Page last updated: 2024-08-16

ro 41-1049 and lazabemide

ro 41-1049 has been researched along with lazabemide in 28 studies

Research

Studies (28)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's25 (89.29)18.2507
2000's3 (10.71)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Fernandes, MH; Pestana, M; Soares-da-Silva, P1
Da Prada, M; Richards, JG; Saura, J; Ulrich, J1
Da Prada, M; Kettler, R; Richards, JG; Saura, J1
Fernandes, MH; Soares-da-Silva, P2
Cesura, AM; Da Prada, M; Imhof, R; Lang, G; Muggli-Maniglio, D1
Da Prada, M; Kettler, R; Richards, JG; Saura Marti, J1
Borroni, E; Colzi, A; d'Agostini, F; Da Prada, M; Kettler, R1
Cesura, AM; Da Prada, M; Imhof, R; Keller, HH; Kettler, R; Kyburz, E; Muggli-Maniglio, D; Richards, JG; Saura Marti, J; Wyss, PC1
Cesura, AM; Chan-Palay, V; Da Prada, M; Huber, G; Löffler, J; Luque, JM; Richards, JG; Saura, J1
Pestana, M; Soares-da-Silva, P1
Fernandes, MH; Soares-da-Silva, P; Vieira-Coelho, MA1
García-Sevilla, JA; Miralles, A; Olmos, G; Ribas, C1
Bryan-Lluka, LJ; Westwood, NN1
García-Sevilla, JA; Sastre, M1
Abell, CW; Da Prada, M; Kwan, SW; Luque, JM; Richards, JG1
Bombi, JA; Mahy, N; Nadal, E; Saura, J; van den Berg, B; Vila, M1
Bleuel, Z; Chen, K; Da Prada, M; Malherbe, P; Mendelowitsch, A; Richards, JG; Saura, J; Shih, JC; Ulrich, J1
Boronat, MA; García-Sevilla, JA; Lizcano, JM; Olmos, G; Ozaita, A; Unzeta, M1
d'Agostini, F; Damsma, G; DaPrada, M; DeBoer, P; Heeringa, MJ1
Guimarães, JT; Soares-Da-Silva, P2
Gundlach, AL; Hosseini, AR; Iakovidis, D; Jackman, GP; King, PR; Louis, WJ; Nero, TL; Suzuki, S1
Gundlach, AL; Hosseini, AR; Jackman, GP; King, PR; Louis, WJ1
Gundlach, AL; King, PR; Louis, WJ1
Asensio, VJ; Esteban, S; García-Sevilla, JA; Miralles, A; Moranta, D; Sastre-Coll, A1
Anderson, NJ; Hudson, AL; Lupo, PA; Nutt, DJ; Robinson, ES1
Anderson, NJ; Hudson, AL; Nutt, DJ; Robinson, ES; Seif, I1

Reviews

1 review(s) available for ro 41-1049 and lazabemide

ArticleYear
From moclobemide to Ro 19-6327 and Ro 41-1049: the development of a new class of reversible, selective MAO-A and MAO-B inhibitors.
    Journal of neural transmission. Supplementum, 1990, Volume: 29

    Topics: Animals; Benzamides; Brain; Enzyme Inhibitors; Moclobemide; Monoamine Oxidase; Picolinic Acids; Rats; Thiazoles

1990

Other Studies

27 other study(ies) available for ro 41-1049 and lazabemide

ArticleYear
Deamination of newly-formed dopamine in rat renal tissues.
    British journal of pharmacology, 1991, Volume: 102, Issue:3

    Topics: 3,4-Dihydroxyphenylacetic Acid; Animals; Deamination; Dopamine; In Vitro Techniques; Kidney; Levodopa; Male; Pargyline; Picolinic Acids; Rats; Rats, Wistar; Thiazoles

1991
Molecular neuroanatomy of monoamine oxidases in human brainstem.
    Psychopharmacology, 1992, Volume: 106 Suppl

    Topics: Aged; Autoradiography; Brain Stem; Chromosome Mapping; Female; Humans; Male; Monoamine Oxidase; Monoamine Oxidase Inhibitors; Nucleic Acid Hybridization; Oligonucleotide Probes; Picolinic Acids; RNA, Messenger; Thiazoles

1992
Quantitative enzyme radioautography with 3H-Ro 41-1049 and 3H-Ro 19-6327 in vitro: localization and abundance of MAO-A and MAO-B in rat CNS, peripheral organs, and human brain.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 1992, Volume: 12, Issue:5

    Topics: Animals; Autoradiography; Binding Sites; Brain; Central Nervous System; Humans; Isoenzymes; Kinetics; Monoamine Oxidase; Monoamine Oxidase Inhibitors; Picolinic Acids; Rats; Thiazoles; Tissue Distribution; Tritium

1992
Role of monoamine oxidase A and B in the deamination of newly-formed dopamine in the rat kidney.
    Journal of neural transmission. Supplementum, 1990, Volume: 32

    Topics: 3,4-Dihydroxyphenylacetic Acid; Animals; Deamination; Dopamine; In Vitro Techniques; Kidney; Levodopa; Male; Monoamine Oxidase; Monoamine Oxidase Inhibitors; Picolinic Acids; Rats; Rats, Inbred Strains; Thiazoles

1990
Monoamine oxidase inhibition by moclobemide and 2-amino-ethyl carboxamide derivatives: mode of action and kinetic characteristics.
    Journal of neural transmission. Supplementum, 1990, Volume: 32

    Topics: Animals; Benzamides; Blood Platelets; Brain; Cell Membrane; Female; Humans; In Vitro Techniques; Kinetics; Moclobemide; Monoamine Oxidase; Monoamine Oxidase Inhibitors; Picolinic Acids; Placenta; Pregnancy; Rats; Thiazoles

1990
Molecular neuroanatomy of MAO-A and MAO-B.
    Journal of neural transmission. Supplementum, 1990, Volume: 32

    Topics: Animals; Autoradiography; Brain; Histocytochemistry; Humans; Monoamine Oxidase; Monoamine Oxidase Inhibitors; Nervous System; Nucleic Acid Hybridization; Picolinic Acids; Rats; Thiazoles

1990
Effect of selective and reversible MAO inhibitors on dopamine outflow in rat striatum: a microdialysis study.
    Journal of neural transmission. Supplementum, 1990, Volume: 32

    Topics: 3,4-Dihydroxyphenylacetic Acid; Animals; Benzamides; Corpus Striatum; Deamination; Dialysis; Dopamine; Homovanillic Acid; Male; Moclobemide; Monoamine Oxidase Inhibitors; Picolinic Acids; Rats; Rats, Inbred Strains; Thiazoles

1990
Effects of MAO-A and MAO-B selective inhibitors Ro 41-1049 and Ro 19-6327 on the deamination of newly formed dopamine in the rat kidney.
    The Journal of pharmacology and experimental therapeutics, 1990, Volume: 255, Issue:3

    Topics: 3,4-Dihydroxyphenylacetic Acid; Animals; Dihydroxyphenylalanine; Dopamine; Isoenzymes; Kidney; Kinetics; Male; Monoamine Oxidase Inhibitors; Norepinephrine; Picolinic Acids; Rats; Rats, Inbred Strains; Thiazoles

1990
Increased monoamine oxidase B activity in plaque-associated astrocytes of Alzheimer brains revealed by quantitative enzyme radioautography.
    Neuroscience, 1994, Volume: 62, Issue:1

    Topics: Aged; Aged, 80 and over; Alzheimer Disease; Astrocytes; Autoradiography; Brain; Female; Humans; Image Processing, Computer-Assisted; Immunohistochemistry; Isoquinolines; Male; Monoamine Oxidase; Monoamine Oxidase Inhibitors; Picolinic Acids; Thiazoles

1994
Effect of type A and B monoamine oxidase selective inhibition by Ro 41-1049 and Ro 19-6327 on dopamine outflow in rat kidney slices.
    British journal of pharmacology, 1994, Volume: 113, Issue:4

    Topics: 3,4-Dihydroxyphenylacetic Acid; Animals; Benserazide; Dopamine; In Vitro Techniques; Isoenzymes; Kidney Cortex; Levodopa; Male; Monoamine Oxidase; Monoamine Oxidase Inhibitors; Pargyline; Picolinic Acids; Rats; Rats, Wistar; Thiazoles

1994
In vivo effects of the monoamine oxidase inhibitors Ro 41-1049 and Ro 19-6327 on the production and fate of renal dopamine.
    Journal of neural transmission. Supplementum, 1994, Volume: 41

    Topics: 3,4-Dihydroxyphenylacetic Acid; Animals; Dopamine; Kidney; Levodopa; Male; Monoamine Oxidase Inhibitors; Picolinic Acids; Rats; Rats, Wistar; Thiazoles; Tissue Distribution

1994
Differential effects of the alkylating agent N-ethoxycarbonyl-2-ethoxy-1,2-dihydroquinoline on brain alpha 2-adrenoceptors and I2-imidazoline sites in vitro and in vivo.
    Journal of neurochemistry, 1993, Volume: 61, Issue:5

    Topics: Animals; Binding Sites; Brain; Cell Membrane; Dioxanes; Idazoxan; Imidazoles; Isoenzymes; Kinetics; Male; Monoamine Oxidase; Neurons; Picolinic Acids; Quinolines; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, alpha-2; Thermodynamics; Thiazoles; Tritium

1993
Types A and B monoamine oxidase contribute to the metabolism of norepinephrine in perfused lungs of rats.
    The Journal of pharmacology and experimental therapeutics, 1993, Volume: 267, Issue:2

    Topics: Animals; Deamination; Female; In Vitro Techniques; Isoenzymes; Kinetics; Lung; Male; Monoamine Oxidase; Monoamine Oxidase Inhibitors; Norepinephrine; Perfusion; Picolinic Acids; Rats; Rats, Wistar; Thiazoles; Vas Deferens

1993
Opposite age-dependent changes of alpha 2A-adrenoceptors and nonadrenoceptor [3H]idazoxan binding sites (I2-imidazoline sites) in the human brain: strong correlation of I2 with monoamine oxidase-B sites.
    Journal of neurochemistry, 1993, Volume: 61, Issue:3

    Topics: Adolescent; Adult; Aged; Aged, 80 and over; Aging; Binding Sites; Brain; Child; Child, Preschool; Dioxanes; Female; Humans; Idazoxan; Imidazoline Receptors; Male; Middle Aged; Monoamine Oxidase; Picolinic Acids; Receptors, Adrenergic, alpha; Receptors, Drug; Thiazoles

1993
Cellular expression of mRNAs encoding monoamine oxidases A and B in the rat central nervous system.
    The Journal of comparative neurology, 1995, Dec-25, Volume: 363, Issue:4

    Topics: Animals; Autoradiography; Biomarkers; Central Nervous System; Histamine; Immunohistochemistry; In Situ Hybridization; Isoenzymes; Male; Monoamine Oxidase; Monoamine Oxidase Inhibitors; Oligonucleotide Probes; Picolinic Acids; Rats; RNA, Messenger; Sulfur Radioisotopes; Thiazoles

1995
Localization of monoamine oxidases in human peripheral tissues.
    Life sciences, 1996, Volume: 59, Issue:16

    Topics: Aged; Aged, 80 and over; Autoradiography; Duodenum; Humans; Isoenzymes; Kidney; Liver; Lung; Monoamine Oxidase; Monoamine Oxidase Inhibitors; Myocardium; Picolinic Acids; Receptors, Adrenergic, beta; Spleen; Thiazoles

1996
Molecular neuroanatomy of human monoamine oxidases A and B revealed by quantitative enzyme radioautography and in situ hybridization histochemistry.
    Neuroscience, 1996, Volume: 70, Issue:3

    Topics: Aged; Aged, 80 and over; Autoradiography; Brain; Female; Histocytochemistry; Humans; In Situ Hybridization; Male; Middle Aged; Monoamine Oxidase; Monoamine Oxidase Inhibitors; Picolinic Acids; Thiazoles

1996
Inhibition of monoamine oxidase A and B activities by imidazol(ine)/guanidine drugs, nature of the interaction and distinction from I2-imidazoline receptors in rat liver.
    British journal of pharmacology, 1997, Volume: 121, Issue:5

    Topics: Animals; Clonidine; Guanidines; Imidazoles; Imidazoline Receptors; Isoenzymes; Kinetics; Liver; Male; Mitochondria, Liver; Monoamine Oxidase; Monoamine Oxidase Inhibitors; Picolinic Acids; Rats; Rats, Sprague-Dawley; Receptors, Drug; Thiazoles

1997
Effect of monoamine oxidase A and B and of catechol-O-methyltransferase inhibition on L-DOPA-induced circling behavior.
    Journal of neural transmission (Vienna, Austria : 1996), 1997, Volume: 104, Issue:6-7

    Topics: Animals; Antiparkinson Agents; Benzophenones; Catechol O-Methyltransferase Inhibitors; Enzyme Inhibitors; Levodopa; Male; Monoamine Oxidase Inhibitors; Motor Activity; Nitrophenols; Oxidopamine; Picolinic Acids; Rats; Rotation; Thiazoles; Tolcapone

1997
Unusual pattern of beta-phenylethylamine deamination in the rat heart.
    Biochemical Society transactions, 1997, Volume: 25, Issue:4

    Topics: Animals; Isoenzymes; Kidney Cortex; Kinetics; Male; Monoamine Oxidase; Monoamine Oxidase Inhibitors; Myocardium; Phenethylamines; Picolinic Acids; Psychotropic Drugs; Rats; Rats, Wistar; Serotonin; Substrate Specificity; Thiazoles

1997
The activity of MAO A and B in rat renal cells and tubules.
    Life sciences, 1998, Volume: 62, Issue:8

    Topics: 3,4-Dihydroxyphenylacetic Acid; Animals; Dopamine; Kidney; Kidney Tubules; Kinetics; Male; Monoamine Oxidase; Monoamine Oxidase Inhibitors; Picolinic Acids; Rats; Rats, Wistar; Thiazoles

1998
[3H]Rilmenidine-labelled imidazoline-receptor binding sites co-localize with [3H]2-(benzofuranyl)-2-imidazoline-labelled imidazoline-receptor binding sites and monoamine oxidase-B in rabbit, but not rat, kidney.
    Journal of the autonomic nervous system, 1998, Oct-15, Volume: 72, Issue:2-3

    Topics: Adrenergic alpha-Agonists; Animals; Autoradiography; Benzofurans; Imidazoles; Imidazoline Receptors; In Vitro Techniques; Isoenzymes; Kidney; Male; Monoamine Oxidase; Monoamine Oxidase Inhibitors; Oxazoles; Picolinic Acids; Rabbits; Rats; Rats, Inbred WKY; Receptors, Drug; Rilmenidine; Species Specificity; Thiazoles

1998
Pharmacology and subcellular distribution of [3H]rilmenidine binding sites in rat brain.
    Journal of the autonomic nervous system, 1998, Oct-15, Volume: 72, Issue:2-3

    Topics: Adrenergic alpha-Agonists; Animals; Binding Sites; Brain; Imidazoles; Imidazoline Receptors; In Vitro Techniques; Male; Membranes; Monoamine Oxidase; Monoamine Oxidase Inhibitors; Oxazoles; Picolinic Acids; Radioligand Assay; Rats; Rats, Inbred WKY; Receptors, Drug; Rilmenidine; Subcellular Fractions; Thiazoles

1998
Identification of imidazoline-receptor binding sites in cortex and medulla of the bovine adrenal gland. Colocalization with MAO-A and MAO-B.
    Annals of the New York Academy of Sciences, 1999, Jun-21, Volume: 881

    Topics: Adrenal Cortex; Adrenal Medulla; Adrenergic beta-Agonists; Animals; Autoradiography; Benzofurans; Binding Sites; Cattle; Clonidine; Imidazoles; Imidazoline Receptors; Isoenzymes; Monoamine Oxidase; Monoamine Oxidase Inhibitors; Oxazoles; Picolinic Acids; Rats; Receptors, Drug; Rilmenidine; Thiazoles; Tritium

1999
High-affinity binding of beta-carbolines to imidazoline I2B receptors and MAO-A in rat tissues: norharman blocks the effect of morphine withdrawal on DOPA/noradrenaline synthesis in the brain.
    European journal of pharmacology, 2005, Aug-22, Volume: 518, Issue:2-3

    Topics: Animals; Benzofurans; Binding, Competitive; Brain; Carbolines; Cerebral Cortex; Dihydroxyphenylalanine; Dose-Response Relationship, Drug; Harmine; Hippocampus; Imidazoles; Imidazoline Receptors; Liver; Male; Monoamine Oxidase; Morphine; Morphine Dependence; Naloxone; Norepinephrine; Picolinic Acids; Radioligand Assay; Rats; Rats, Sprague-Dawley; Receptors, Drug; Substance Withdrawal Syndrome; Thiazoles; Tritium; Tyrosine 3-Monooxygenase

2005
Characterisation of imidazoline I2 binding sites in pig brain.
    European journal of pharmacology, 2005, Sep-05, Volume: 519, Issue:1-2

    Topics: Animals; Benzofurans; Binding Sites; Binding, Competitive; Brain; Carbolines; Clonidine; Dose-Response Relationship, Drug; Female; Idazoxan; Imidazoles; Imidazoline Receptors; Kinetics; Male; Monoamine Oxidase Inhibitors; Picolinic Acids; Radioligand Assay; Receptors, Drug; Swine; Thiazoles; Tritium

2005
Autoradiographical distribution of imidazoline binding sites in monoamine oxidase A deficient mice.
    Journal of neurochemistry, 2006, Volume: 96, Issue:6

    Topics: Animals; Autoradiography; Benzofurans; Binding Sites; Binding, Competitive; Brain; Cell Membrane; Epithelial Cells; Harmine; Idazoxan; Imidazoles; Imidazoline Receptors; Imidazolines; Iodine Radioisotopes; Kidney; Mice; Mice, Inbred C3H; Mice, Knockout; Monoamine Oxidase; Neurons; Picolinic Acids; Radioligand Assay; Receptors, Drug; Thiazoles

2006