Page last updated: 2024-09-03

rmi 12330a and nifedipine

rmi 12330a has been researched along with nifedipine in 6 studies

Compound Research Comparison

Studies
(rmi 12330a)
Trials
(rmi 12330a)
Recent Studies (post-2010)
(rmi 12330a)
Studies
(nifedipine)
Trials
(nifedipine)
Recent Studies (post-2010) (nifedipine)
14102416,0242,4961,505

Protein Interaction Comparison

ProteinTaxonomyrmi 12330a (IC50)nifedipine (IC50)
perilipin-5Homo sapiens (human)7.133
perilipin-1Homo sapiens (human)9.619
1-acylglycerol-3-phosphate O-acyltransferase ABHD5 isoform aHomo sapiens (human)8.376
Voltage-dependent L-type calcium channel subunit alpha-1CCavia porcellus (domestic guinea pig)0.0429
Voltage-dependent L-type calcium channel subunit alpha-1FHomo sapiens (human)0.035
Cytochrome P450 1A2Homo sapiens (human)0.3
Cytochrome P450 3A4Homo sapiens (human)10
Adenosine receptor A3Homo sapiens (human)7.214
Cytochrome P450 2C9 Homo sapiens (human)3.06
5-hydroxytryptamine receptor 2ARattus norvegicus (Norway rat)10
Alpha-1B adrenergic receptorRattus norvegicus (Norway rat)7.214
Voltage-dependent L-type calcium channel subunit alpha-1CRattus norvegicus (Norway rat)0.0385
Potassium voltage-gated channel subfamily A member 5Homo sapiens (human)6.1
3-oxo-5-alpha-steroid 4-dehydrogenase 1 Rattus norvegicus (Norway rat)1.12
Adenosine receptor A1Homo sapiens (human)7.701
3-oxo-5-alpha-steroid 4-dehydrogenase 2Rattus norvegicus (Norway rat)1.12
C-C chemokine receptor type 2Homo sapiens (human)2.191
Alpha-1A adrenergic receptorRattus norvegicus (Norway rat)7.214
Cytochrome P450 2J2Homo sapiens (human)3.06
Voltage-dependent L-type calcium channel subunit alpha-1D Homo sapiens (human)0.4733
Voltage-dependent L-type calcium channel subunit alpha-1CMus musculus (house mouse)1.2
Voltage-dependent L-type calcium channel subunit alpha-1SMus musculus (house mouse)1.2
Voltage-dependent L-type calcium channel subunit alpha-1SHomo sapiens (human)0.035
Voltage-dependent L-type calcium channel subunit alpha-1CHomo sapiens (human)0.0394
Myosin light chain kinase, smooth muscleHomo sapiens (human)2.02
Potassium channel subfamily K member 2 Bos taurus (cattle)8.2
Indoleamine 2,3-dioxygenase 2Mus musculus (house mouse)1.5
Voltage-dependent L-type calcium channel subunit alpha-1DMus musculus (house mouse)1.2
Voltage-dependent L-type calcium channel subunit alpha-1FMus musculus (house mouse)1.2

Research

Studies (6)

TimeframeStudies, this research(%)All Research%
pre-19901 (16.67)18.7374
1990's0 (0.00)18.2507
2000's3 (50.00)29.6817
2010's2 (33.33)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Jaros, JA; Lee, HR; Roeske, WR; Ursillo, R; Wiech, NL; Yamamura, HI1
Fukushima, Y; Hikichi, H; Hisa, H; Kawashima, H; Kimura, T; Nagayama, T; Satoh, S; Suzuki-Kusaba, M; Yoshida, M1
Chu, MM; Lee, EK; Lin, HR; Wong, AO; Xiao, D1
Aguilar, R; Bellido, C; Garrido-Gracia, JC; Sánchez-Criado, JE1
Anderson, C; Haynes, JM; Oliver, VL; Ventura, S1
Odnoshivkina, IuG; Petrov, AM; Zefirov, AL1

Other Studies

6 other study(ies) available for rmi 12330a and nifedipine

ArticleYear
Potent enhancement of [3H]nitrendipine binding in rat cerebral cortical and cardiac homogenates: a putative mechanism for the action of MDL 12,330A.
    The Journal of pharmacology and experimental therapeutics, 1985, Volume: 233, Issue:3

    Topics: Animals; Calcium Channel Blockers; Cerebral Cortex; Half-Life; Heart; Imines; In Vitro Techniques; Kinetics; Male; Myocardium; Nifedipine; Nitrendipine; Rats; Rats, Inbred Strains; Temperature; Tritium

1985
Role of calcium channels and adenylate cyclase in the PACAP-induced adrenal catecholamine secretion.
    American journal of physiology. Regulatory, integrative and comparative physiology, 2001, Volume: 281, Issue:2

    Topics: Adenylyl Cyclases; Adrenal Glands; Animals; Calcium; Calcium Channel Blockers; Calcium Channels; Catecholamines; Epinephrine; Imines; In Vitro Techniques; Male; Neuropeptides; Nifedipine; Norepinephrine; omega-Conotoxin GVIA; omega-Conotoxins; Pituitary Adenylate Cyclase-Activating Polypeptide; Rats; Rats, Wistar

2001
Regulation of growth hormone release in common carp pituitary cells by pituitary adenylate cyclase-activating polypeptide: signal transduction involves cAMP- and calcium-dependent mechanisms.
    Neuroendocrinology, 2002, Volume: 76, Issue:5

    Topics: 1-Methyl-3-isobutylxanthine; Animals; Calcimycin; Calcium; Calcium Channel Blockers; Calcium Channels, L-Type; Carps; Colforsin; Cyclic AMP; Cyclic AMP-Dependent Protein Kinases; Dose-Response Relationship, Drug; Enzyme Activators; Enzyme Inhibitors; Growth Hormone; Imines; In Vitro Techniques; Ionophores; Isoquinolines; Neuropeptides; Neurotransmitter Agents; Nifedipine; Phosphodiesterase Inhibitors; Pituitary Adenylate Cyclase-Activating Polypeptide; Pituitary Gland; Signal Transduction; Sulfonamides; Vasoactive Intestinal Peptide

2002
Protein kinase C cross-talk with gonadotrope progesterone receptor is involved in GnRH-induced LH secretion.
    Journal of physiology and biochemistry, 2006, Volume: 62, Issue:1

    Topics: 8-Bromo Cyclic Adenosine Monophosphate; Animals; Bodily Secretions; Cells, Cultured; Chelating Agents; Colforsin; Egtazic Acid; Enzyme Inhibitors; Female; Gonadotropin-Releasing Hormone; Imines; Indoles; Ionomycin; Luteinizing Hormone; Maleimides; Mifepristone; Nifedipine; Pituitary Gland, Anterior; Protein Kinase C; Rats; Rats, Wistar; Receptors, Progesterone; Signal Transduction; Tetradecanoylphorbol Acetate

2006
Androgens regulate adenylate cyclase activity and intracellular calcium in stromal cells derived from human prostate.
    The Prostate, 2010, Volume: 70, Issue:11

    Topics: Adenylyl Cyclase Inhibitors; Adenylyl Cyclases; Aged; Androgen Antagonists; Androgens; Calcium; Cyclic AMP; Enzyme Inhibitors; Flutamide; Humans; Imines; Immunohistochemistry; Male; Microscopy, Fluorescence; Nifedipine; Prostatic Hyperplasia; Ryanodine; Stromal Cells

2010
[Mechanism of the slow inotropic response of the mouse atrium mediated by the beta2-adrenoreceptor].
    Rossiiskii fiziologicheskii zhurnal imeni I.M. Sechenova, 2011, Volume: 97, Issue:11

    Topics: Adenylyl Cyclases; Adrenergic beta-2 Receptor Agonists; Animals; Atrial Function; Calcium; Cyclic AMP; Cyclic AMP-Dependent Protein Kinases; Fenoterol; Humans; Imines; Mice; Myocardial Contraction; Myocytes, Cardiac; NG-Nitroarginine Methyl Ester; Nifedipine; Nitric Oxide; Nitric Oxide Synthase; Receptors, Adrenergic, beta-2; Signal Transduction; Thionucleotides

2011