Page last updated: 2024-08-16

ritanserin and prazosin

ritanserin has been researched along with prazosin in 31 studies

Research

Studies (31)

TimeframeStudies, this research(%)All Research%
pre-19908 (25.81)18.7374
1990's15 (48.39)18.2507
2000's7 (22.58)29.6817
2010's1 (3.23)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Arnt, J; Boeck, V; Bøgesø, KP; Christensen, AV; Hyttel, J; Jensen, KG1
Janssen, CG; Laduron, PM; Thijssen, JB; Van Dun, J; Wouters, W1
Artursson, P; Bergström, CA; Hoogstraate, J; Matsson, P; Norinder, U; Pedersen, JM1
Nakamura, H; Suzukawa, M1
Bouysset, F; Laubie, M; Schmitt, H; Vayssettes-Courchay, C; Verbeuren, TJ1
Backus, LI; Grahame-Smith, DG; Sharp, T1
Jackson, DA; White, SR1
Ball, SG; Robertson, JI; Stott, DJ1
Gradin, K; Hedner, T; Persson, B; Pettersson, A3
Ramage, AG1
Smits, J; Struyker Boudier, H; van Dorsten, F1
Deutch, AY; Duman, RS; Ongür, D1
Arnt, J1
Benington, JH; Heller, HC1
Hong, E; López-Muñoz, FJ; Terrón, JA; Villalón, CM1
Bennie, J; Carroll, S; Dow, RC; Fink, G; Williams, BC1
Bietti, G; Borsini, F; Ceci, A; Donetti, A1
Kleven, MS; Koek, W; Prinssen, EP1
Bertolino, F; Fauré, P; John, GW; Valentin, JP; Vieu, S1
Marwood, JF; Okoro, EO1
Depoortere, R; Perrault, G; Sanger, DJ1
Del Bel, EA; Guimarães, FS; Nucci-da-Silva, LP1
Chen, J; Purdy, RE; Yildiz, O1
Fernández, MM; Martín, ML; Morán, A; San Román, L1
Matsushima, K; Tozawa, Y1
Calama, E; Martín, ML; Morán, A; Ortiz de Urbina, AV; San Román, L1
Fu, YJ; Miao, CY; Shu, H; Su, DF; Wang, MW1
Centurión, D; Gupta, S; Mehrotra, S; Saxena, PR; VandenBrink, AM; Villalón, CM1
Chen, Y; Fan, S; Hu, Z; Jia, X; Qi, A; Wang, T; Xia, J; Xiong, J; Yan, J; Yang, N; Ye, J1

Reviews

1 review(s) available for ritanserin and prazosin

ArticleYear
Antihypertensive mode of action of ketanserin.
    Journal of cardiovascular pharmacology, 1987, Volume: 10 Suppl 3

    Topics: Adrenergic alpha-Antagonists; Aldosterone; Animals; Antihypertensive Agents; Blood Pressure; Carcinoid Heart Disease; Humans; Ketanserin; Piperidines; Prazosin; Ritanserin

1987

Other Studies

30 other study(ies) available for ritanserin and prazosin

ArticleYear
Antihypertensive activity in a series of 1-piperazino-3-phenylindans with potent 5-HT2-antagonistic activity.
    Journal of medicinal chemistry, 1988, Volume: 31, Issue:12

    Topics: Animals; Antihypertensive Agents; Antipsychotic Agents; Blood Pressure; Chemical Phenomena; Chemistry; Dopamine; Imidazoles; Ketanserin; Norepinephrine; Phenylephrine; Piperazines; Rats; Rats, Inbred SHR; Serotonin Antagonists; Structure-Activity Relationship

1988
In vitro labeling of serotonin-S2 receptors: synthesis and binding characteristics of [3H]-7-aminoketanserin.
    Journal of medicinal chemistry, 1986, Volume: 29, Issue:9

    Topics: Animals; Binding, Competitive; Brain; Chemical Phenomena; Chemistry; Frontal Lobe; Guinea Pigs; Ketanserin; Kinetics; Piperidines; Rats; Rats, Inbred Strains; Receptors, Serotonin

1986
Prediction and identification of drug interactions with the human ATP-binding cassette transporter multidrug-resistance associated protein 2 (MRP2; ABCC2).
    Journal of medicinal chemistry, 2008, Jun-12, Volume: 51, Issue:11

    Topics: Administration, Oral; Animals; Antineoplastic Agents; Antipsychotic Agents; Antiviral Agents; ATP Binding Cassette Transporter, Subfamily B; ATP Binding Cassette Transporter, Subfamily B, Member 1; ATP Binding Cassette Transporter, Subfamily G, Member 2; ATP-Binding Cassette Transporters; Biological Transport; Cell Line; Computer Simulation; Cytochrome P-450 Enzyme System; Drug-Related Side Effects and Adverse Reactions; Estradiol; Humans; Insecta; Liver; Models, Molecular; Multidrug Resistance-Associated Protein 2; Multidrug Resistance-Associated Proteins; Neoplasm Proteins; Pharmaceutical Preparations; Pharmacology; Structure-Activity Relationship

2008
Effects of ketanserin tartrate on 3-hydroxy, 3-methylglutaryl coenzyme A reductase activity in cultured human skin fibroblasts.
    Cardiovascular drugs and therapy, 1990, Volume: 4 Suppl 1

    Topics: Adrenergic alpha-Antagonists; Cells, Cultured; Fibroblasts; Humans; Hydroxymethylglutaryl CoA Reductases; Ketanserin; Piperidines; Prazosin; Ritanserin; Serotonin Antagonists

1990
The cardiovascular effects of quipazine are mediated by peripheral 5-HT2 and 5-HT3 receptors in anaesthetized rats.
    European journal of pharmacology, 1990, Aug-02, Volume: 184, Issue:1

    Topics: Amidines; Anesthesia; Animals; Blood Pressure; Carotid Body; Denervation; Heart Rate; Hemodynamics; Hexamethonium Compounds; In Vitro Techniques; Indoles; Lung; Male; Myocardium; Piperidines; Prazosin; Pressoreceptors; Propanolamines; Quipazine; Rats; Rats, Inbred Strains; Receptors, Serotonin; Renin-Angiotensin System; Ritanserin; Sympathetic Nervous System; Thiophenes; Tropisetron; Vagotomy

1990
Behavioural evidence for a functional interaction between central 5-HT2 and 5-HT1A receptors.
    British journal of pharmacology, 1990, Volume: 100, Issue:4

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Apomorphine; Behavior, Animal; Central Nervous System; Dose-Response Relationship, Drug; Haloperidol; Ketanserin; Male; Methoxydimethyltryptamines; Piperidines; Prazosin; Pyrimidines; Quinolines; Rats; Rats, Inbred Strains; Receptors, Serotonin; Ritanserin; Serotonin; Stereotyped Behavior; Tetrahydronaphthalenes

1990
Receptor subtypes mediating facilitation by serotonin of excitability of spinal motoneurons.
    Neuropharmacology, 1990, Volume: 29, Issue:9

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Amphetamines; Animals; In Vitro Techniques; Injections, Intravenous; Iontophoresis; Ketanserin; Male; Methysergide; Microelectrodes; Motor Neurons; Piperidines; Prazosin; Quipazine; Rats; Rats, Inbred Strains; Receptors, Serotonin; Ritanserin; Serotonin; Serotonin Antagonists; Spinal Cord; Tetrahydronaphthalenes

1990
Antihypertensive effects of ketanserin and ritanserin in the spontaneously hypertensive rat.
    Journal of cardiovascular pharmacology, 1988, Volume: 11 Suppl 1

    Topics: Animals; Antihypertensive Agents; Blood Pressure; Heart Rate; Hypertension; Ketanserin; Male; Phenylephrine; Piperidines; Prazosin; Rats; Rats, Inbred SHR; Receptors, Adrenergic, alpha; Receptors, Serotonin; Ritanserin; Serotonin; Sympathetic Nervous System

1988
Are drugs that act both on serotonin receptors and alpha 1-adrenoceptors more potent hypotensive agents than those that act only on alpha 1-adrenoceptors?
    Journal of cardiovascular pharmacology, 1988, Volume: 11 Suppl 1

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Blood Pressure; Cats; Cinanserin; Ergolines; Ketanserin; Male; Metergoline; Piperidines; Prazosin; Receptors, Adrenergic, alpha; Receptors, Serotonin; Ritanserin; Serotonin Antagonists; Sympathetic Nervous System; Tetrahydronaphthalenes

1988
Chronic 5-HT2 receptor blockade with ritanserin does not reduce blood pressure in the spontaneously hypertensive rat.
    Journal of neural transmission, 1985, Volume: 64, Issue:2

    Topics: Animals; Blood Pressure; Decerebrate State; Dose-Response Relationship, Drug; Electric Stimulation; Heart Rate; Hypertension; Ketanserin; Male; Phenylephrine; Piperidines; Prazosin; Rats; Rats, Inbred SHR; Receptors, Serotonin; Ritanserin; Time Factors

1985
Antihypertensive mechanism of action of ketanserin and some ketanserin analogues in the spontaneously hypertensive rat.
    Naunyn-Schmiedeberg's archives of pharmacology, 1985, Volume: 329, Issue:4

    Topics: Animals; Blood Pressure; Dose-Response Relationship, Drug; Electric Stimulation; Hypertension; Ketanserin; Phenylephrine; Piperidines; Prazosin; Pyrimidines; Rats; Rats, Inbred SHR; Receptors, Adrenergic, alpha; Ritanserin; Sympathetic Nervous System

1985
Interference of ketanserin with baroreflex control of the circulation in the conscious spontaneously hypertensive rat.
    Drugs, 1988, Volume: 36 Suppl 1

    Topics: Animals; Blood Pressure; Heart Rate; Hypertension; Ketanserin; Male; Piperidines; Prazosin; Pressoreceptors; Rats; Rats, Inbred SHR; Ritanserin; Serotonin Antagonists

1988
Antipsychotic drugs induce Fos protein in the thalamic paraventricular nucleus: a novel locus of antipsychotic drug action.
    Neuroscience, 1995, Volume: 66, Issue:2

    Topics: Animals; Antipsychotic Agents; Blotting, Western; Clozapine; Haloperidol; Immunohistochemistry; Male; Muscarinic Antagonists; Prazosin; Proto-Oncogene Proteins c-fos; Rats; Rats, Sprague-Dawley; Ritanserin; Scopolamine; Serotonin Antagonists; Sulpiride; Thalamic Nuclei

1995
Differential effects of classical and newer antipsychotics on the hypermotility induced by two dose levels of D-amphetamine.
    European journal of pharmacology, 1995, Sep-05, Volume: 283, Issue:1-3

    Topics: Animals; Antipsychotic Agents; Clozapine; Dextroamphetamine; Dose-Response Relationship, Drug; Fluphenazine; Haloperidol; Imidazoles; Indoles; Locomotion; Male; Motor Activity; Prazosin; Rats; Rats, Wistar; Ritanserin

1995
Monoaminergic and cholinergic modulation of REM-sleep timing in rats.
    Brain research, 1995, May-29, Volume: 681, Issue:1-2

    Topics: Animals; Biogenic Monoamines; Cholinergic Antagonists; Electroencephalography; Male; Metergoline; Parasympathetic Nervous System; Prazosin; Quinuclidinyl Benzilate; Rats; Rats, Wistar; Ritanserin; Serotonin Antagonists; Sleep, REM; Sympatholytics

1995
Inhibition of serotonin-induced increase in canine external carotid blood flow by drugs that decrease the sympathetic outflow.
    Journal of autonomic pharmacology, 1994, Volume: 14, Issue:3

    Topics: Animals; Blood Pressure; Carotid Arteries; Dioxanes; Dogs; Dose-Response Relationship, Drug; Female; Heart Rate; Infusions, Intra-Arterial; Injections, Intravenous; Ketanserin; Male; Mecamylamine; Methiothepin; Prazosin; Receptors, Serotonin; Regional Blood Flow; Regression Analysis; Ritanserin; Serotonin; Spiro Compounds; Vascular Resistance

1994
A central 5-HT2 receptor mechanism plays a key role in the proestrous surge of luteinizing hormone in the rat.
    Psychoneuroendocrinology, 1994, Volume: 19, Issue:4

    Topics: Animals; Female; Ketanserin; Luteinizing Hormone; Prazosin; Proestrus; Rats; Rats, Wistar; Receptors, Serotonin; Ritanserin

1994
BIMT 17, a 5-HT1A receptor agonist/5-HT2A receptor antagonist, directly activates postsynaptic 5-HT inhibitory responses in the rat cerebral cortex.
    Naunyn-Schmiedeberg's archives of pharmacology, 1995, Volume: 352, Issue:3

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Adrenergic beta-Antagonists; Analysis of Variance; Animals; Antidepressive Agents; Benzimidazoles; Binding, Competitive; Buspirone; Cerebral Cortex; Dose-Response Relationship, Drug; In Vitro Techniques; Iontophoresis; Male; Microelectrodes; Neurons; Piperazines; Prazosin; Propanolamines; Rats; Rats, Sprague-Dawley; Receptors, Serotonin; Ritanserin; Serotonin Antagonists; Serotonin Receptor Agonists; Thiophenes

1995
Effects of dopamine antagonists in a two-way active avoidance procedure in rats: interactions with 8-OH-DPAT, ritanserin, and prazosin.
    Psychopharmacology, 1996, Volume: 128, Issue:2

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Adrenergic alpha-Antagonists; Animals; Avoidance Learning; Dopamine Antagonists; Dose-Response Relationship, Drug; Haloperidol; Male; Prazosin; Raclopride; Rats; Rats, Sprague-Dawley; Ritanserin; Salicylamides; Serotonin Agents

1996
Differential involvement of serotonin 2A/C and thromboxane A2/prostanoid receptors in high- vs. low-shear rate arterial thrombosis in rabbits.
    The Journal of pharmacology and experimental therapeutics, 1997, Volume: 280, Issue:2

    Topics: Animals; Arteriovenous Shunt, Surgical; Aspirin; Blood Pressure; Bridged Bicyclo Compounds, Heterocyclic; Carotid Arteries; Carotid Stenosis; Endothelium, Vascular; Fatty Acids, Unsaturated; Heart Rate; Hemodynamics; Hydrazines; Jugular Veins; Ketanserin; Male; Oxadiazoles; Piperazines; Platelet Aggregation; Prazosin; Rabbits; Receptor, Serotonin, 5-HT2A; Receptor, Serotonin, 5-HT2C; Receptors, Prostaglandin; Receptors, Serotonin; Receptors, Thromboxane; Ritanserin; Serotonin Antagonists; Stress, Mechanical

1997
Effects of 5HT2 receptor antagonists on responses to potassium depolarization in rat isolated aorta.
    Clinical and experimental pharmacology & physiology, 1997, Volume: 24, Issue:1

    Topics: Animals; Aorta, Thoracic; Cinnarizine; Cyproheptadine; Diltiazem; Drug Synergism; Felodipine; Female; In Vitro Techniques; Ketanserin; Male; Mianserin; Muscle Contraction; Nifedipine; Potassium; Prazosin; Rats; Rats, Sprague-Dawley; Receptors, Serotonin; Reproducibility of Results; Ritanserin; Serotonin Antagonists; Verapamil

1997
Some, but not all, antipsychotic drugs potentiate a low level of prepulse inhibition shown by rats of the Wistar strain.
    Behavioural pharmacology, 1997, Volume: 8, Issue:4

    Topics: Adrenergic alpha-Antagonists; Animals; Antipsychotic Agents; Behavior, Animal; Benzazepines; Benzodiazepines; Clozapine; Haloperidol; Imidazoles; Indoles; Injections, Intraperitoneal; Male; Neural Inhibition; Olanzapine; Pirenzepine; Prazosin; Rats; Rats, Wistar; Reflex, Startle; Remoxipride; Risperidone; Ritanserin; Serotonin Antagonists

1997
Serotonin modulation of catalepsy induced by N(G)-nitro-L-arginine in mice.
    European journal of pharmacology, 1999, Aug-20, Volume: 379, Issue:1

    Topics: Adrenergic alpha-Antagonists; Animals; Bridged Bicyclo Compounds, Heterocyclic; Catalepsy; Dose-Response Relationship, Drug; Drug Synergism; Enzyme Inhibitors; Indoles; Ketanserin; Male; Mice; Nitric Oxide; Nitric Oxide Synthase; Nitroarginine; Piperazines; Prazosin; Ritanserin; Serotonin Antagonists; Time Factors

1999
Phenylephrine precontraction increases the sensitivity of rabbit femoral artery to serotonin by enabling 5-HT1-like receptors.
    Journal of cardiovascular pharmacology, 2000, Volume: 35, Issue:6

    Topics: Animals; Dose-Response Relationship, Drug; Femoral Artery; In Vitro Techniques; Oxadiazoles; Phenylephrine; Piperazines; Prazosin; Rabbits; Receptors, Serotonin; Ritanserin; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Specific Pathogen-Free Organisms; Sumatriptan; Vasoconstriction

2000
Mesenteric vasoconstrictor response to 5-hydroxytryptamine in the in situ blood autoperfused rat mesentery: involvement of 5-HT(2B) and/or 5-HT(2C) receptor activation.
    European journal of pharmacology, 2000, Aug-04, Volume: 401, Issue:2

    Topics: Amphetamines; Animals; Biguanides; Dose-Response Relationship, Drug; Enalapril; Indoles; Indomethacin; Male; Mesenteric Arteries; Mesentery; Perfusion; Piperazines; Prazosin; Propranolol; Pyridines; Rats; Rats, Wistar; Receptor, Serotonin, 5-HT2B; Receptor, Serotonin, 5-HT2C; Receptors, Serotonin; Ritanserin; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Splanchnic Circulation; Vasoconstriction

2000
Peripheral 5-HT(2A)-receptor-mediated formation of an inhibitor of atrial natriuretic peptide binding involves inflammation.
    European journal of pharmacology, 2002, Apr-05, Volume: 440, Issue:1

    Topics: Adrenergic alpha-Antagonists; alpha-Methyltyrosine; Animals; Atrial Natriuretic Factor; Catecholamines; Cyclooxygenase Inhibitors; Dexamethasone; Ditiocarb; Dopamine beta-Hydroxylase; Dose-Response Relationship, Drug; Endothelium, Vascular; Humans; Indomethacin; Inflammation; Isatin; Ketanserin; Muscle, Smooth; Prazosin; Propranolol; Protein Binding; Rats; Rats, Wistar; Reactive Oxygen Species; Receptor, Angiotensin, Type 1; Receptor, Serotonin, 5-HT2A; Receptors, Angiotensin; Receptors, Serotonin; Reserpine; Ritanserin; Serotonin; Serotonin Receptor Agonists; Tyrosine 3-Monooxygenase; Urination; Vascular Resistance; Yohimbine

2002
Vasoconstrictor responses to 5-hydroxytryptamine in the autoperfused hindquarters of spontaneously hypertensive rats.
    Pharmacology, 2004, Volume: 71, Issue:2

    Topics: Animals; Dose-Response Relationship, Drug; Hindlimb; Indoles; Injections, Intra-Arterial; Injections, Intravenous; Male; Perfusion; Piperazines; Prazosin; Pyridines; Rats; Rats, Inbred SHR; Rats, Wistar; Receptor, Serotonin, 5-HT1A; Receptor, Serotonin, 5-HT2A; Receptor, Serotonin, 5-HT2B; Receptor, Serotonin, 5-HT2C; Receptors, Serotonin, 5-HT2; Regional Blood Flow; Ritanserin; Serotonin; Serotonin 5-HT1 Receptor Antagonists; Serotonin 5-HT2 Receptor Agonists; Serotonin 5-HT2 Receptor Antagonists; Serotonin Receptor Agonists; Spiperone; Thiophenes; Vasoconstriction

2004
Restoration of baroreflex function by ketanserin is not blood pressure dependent in conscious freely moving rats.
    Journal of hypertension, 2004, Volume: 22, Issue:6

    Topics: Animals; Antihypertensive Agents; Baroreflex; Blood Pressure; Female; Ketanserin; Male; Myocardial Infarction; Prazosin; Rats; Rats, Inbred SHR; Rats, Sprague-Dawley; Ritanserin; Time Factors

2004
A61603-induced contractions of the porcine meningeal artery are mediated by alpha1- and alpha2-adrenoceptors.
    Basic & clinical pharmacology & toxicology, 2007, Volume: 100, Issue:4

    Topics: Adrenergic alpha-1 Receptor Agonists; Adrenergic alpha-2 Receptor Agonists; Adrenergic alpha-Antagonists; Alkaloids; Animals; Benzophenanthridines; Colforsin; Dose-Response Relationship, Drug; Female; Forecasting; Imidazoles; In Vitro Techniques; Meningeal Arteries; Methiothepin; Norepinephrine; Oxadiazoles; Phenylephrine; Piperazines; Potassium Chloride; Prazosin; Protein Kinase C; Receptors, Adrenergic, alpha-1; Receptors, Adrenergic, alpha-2; Ritanserin; Serotonin 5-HT1 Receptor Antagonists; Serotonin Antagonists; Swine; Tetrahydronaphthalenes; Vasoconstriction; Yohimbine

2007
Arousal effects of orexin A on acute alcohol intoxication-induced coma in rats.
    Neuropharmacology, 2012, Volume: 62, Issue:2

    Topics: Alcoholic Intoxication; Animals; Arousal; Benzoxazoles; Brain; Coma; Consciousness; Electroencephalography; Ethanol; Female; Intracellular Signaling Peptides and Proteins; Naphthyridines; Neurons; Neuropeptides; Orexins; Prazosin; Pyrilamine; Rats; Rats, Sprague-Dawley; Receptors, Neuropeptide; Ritanserin; Urea

2012