Page last updated: 2024-09-05

ro 5-3438 and chlordesmethyldiazepam

ro 5-3438 has been researched along with chlordesmethyldiazepam in 4 studies

Compound Research Comparison

Studies
(ro 5-3438)
Trials
(ro 5-3438)
Recent Studies (post-2010)
(ro 5-3438)
Studies
(chlordesmethyldiazepam)
Trials
(chlordesmethyldiazepam)
Recent Studies (post-2010) (chlordesmethyldiazepam)
7001603

Protein Interaction Comparison

ProteinTaxonomyro 5-3438 (IC50)chlordesmethyldiazepam (IC50)
Gamma-aminobutyric acid receptor subunit piHomo sapiens (human)0.0028
Gamma-aminobutyric acid receptor subunit deltaHomo sapiens (human)0.0028
Gamma-aminobutyric acid receptor subunit alpha-1Homo sapiens (human)0.0028
Gamma-aminobutyric acid receptor subunit beta-1Homo sapiens (human)0.0028
Gamma-aminobutyric acid receptor subunit gamma-2Homo sapiens (human)0.0028
Gamma-aminobutyric acid receptor subunit beta-3Homo sapiens (human)0.0028
Gamma-aminobutyric acid receptor subunit alpha-5Homo sapiens (human)0.0028
Gamma-aminobutyric acid receptor subunit alpha-3Homo sapiens (human)0.0028
Gamma-aminobutyric acid receptor subunit alpha-2Homo sapiens (human)0.0028
Gamma-aminobutyric acid receptor subunit beta-2Homo sapiens (human)0.0028
Gamma-aminobutyric acid receptor subunit alpha-4Homo sapiens (human)0.0028
Gamma-aminobutyric acid receptor subunit epsilonHomo sapiens (human)0.0028
Gamma-aminobutyric acid receptor subunit alpha-6Homo sapiens (human)0.0028
Gamma-aminobutyric acid receptor subunit gamma-1Homo sapiens (human)0.0028
Gamma-aminobutyric acid receptor subunit gamma-3Homo sapiens (human)0.0028
Gamma-aminobutyric acid receptor subunit thetaHomo sapiens (human)0.0028

Research

Studies (4)

TimeframeStudies, this research(%)All Research%
pre-19901 (25.00)18.7374
1990's3 (75.00)18.2507
2000's0 (0.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Blair, T; Webb, GA1
Aoyama, T; Ichikawa, H; Suzuki, Y1
Johnston, GA; Maddalena, DJ1
Karplus, M; So, SS1

Reviews

1 review(s) available for ro 5-3438 and chlordesmethyldiazepam

ArticleYear
Neural networks applied to quantitative structure-activity relationship analysis.
    Journal of medicinal chemistry, 1990, Volume: 33, Issue:9

    Topics: Animals; Azirines; Benzodiazepines; Carbazilquinone; Nerve Net; Nervous System; Regression Analysis; Structure-Activity Relationship

1990

Other Studies

3 other study(ies) available for ro 5-3438 and chlordesmethyldiazepam

ArticleYear
Electronic factors in the structure-activity relationship of some 1,4-benzodiazepin-2-ones.
    Journal of medicinal chemistry, 1977, Volume: 20, Issue:9

    Topics: Benzodiazepinones; Electrochemistry; Structure-Activity Relationship

1977
Prediction of receptor properties and binding affinity of ligands to benzodiazepine/GABAA receptors using artificial neural networks.
    Journal of medicinal chemistry, 1995, Feb-17, Volume: 38, Issue:4

    Topics: Binding Sites; Ligands; Neural Networks, Computer; Predictive Value of Tests; Receptors, GABA-A; Structure-Activity Relationship

1995
Genetic neural networks for quantitative structure-activity relationships: improvements and application of benzodiazepine affinity for benzodiazepine/GABAA receptors.
    Journal of medicinal chemistry, 1996, Dec-20, Volume: 39, Issue:26

    Topics: Algorithms; Benzodiazepines; Models, Genetic; Nerve Net; Protein Binding; Receptors, GABA-A; Structure-Activity Relationship

1996