Page last updated: 2024-09-03

rmi 12330a and h 89

rmi 12330a has been researched along with h 89 in 11 studies

Compound Research Comparison

Studies
(rmi 12330a)
Trials
(rmi 12330a)
Recent Studies (post-2010)
(rmi 12330a)
Studies
(h 89)
Trials
(h 89)
Recent Studies (post-2010) (h 89)
1410241,6190409

Protein Interaction Comparison

ProteinTaxonomyrmi 12330a (IC50)h 89 (IC50)
Rho-associated protein kinase 2Homo sapiens (human)1.9504
Ribosomal protein S6 kinase alpha-5Homo sapiens (human)0.12
cAMP-dependent protein kinase catalytic subunit alphaBos taurus (cattle)0.073
cAMP-dependent protein kinase catalytic subunit alpha Mus musculus (house mouse)0.381
cAMP-dependent protein kinase catalytic subunit alphaHomo sapiens (human)0.6365
cAMP-dependent protein kinase catalytic subunit gammaHomo sapiens (human)0.6365
cAMP-dependent protein kinase catalytic subunit betaHomo sapiens (human)0.6365
Ribosomal protein S6 kinase beta-1Homo sapiens (human)0.08
RAC-alpha serine/threonine-protein kinaseHomo sapiens (human)1.9886
RAC-beta serine/threonine-protein kinaseHomo sapiens (human)0.5417
Rho-associated protein kinase 2Rattus norvegicus (Norway rat)0.27
RAC-gamma serine/threonine-protein kinaseHomo sapiens (human)0.3207

Research

Studies (11)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's1 (9.09)18.2507
2000's8 (72.73)29.6817
2010's2 (18.18)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Dun, NJ; Dun, SL; Leung, GP; Wong, PY1
Dohovics, R; Hermann, A; Janáky, R; Oja, SS; Saransaari, P; Varga, V1
Chu, MM; Lee, EK; Lin, HR; Wong, AO; Xiao, D1
Azad, SC; DeBock, F; Hapfelmeier, G; Kurz, J; Parsons, CG; Rammes, G; Zieglgänsberger, W1
Kageyama, K; Suda, T1
Cao, C; Cho, KW; Han, JH; Kim, SH; Kim, SZ1
Bie, B; Pan, ZZ; Peng, Y; Zhang, Y1
Babcock, DF; Carlson, AE; Conti, M; Hille, B; McKnight, GS; Schuh, SM1
Azuma, M; Matsuda, K; Nejigaki, Y; Shioda, S; Takahashi, A; Tanaka, M; Uchiyama, M1
Cheung, CS; Hao, Y; Ko, WH; Yip, WC1
Tang, X; Xue, H1

Other Studies

11 other study(ies) available for rmi 12330a and h 89

ArticleYear
Serotonin via 5-HT1B and 5-HT2B receptors stimulates anion secretion in the rat epididymal epithelium.
    The Journal of physiology, 1999, Sep-15, Volume: 519 Pt 3

    Topics: Animals; Anions; Chelating Agents; Colforsin; Culture Techniques; Cyclic AMP; Egtazic Acid; Enzyme Inhibitors; Epididymis; Epithelium; Imines; Isoquinolines; Male; Rats; Rats, Sprague-Dawley; Receptor, Serotonin, 5-HT1B; Receptor, Serotonin, 5-HT2B; Receptors, Serotonin; Serotonin; Sulfonamides; Thapsigargin

1999
Regulation of glutamatergic neurotransmission in the striatum by presynaptic adenylyl cyclase-dependent processes.
    Neurochemistry international, 2003, Volume: 42, Issue:1

    Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Adenylyl Cyclase Inhibitors; Adenylyl Cyclases; Adrenergic beta-Antagonists; alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Animals; Bucladesine; Calcium; Calmodulin; Corpus Striatum; Cyclic AMP; Cyclic AMP-Dependent Protein Kinases; Enzyme Inhibitors; Feedback; Female; Glutamic Acid; Imidazoles; Imines; Isoenzymes; Isoproterenol; Isoquinolines; Kainic Acid; Male; Mice; N-Methylaspartate; Nerve Tissue Proteins; Propranolol; Receptors, Adrenergic, beta; Receptors, AMPA; Receptors, Glutamate; Receptors, Kainic Acid; Receptors, Presynaptic; Second Messenger Systems; Sulfonamides; Synaptic Transmission; Trifluoperazine

2003
Regulation of growth hormone release in common carp pituitary cells by pituitary adenylate cyclase-activating polypeptide: signal transduction involves cAMP- and calcium-dependent mechanisms.
    Neuroendocrinology, 2002, Volume: 76, Issue:5

    Topics: 1-Methyl-3-isobutylxanthine; Animals; Calcimycin; Calcium; Calcium Channel Blockers; Calcium Channels, L-Type; Carps; Colforsin; Cyclic AMP; Cyclic AMP-Dependent Protein Kinases; Dose-Response Relationship, Drug; Enzyme Activators; Enzyme Inhibitors; Growth Hormone; Imines; In Vitro Techniques; Ionophores; Isoquinolines; Neuropeptides; Neurotransmitter Agents; Nifedipine; Phosphodiesterase Inhibitors; Pituitary Adenylate Cyclase-Activating Polypeptide; Pituitary Gland; Signal Transduction; Sulfonamides; Vasoactive Intestinal Peptide

2002
Alpha2-adrenoreceptor activation inhibits LTP and LTD in the basolateral amygdala: involvement of Gi/o-protein-mediated modulation of Ca2+-channels and inwardly rectifying K+-channels in LTD.
    The European journal of neuroscience, 2003, Volume: 17, Issue:7

    Topics: 3',5'-Cyclic-AMP Phosphodiesterases; Adenylyl Cyclase Inhibitors; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Amygdala; Animals; Barium; Cadmium; Calcium Channel Blockers; Calcium Channels; Clonidine; Colforsin; Cyclic Nucleotide Phosphodiesterases, Type 4; Electric Stimulation; Enzyme Inhibitors; Excitatory Postsynaptic Potentials; Heterotrimeric GTP-Binding Proteins; Imines; In Vitro Techniques; Isoquinolines; Long-Term Potentiation; Long-Term Synaptic Depression; Membrane Potentials; Mice; Norepinephrine; omega-Agatoxin IVA; omega-Conotoxins; Patch-Clamp Techniques; Pertussis Toxin; Piperazines; Potassium Channel Blockers; Potassium Channels, Inwardly Rectifying; Pyridines; Receptors, Adrenergic, alpha-2; Serotonin Antagonists; Sulfonamides; Yohimbine

2003
Urocortin-related peptides increase interleukin-6 output via cyclic adenosine 5'-monophosphate-dependent pathways in A7r5 aortic smooth muscle cells.
    Endocrinology, 2003, Volume: 144, Issue:6

    Topics: Animals; Aorta; Cells, Cultured; Corticotropin-Releasing Hormone; Cyclic AMP; Cyclic AMP-Dependent Protein Kinases; Enzyme Inhibitors; Flavonoids; Imidazoles; Imines; Indoles; Interleukin-6; Isoquinolines; Maleimides; MAP Kinase Signaling System; Mitogen-Activated Protein Kinases; Muscle, Smooth, Vascular; Protein Kinase C; Pyridines; Rats; Sulfonamides; Urocortins

2003
Diverse regulation of atrial natriuretic peptide secretion by serotonin receptor subtypes.
    Cardiovascular research, 2003, Aug-01, Volume: 59, Issue:2

    Topics: Adenylyl Cyclase Inhibitors; Alkaloids; Aminobenzoates; Animals; Atrial Natriuretic Factor; Benzophenanthridines; Benzothiazoles; Calcium; Carbazoles; Cyclic AMP-Dependent Protein Kinases; Depression, Chemical; Dose-Response Relationship, Drug; Heart; Heart Atria; Imines; Indoles; Isoquinolines; Ketanserin; Male; Myocytes, Cardiac; Neomycin; para-Aminobenzoates; Perfusion; Phenanthridines; Piperazines; Piperidines; Protein Kinase C; Pyrroles; Rats; Rats, Sprague-Dawley; Receptors, Serotonin; Receptors, Serotonin, 5-HT4; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Staurosporine; Sulfonamides; Thiazoles; Type C Phospholipases

2003
cAMP-mediated mechanisms for pain sensitization during opioid withdrawal.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 2005, Apr-13, Volume: 25, Issue:15

    Topics: 2-Amino-5-phosphonovalerate; 6-Cyano-7-nitroquinoxaline-2,3-dione; 8-Bromo Cyclic Adenosine Monophosphate; Adenylyl Cyclases; Animals; Animals, Newborn; Behavior, Animal; Blotting, Western; Colforsin; Cyclic AMP; Dose-Response Relationship, Radiation; Drug Administration Schedule; Drug Interactions; Electric Stimulation; Enzyme Inhibitors; Excitatory Amino Acid Antagonists; Excitatory Postsynaptic Potentials; Gene Expression Regulation; Imines; In Vitro Techniques; Isoquinolines; Male; Membrane Potentials; Microinjections; Morphine; Naloxone; Narcotic Antagonists; Narcotics; Opioid-Related Disorders; Oxidoreductases; Pain; Pain Measurement; Patch-Clamp Techniques; Pyrimidines; Raphe Nuclei; Rats; Rats, Wistar; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Sulfonamides

2005
Signaling pathways for modulation of mouse sperm motility by adenosine and catecholamine agonists.
    Biology of reproduction, 2006, Volume: 74, Issue:3

    Topics: Adenine; Adenosine; Adenylyl Cyclases; Animals; Calcium; Catecholamines; Cyclic AMP; Cyclic AMP-Dependent Protein Kinase Catalytic Subunits; Dideoxyadenosine; Enzyme Inhibitors; Imines; Isoquinolines; Male; Mice; Mice, Inbred C57BL; Mice, Knockout; Protein Kinase Inhibitors; Signal Transduction; Sperm Motility; Sperm Tail; Sulfonamides

2006
Pituitary adenylate cyclase-activating polypeptide induces somatolactin release from cultured goldfish pituitary cells.
    Peptides, 2009, Volume: 30, Issue:7

    Topics: Adenylyl Cyclase Inhibitors; Adenylyl Cyclases; Animals; Calmodulin; Cells, Cultured; Enzyme Inhibitors; Estrenes; Female; Fish Proteins; Glycoproteins; Goldfish; Growth Substances; Imidazoles; Imines; Immunoblotting; Indoles; Intracellular Signaling Peptides and Proteins; Isoquinolines; Male; Maleimides; Phosphoinositide Phospholipase C; Pituitary Adenylate Cyclase-Activating Polypeptide; Pituitary Gland; Pituitary Hormones; Protein Kinase C; Pyrrolidinones; Receptors, Pituitary Adenylate Cyclase-Activating Polypeptide; Signal Transduction; Sulfonamides; Vasoactive Intestinal Peptide

2009
Nobiletin Stimulates Chloride Secretion in Human Bronchial Epithelia via a cAMP/PKA-Dependent Pathway.
    Cellular physiology and biochemistry : international journal of experimental cellular physiology, biochemistry, and pharmacology, 2015, Volume: 37, Issue:1

    Topics: Adenylyl Cyclases; Bronchi; Calcium; Cell Line; Chlorides; Cyclic AMP; Cyclic AMP-Dependent Protein Kinases; Cystic Fibrosis; Cystic Fibrosis Transmembrane Conductance Regulator; Epithelial Cells; Flavones; Humans; Imines; Ion Transport; Isoquinolines; Respiratory Mucosa; Signal Transduction; Sulfonamides

2015
Effect of vasopressin on Na(+)-K(+)-2Cl(-) cotransporter (NKCC) and the signaling mechanisms on the murine late distal colon.
    European journal of pharmacology, 2016, Jan-15, Volume: 771

    Topics: Animals; Calcium Signaling; Chelating Agents; Colon; Cyclic AMP; Cyclic AMP-Dependent Protein Kinases; Egtazic Acid; Imines; Isoquinolines; Male; Mice; Mice, Inbred C57BL; Phosphorylation; RNA, Small Interfering; Solute Carrier Family 12, Member 1; Solute Carrier Family 12, Member 2; Sulfonamides; Vasopressins; Water Deprivation

2016