8

    Topics: Adrenal Cortex Hormones; Animals; Benzodiazepinones; Binding, Competitive; Clonazepam; Hormones; In Vitro Techniques; Male; Prostaglandins; Radioligand Assay; Rats; Rats, Inbred Strains; Receptors, GABA-A; Thyroxine

1986
Central- and peripheral-type benzodiazepine receptors.
    Advances in biochemical psychopharmacology, 1986, Volume: 41

    Topics: Animals; Benzodiazepinones; Binding, Competitive; Brain; Clonazepam; Convulsants; Flunitrazepam; Kidney; Kinetics; Membranes; Muscimol; Rats; Receptors, GABA-A; Subcellular Fractions; Tissue Distribution

1986
Pyrazolo[4,5-c]quinolines. 3. Synthesis, receptor binding, and 13C NMR study.
    Journal of pharmaceutical sciences, 1986, Volume: 75, Issue:12

    Topics: Animals; Benzodiazepinones; Binding, Competitive; Brain; Cattle; Chemical Phenomena; Chemistry; Clonazepam; Flunitrazepam; In Vitro Techniques; Magnetic Resonance Spectroscopy; Pyrazoles; Quinolines; Receptors, GABA-A

1986
Coexistence of central and peripheral benzodiazepine binding sites in the human pineal gland.
    Life sciences, 1987, Apr-13, Volume: 40, Issue:15

    Topics: Aged; Benzodiazepinones; Binding, Competitive; Cell Membrane; Clonazepam; Female; Flumazenil; Flunitrazepam; Humans; Isoquinolines; Male; Middle Aged; Pineal Gland; Receptors, GABA-A

1987
Benzodiazepine receptor affinity alterations at physiologic temperature after chronic clonazepam exposure.
    Brain & development, 1987, Volume: 9, Issue:1

    Topics: Animals; Benzodiazepinones; Body Temperature; Cells, Cultured; Cerebral Cortex; Clonazepam; Convulsants; Flunitrazepam; Kinetics; Mice; Receptors, GABA-A; Time Factors

1987
Peripheral benzodiazepines enhance the respiratory burst of macrophage-like P388D1 cells stimulated by arachidonic acid.
    International journal of immunopharmacology, 1987, Volume: 9, Issue:3

    Topics: Animals; Arachidonic Acid; Arachidonic Acids; Benzodiazepinones; Cell Line; Clonazepam; Diazepam; Isoquinolines; Kinetics; Macrophages; Receptors, GABA-A; Superoxides

1987
Diazepam-sensitive specific binding of phenytoin in rat brain.
    Journal of receptor research, 1986, Volume: 6, Issue:3-4

    Topics: Animals; Benzodiazepinones; Binding Sites; Cell Membrane; Cerebral Cortex; Clonazepam; Diazepam; Flumazenil; Male; Phenytoin; Rats; Rats, Inbred Strains

1986
Inhibition of cell proliferation of human gliomas by benzodiazepines in vitro.
    Acta neurologica Scandinavica, 1988, Volume: 77, Issue:3

    Topics: Astrocytoma; Benzodiazepines; Benzodiazepinones; Cell Division; Clonazepam; Diazepam; Female; Flumazenil; Glioma; Humans; Male; Middle Aged; Thymidine; Tumor Cells, Cultured

1988
Central administration of benzodiazepines alters water absorption by the rat ileum in vivo.
    Gastroenterology, 1987, Volume: 93, Issue:2

    Topics: Animals; Benzodiazepines; Benzodiazepinones; Clonazepam; Diazepam; Ileum; Injections, Intraventricular; Intestinal Absorption; Lorazepam; Male; Nifedipine; Nitrendipine; Rats; Rats, Inbred Strains; Water

1987
Benzodiazepine Ro 5-4864 increases coronary flow.
    European journal of pharmacology, 1987, Nov-03, Volume: 143, Issue:1

    Topics: Animals; Benzodiazepinones; Clonazepam; Convulsants; Coronary Circulation; Heart Rate; In Vitro Techniques; Isoquinolines; Male; Muscle Contraction; Rats; Rats, Inbred Strains

1987
Electrophysiological and pharmacological characterization of peripheral benzodiazepine receptors in a guinea pig heart preparation.
    Life sciences, 1984, Aug-27, Volume: 35, Issue:9

    Topics: Action Potentials; Animals; Benzodiazepinones; Clonazepam; Convulsants; Diazepam; Dose-Response Relationship, Drug; Electric Stimulation; Flumazenil; Guinea Pigs; Heart; In Vitro Techniques; Isoquinolines; Myocardial Contraction; Myocardium; Receptors, Cell Surface; Receptors, GABA-A

1984
Autoradiographic localisation of benzodiazepine receptors in the rat pituitary gland.
    European journal of pharmacology, 1984, Jul-20, Volume: 102, Issue:3-4

    Topics: Animals; Autoradiography; Benzodiazepinones; Clonazepam; Flumazenil; gamma-Aminobutyric Acid; In Vitro Techniques; Male; Pituitary Gland; Rats; Rats, Inbred Strains; Receptors, GABA-A

1984
Flunitrazepam binding to intact and homogenized astrocytes and neurons in primary cultures.
    Journal of neurochemistry, 1984, Volume: 43, Issue:5

    Topics: Animals; Astrocytes; Benzodiazepinones; Cells, Cultured; Clonazepam; Diazepam; Flunitrazepam; Kinetics; Mice; Neurons; Receptors, GABA-A; Temperature

1984
Autoradiographic localization of benzodiazepine receptors in the rat kidney.
    The American journal of physiology, 1984, Volume: 247, Issue:5 Pt 2

    Topics: Animals; Autoradiography; Benzodiazepinones; Clonazepam; Diazepam; Flunitrazepam; Kidney; Kidney Tubules, Distal; Loop of Henle; Male; Mucoproteins; Rats; Rats, Inbred Strains; Receptors, GABA-A; Tritium; Uromodulin

1984
Benzodiazepine binding sites in human myometrium.
    International journal of tissue reactions, 1984, Volume: 6, Issue:5

    Topics: Adult; Benzodiazepinones; Binding Sites; Cell Membrane; Clonazepam; Diazepam; Female; Flunitrazepam; Humans; In Vitro Techniques; Lorazepam; Middle Aged; Myometrium; Receptors, GABA-A

1984
Analysis of benzodiazepine binding sites in rat pituitary gland.
    Brain research, 1984, Dec-10, Volume: 323, Issue:2

    Topics: Animals; Benzodiazepinones; Binding, Competitive; Clonazepam; Diazepam; Flunitrazepam; gamma-Aminobutyric Acid; In Vitro Techniques; Male; Pituitary Gland; Rats; Rats, Inbred Strains; Receptors, GABA-A

1984
Binding of [3H]flunitrazepam to the LM cell, a transformed murine fibroblast.
    Biochemical pharmacology, 1983, Jul-15, Volume: 32, Issue:14

    Topics: Animals; Anti-Anxiety Agents; Benzodiazepinones; Binding Sites; Cell Line; Cell Membrane; Choline; Clonazepam; Culture Media; Cyclic AMP; Flunitrazepam; Kinetics; Mice; Neoplasms, Experimental; Phospholipids

1983
Properties of [3H]diazepam binding sites on rat blood platelets.
    Life sciences, 1980, Nov-17, Volume: 27, Issue:20

    Topics: Animals; Benzodiazepinones; Blood Platelets; Clonazepam; Diazepam; Hydrogen-Ion Concentration; Kinetics; Male; Rats; Receptors, Drug; Receptors, GABA-A; Temperature

1980
Peripheral benzodiazepine binding sites: effect of PK 11195, 1-(2-chlorophenyl)-N-methyl-N-(1-methylpropyl)-3-isoquinolinecarboxamide. I. In vitro studies.
    Life sciences, 1983, Apr-18, Volume: 32, Issue:16

    Topics: Adrenal Glands; Animals; Benzodiazepinones; Blood Platelets; Brain; Clonazepam; Diazepam; In Vitro Techniques; Isoquinolines; Kidney; Male; Myocardium; Rats; Rats, Inbred Strains; Receptors, Cell Surface; Receptors, GABA-A; Tissue Distribution

1983
Peripheral benzodiazepine binding sites: effect of PK 11195, 1-(2-chlorophenyl)-N-methyl-(1-methylpropyl)-3 isoquinolinecarboxamide. II. In vivo studies.
    Life sciences, 1983, Apr-18, Volume: 32, Issue:16

    Topics: Animals; Benzodiazepinones; Brain; Clonazepam; Diazepam; Isoquinolines; Kidney; Kinetics; Male; Mice; Myocardium; Receptors, Cell Surface; Receptors, GABA-A

1983
Development and differentiation of the benzodiazepine receptor in cultures of fetal mouse spinal cord.
    Brain research, 1983, Volume: 283, Issue:2-3

    Topics: Animals; Benzodiazepinones; Cell Differentiation; Clonazepam; Diazepam; Fetus; Flunitrazepam; Kinetics; Mice; Neurons; Receptors, Cell Surface; Receptors, GABA-A; Spinal Cord

1983
Differentiation between two ligands for peripheral benzodiazepine binding sites, [3H]RO5-4864 and [3H]PK 11195, by thermodynamic studies.
    Life sciences, 1983, Aug-01, Volume: 33, Issue:5

    Topics: Animals; Benzodiazepinones; Clonazepam; Diazepam; Dipyridamole; Isoquinolines; Ligands; Male; Membranes; Myocardium; Rats; Receptors, Cell Surface; Receptors, GABA-A; Thermodynamics

1983
Benzodiazepine receptors along the nephron: [3H]PK 11195 binding in rat tubules.
    FEBS letters, 1984, Apr-24, Volume: 169, Issue:2

    Topics: Animals; Benzodiazepinones; Clonazepam; Dose-Response Relationship, Drug; Isoquinolines; Kidney Tubules; Male; Nephrons; Rats; Rats, Inbred Strains; Receptors, Cell Surface; Receptors, GABA-A; Tissue Distribution

1984
Receptors for psychoactive drugs: autoradiographic visualization of benzodiazepine binding sites.
    Acta histochemica. Supplementband, 1984, Volume: 29

    Topics: Animals; Autoradiography; Benzodiazepinones; Binding Sites; Brain; Brain Chemistry; Clonazepam; Convulsants; Rats; Receptors, Cell Surface; Receptors, GABA-A

1984
Specific binding of [3H]diazepam in mouse glioblastoma: the influence of clonazepam and Ro 5-4864 on [3H]diazepam binding.
    Neuroscience letters, 1984, Dec-21, Volume: 52, Issue:3

    Topics: Animals; Benzodiazepinones; Binding Sites; Cell Line; Clonazepam; Diazepam; Glioma; Mice; Neuroglia

1984
[3H]diazepam binding sites on chick neurons in primary culture.
    Neuroscience letters, 1983, Aug-19, Volume: 39, Issue:1

    Topics: Animals; Benzodiazepinones; Binding Sites; Binding, Competitive; Cells, Cultured; Chick Embryo; Clonazepam; Diazepam; gamma-Aminobutyric Acid; Neurons; Pentobarbital; Telencephalon

1983
Properties of [3H]diazepam binding sites on cultured murine glia and neurons.
    Brain research, 1984, Volume: 316, Issue:1

    Topics: Animals; Animals, Newborn; Benzodiazepinones; Binding Sites; Cells, Cultured; Cerebral Cortex; Clonazepam; Diazepam; Kinetics; Mice; Neuroglia; Neurons

1984
Vascular and tubular actions of diazepam in isolated and perfused rat kidney.
    European journal of pharmacology, 1995, Apr-04, Volume: 276, Issue:3

    Topics: Animals; Benzodiazepinones; Biological Transport, Active; Blood Vessels; Clonazepam; Convulsants; Diazepam; Diuresis; In Vitro Techniques; Kidney Function Tests; Kidney Tubules; Male; Muscle Contraction; Muscle Relaxation; Muscle, Smooth, Vascular; Natriuresis; Norepinephrine; Potassium Chloride; Rats; Rats, Wistar; Renal Circulation

1995
Mitochondrial benzodiazepine receptor linked to inner membrane ion channels by nanomolar actions of ligands.
    Proceedings of the National Academy of Sciences of the United States of America, 1993, Feb-15, Volume: 90, Issue:4

    Topics: Animals; Benzodiazepinones; Clonazepam; Convulsants; Flumazenil; Intracellular Membranes; Ion Channels; Isoquinolines; Male; Membrane Potentials; Mitochondria, Heart; Protoporphyrins; Rats; Rats, Sprague-Dawley; Receptors, GABA-A; Submitochondrial Particles

1993
Differential effects of 4'-chlorodiazepam on expressed human GABAA receptors.
    Journal of neurochemistry, 1995, Volume: 64, Issue:2

    Topics: Benzodiazepinones; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cell Line; Clonazepam; Flumazenil; Humans; Quinolines; Receptors, GABA; Transfection

1995
Modification of the photodynamic action of delta-aminolaevulinic acid (ALA) on rat pancreatoma cells by mitochondrial benzodiazepine receptor ligands.
    British journal of cancer, 1995, Volume: 71, Issue:2

    Topics: Aminolevulinic Acid; Animals; Benzodiazepines; Benzodiazepinones; Cell Division; Cell Survival; Clonazepam; Flumazenil; Isoquinolines; Ligands; Mitochondria; Oxygen; Pancreatic Neoplasms; Photochemotherapy; Protoporphyrins; Radiation-Protective Agents; Radiation-Sensitizing Agents; Rats; Receptors, GABA-A; Singlet Oxygen; Tumor Cells, Cultured

1995
Effect of peripheral benzodiazepine receptor ligands on lipopolysaccharide-induced tumor necrosis factor activity in thioglycolate-treated mice.
    Antimicrobial agents and chemotherapy, 1994, Volume: 38, Issue:4

    Topics: Animals; Benzodiazepinones; Clonazepam; GABA-A Receptor Antagonists; Isoquinolines; Ligands; Lipopolysaccharides; Macrophages, Peritoneal; Male; Mice; Mice, Inbred C3H; Midazolam; Receptors, GABA-A; Thioglycolates; Tumor Necrosis Factor-alpha

1994
In vitro inhibition of cellular immune responses by benzodiazepines and PK 11195. Effects on mitogen- and alloantigen-driven lymphocyte proliferation and on IL-1, IL-2 synthesis and IL-2 receptor expression.
    Immunopharmacology and immunotoxicology, 1993, Volume: 15, Issue:5

    Topics: Animals; B-Lymphocytes; Benzodiazepines; Benzodiazepinones; Clonazepam; Diazepam; Female; Flumazenil; Immunity, Cellular; In Vitro Techniques; Interleukin-1; Interleukin-2; Isoquinolines; Lymphocyte Activation; Male; Mice; Mice, Inbred A; Mice, Inbred C57BL; Neuroimmunomodulation; Receptors, GABA-A; T-Lymphocytes

1993
The specific binding of the platelet-activating factor (PAF) receptor antagonist WEB 2086 and the benzodiazepine flunitrazepam to rat hepatocytes.
    Life sciences, 1996, Volume: 58, Issue:5

    Topics: Animals; Anti-Anxiety Agents; Anticonvulsants; Azepines; Benzodiazepinones; Bicuculline; Cells, Cultured; Clonazepam; Convulsants; Flunitrazepam; Kinetics; Liver; Male; Platelet Aggregation Inhibitors; Platelet Membrane Glycoproteins; Rats; Rats, Sprague-Dawley; Receptors, Cell Surface; Receptors, G-Protein-Coupled; Triazoles; Tritium

1996
Prevention of ACTH- and adrenalectomy-induced muricidal behavior: by benzodiazepinic ligands.
    Peptides, 1997, Volume: 18, Issue:2

    Topics: Adrenalectomy; Adrenocorticotropic Hormone; Aggression; Animals; Benzodiazepinones; Clonazepam; Flumazenil; GABA Modulators; Isoquinolines; Male; Mice; Muscimol; Rats; Rats, Wistar; Receptors, GABA-A; Time Factors

1997
Synthesis and biology of a 7-nitro-2,1,3-benzoxadiazol-4-yl derivative of 2-phenylindole-3-acetamide: a fluorescent probe for the peripheral-type benzodiazepine receptor.
    Journal of medicinal chemistry, 1997, Aug-01, Volume: 40, Issue:16

    Topics: 4-Chloro-7-nitrobenzofurazan; Animals; Benzodiazepinones; Biological Transport; Cholesterol; Clonazepam; Fluorescent Dyes; Hypolipidemic Agents; Indoleacetic Acids; Isoquinolines; Ligands; Male; Mice; Microscopy, Fluorescence; Mitochondria; Rats; Receptors, GABA-A; Tumor Cells, Cultured

1997
Effects of peripheral-type benzodiazepine receptor antisense knockout on MA-10 Leydig cell proliferation and steroidogenesis.
    The Journal of biological chemistry, 1998, Mar-06, Volume: 273, Issue:10

    Topics: Algestone; Androstenedione; Animals; Benzodiazepinones; Cell Division; Clonazepam; Cyclic AMP; DNA, Antisense; GABA-A Receptor Antagonists; Isoquinolines; Leydig Cells; Male; Mice; Plasmids; Progesterone; Protein Binding; Receptors, GABA-A; RNA, Messenger; Transfection; Tumor Cells, Cultured

1998
Characterization of binding sites for the omega3 receptor ligands [3H]PK11195 and [3H]RO5-4864 in human brain.
    European journal of pharmacology, 1997, Dec-04, Volume: 340, Issue:1

    Topics: Allosteric Regulation; Benzodiazepines; Benzodiazepinones; Binding Sites; Binding, Competitive; Clonazepam; Convulsants; Detergents; Diazepam; Dithiothreitol; Female; Histidine; Humans; Isoquinolines; Ligands; Male; Occipital Lobe; Receptors, GABA-A; Sulfhydryl Reagents; Tritium

1997
Modulation of intracellular calcium in human neutrophils by peripheral benzodiazepine receptor ligands.
    Journal of chemotherapy (Florence, Italy), 1998, Volume: 10, Issue:2

    Topics: Anti-Anxiety Agents; Benzodiazepinones; Calcium; Clonazepam; Cytosol; Diazepam; Drug Antagonism; GABA Modulators; Humans; Isoquinolines; Neutrophils; Receptors, GABA-A

1998
Antiproliferative and differentiating effects of benzodiazepine receptor ligands on B16 melanoma cells.
    Biochemical pharmacology, 1998, Oct-15, Volume: 56, Issue:8

    Topics: Animals; Antineoplastic Agents; Benzodiazepinones; Cell Cycle; Cell Differentiation; Cell Division; Clonazepam; Diazepam; GABA Agents; gamma-Glutamyltransferase; Isoquinolines; Melanoma, Experimental; Mice; Nucleotides; Phenotype; Tumor Cells, Cultured

1998
Inhibitory regulation of amylase release in rat parotid acinar cells by benzodiazepine receptors.
    European journal of pharmacology, 1998, Oct-23, Volume: 359, Issue:2-3

    Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Amylases; Animals; Atropine; Benzodiazepinones; Carbachol; Clonazepam; Diazepam; Dose-Response Relationship, Drug; Flumazenil; GABA Modulators; GABA-A Receptor Agonists; GABA-A Receptor Antagonists; Isoproterenol; Male; Muscarinic Agonists; Muscarinic Antagonists; Parotid Gland; Propranolol; Rats; Rats, Wistar; Receptors, GABA-A

1998
Effect of benzodiazepines and neurosteroids on ammonia-induced swelling in cultured astrocytes.
    Journal of neuroscience research, 1998, Dec-01, Volume: 54, Issue:5

    Topics: Ammonia; Astrocytes; Atrial Natriuretic Factor; Benzodiazepines; Benzodiazepinones; Brain Edema; Cell Size; Clonazepam; Dehydroepiandrosterone Sulfate; Desoxycorticosterone; Diazepam; Diazepam Binding Inhibitor; Flumazenil; GABA-A Receptor Agonists; GABA-A Receptor Antagonists; Isoquinolines; Nerve Tissue Proteins; Neuropeptides; Peptide Fragments; Pregnanolone; Pregnenolone; Protoporphyrins; Receptors, GABA-A; Steroids; Up-Regulation

1998
Benzodiazepine receptor agonists modulate thymocyte apoptosis through reduction of the mitochondrial transmembrane potential.
    Japanese journal of pharmacology, 1999, Volume: 79, Issue:2

    Topics: Animals; Apoptosis; Benzodiazepines; Benzodiazepinones; Binding Sites; Caspase Inhibitors; Cells, Cultured; Clonazepam; Dexamethasone; Diazepam; Drug Interactions; Drug Synergism; Etoposide; GABA-A Receptor Agonists; Male; Membrane Potentials; Mice; Mice, Inbred BALB C; Mitochondria; Protease Inhibitors; Protein Biosynthesis; Proteins; RNA, Messenger; Thymus Gland

1999
Central and peripheral benzodiazepine ligands prevent mitochondrial damage induced by noise exposure in the rat myocardium: an ultrastructural study.
    The Anatomical record, 1999, 07-01, Volume: 255, Issue:3

    Topics: Animals; Benzodiazepines; Benzodiazepinones; Clonazepam; Diazepam; GABA Modulators; Isoquinolines; Male; Microscopy, Electron; Microscopy, Electron, Scanning; Mitochondria, Heart; Myocardium; Noise; Rats; Rats, Wistar; Time Factors

1999
Peripheral benzodiazepine receptor agonists exhibit potent antiapoptotic activities.
    Biochemical and biophysical research communications, 1999, Nov-19, Volume: 265, Issue:2

    Topics: Apoptosis; Benzodiazepinones; Clonazepam; Diazepam; Flunitrazepam; GABA-A Receptor Agonists; GABA-A Receptor Antagonists; Humans; Isoquinolines; Jurkat Cells; Kinetics; Ligands; Receptors, GABA-A; Transfection; Tumor Necrosis Factor-alpha; U937 Cells

1999
2-Arylpyrazolo[1,5-a]pyrimidin-3-yl acetamides. New potent and selective peripheral benzodiazepine receptor ligands.
    Bioorganic & medicinal chemistry, 2001, Volume: 9, Issue:10

    Topics: Acetamides; Animals; Benzodiazepinones; Binding Sites; Cerebral Cortex; Clonazepam; Flumazenil; Glioma; Intracellular Membranes; Isoquinolines; Kidney; Ligands; Magnetic Resonance Spectroscopy; Molecular Structure; Pyrazoles; Pyrimidines; Rats; Receptors, GABA-A; Structure-Activity Relationship; Thermodynamics; Tumor Cells, Cultured

2001
Diazepam inhibits HIV-1 Tat-induced migration of human microglia.
    Journal of neurovirology, 2001, Volume: 7, Issue:5

    Topics: Adjuvants, Immunologic; Benzodiazepinones; Calcium Signaling; Chemotaxis; Clonazepam; Diazepam; Gene Products, tat; HIV-1; Humans; Microglia; Nerve Tissue Proteins; Receptors, CCR5; Receptors, GABA-A; tat Gene Products, Human Immunodeficiency Virus; Up-Regulation

2001
Effect of midazolam on interleukin-6 mRNA expression in human peripheral blood mononuclear cells in the absence of lipopolysaccharide.
    Cytokine, 2001, Sep-21, Volume: 15, Issue:6

    Topics: Anti-Anxiety Agents; Anticonvulsants; Benzodiazepinones; Binding, Competitive; Cell Survival; Cells, Cultured; Clonazepam; Convulsants; DNA, Complementary; Dose-Response Relationship, Drug; GABA-A Receptor Agonists; Humans; Interleukin-6; Leukocytes, Mononuclear; Ligands; Lipopolysaccharides; Midazolam; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Time Factors

2001
Effects on free radical generation by ligands of the peripheral benzodiazepine receptor in cultured neural cells.
    Journal of neurochemistry, 2002, Volume: 83, Issue:5

    Topics: Animals; Antioxidants; Astrocytes; Benzodiazepinones; Binding, Competitive; Cells, Cultured; Clonazepam; Cyclosporine; Dose-Response Relationship, Drug; Free Radicals; Isoquinolines; Ligands; Microglia; Mitochondria; Neurons; Protoporphyrins; Rats; Receptors, GABA-A

2002
Effects of peripheral-type benzodiazepine receptor ligands on Ehrlich tumor cell proliferation.
    European journal of pharmacology, 2006, Nov-21, Volume: 550, Issue:1-3

    Topics: Animals; Benzodiazepinones; Carcinoma, Ehrlich Tumor; Cell Cycle; Cell Division; Cell Proliferation; Clonazepam; Flow Cytometry; GABA Modulators; Immunohistochemistry; Isoquinolines; Ligands; Mice; Receptors, GABA-A

2006
Characterization of two classes of benzodiazepine binding sites in Schistosoma mansoni.
    Parasitology, 2007, Volume: 134, Issue:Pt 7

    Topics: Animals; Benzodiazepines; Benzodiazepinones; Binding Sites; Clonazepam; Diazepam; Flunitrazepam; GABA Agonists; GABA Modulators; Inhibitory Concentration 50; Isoquinolines; Ligands; Male; Pyridines; Rats; Rats, Wistar; Receptors, GABA-A; Schistosoma mansoni; Synaptosomes; Temperature; Time Factors; Tritium; Zolpidem

2007
Allosteric modulation by benzodiazepines of GABA-gated chloride channels of an identified insect motor neurone.
    Invertebrate neuroscience : IN, 2009, Volume: 9, Issue:2

    Topics: Animals; Benzodiazepines; Benzodiazepinones; Chloride Channels; Clonazepam; Diazepam; Dose-Response Relationship, Drug; Evoked Potentials; GABA Modulators; gamma-Aminobutyric Acid; Glutamic Acid; In Vitro Techniques; Insect Proteins; Male; Membrane Potentials; Microelectrodes; Motor Neurons; Periplaneta

2009
Investigation into mechanisms mediating the inhibitory effect of 1,4-benzodiazepines on mast cells by gene expression profiling.
    Life sciences, 2013, Mar-14, Volume: 92, Issue:6-7

    Topics: Adult; Aged; Benzodiazepinones; Clonazepam; Female; Flunitrazepam; Gene Expression; Gene Expression Profiling; HL-60 Cells; Humans; Male; Mast Cells; Mastocytosis; Microarray Analysis; Middle Aged; Polymerase Chain Reaction

2013
Acute chloroquine poisoning: A comprehensive experimental toxicology assessment of the role of diazepam.
    British journal of pharmacology, 2020, Volume: 177, Issue:21

    Topics: Animals; Arrhythmias, Cardiac; Benzodiazepinones; Cardiotoxicity; Chloroquine; Clonazepam; Coronavirus Infections; COVID-19; Diazepam; Dose-Response Relationship, Drug; Drug Overdose; Electrocardiography; Female; Hypokalemia; Male; Pandemics; Pneumonia, Viral; Rabbits; Random Allocation; Rats; Rats, Wistar

2020