Page last updated: 2024-08-16

ritanserin and pyrimidinones

ritanserin has been researched along with pyrimidinones in 7 studies

Research

Studies (7)

TimeframeStudies, this research(%)All Research%
pre-19904 (57.14)18.7374
1990's1 (14.29)18.2507
2000's0 (0.00)29.6817
2010's2 (28.57)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Awouters, FH; Janssen, PA; Meert, TF; Megens, AA; Niemegeers, CJ; Schellekens, KH1
Cohen, ML; Kurz, KD; Schenck, KW1
Gelders, YG1
Gommeren, W; Laduron, PM; Leysen, JE; van Gompel, P1
Gommeren, W; Janssen, PA; Leysen, JE; Van Gompel, P; Woestenborghs, R1
Boroda, S; Harris, TE; Niccum, M; Purow, BW; Raje, V1
Baldanzi, G; Bertoni, A; Capello, D; Fresu, LG; Gesu, A; Graziani, A; Massarotti, A; Ruffo, E; Snow, AL; Talmon, M; Tron, GC; Varma, KSS; Velnati, S1

Trials

1 trial(s) available for ritanserin and pyrimidinones

ArticleYear
Thymosthenic agents, a novel approach in the treatment of schizophrenia.
    The British journal of psychiatry. Supplement, 1989, Issue:5

    Topics: Brain; Butyrophenones; Humans; Isoxazoles; Piperidines; Pyrimidinones; Randomized Controlled Trials as Topic; Receptors, Serotonin; Risperidone; Ritanserin; Schizophrenia; Schizophrenic Psychology; Serotonin Antagonists

1989

Other Studies

6 other study(ies) available for ritanserin and pyrimidinones

ArticleYear
Pharmacological profile of the new potent neuroleptic ocaperidone (R 79,598).
    The Journal of pharmacology and experimental therapeutics, 1992, Volume: 260, Issue:1

    Topics: Animals; Antiemetics; Antipsychotic Agents; Apomorphine; Behavior, Animal; Body Temperature; Dogs; Dopamine Agents; Dopamine Antagonists; Eating; Female; Haloperidol; Isoxazoles; Lethal Dose 50; Locomotion; Male; Mice; Motor Activity; Muscles; Neurotransmitter Agents; Piperidines; Posture; Pyrimidinones; Rats; Rats, Inbred Strains; Risperidone; Ritanserin; Serotonin; Serotonin Antagonists; Synaptic Transmission

1992
5-HT2-receptor antagonists: alpha 1- vs. 5-HT2-receptor blocking properties in blood vessels.
    Journal of cardiovascular pharmacology, 1988, Volume: 11 Suppl 1

    Topics: Adrenergic alpha-Antagonists; Animals; Blood Pressure; Ergolines; Ketanserin; Male; Muscle Contraction; Muscle, Smooth, Vascular; Phentolamine; Piperidines; Pyrimidinones; Rats; Rats, Inbred SHR; Rats, Inbred Strains; Receptors, Adrenergic, alpha; Receptors, Serotonin; Ritanserin; Serotonin Antagonists; Spiperone

1988
Differential regulation of dopamine-D2 and serotonin-S2 receptors by chronic treatment with the serotonin-S2 antagonists, ritanserin, and setoperone.
    Psychopharmacology series, 1987, Volume: 3

    Topics: Animals; Brain; Corpus Striatum; Frontal Lobe; Male; Piperidines; Pyrimidinones; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Dopamine D2; Receptors, Serotonin; Ritanserin; Serotonin Antagonists

1987
Down regulation of serotonin-S2 receptor sites in rat brain by chronic treatment with the serotonin-S2 antagonists: ritanserin and setoperone.
    Psychopharmacology, 1986, Volume: 88, Issue:4

    Topics: Animals; Brain; Corpus Striatum; Frontal Lobe; Ketanserin; Male; Piperidines; Pyrimidinones; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Dopamine D2; Receptors, Neurotransmitter; Receptors, Serotonin; Ritanserin

1986
Dual activities of ritanserin and R59022 as DGKα inhibitors and serotonin receptor antagonists.
    Biochemical pharmacology, 2017, Jan-01, Volume: 123

    Topics: Adenosine Triphosphate; Diacylglycerol Kinase; Electrophoresis, Polyacrylamide Gel; Enzyme Inhibitors; HEK293 Cells; HeLa Cells; Humans; Kinetics; Pyrimidinones; Ritanserin; Thiazoles

2017
Identification of a novel DGKα inhibitor for XLP-1 therapy by virtual screening.
    European journal of medicinal chemistry, 2019, Feb-15, Volume: 164

    Topics: Cell Death; Computer Simulation; Diacylglycerol Kinase; Drug Evaluation, Preclinical; Humans; Lymphoproliferative Disorders; Piperidines; Protein Kinase Inhibitors; Pyrimidinones; Quinazolinones; Ritanserin; Thiazoles

2019