ro 31-7549 and staurosporine

ro 31-7549 has been researched along with staurosporine in 13 studies

Research

Studies (13)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's10 (76.92)18.2507
2000's3 (23.08)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Bit, RA; Davis, PD; Elliott, LH; Harris, W; Hill, CH; Keech, E; Kumar, H; Lawton, G; Maw, A; Nixon, JS1
Bullock, AN; Debreczeni, JE; Fedorov, OY; Knapp, S; Marsden, BD; Nelson, A1
Bergstrand, H; Karabelas, K; Lundquist, B; Michelsen, P1
Gilfillan, AM; Lin, P1
Beaven, MA; Jelsema, CL; Yamada, K1
Carew, MA; Paleolog, EM; Pearson, JD1
Dieter, P; Fitzke, E1
Corvaia, N; Coutant, KD; Ryder, NS1
Deisher, TA; Harlan, JM; Pohlman, TH; Sato, TT1
Nixon, JS; Parker, PJ; Wilkinson, SE1
Chock, PB; Huang, CY; Tekle, E; Zhu, DM1
Edvinsson, L; Hansen-Schwartz, J; Svensson, CL; Xu, CB1
Bork, S; Das, S; Igarashi, I; Okubo, K; Yokoyama, N1

Other Studies

13 other study(ies) available for ro 31-7549 and staurosporine

ArticleYear
Inhibitors of protein kinase C. 3. Potent and highly selective bisindolylmaleimides by conformational restriction.
    Journal of medicinal chemistry, 1993, Jan-08, Volume: 36, Issue:1

    Topics: Alkaloids; Animals; Humans; Maleimides; Mice; Models, Molecular; Molecular Conformation; Protein Kinase C; Rabbits; Rats; Staurosporine; Stereoisomerism; Structure-Activity Relationship

1993
Structural basis of inhibitor specificity of the human protooncogene proviral insertion site in moloney murine leukemia virus (PIM-1) kinase.
    Journal of medicinal chemistry, 2005, Dec-01, Volume: 48, Issue:24

    Topics: Antineoplastic Agents; Crystallization; Crystallography, X-Ray; Flavonoids; Humans; Imidazoles; Indoles; Maleimides; Models, Molecular; Molecular Structure; Moloney murine leukemia virus; Phosphorylation; Protein Binding; Proto-Oncogene Proteins c-pim-1; Proviruses; Pyrazoles; Pyridazines; Pyrimidines; Structure-Activity Relationship

2005
Modulation of human basophil histamine release by protein kinase C inhibitors differs with secretagogue and with inhibitor.
    The Journal of pharmacology and experimental therapeutics, 1992, Volume: 260, Issue:3

    Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Alkaloids; Basophils; Calcimycin; Glyceryl Ethers; Histamine Release; Humans; Indoles; Isoquinolines; Maleimides; Mannitol; Palmitoylcarnitine; Piperazines; Polymyxin B; Protein Kinase C; Sphingosine; Staurosporine; Sulfonamides; Tetradecanoylphorbol Acetate

1992
The role of calcium and protein kinase C in the IgE-dependent activation of phosphatidylcholine-specific phospholipase D in a rat mast (RBL 2H3) cell line.
    European journal of biochemistry, 1992, Jul-01, Volume: 207, Issue:1

    Topics: Alkaloids; Animals; Calcium; Cell Line; Enzyme Activation; Histamine Release; Immunoglobulin E; Indoles; Ionomycin; Kinetics; Maleimides; Mast Cells; Phospholipase D; Protein Kinase C; Rats; Staurosporine; Terpenes; Tetradecanoylphorbol Acetate; Thapsigargin

1992
Certain inhibitors of protein serine/threonine kinases also inhibit tyrosine phosphorylation of phospholipase C gamma 1 and other proteins and reveal distinct roles for tyrosine kinase(s) and protein kinase C in stimulated, rat basophilic RBL-2H3 cells.
    Journal of immunology (Baltimore, Md. : 1950), 1992, Aug-01, Volume: 149, Issue:3

    Topics: Alkaloids; Androstadienes; Angiotensin I; Animals; Antigens; Arachidonic Acid; Basophils; Calcimycin; Carbazoles; Exocytosis; In Vitro Techniques; Indoles; Inositol Phosphates; Leukemia, Experimental; Maleimides; Phosphorylation; Phosphotyrosine; Protein Kinase C; Protein Kinase Inhibitors; Protein Serine-Threonine Kinases; Protein-Tyrosine Kinases; Rats; Serotonin; Staurosporine; Tumor Cells, Cultured; Type C Phospholipases; Tyrosine; Wortmannin

1992
The roles of protein kinase C and intracellular Ca2+ in the secretion of von Willebrand factor from human vascular endothelial cells.
    The Biochemical journal, 1992, Sep-01, Volume: 286 ( Pt 2)

    Topics: Adenosine Triphosphate; Alkaloids; Calcimycin; Calcium; Cations, Divalent; Cells, Cultured; Endothelium, Vascular; Enzyme Activation; Humans; Indoles; Maleimides; Protein Kinase C; Signal Transduction; Staurosporine; Tetradecanoylphorbol Acetate; von Willebrand Factor

1992
RO 31-8220 and RO 31-7549 show improved selectivity for protein kinase C over staurosporine in macrophages.
    Biochemical and biophysical research communications, 1991, Nov-27, Volume: 181, Issue:1

    Topics: Alkaloids; Animals; Cells, Cultured; Dinoprostone; Indoles; Kinetics; Macrophages; Maleimides; Protein Kinase C; Staurosporine; Tetradecanoylphorbol Acetate

1991
Bradykinin induces tyrosine phosphorylation of epidermal growth factor-receptor and focal adhesion proteins in human keratinocytes.
    Biochemical and biophysical research communications, 1995, May-25, Volume: 210, Issue:3

    Topics: Alkaloids; Bradykinin; Cell Adhesion Molecules; Cell Line; Chromatography, Affinity; Cytoskeletal Proteins; Electrophoresis, Polyacrylamide Gel; ErbB Receptors; Focal Adhesion Kinase 1; Focal Adhesion Protein-Tyrosine Kinases; Genistein; Humans; Immunoblotting; Indoles; Isoflavones; Keratinocytes; Maleimides; Molecular Weight; Paxillin; Phosphoproteins; Phosphotyrosine; Protein Kinase C; Protein-Tyrosine Kinases; Receptor, Insulin; Receptors, Bradykinin; Staurosporine; Tyrosine

1995
A protein kinase C agonist, selective for the beta I isozyme, induces E-selectin and VCAM-1 expression on HUVEC but does not translocate PKC.
    Biochemical and biophysical research communications, 1993, Jun-30, Volume: 193, Issue:3

    Topics: Alkaloids; Base Sequence; Cell Adhesion Molecules; Cell Membrane; Cells, Cultured; Cytosol; E-Selectin; Endothelium, Vascular; Humans; Indoles; Isoenzymes; Kinetics; Maleimides; Membrane Glycoproteins; Molecular Sequence Data; NF-kappa B; Oligonucleotide Probes; Phorbol Esters; Promoter Regions, Genetic; Protein Kinase C; Staurosporine; Tetradecanoylphorbol Acetate; Tumor Necrosis Factor-alpha; Umbilical Veins; Vascular Cell Adhesion Molecule-1

1993
Isoenzyme specificity of bisindolylmaleimides, selective inhibitors of protein kinase C.
    The Biochemical journal, 1993, Sep-01, Volume: 294 ( Pt 2)

    Topics: Adenosine Triphosphate; Alkaloids; Animals; Binding Sites; Binding, Competitive; Brain; Indoles; Isoenzymes; Maleimides; Molecular Conformation; Protein Kinase C; Rats; Staurosporine; Structure-Activity Relationship

1993
Reversible phosphorylation as a controlling factor for sustaining calcium oscillations in HeLa cells: Involvement of calmodulin-dependent kinase II and a calyculin A-inhibitable phosphatase.
    Biochemistry, 1996, Jun-04, Volume: 35, Issue:22

    Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Alkaloids; Amino Acid Sequence; Binding Sites; Calcium; Calcium Channels; Calcium-Calmodulin-Dependent Protein Kinase Type 2; Calcium-Calmodulin-Dependent Protein Kinases; Calcium-Transporting ATPases; Enzyme Inhibitors; Ethers, Cyclic; HeLa Cells; Histamine; Humans; Indoles; Inositol 1,4,5-Trisphosphate; Inositol 1,4,5-Trisphosphate Receptors; Isoquinolines; Maleimides; Marine Toxins; Molecular Sequence Data; Okadaic Acid; Oxazoles; Phosphoprotein Phosphatases; Phosphorylation; Piperazines; Protein Kinase C; Receptors, Cytoplasmic and Nuclear; Ryanodine; Spectrometry, Fluorescence; Staurosporine; Sulfonamides

1996
Protein kinase mediated upregulation of endothelin A, endothelin B and 5-hydroxytryptamine 1B/1D receptors during organ culture in rat basilar artery.
    British journal of pharmacology, 2002, Volume: 137, Issue:1

    Topics: Animals; Basilar Artery; Cyclic AMP-Dependent Protein Kinases; Indoles; Isoquinolines; Male; Maleimides; Muscle Contraction; Muscle, Smooth, Vascular; Organ Culture Techniques; Protein Kinase C; Rats; Rats, Inbred WKY; Receptor, Endothelin A; Receptor, Endothelin B; Receptor, Serotonin, 5-HT1B; Receptor, Serotonin, 5-HT1D; Receptors, Endothelin; Receptors, Serotonin; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Staurosporine; Sulfonamides; Up-Regulation

2002
Effects of protein kinase inhibitors on the in vitro growth of Babesia bovis.
    Parasitology, 2006, Volume: 132, Issue:Pt 6

    Topics: Animals; Babesia bovis; Benzylamines; Cattle; Cells, Cultured; Enzyme Inhibitors; Erythrocytes; Indoles; Maleimides; Protein Kinase Inhibitors; Staurosporine; Sulfonamides; Time Factors

2006