Page last updated: 2024-08-16

ro 15-4513 and ro 14-7437

ro 15-4513 has been researched along with ro 14-7437 in 7 studies

Research

Studies (7)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's6 (85.71)18.2507
2000's1 (14.29)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Cook, JM; Harris, B; Liu, R; Skolnick, P; Zhang, P; Zhang, W1
Ananthan, S; Clayton, SD; Ealick, SE; Evoniuk, GE; Skolnick, P; Wong, G1
de Costa, BR; Dominguez, C; Gu, ZQ; Rice, KC; Skolnick, P; Wong, G1
Ananthan, S; Cook, JM; Gu, ZQ; Hunkeler, W; Koehler, KF; Schönholzer, P; Skolnick, P; Wong, G; Zhang, W1
Cook, JM; Dayer, CA; He, X; Huang, Q; Liu, R; Ma, C; McKernan, R; Wenger, GR; Yu, S1
Gu, ZQ; Harris, BD; Moody, EJ; Skolnick, P1
Ferenci, P; Herneth, A; Püspök, A; Steindl, P1

Other Studies

7 other study(ies) available for ro 15-4513 and ro 14-7437

ArticleYear
Synthesis of novel imidazobenzodiazepines as probes of the pharmacophore for "diazepam-insensitive" GABAA receptors.
    Journal of medicinal chemistry, 1995, May-12, Volume: 38, Issue:10

    Topics: Affinity Labels; Animals; Azides; Benzodiazepines; Diazepam; Male; Molecular Probes; Radioligand Assay; Rats; Rats, Sprague-Dawley; Receptors, GABA-A; Structure-Activity Relationship

1995
Synthesis and structure-activity relationships of 3,5-disubstituted 4,5-dihydro-6H-imidazo[1,5-a][1,4]benzodiazepin-6-ones at diazepam-sensitive and diazepam-insensitive benzodiazepine receptors.
    Journal of medicinal chemistry, 1993, Feb-19, Volume: 36, Issue:4

    Topics: Animals; Benzodiazepinones; Binding Sites; Cell Membrane; Cerebellum; Cerebral Cortex; Crystallization; Diazepam; Male; Mice; Models, Molecular; Molecular Structure; Receptors, GABA-A; Structure-Activity Relationship; X-Ray Diffraction

1993
Synthesis and evaluation of imidazo[1,5-a][1,4]benzodiazepine esters with high affinities and selectivities at "diazepam-insensitive" benzodiazepine receptors.
    Journal of medicinal chemistry, 1993, Apr-16, Volume: 36, Issue:8

    Topics: Animals; Benzodiazepines; Binding Sites; Brain; Esters; Imidazoles; Male; Rats; Rats, Sprague-Dawley; Receptors, GABA-A

1993
Synthetic and computer-assisted analysis of the structural requirements for selective, high-affinity ligand binding to diazepam-insensitive benzodiazepine receptors.
    Journal of medicinal chemistry, 1993, Jun-25, Volume: 36, Issue:13

    Topics: Animals; Azepines; Benzodiazepines; Cerebellum; Computer Simulation; Diazepam; In Vitro Techniques; Ligands; Male; Models, Molecular; Molecular Conformation; Rats; Rats, Sprague-Dawley; Receptors, GABA-A; Structure-Activity Relationship; X-Ray Diffraction

1993
Pharmacophore/receptor models for GABA(A)/BzR subtypes (alpha1beta3gamma2, alpha5beta3gamma2, and alpha6beta3gamma2) via a comprehensive ligand-mapping approach.
    Journal of medicinal chemistry, 2000, Jan-13, Volume: 43, Issue:1

    Topics: Animals; Benzodiazepines; Carbolines; Cell Line; Columbidae; Conditioning, Operant; Crystallography, X-Ray; Humans; Indoles; Ligands; Male; Models, Molecular; Pyrimidines; Quinolones; Radioligand Assay; Receptors, GABA-A; Saimiri; Stereoisomerism; Structure-Activity Relationship

2000
Contribution of "diazepam-insensitive" GABAA receptors to the alcohol antagonist properties of Ro 15-4513 and related imidazobenzodiazepines.
    Pharmacology, biochemistry, and behavior, 1995, Volume: 52, Issue:1

    Topics: Alcohol Deterrents; Animals; Azides; Behavior, Animal; Benzodiazepines; Carbolines; Cerebellum; Diazepam; Dose-Response Relationship, Drug; GABA Antagonists; GABA Modulators; GABA-A Receptor Antagonists; Male; Mice; Mice, Inbred Strains

1995
Hepatic encephalopathy in rats with thioacetamide-induced acute liver failure is not mediated by endogenous benzodiazepines.
    Gastroenterology, 1993, Volume: 105, Issue:3

    Topics: Animals; Azides; Benzodiazepines; Carbolines; Convulsants; Flunitrazepam; Hepatic Encephalopathy; Liver Failure, Acute; Male; Rats; Rats, Sprague-Dawley; Thioacetamide

1993