Page last updated: 2024-09-03

ro 22-1319 and metoclopramide

ro 22-1319 has been researched along with metoclopramide in 2 studies

Compound Research Comparison

Studies
(ro 22-1319)
Trials
(ro 22-1319)
Recent Studies (post-2010)
(ro 22-1319)
Studies
(metoclopramide)
Trials
(metoclopramide)
Recent Studies (post-2010) (metoclopramide)
23305,0441,216623

Protein Interaction Comparison

ProteinTaxonomyro 22-1319 (IC50)metoclopramide (IC50)
5-hydroxytryptamine receptor 4Cavia porcellus (domestic guinea pig)2.383
MyeloperoxidaseHomo sapiens (human)0.35
Alpha-2A adrenergic receptorHomo sapiens (human)2.721
Cytochrome P450 2D6Homo sapiens (human)0.8
D(2) dopamine receptorHomo sapiens (human)0.127
Alpha-1B adrenergic receptorRattus norvegicus (Norway rat)7.8
5-hydroxytryptamine receptor 1ARattus norvegicus (Norway rat)7.8
Alpha-2B adrenergic receptorRattus norvegicus (Norway rat)7.7
Alpha-2C adrenergic receptorRattus norvegicus (Norway rat)7.7
Alpha-2A adrenergic receptorRattus norvegicus (Norway rat)7.7
Alpha-1D adrenergic receptorRattus norvegicus (Norway rat)7.8
5-hydroxytryptamine receptor 2AHomo sapiens (human)3.675
5-hydroxytryptamine receptor 2CHomo sapiens (human)2.383
5-hydroxytryptamine receptor 1BRattus norvegicus (Norway rat)7.8
5-hydroxytryptamine receptor 1DRattus norvegicus (Norway rat)7.8
5-hydroxytryptamine receptor 1FRattus norvegicus (Norway rat)7.8
D(3) dopamine receptorHomo sapiens (human)0.2
5-hydroxytryptamine receptor 3ARattus norvegicus (Norway rat)0.88
5-hydroxytryptamine receptor 2BHomo sapiens (human)0.63
Alpha-1A adrenergic receptorRattus norvegicus (Norway rat)7.8
D(2) dopamine receptorRattus norvegicus (Norway rat)0.6237
5-hydroxytryptamine receptor 3BRattus norvegicus (Norway rat)0.88

Research

Studies (2)

TimeframeStudies, this research(%)All Research%
pre-19902 (100.00)18.7374
1990's0 (0.00)18.2507
2000's0 (0.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Collin, S; Durant, F; Evrard, G; Vanderveken, D; Vercauteren, DP1
Molloy, AG; O'Boyle, KM; Pugh, MT; Waddington, JL1

Other Studies

2 other study(ies) available for ro 22-1319 and metoclopramide

ArticleYear
Structural requirements of Na+-dependent antidopaminergic agents: Tropapride, Piquindone, Zetidoline, and Metoclopramide. Comparison with Na+-independent ligands.
    Journal of computer-aided molecular design, 1989, Volume: 3, Issue:1

    Topics: Computer Graphics; Dopamine Antagonists; Imidazoles; Isoquinolines; Metoclopramide; Models, Molecular; Motion; Nortropanes; Receptors, Dopamine; Sodium; Structure-Activity Relationship

1989
Locomotor behaviors in response to new selective D-1 and D-2 dopamine receptor agonists, and the influence of selective antagonists.
    Pharmacology, biochemistry, and behavior, 1986, Volume: 25, Issue:1

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Benzazepines; Flupenthixol; Isoquinolines; Male; Metoclopramide; Motor Activity; Phenethylamines; Rats; Rats, Inbred Strains; Receptors, Dopamine; Stimulation, Chemical

1986