Page last updated: 2024-09-03

ro 32-0432 and rottlerin

ro 32-0432 has been researched along with rottlerin in 5 studies

Compound Research Comparison

Studies
(ro 32-0432)
Trials
(ro 32-0432)
Recent Studies (post-2010)
(ro 32-0432)
Studies
(rottlerin)
Trials
(rottlerin)
Recent Studies (post-2010) (rottlerin)
560135561202

Protein Interaction Comparison

ProteinTaxonomyro 32-0432 (IC50)rottlerin (IC50)
Eukaryotic elongation factor 2 kinaseHomo sapiens (human)5.3
B2 bradykinin receptorCavia porcellus (domestic guinea pig)1.2
Ubiquitin carboxyl-terminal hydrolase 1Homo sapiens (human)8
Beta-lactamaseEscherichia coli K-121.5
Malate dehydrogenaseThermus thermophilus0.7
5-hydroxytryptamine receptor 1ARattus norvegicus (Norway rat)1.2
MAP kinase-activated protein kinase 2Homo sapiens (human)5.4
Protein kinase C delta typeHomo sapiens (human)3
MAP kinase-activated protein kinase 5Homo sapiens (human)1.9
WD repeat-containing protein 48Homo sapiens (human)8
RuvB-like 1Homo sapiens (human)10

Research

Studies (5)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's4 (80.00)29.6817
2010's1 (20.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Akao, Y; Iinuma, M; Itoh, T; Nozawa, Y; Ohguchi, K1
Curtis, JL; Hu, B; Polak, T; Punturieri, A; Sonstein, J; Todt, JC1
Fresco, P; Gonçalves, J; Pinto, E; Saraiva, L1
Brown, Z; Cronshaw, DG; Kouroumalis, A; Parry, R; Ward, SG; Webb, A1
Liu, W; Liu, XC; Liu, ZC; Tang, SB; Yu, EH; Zhu, BH1

Other Studies

5 other study(ies) available for ro 32-0432 and rottlerin

ArticleYear
Inhibitory effect of xanthones isolated from the pericarp of Garcinia mangostana L. on rat basophilic leukemia RBL-2H3 cell degranulation.
    Bioorganic & medicinal chemistry, 2008, Apr-15, Volume: 16, Issue:8

    Topics: Animals; Calcium; Cell Degranulation; Cell Line, Tumor; Enzyme Activation; Extracellular Signal-Regulated MAP Kinases; Garcinia mangostana; Histamine; Immunoglobulin E; Intracellular Signaling Peptides and Proteins; Leukemia, Basophilic, Acute; MAP Kinase Signaling System; Molecular Structure; Phosphatidylinositol 3-Kinases; Phospholipase C gamma; Protein-Tyrosine Kinases; Rats; Reactive Oxygen Species; Receptors, IgE; Structure-Activity Relationship; Syk Kinase; Xanthones

2008
Activation of protein kinase C beta II by the stereo-specific phosphatidylserine receptor is required for phagocytosis of apoptotic thymocytes by resident murine tissue macrophages.
    The Journal of biological chemistry, 2002, Sep-27, Volume: 277, Issue:39

    Topics: Acetophenones; Animals; Apoptosis; Benzopyrans; Blotting, Western; Cell Adhesion; Dose-Response Relationship, Drug; Enzyme Activation; Female; Flow Cytometry; Immunoblotting; Indoles; Inhibitory Concentration 50; Isoenzymes; Liposomes; Macrophages; Mice; Mice, Inbred C57BL; Myristic Acid; Phagocytosis; Protein Isoforms; Protein Kinase C; Protein Kinase C beta; Protein Transport; Pyrroles; Receptors, Cell Surface; Reverse Transcriptase Polymerase Chain Reaction; RNA; Tetradecanoylphorbol Acetate; Thymus Gland; Time Factors

2002
Isoform-selectivity of PKC inhibitors acting at the regulatory and catalytic domain of mammalian PKC-alpha, -betaI, -delta, -eta and -zeta.
    Journal of enzyme inhibition and medicinal chemistry, 2003, Volume: 18, Issue:6

    Topics: Acetophenones; Alkaloids; Animals; Benzophenanthridines; Benzopyrans; Catalysis; Enzyme Inhibitors; Escherichia coli; Indoles; Isoenzymes; Phenanthridines; Piperidines; Protein Kinase C; Protein Kinase C beta; Protein Kinase C-alpha; Protein Kinase C-delta; Pyrroles; Saccharomyces cerevisiae; Sphingosine; Tamoxifen; Yeasts

2003
Evidence that phospholipase-C-dependent, calcium-independent mechanisms are required for directional migration of T-lymphocytes in response to the CCR4 ligands CCL17 and CCL22.
    Journal of leukocyte biology, 2006, Volume: 79, Issue:6

    Topics: Acetophenones; Benzopyrans; Calcium; Calcium Channels; Calcium Signaling; Catalytic Domain; Cell Line, Tumor; Chemokine CCL17; Chemokine CCL22; Chemokines, CC; Chemotaxis; Chromones; Diglycerides; Estrenes; Humans; Indoles; Inositol 1,4,5-Trisphosphate; Inositol 1,4,5-Trisphosphate Receptors; Leukemia-Lymphoma, Adult T-Cell; Morpholines; Pertussis Toxin; Phosphatidylinositol 3-Kinases; Phosphatidylinositol Diacylglycerol-Lyase; Phosphoinositide-3 Kinase Inhibitors; Phosphorylation; Phosphothreonine; Protein Processing, Post-Translational; Pyrroles; Pyrrolidinones; Receptors, CCR4; Receptors, Chemokine; Receptors, Cytoplasmic and Nuclear; Recombinant Fusion Proteins; T-Lymphocytes; Th2 Cells

2006
Translocation of protein kinase C δ contributes to the moderately high glucose-, but not hypoxia-induced proliferation in primary cultured human retinal endothelial cells.
    Molecular medicine reports, 2014, Volume: 9, Issue:5

    Topics: Acetophenones; Benzopyrans; Cell Proliferation; Cells, Cultured; Endothelial Cells; Gene Expression; Glucose; Humans; Hypoxia; Indoles; Primary Cell Culture; Protein Kinase C-delta; Protein Transport; Pyrroles; Retinal Pigment Epithelium

2014