ro 15-4513 has been researched along with ro 15-3505 in 7 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 0 (0.00) | 18.7374 |
1990's | 5 (71.43) | 18.2507 |
2000's | 2 (28.57) | 29.6817 |
2010's | 0 (0.00) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
---|---|
Cook, JM; Harris, B; Liu, R; Skolnick, P; Zhang, P; Zhang, W | 1 |
Ananthan, S; Clayton, SD; Ealick, SE; Evoniuk, GE; Skolnick, P; Wong, G | 1 |
de Costa, BR; Dominguez, C; Gu, ZQ; Rice, KC; Skolnick, P; Wong, G | 1 |
Ananthan, S; Cook, JM; Gu, ZQ; Hunkeler, W; Koehler, KF; Schönholzer, P; Skolnick, P; Wong, G; Zhang, W | 1 |
Bennett, DW; Cook, JM; Gan, T; He, X; Huang, Q; Liu, R; McKernan, R; Zhang, P | 1 |
Cook, JM; Dayer, CA; He, X; Huang, Q; Liu, R; Ma, C; McKernan, R; Wenger, GR; Yu, S | 1 |
Clayton, T; Cook, J; DeLorey, TM; Furtmüller, R; Halliwell, RF; Harris, D; Huck, S; Sahbaie, P; Sieghart, W | 1 |
7 other study(ies) available for ro 15-4513 and ro 15-3505
Article | Year |
---|---|
Synthesis of novel imidazobenzodiazepines as probes of the pharmacophore for "diazepam-insensitive" GABAA receptors.
Topics: Affinity Labels; Animals; Azides; Benzodiazepines; Diazepam; Male; Molecular Probes; Radioligand Assay; Rats; Rats, Sprague-Dawley; Receptors, GABA-A; Structure-Activity Relationship | 1995 |
Synthesis and structure-activity relationships of 3,5-disubstituted 4,5-dihydro-6H-imidazo[1,5-a][1,4]benzodiazepin-6-ones at diazepam-sensitive and diazepam-insensitive benzodiazepine receptors.
Topics: Animals; Benzodiazepinones; Binding Sites; Cell Membrane; Cerebellum; Cerebral Cortex; Crystallization; Diazepam; Male; Mice; Models, Molecular; Molecular Structure; Receptors, GABA-A; Structure-Activity Relationship; X-Ray Diffraction | 1993 |
Synthesis and evaluation of imidazo[1,5-a][1,4]benzodiazepine esters with high affinities and selectivities at "diazepam-insensitive" benzodiazepine receptors.
Topics: Animals; Benzodiazepines; Binding Sites; Brain; Esters; Imidazoles; Male; Rats; Rats, Sprague-Dawley; Receptors, GABA-A | 1993 |
Synthetic and computer-assisted analysis of the structural requirements for selective, high-affinity ligand binding to diazepam-insensitive benzodiazepine receptors.
Topics: Animals; Azepines; Benzodiazepines; Cerebellum; Computer Simulation; Diazepam; In Vitro Techniques; Ligands; Male; Models, Molecular; Molecular Conformation; Rats; Rats, Sprague-Dawley; Receptors, GABA-A; Structure-Activity Relationship; X-Ray Diffraction | 1993 |
Predictive models for GABAA/benzodiazepine receptor subtypes: studies of quantitative structure-activity relationships for imidazobenzodiazepines at five recombinant GABAA/benzodiazepine receptor subtypes [alphaxbeta3gamma2 (x = 1-3, 5, and 6)] via compar
Topics: Animals; Benzodiazepines; Cell Line; Crystallography, X-Ray; Humans; Ligands; Mice; Models, Molecular; Radioligand Assay; Receptors, GABA-A; Recombinant Proteins; Regression Analysis; Structure-Activity Relationship | 1998 |
Pharmacophore/receptor models for GABA(A)/BzR subtypes (alpha1beta3gamma2, alpha5beta3gamma2, and alpha6beta3gamma2) via a comprehensive ligand-mapping approach.
Topics: Animals; Benzodiazepines; Carbolines; Cell Line; Columbidae; Conditioning, Operant; Crystallography, X-Ray; Humans; Indoles; Ligands; Male; Models, Molecular; Pyrimidines; Quinolones; Radioligand Assay; Receptors, GABA-A; Saimiri; Stereoisomerism; Structure-Activity Relationship | 2000 |
Selective influence on contextual memory: physiochemical properties associated with selectivity of benzodiazepine ligands at GABAA receptors containing the alpha5 subunit.
Topics: Animals; Behavior, Animal; Benzodiazepines; Chemical Phenomena; Chemistry, Physical; Computer Simulation; Databases, Factual; Electrophysiology; Female; Ligands; Male; Memory; Mice; Models, Molecular; Molecular Structure; Oocytes; Protein Isoforms; Protein Subunits; Quantitative Structure-Activity Relationship; Receptors, GABA-A; Structure-Activity Relationship; Xenopus laevis | 2008 |