Page last updated: 2024-09-04

ro 03-7410 and quinidine

ro 03-7410 has been researched along with quinidine in 1 studies

Compound Research Comparison

Studies
(ro 03-7410)
Trials
(ro 03-7410)
Recent Studies (post-2010)
(ro 03-7410)
Studies
(quinidine)
Trials
(quinidine)
Recent Studies (post-2010) (quinidine)
5116,608387594

Protein Interaction Comparison

ProteinTaxonomyro 03-7410 (IC50)quinidine (IC50)
Voltage-dependent L-type calcium channel subunit alpha-1FHomo sapiens (human)6.4
CholinesteraseHomo sapiens (human)1.23
ATP-dependent translocase ABCB1Mus musculus (house mouse)10
ATP-dependent translocase ABCB1Homo sapiens (human)3.32
Cytochrome P450 2D26Rattus norvegicus (Norway rat)2.8
Cytochrome P450 2D6Homo sapiens (human)0.3532
Potassium voltage-gated channel subfamily A member 5Homo sapiens (human)7.3
CholinesteraseEquus caballus (horse)7.37
Voltage-dependent L-type calcium channel subunit alpha-1D Homo sapiens (human)6.4
Potassium voltage-gated channel subfamily H member 2Homo sapiens (human)0.7882
Voltage-dependent L-type calcium channel subunit alpha-1SHomo sapiens (human)6.4
Voltage-dependent L-type calcium channel subunit alpha-1CHomo sapiens (human)6.4
Sodium channel protein type 5 subunit alphaHomo sapiens (human)6.9
Potassium voltage-gated channel subfamily D member 2Rattus norvegicus (Norway rat)2.2

Research

Studies (1)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's1 (100.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Margolis, JM; Obach, RS1

Other Studies

1 other study(ies) available for ro 03-7410 and quinidine

ArticleYear
Impact of nonspecific binding to microsomes and phospholipid on the inhibition of cytochrome P4502D6: implications for relating in vitro inhibition data to in vivo drug interactions.
    Drug metabolism and disposition: the biological fate of chemicals, 2003, Volume: 31, Issue:5

    Topics: Benzylamines; Bridged Bicyclo Compounds, Heterocyclic; Cytochrome P-450 CYP2D6; Cytochrome P-450 CYP2D6 Inhibitors; Drug Interactions; Enzyme Inhibitors; Ethanolamines; Fluoxetine; Humans; Imipramine; In Vitro Techniques; Microsomes; Phospholipids; Protein Binding; Quinidine

2003