ritanserin has been researched along with piperidines in 200 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 100 (50.00) | 18.7374 |
1990's | 91 (45.50) | 18.2507 |
2000's | 5 (2.50) | 29.6817 |
2010's | 4 (2.00) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
---|---|
Awouters, FH; Janssen, PA; Meert, TF; Megens, AA; Niemegeers, CJ; Schellekens, KH | 1 |
Humphreys, TM; Schmidt, CJ; Sorensen, SM; Taylor, VL | 1 |
Ashby, CR; Edwards, E; Wang, RY | 1 |
Bernardi, M; Di Sarra, B; Montecchiani, G; Re, L; Rossini, L; Tonnini, C | 1 |
Alterwain, P; Monti, JM | 1 |
Devaud, LL; Hollingsworth, EB | 1 |
Almeida, SS; de Oliveira, LM; Graeff, FG | 2 |
Arends, J; Declerck, AC; Kamphuisen, HA; Lammers, GJ; Schouwink, G; Troost, J | 1 |
Hajdukovic, R; Mitler, MM | 1 |
Brazell, C; Campbell, IC; Mitchell, S; Stahl, SM; Twist, EC | 1 |
Neal, BS; Sparber, SB | 1 |
Den Boer, JA; Westenberg, HG | 2 |
Awouters, F; Janssen, PA; Megens, AA; Niemegeers, CJ | 1 |
Kidd, EJ; Leysen, JE; Marsden, CA | 1 |
Allen, AD; Barrett, RJ; Taylor, DR; Wright, KF | 1 |
Bogdanov, MB; Gaĭnetdinov, RR; Kudrin, VS; Medvedev, OS; Val'dman, AV | 1 |
Ohno, M; Watanabe, S; Yamamoto, T | 1 |
Gorzalka, BB; Watson, NV | 1 |
Brownfield, MS; Rittenhouse, PA; Saydoff, JA; van de Kar, LD | 1 |
Barnes, M; Lee, MA; Meltzer, HY; Nash, JF | 1 |
Abbate, GM; Nieduzak, TR; Schmidt, CJ; Taylor, VL | 1 |
Bersani, G; Ciani, N; Grispini, A; Marini, S; Pasini, A; Pozzi, F | 1 |
Idzikowski, C; James, RJ; Mills, FJ | 1 |
Linnoila, M; Wozniak, KM | 1 |
Beczkowska, IW; Bodnar, RJ | 1 |
Campbell, IC; Corn, TH; Mitchell, SN; Twist, EC | 1 |
Blanchard, JC; Comte, MT; Doble, A; Gueremy, C; Huon, C; Malleron, JL; Peyronel, JF; Piot, O; Truchon, A; Zundel, JL | 1 |
Deakin, JF; Guimarães, FS; Hensman, R; Wang, M | 1 |
D'Urso, R; Falaschi, P; Melis, GB; Proietti, A; Rocco, A; Rosa, M | 1 |
Bizzi, A; Garattini, S; Grignaschi, G; Neill, JC; Padura, IM; Samanin, R | 1 |
Heykants, J; Huang, ML; Koch, S; Kokot, F; Kuska, J; Van Peer, A; Zazgornik, J | 1 |
Fink, H; Morgenstern, R; Ott, T; Schremmer, C | 1 |
Dahlitz, M; Idzikowski, C; James, R; Parkes, JD; Wells, P | 1 |
Borsini, F; D'Aranno, V; Lecci, A; Mancinelli, A; Meli, A; Stasi, MA; Volterra, G | 1 |
Ehrmann, H; Fleischhacker, WW; Kane, JM; Miller, CH | 1 |
Nakamura, H; Suzukawa, M | 1 |
Giroux, L; Huet, PM; Mastai, R; Semret, M | 1 |
Aghajanian, GK; Sheldon, PW | 1 |
Markianos, M; Papadimitriou, G; Papakostas, Y; Stefanis, C | 1 |
Broekkamp, CL; Jenck, F; Van Delft, AM | 1 |
Mück-Seler, D; Pericić, D | 1 |
Argenio, GF; Bernini, GP; Birindelli, R; Del Corso, C; Franchi, F; Luisi, M; Vivaldi, MS | 1 |
Gustafsson, U; Harrison, DK; Lewis, DH; Sjöberg, F; Thorborg, P | 1 |
Dewar, KM; Lima, L; Reader, TA | 1 |
el-Mahdy, SA | 1 |
Folts, JD; Noble, MI; Torr, S | 1 |
Cowen, PJ; da Roza Davis, JM; Fernando, AI; Sharpley, AL; Solomon, RA | 1 |
Glowinski, J; Godbout, R; Mantz, J; Tassin, JP; Thierry, AM | 1 |
Blandini, F; Cerutti, G; Facchinetti, F; Granella, F; Manzoni, GC; Nappi, G; Ruiz, L; Sandrini, G | 1 |
Bouysset, F; Laubie, M; Schmitt, H; Vayssettes-Courchay, C; Verbeuren, TJ | 1 |
Brammer, MJ; Campbell, IC; Corn, TH; Stephenson, JD; Twist, EC | 1 |
Loo, H; Sechter, D | 1 |
Cohen, ML; Mann, JJ; McBride, PA; Nimchinsky, E | 1 |
Hietala, J; Koulu, M; Lappalainen, J; Syvälahti, E | 1 |
Bersani, G; Ciani, N; Grispini, A; Marini, S; Pasini, A; Valducci, M | 1 |
Baudrie, V; Chaouloff, F; Laude, D | 1 |
Bendotti, C; Neill, JC; Samanin, R | 1 |
Abe, Y; Iwao, H; Kiyomoto, H; Shoji, T; Tamaki, T | 1 |
Netter, P; Rammsayer, T | 3 |
Geyer, MA; Tapson, GS; Wing, LL | 1 |
Dreteler, GH; Saxena, PR; Wouters, W | 1 |
Carlsson, S; Hoffmann, P; Skarphedinsson, JO; Thorén, P | 1 |
Backus, LI; Grahame-Smith, DG; Sharp, T | 1 |
Demetrikopoulos, MK; Flaherty, CF; Grigson, PS; Krauss, KL; Rowan, GA; Weaver, MS | 1 |
Blöchl-Daum, B; Brenner, B; Eichler, HG; Kyrle, PA; Lechner, K; Schneider, B; Speiser, W; Wagner, B | 1 |
Bjorvatn, B; Ursin, R | 1 |
Jackson, DA; White, SR | 1 |
Cowen, PJ; Gartside, SE | 1 |
Coker, SJ; Ellis, AM | 1 |
Ball, SG; Robertson, JI; Stott, DJ | 1 |
Ball, SG; Hosie, J; Robertson, JI; Stott, DJ | 1 |
Ishikawa, K; Kameyama, T; Nabeshima, T; Yamaguchi, K; Yoshida, S | 1 |
Gradin, K; Hedner, T; Persson, B; Pettersson, A | 3 |
Cohen, ML; Kurz, KD; Schenck, KW | 1 |
Ramage, AG | 2 |
Hedner, T; Persson, B | 1 |
Reneman, RS; van der Starre, PJ | 1 |
de Chaffoy de Courcelles, D; Eens, A; Gommeren, W; Janssen, PA; Leysen, JE; Stoof, JC | 1 |
Blauw, GJ; Chang, PC; van Brummelen, P; van Zwieten, PA; Vermeij, P | 1 |
Goossens, JG; van Wauwe, JP | 1 |
Gelders, YG | 1 |
de Bruyckere, K; Janssen, PF; Leysen, JE; Schotte, A | 1 |
Huet, PM; Mastaï, R; Rocheleau, B | 1 |
Cooper, SJ; Neill, JC | 1 |
Lund, N; Thorborg, P | 1 |
Bruinvels, J; Ketelaars, CE | 1 |
Itoh, K; Kameyama, T; Kawashima, K; Nabeshima, T | 1 |
Allal, G; Crichlow, EC; Ruckebusch, Y | 1 |
Argenio, GF; Bernini, GP; Del Corso, C; Franchi, F; Luisi, M; Sgrò, M; Vivaldi, MS | 1 |
Barber, A; Harting, J; Wolf, HP | 1 |
Heykants, J; Lenoir, H; Timmerman, P; Woestenborghs, R | 1 |
Bloomquist, WL; Cohen, ML; Fuller, RW; Snoddy, HD | 1 |
Adam, K; Oswald, I | 1 |
Molcan, J; Náhunek, K; Svestka, J; Vinar, O; Zapletálek, M | 1 |
Dugovic, C; Leysen, JE; Wauquier, A | 1 |
Colpaert, FC; Koek, W; Lategan, A | 1 |
Audi, EA; de-Oliveira, CE; Graeff, FG | 1 |
Dugovic, C; Janssen, PF; Leysen, JE; Wauquier, A | 1 |
Arnt, J; Hyttel, J | 1 |
Amoroso, S; Annunziato, L; Basile, V; Canzoniero, L; Di Renzo, G; Fatatis, A; Taglialatela, M | 1 |
Dugovic, C; Janssen, PA; Leysen, JE; Marrannes, R; Wauquier, A | 1 |
Grenhoff, J; Svensson, TH; Ugedo, L | 1 |
Kameyama, T; Kawashima, K; Nabeshima, T | 1 |
Chau, NP; Levenson, J; Pithois-Merli, I; Simon, AC | 1 |
Bennett, GW; Fone, KC; Johnson, JV; Marsden, CA | 1 |
Barone, D; Bendotti, C; Caccia, S; Garattini, S; Mennini, T; Samanin, R | 1 |
Hatano, K; Hatazawa, J; Ido, T; Ishiwata, K; Itoh, M; Kawashima, K | 1 |
Altamura, AC; Colacurcio, F; Marini, S | 1 |
Grenhoff, J; Svensson, TH; Tung, CS | 1 |
Kumasaka, Y; Ueki, S; Yamamoto, T | 1 |
Alling, C; Hansson, E; Simonsson, P | 1 |
Furukawa, H; Ishikawa, K; Kameyama, T; Nabeshima, T; Yamaguchi, K | 4 |
Gommeren, W; Janssen, PF; Laduron, PM; Leysen, JE; Van Gompel, P; Wynants, J | 1 |
Colpaert, FC; Janssen, PA; Meert, TF; Niemegeers, CJ | 1 |
Batink, HD; Boddeke, E; Doods, HN; Hugtenburg, JG; Korstanje, C; Sprenkels, R; Thoolen, MJ; Van Zwieten, PA | 1 |
Gardner, CR | 1 |
Forsman, A; Larsson, M | 1 |
Hedner, T; Persson, B; Pettersson, A | 1 |
Hewson, G; Hill, RG; Hughes, J; Leighton, GE | 1 |
Gommeren, W; Laduron, PM; Leysen, JE; van Gompel, P | 1 |
Dugovic, C; Wauquier, A | 1 |
Facchinetti, F; Genazzani, AR; Marini, S; Martignoni, E; Nappi, G; Petraglia, F; Sandrini, G | 1 |
Gommeren, W; Janssen, PA; Leysen, JE; Van Gompel, P; Woestenborghs, R | 1 |
Glennard, R; Idzikowski, C; Mills, FJ | 1 |
Delwaide, PJ; Maertens de Noordhout, A | 1 |
Barone, JA; Bierman, RH; Colaizzi, JL; Cornish, JW; Drake, ND; Hsuan, A | 1 |
Byrne, JH; Ocorr, KA | 1 |
Aghajanian, GK; Rasmussen, K | 1 |
Alfonsi, E; De Rysky, C; Facchinetti, F; Marini, S; Nappi, G; Sandrini, G | 1 |
Costall, B; Kelly, ME; Naylor, RJ; Tan, CC; Tattersall, FD | 1 |
Jandhyala, BS; Kivlighn, SD | 1 |
Laguzzi, R; Shvaloff, A | 1 |
De Clerck, F; De Ridder, W; Van Gorp, L; Van Nueten, JM | 1 |
Marini, S; Massi, M | 1 |
Bressa, GM; Gregori, S; Marini, S | 1 |
Gelders, Y; Hoppenbrowers, ML; Vanden Bussche, G | 1 |
Frenken, M; Kaumann, AJ | 1 |
Bagdy, G; Hill, J; Murphy, DL; Szemeredi, K; Zukowska-Grojec, Z | 1 |
Janssen, PA | 2 |
Jappay, E; Pranzatelli, MR; Snodgrass, SR | 1 |
Davies, MF; Deisz, RA; Peroutka, SJ; Prince, DA | 1 |
Alling, C; Simonsson, P | 1 |
Davis, M | 1 |
Cowen, PJ; Idzikowski, C; Mills, FJ; Nutt, D | 1 |
Coghlan, JP; Denton, DA; Nelson, M; Scoggins, BA; Tresham, JJ; Whitworth, JA | 1 |
Breeding, M; Sanders-Bush, E | 1 |
Ball, SG; Hosie, J; Lowe, GD; Saniabadi, AR; Stott, DJ | 1 |
Gibb, JW; Hanson, GR; Johnson, M | 1 |
Arriaga, F; Lara, E; Largo, R; Leitao, JN; Paiva, T; Wauquier, A | 1 |
Nomikos, GG; Spyraki, C | 1 |
Fletcher, PJ | 1 |
Smits, J; Struyker Boudier, H; van Dorsten, F | 1 |
Borbély, AA; Tobler, I; Trachsel, L | 1 |
Klieser, E; Strauss, WH | 1 |
Geyer, MA; Tapson, GS | 1 |
Furukawa, H; Hiramatsu, M; Ishizaki, K; Itoh, K; Kasugai, M; Katoh, A; Kawashima, K; Nabeshima, T; Ogawa, S; Yamaguchi, K | 1 |
Griez, E; Lousberg, H; Pols, H | 1 |
Ceulemans, DL; Gelders, YG; Hoppenbrouwers, ML; Reyntjens, AJ | 1 |
Ciccocioppo, R; Massi, M; Panocka, I; Pompei, P | 1 |
Lindström, E; von Knorring, L | 1 |
Jahnová, E | 1 |
Furukawa, H; Hasegawa, T; Kitaichi, K; Nabeshima, T; Yamada, K | 1 |
Bruns, GC; Dage, RC; Hsieh, CP; Sakai, K | 1 |
Furukawa, H; Hasegawa, T; Kitaichi, K; Nabeshima, T; Ogita, K; Yamada, K; Yoneda, Y | 1 |
Fadayel, GM; Schmidt, CJ | 1 |
Araki, H; Ogawa, S; Okuyama, S; Otomo, S | 1 |
Aghajanian, GK; Marek, GJ | 1 |
Dudley, MW; Kehne, JH; Ketteler, HJ; McCloskey, TC; Schmidt, CJ; Sullivan, CK | 1 |
Ashby, CR; Edwards, E; Hampton, E; Wang, RY; Zhang, J | 1 |
Assié, MB; Kleven, MS; Koek, W | 1 |
Carlsson, A; Carlsson, ML; Martin, P; Waters, N | 1 |
Kaisar, M; Naylor, RJ; Tuladhar, BR | 1 |
Beleta, J; Bernabeu, E; Bou, J; Cortijo, J; Domènech, T; Fernández, AG; Martí-Cabrera, M; Morcillo, EJ; Palacios, JM | 1 |
Harvey, JA; Romano, AG; Welsh, SE | 1 |
Adamkiewicz, M; Buczko, W; Malyszko, J; Mysliwiec, M; Pawlak, D; Takada, A | 1 |
Kulkarni, SK; Ninan, I | 1 |
Harvey, JA; Hood, H; Romano, AG; Welsh, SE | 1 |
Gallate, JE; McGregor, IS | 1 |
Alsayegh, L; Backstrom, JR; Berry, SA; Friedman, L; Roth, BL; Sanders-Bush, E; Willins, DL | 1 |
Heron-Maxwell, CL; O'Neill, MF; Shaw, G | 1 |
Naylor, RJ; Tuladhar, BR; Womack, MD | 1 |
Colado, MI; Elliott, JM; Esteban, B; Green, AR; Mechan, AO; O'Shea, E | 1 |
Feuerbach, D; Loetscher, E; Mahé, C; Müller, W; Schoeffter, P; Seiler, MP | 1 |
France, CP; Li, JX; Rice, KC | 1 |
France, CP; Javors, MA; Koek, W; Li, JX; Rice, KC; Unzeitig, A | 1 |
Chaki, S; Fukumoto, K; Iijima, M | 1 |
Amato, D; Carey, RJ; de Souza Silva, MA; Groos, D; Huston, JP; Lauber, AC; Müller, CP; Pum, ME | 1 |
Audia, A; Bhat, KP | 1 |
Baldanzi, G; Bertoni, A; Capello, D; Fresu, LG; Gesu, A; Graziani, A; Massarotti, A; Ruffo, E; Snow, AL; Talmon, M; Tron, GC; Varma, KSS; Velnati, S | 1 |
2 review(s) available for ritanserin and piperidines
Article | Year |
---|---|
Antihypertensive mode of action of ketanserin.
Topics: Adrenergic alpha-Antagonists; Aldosterone; Animals; Antihypertensive Agents; Blood Pressure; Carcinoid Heart Disease; Humans; Ketanserin; Piperidines; Prazosin; Ritanserin | 1987 |
Ritanserin (R 55667) an original thymosthenic.
Topics: Humans; Mental Disorders; Piperidines; Ritanserin; Serotonin Antagonists | 1986 |
33 trial(s) available for ritanserin and piperidines
Article | Year |
---|---|
Ritanserin, a 5-HT2 receptor blocker, as add-on treatment in narcolepsy.
Topics: Adolescent; Adult; Animals; Circadian Rhythm; Double-Blind Method; Histamine H2 Antagonists; Humans; Middle Aged; Narcolepsy; Piperidines; Placebos; Ritanserin; Sleep | 1991 |
Relative efficacy of drugs for the treatment of sleepiness in narcolepsy.
Topics: Adult; Arousal; Benzhydryl Compounds; Central Nervous System Stimulants; Codeine; Dextroamphetamine; Female; Humans; Male; Methylphenidate; Modafinil; Narcolepsy; Pemoline; Piperidines; Protriptyline; Reaction Time; Ritanserin; Sleep Stages; Sodium Oxybate; Viloxazine; Wakefulness | 1991 |
Serotonin function in panic disorder: a double blind placebo controlled study with fluvoxamine and ritanserin.
Topics: Adult; beta-Endorphin; Blood Platelets; Double-Blind Method; Fear; Female; Fluvoxamine; Humans; Hydrocortisone; Hydroxyindoleacetic Acid; Male; Melatonin; Mental Disorders; Methoxyhydroxyphenylglycol; Norepinephrine; Oximes; Panic; Piperidines; Psychiatric Status Rating Scales; Randomized Controlled Trials as Topic; Ritanserin; Serotonin | 1990 |
5-HT2 receptor antagonism in dysthymic disorder: a double-blind placebo-controlled study with ritanserin.
Topics: Adult; Depressive Disorder; Double-Blind Method; Female; Humans; Male; Middle Aged; Personality Inventory; Piperidines; Placebos; Psychiatric Status Rating Scales; Receptors, Serotonin; Ritanserin; Serotonin Antagonists | 1991 |
A dose-response study examining the effects of ritanserin on human slow wave sleep.
Topics: Adolescent; Adult; Diazepam; Dose-Response Relationship, Drug; Double-Blind Method; Electroencephalography; Electromyography; Female; Humans; Male; Piperidines; Ritanserin; Sleep Stages; Sleep, REM | 1991 |
Effects of ritanserin on aversive classical conditioning in humans.
Topics: Adult; Conditioning, Classical; Female; Galvanic Skin Response; Humans; Male; Personality Tests; Piperidines; Receptors, Serotonin; Ritanserin; Serotonin Antagonists | 1991 |
Effect of ritanserin, specific 5HT-2 antagonist, on PRL secretion in normal subjects and in different hyperprolactinaemic conditions.
Topics: Adenoma; Female; Follicular Phase; Humans; Hyperprolactinemia; Piperidines; Pituitary Neoplasms; Postpartum Period; Pregnancy; Prolactin; Ritanserin; Serotonin Antagonists; Single-Blind Method; Sulpiride | 1991 |
Pharmacokinetics of ritanserin in patients undergoing hemodialysis.
Topics: Administration, Oral; Adult; Female; Half-Life; Humans; Kidney Failure, Chronic; Male; Middle Aged; Piperidines; Renal Dialysis; Ritanserin; Uremia | 1991 |
Treatment of neuroleptic induced akathisia with the 5-HT2 antagonist ritanserin.
Topics: Administration, Oral; Adult; Akathisia, Drug-Induced; Antipsychotic Agents; Female; Humans; Male; Piperidines; Psychomotor Agitation; Ritanserin; Serotonin Antagonists | 1990 |
Impaired growth hormone response to insulin-induced hypoglycaemia in obese patients: restoration blocked by ritanserin after fenfluramine administration.
Topics: Adult; Blood Glucose; Female; Fenfluramine; Growth Hormone; Humans; Hypoglycemia; Insulin; Middle Aged; Obesity; Piperidines; Random Allocation; Ritanserin; Serotonin Antagonists; Time Factors | 1990 |
A new 5-HT2 antagonist (ritanserin) in the treatment of chronic headache with depression. A double-blind study vs amitriptyline.
Topics: Adult; Amitriptyline; Chronic Disease; Depression; Double-Blind Method; Female; Headache; Humans; Male; Piperidines; Ritanserin | 1990 |
5-HT2 antagonist ritanserin in neuroleptic-induced parkinsonism: a double-blind comparison with orphenadrine and placebo.
Topics: Adolescent; Adult; Double-Blind Method; Female; Humans; Male; Middle Aged; Orphenadrine; Parkinson Disease, Secondary; Piperidines; Psychiatric Status Rating Scales; Ritanserin; Serotonin Antagonists | 1990 |
Effect of ritanserin, a 5-hydroxytryptamine2-receptor antagonist, on platelet function and thrombin generation at the site of plug formation in vivo.
Topics: Adult; beta-Thromboglobulin; Bleeding Time; Blood Platelets; Double-Blind Method; Fibrinopeptide A; Humans; Piperidines; Platelet Aggregation; Platelet Aggregation Inhibitors; Ritanserin; Serotonin Antagonists; Thrombin; Thromboxane B2 | 1990 |
Does acute serotonergic type-2 antagonism reduce blood pressure? Comparative effects of single doses of ritanserin and ketanserin in essential hypertension.
Topics: Adult; Affect; Aged; Blood Pressure; Female; Heart Rate; Humans; Hypertension; Ketanserin; Male; Middle Aged; Piperidines; Receptors, Serotonin; Ritanserin | 1987 |
Experience with ketanserin and ritanserin in hypertensive patients.
Topics: Antihypertensive Agents; Blood Pressure; Clinical Trials as Topic; Double-Blind Method; Female; Humans; Hypertension; Ketanserin; Male; Middle Aged; Piperidines; Ritanserin | 1988 |
The alpha-adrenergic receptor blocking effect of ketanserin and the interaction between alpha-adrenergic and S2-serotonergic receptor blockade.
Topics: Adrenergic alpha-Antagonists; Blood Pressure; Droperidol; Female; Humans; Ketanserin; Male; Middle Aged; Phentolamine; Phenylephrine; Piperidines; Receptors, Adrenergic, alpha; Receptors, Serotonin; Ritanserin | 1988 |
Thymosthenic agents, a novel approach in the treatment of schizophrenia.
Topics: Brain; Butyrophenones; Humans; Isoxazoles; Piperidines; Pyrimidinones; Randomized Controlled Trials as Topic; Receptors, Serotonin; Risperidone; Ritanserin; Schizophrenia; Schizophrenic Psychology; Serotonin Antagonists | 1989 |
Serotoninergic effects on sensory and motor responses in extraverts and introverts.
Topics: Adult; Arousal; Extraversion, Psychological; Flicker Fusion; Fluoxetine; Humans; Introversion, Psychological; Male; Piperidines; Psychomotor Performance; Reaction Time; Ritanserin; Serotonin | 1989 |
Serotonin-influencing drugs in the treatment of panic disorder.
Topics: Adolescent; Adult; Aged; Agoraphobia; Brain; Clinical Trials as Topic; Fear; Female; Fluvoxamine; Humans; Male; Middle Aged; Oximes; Panic; Phobic Disorders; Piperidines; Psychological Tests; Random Allocation; Receptors, Serotonin; Ritanserin | 1989 |
Comparative haemodynamic effects of ketanserin and ritanserin in the proximal and distal upper limb circulations of hypertensive patients.
Topics: Arm; Blood Pressure; Brachial Artery; Double-Blind Method; Hand; Humans; Hypertension; Ketanserin; Middle Aged; Piperidines; Regional Blood Flow; Rheology; Ritanserin; Serotonin Antagonists; Vascular Resistance | 1989 |
Ritanserin versus lorazepam: a double-blind, cross-over study of reaction times in healthy volunteers.
Topics: Acoustic Stimulation; Adult; Double-Blind Method; Female; Hemodynamics; Histamine H2 Antagonists; Humans; Lorazepam; Male; Photic Stimulation; Piperidines; Random Allocation; Reaction Time; Ritanserin | 1989 |
Chronic 5-HT2-receptor blockade by ritanserin does not reduce blood pressure in patients with essential hypertension.
Topics: Aged; Clinical Trials as Topic; Double-Blind Method; Female; Histamine H2 Antagonists; Humans; Hypertension; Ketanserin; Male; Middle Aged; Piperidines; Ritanserin; Time Factors | 1987 |
5-Hydroxytryptamine-2 antagonist increases human slow wave sleep.
Topics: Adult; Double-Blind Method; Humans; Male; Piperidines; Reaction Time; Ritanserin; Serotonin; Serotonin Antagonists; Sleep; Sleep Stages; Stimulation, Chemical | 1986 |
Safety evaluation of ritanserin--an investigational serotonin antagonist.
Topics: Adolescent; Adult; Blood Pressure; Dose-Response Relationship, Drug; Double-Blind Method; Drug Evaluation; Humans; Male; Piperidines; Ritanserin; Serotonin Antagonists | 1986 |
Evidence for serotonin-S2 receptor involvement in analgesia in humans.
Topics: Adult; Analgesia; Double-Blind Method; Humans; Male; Naloxone; Piperidines; Receptors, Serotonin; Reflex; Ritanserin; Sensory Thresholds; Serotonin Antagonists | 1986 |
Serotonin S2 receptors blockage and generalized anxiety disorders. A double-blind study on ritanserin and lorazepam.
Topics: Adolescent; Adult; Aged; Anxiety Disorders; Double-Blind Method; Female; Humans; Lorazepam; Male; Piperidines; Random Allocation; Receptors, Serotonin; Ritanserin; Serotonin Antagonists | 1987 |
Does ritanserin, a potent serotonin-S2 antagonist, restore energetic functions during the night?
Topics: Clinical Trials as Topic; Depressive Disorder; Humans; Piperidines; Ritanserin; Schizophrenia; Serotonin Antagonists; Sleep | 1987 |
The relevance of pharmacological studies to sleep research in psychiatry.
Topics: Clinical Trials as Topic; Humans; Mental Disorders; Piperidines; Ritanserin; Serotonin Antagonists; Sleep | 1988 |
The effects of the 5 HT2 antagonist ritanserin on blood pressure and serotonin-induced platelet aggregation in patients with untreated essential hypertension.
Topics: Aged; Blood Pressure; Double-Blind Method; Electrocardiography; Female; Forearm; Heart Rate; Humans; Hypertension; Male; Middle Aged; Piperidines; Platelet Aggregation; Random Allocation; Regional Blood Flow; Ritanserin; Serotonin; Serotonin Antagonists | 1988 |
Effects of ritanserin on sleep disturbances of dysthymic patients.
Topics: Adult; Depressive Disorder; Female; Humans; Male; Middle Aged; Piperidines; Psychiatric Status Rating Scales; Ritanserin; Serotonin Antagonists; Sleep Stages; Sleep Wake Disorders; Sleep, REM | 1988 |
Effects of changes in brain 5-HT activity on indicators of cortical arousal.
Topics: Adult; Arousal; Attention; Cerebral Cortex; Double-Blind Method; Fluoxetine; Humans; Male; Piperidines; Receptors, Serotonin; Ritanserin; Serotonin; Serotonin Antagonists | 1988 |
The influence of ritanserin, a serotonin antagonist, in anxiety disorders: a double-blind placebo-controlled study versus lorazepam.
Topics: Adult; Anxiety Disorders; Clinical Trials as Topic; Double-Blind Method; Female; Humans; Lorazepam; Male; Piperidines; Psychological Tests; Ritanserin; Serotonin Antagonists | 1985 |
Symptoms in schizophrenic syndromes in relation to age, sex, duration of illness and number of previous hospitalizations.
Topics: Adult; Age Factors; Age of Onset; Aged; Antipsychotic Agents; Female; Haloperidol; Hospitalization; Hospitals, Psychiatric; Humans; Isoxazoles; Male; Middle Aged; Patient Admission; Piperidines; Risperidone; Ritanserin; Schizophrenia; Schizophrenic Psychology; Sex Factors | 1994 |
165 other study(ies) available for ritanserin and piperidines
Article | Year |
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Pharmacological profile of the new potent neuroleptic ocaperidone (R 79,598).
Topics: Animals; Antiemetics; Antipsychotic Agents; Apomorphine; Behavior, Animal; Body Temperature; Dogs; Dopamine Agents; Dopamine Antagonists; Eating; Female; Haloperidol; Isoxazoles; Lethal Dose 50; Locomotion; Male; Mice; Motor Activity; Muscles; Neurotransmitter Agents; Piperidines; Posture; Pyrimidinones; Rats; Rats, Inbred Strains; Risperidone; Ritanserin; Serotonin; Serotonin Antagonists; Synaptic Transmission | 1992 |
5-HT2 receptor antagonists reverse amphetamine-induced slowing of dopaminergic neurons by interfering with stimulated dopamine synthesis.
Topics: Action Potentials; Amphetamines; Animals; Apomorphine; Carbidopa; Dopamine; Dopamine Antagonists; Fenclonine; Levodopa; Male; Neurons; Piperidines; Rats; Rats, Inbred Strains; Ritanserin | 1992 |
Action of serotonin in the medial prefrontal cortex: mediation by serotonin3-like receptors.
Topics: Analysis of Variance; Animals; Benzamides; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Frontal Lobe; Indoles; Injections, Intravenous; Iontophoresis; Male; Metergoline; Pindolol; Piperidines; Rats; Rats, Inbred Strains; Receptors, Serotonin; Ritanserin; Serotonin; Serotonin Antagonists; Spiperone; Tropisetron | 1992 |
[Persistence of the control of the fluctuations of heart rate in the anesthetized and pithed adult rat. Effect of enteraminergic drugs].
Topics: Anesthesia; Animals; Decerebrate State; Depression, Chemical; Dose-Response Relationship, Drug; Ether; Female; Granisetron; Heart Rate; Indazoles; Male; Piperidines; Rats; Ritanserin; Serotonin Antagonists | 1991 |
Ritanserin decreases alcohol intake in chronic alcoholics.
Topics: Adult; Affect; Alcoholism; Humans; Male; Middle Aged; Piperidines; Ritanserin; Serotonin Antagonists; Sleep | 1991 |
Effects of the 5-HT2 receptor antagonist, ritanserin, on biogenic amines in the rat nucleus accumbens.
Topics: Animals; Antipsychotic Agents; Dialysis; Dopamine; Male; Nucleus Accumbens; Piperidines; Rats; Rats, Inbred Strains; Ritanserin; Serotonin; Serotonin Antagonists; Synaptic Transmission | 1991 |
Early life protein malnutrition changes exploration of the elevated plus-maze and reactivity to anxiolytics.
Topics: Animals; Anti-Anxiety Agents; Anxiety; Diazepam; Dose-Response Relationship, Drug; Exploratory Behavior; Male; Piperidines; Propanolamines; Protein-Energy Malnutrition; Pyrimidines; Rats; Rats, Inbred Strains; Ritanserin | 1991 |
5HT2 receptor changes in rat cortex and platelets following chronic ritanserin and clorgyline administration.
Topics: Animals; Blood Platelets; Cerebral Cortex; Clorgyline; Homovanillic Acid; Hydroxyindoleacetic Acid; Ketanserin; Lysergic Acid Diethylamide; Male; Norepinephrine; Piperidines; Propylamines; Rats; Rats, Inbred Strains; Receptors, Serotonin; Ritanserin; Serotonin | 1990 |
The serotonin2 antagonist ritanserin blocks quasi-morphine withdrawal at a time when mianserin is no longer effective.
Topics: 1-Methyl-3-isobutylxanthine; Animals; Conditioning, Operant; Male; Mianserin; Morphine Dependence; Naloxone; Piperidines; Rats; Reinforcement Schedule; Ritanserin; Serotonin Antagonists; Substance Withdrawal Syndrome | 1990 |
Functional interaction between serotonin-S2 and dopamine-D2 neurotransmission as revealed by selective antagonism of hyper-reactivity to tryptamine and apomorphine.
Topics: Animals; Antipsychotic Agents; Apomorphine; Dopamine; Dose-Response Relationship, Drug; Drug Interactions; Haloperidol; Injections, Intravenous; Isoxazoles; Male; Piperidines; Rats; Rats, Inbred Strains; Risperidone; Ritanserin; Seizures; Serotonin; Serotonin Antagonists; Synaptic Transmission; Tryptamines | 1990 |
Chronic 5-HT2 receptor antagonist treatment alters 5-HT1A autoregulatory control of 5-HT release in rat brain in vivo.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Brain Chemistry; Cerebral Cortex; Chromatography, High Pressure Liquid; Hydroxyindoleacetic Acid; Piperidines; Rats; Rats, Inbred Strains; Receptors, Serotonin; Ritanserin; Serotonin Antagonists; Tetrahydronaphthalenes | 1990 |
Cardiovascular and renal actions of AHR-16303B, an antagonist of 5-HT2 receptors and calcium channels, in hypertensive and normotensive rats.
Topics: Administration, Oral; Animals; Blood Pressure; Calcium Channel Blockers; Cardiovascular System; Dose-Response Relationship, Drug; Heart Rate; Hypertension; Injections, Intravenous; Kidney; Male; Piperidines; Propiophenones; Rats; Rats, Inbred SHR; Rats, Inbred Strains; Ritanserin; Serotonin Antagonists; Verapamil | 1991 |
[Study by the intracerebral microdialysis method of the effects of atypical neuroleptics and anxiolytics on striatal release and metabolism of dopamine in awake rats].
Topics: Animals; Anti-Anxiety Agents; Antipsychotic Agents; Brain Chemistry; Buspirone; Corpus Striatum; Dialysis; Dopamine; In Vitro Techniques; Isoxazoles; Male; Methoxydimethyltryptamines; Piperidines; Rats; Rats, Inbred Strains; Risperidone; Ritanserin; Sulpiride; Wakefulness | 1991 |
Blockade of 5-HT2 receptors protects against impairment of working memory following transient forebrain ischemia in the rat.
Topics: Animals; Cinanserin; Ischemic Attack, Transient; Male; Memory; Piperidines; Rats; Rats, Inbred Strains; Ritanserin; Serotonin Antagonists | 1991 |
DOI-induced inhibition of copulatory behavior in male rats: reversal by 5-HT2 antagonists.
Topics: Amphetamines; Animals; Copulation; Ejaculation; Female; Ketanserin; Male; Piperidines; Rats; Rats, Inbred Strains; Ritanserin; Serotonin Antagonists; Tranquilizing Agents | 1991 |
Enhanced serotonergic transmission stimulates oxytocin secretion in conscious male rats.
Topics: Animals; Male; Oxytocin; Piperazines; Piperidines; Rats; Rats, Inbred Strains; Receptors, Serotonin; Ritanserin; Serotonin; Synaptic Transmission | 1991 |
Inhibitory effect of ritanserin on the 5-hydroxytryptophan-mediated cortisol, ACTH and prolactin secretion in humans.
Topics: 5-Hydroxytryptophan; Adrenocorticotropic Hormone; Adult; Humans; Hydrocortisone; Male; Piperidines; Prolactin; Ritanserin; Serotonin Antagonists | 1991 |
5-HT2 antagonists stereoselectively prevent the neurotoxicity of 3,4-methylenedioxymethamphetamine by blocking the acute stimulation of dopamine synthesis: reversal by L-dopa.
Topics: 3,4-Dihydroxyphenylacetic Acid; 3,4-Methylenedioxyamphetamine; Animals; Anti-Arrhythmia Agents; Brain; Corpus Striatum; Dopamine; Dose-Response Relationship, Drug; Drug Synergism; Haloperidol; Homovanillic Acid; Levodopa; Male; Nomifensine; Piperidines; Rats; Rats, Inbred Strains; Ritanserin; Serotonin Antagonists; Stereoisomerism; Time Factors | 1991 |
Hyperglycemic properties of serotonin receptor antagonists.
Topics: Animals; Blood Glucose; Male; Metergoline; Methysergide; Mice; Piperidines; Receptors, Serotonin; Ritanserin; Serotonin Antagonists; Tropanes | 1991 |
Naloxone and serotonin receptor subtype antagonists: interactive effects upon deprivation-induced intake.
Topics: Animals; Drug Interactions; Feeding Behavior; Food Deprivation; Indoles; Ketanserin; Male; Methysergide; Naloxone; Piperidines; Rats; Rats, Inbred Strains; Ritanserin; Serotonin Antagonists; Tropisetron | 1991 |
Effect of chronic ritanserin or clorgyline on amine and metabolite levels in rat frontal cortex.
Topics: Amines; Animals; Cerebral Cortex; Clorgyline; In Vitro Techniques; Male; Monoamine Oxidase; Piperidines; Rats; Rats, Inbred Strains; Receptors, Serotonin; Ritanserin; Serotonin Antagonists | 1991 |
Naphthosultam derivatives: a new class of potent and selective 5-HT2 antagonists.
Topics: Animals; Behavior, Animal; Chemical Phenomena; Chemistry; Cyclic S-Oxides; Male; Mescaline; Mice; Molecular Structure; Naphthalenes; Piperidines; Rats; Rats, Inbred Strains; Receptors, Serotonin; Ritanserin; Serotonin Antagonists; Structure-Activity Relationship; Thiazoles | 1991 |
Role of 5-HT receptors in the effect of d-fenfluramine on gastric emptying and feeding behaviour as examined in the runway test.
Topics: Animals; Behavior, Animal; Feeding Behavior; Fenfluramine; Gastric Emptying; Male; Metergoline; Piperidines; Proglumide; Rats; Receptors, Serotonin; Ritanserin; Serotonin Antagonists | 1991 |
Atypical neuroleptics suppress dopaminergic behavioral supersensitivity.
Topics: Animals; Antipsychotic Agents; Apomorphine; Behavior, Animal; Clozapine; Cyproheptadine; Haloperidol; Male; Piperidines; Rats; Rats, Inbred Strains; Receptors, Dopamine; Ritanserin; Serotonin Antagonists; Sulpiride; Thioridazine | 1990 |
Treatment of insomnia with ritanserin.
Topics: Adult; Female; Humans; Piperidines; Ritanserin; Serotonin Antagonists; Sleep Initiation and Maintenance Disorders | 1990 |
Decreased reactivity to anxiolytics caused by early protein malnutrition in rats.
Topics: Animals; Anti-Anxiety Agents; Body Weight; Diazepam; Diet; Dose-Response Relationship, Drug; Hypertonic Solutions; Lactation; Male; Piperidines; Propanolamines; Protein-Energy Malnutrition; Pyrimidines; Rats; Rats, Inbred Strains; Ritanserin | 1990 |
Effect of serotoninergic drugs on stress-induced hyperthermia (SIH) in mice.
Topics: 5,7-Dihydroxytryptamine; 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Anti-Anxiety Agents; Body Temperature Regulation; Buspirone; Diazepam; Ergolines; Fenclonine; Fever; Flumazenil; Imidazoles; Male; Mice; Ondansetron; Piperazines; Piperidines; Ritanserin; Serotonin; Serotonin Antagonists; Stress, Psychological; Tetrahydronaphthalenes | 1990 |
Effects of ketanserin tartrate on 3-hydroxy, 3-methylglutaryl coenzyme A reductase activity in cultured human skin fibroblasts.
Topics: Adrenergic alpha-Antagonists; Cells, Cultured; Fibroblasts; Humans; Hydroxymethylglutaryl CoA Reductases; Ketanserin; Piperidines; Prazosin; Ritanserin; Serotonin Antagonists | 1990 |
Ritanserin decreases portal pressure in conscious and unrestrained cirrhotic rats.
Topics: Animals; Consciousness; Depression, Chemical; Hemodynamics; Hypertension, Portal; Liver Cirrhosis, Experimental; Male; Piperidines; Rats; Rats, Inbred Strains; Ritanserin; Serotonin Antagonists; Splanchnic Circulation | 1990 |
Serotonin (5-HT) induces IPSPs in pyramidal layer cells of rat piriform cortex: evidence for the involvement of a 5-HT2-activated interneuron.
Topics: Animals; Cerebral Cortex; Evoked Potentials; In Vitro Techniques; Interneurons; Male; Neural Inhibition; Piperidines; Rats; Rats, Inbred Strains; Ritanserin; Serotonin; Spiperone | 1990 |
Ritanserin, a 5-HT2 receptor antagonist, does not modify ECT-induced prolactin release.
Topics: Aged; Depressive Disorder; Electroconvulsive Therapy; Female; Humans; Middle Aged; Piperidines; Prolactin; Ritanserin; Serotonin Antagonists | 1990 |
5-HT1C receptors in the serotonergic control of periaqueductal gray induced aversion in rats.
Topics: Amphetamines; Animals; Cyproheptadine; Indoles; Ketanserin; Male; Periaqueductal Gray; Piperazines; Piperidines; Rats; Rats, Inbred Strains; Receptors, Serotonin; Reinforcement, Psychology; Ritanserin; Serotonin; Serotonin Antagonists | 1990 |
Do imipramine and dihydroergosine possess two components--one stimulating 5-HT1 and the other inhibiting 5-HT2 receptors?
Topics: Animals; Brain; Ergotamines; Imipramine; Male; Mice; Mice, Inbred CBA; Motor Activity; Piperidines; Propranolol; Radioligand Assay; Rats; Rats, Inbred Strains; Ritanserin; Serotonin Antagonists; Syndrome | 1990 |
Effect of hyperoxemia and ritanserin on skeletal muscle microflow.
Topics: Animals; Arteries; Blood Flow Velocity; Capillaries; Hydrogen; Lasers; Muscles; Oxygen; Piperidines; Rabbits; Ritanserin; Serotonin Antagonists | 1990 |
[3H]ketanserin binds to non-5-HT2 sites in rabbit cerebral cortex and neostriatum.
Topics: Animals; Binding, Competitive; Caudate Nucleus; Cell Membrane; Cerebral Cortex; Corpus Striatum; Frontal Lobe; Ketanserin; Kinetics; Male; Methysergide; Mianserin; Piperidines; Putamen; Rabbits; Receptors, Serotonin; Ritanserin; Serotonin; Serotonin Antagonists | 1990 |
5-Hydroxytryptamine (serotonin) enhances ventricular arrhythmias induced by acute coronary artery ligation in rats.
Topics: Animals; Arrhythmias, Cardiac; Coronary Vessels; Dose-Response Relationship, Drug; Heart Ventricles; Ligation; Male; Piperidines; Rats; Rats, Inbred Strains; Receptors, Serotonin; Ritanserin; Serotonin; Serotonin Antagonists | 1990 |
Inhibition of acute platelet thrombosis formation in stenosed canine coronary arteries by specific serotonin 5HT2 receptor antagonist ritanserin.
Topics: Animals; Coronary Disease; Coronary Thrombosis; Dogs; Dose-Response Relationship, Drug; Epinephrine; Female; Male; Piperidines; Platelet Aggregation; Platelet Aggregation Inhibitors; Receptors, Serotonin; Ritanserin; Serotonin Antagonists | 1990 |
Dose-related effects of selective 5-HT2 receptor antagonists on slow wave sleep in humans.
Topics: Adult; Dose-Response Relationship, Drug; Electroencephalography; Female; Humans; Male; Piperidines; Quinolines; Receptors, Serotonin; Ritanserin; Serotonin Antagonists; Sleep | 1990 |
Inhibition of spontaneous and evoked unit activity in the rat medial prefrontal cortex by mesencephalic raphe nuclei.
Topics: 5,7-Dihydroxytryptamine; Animals; Brain; Cerebral Cortex; Electric Stimulation; Evoked Potentials; Ketanserin; Male; Membrane Potentials; Neurons; Piperidines; Raphe Nuclei; Rats; Rats, Inbred Strains; Ritanserin; Serotonin | 1990 |
The cardiovascular effects of quipazine are mediated by peripheral 5-HT2 and 5-HT3 receptors in anaesthetized rats.
Topics: Amidines; Anesthesia; Animals; Blood Pressure; Carotid Body; Denervation; Heart Rate; Hemodynamics; Hexamethonium Compounds; In Vitro Techniques; Indoles; Lung; Male; Myocardium; Piperidines; Prazosin; Pressoreceptors; Propanolamines; Quipazine; Rats; Rats, Inbred Strains; Receptors, Serotonin; Renin-Angiotensin System; Ritanserin; Sympathetic Nervous System; Thiophenes; Tropisetron; Vagotomy | 1990 |
The effect of chronic ritanserin and clorgyline administration on 5-HT2 receptor linked inositol phospholipid hydrolysis.
Topics: Animals; Cerebral Cortex; Clorgyline; Hydrolysis; Phosphatidylinositols; Piperidines; Rats; Rats, Inbred Strains; Receptors, Serotonin; Ritanserin; Serotonin; Serotonin Antagonists | 1990 |
[5 HT2 antagonists and carpipramine].
Topics: Anti-Anxiety Agents; Benzodiazepines; Cerebral Cortex; Dibenzazepines; Humans; Piperidines; Psychotropic Drugs; Receptors, Serotonin; Ritanserin; Serotonin Antagonists; Sleep | 1990 |
Inhibition of serotonin-amplified human platelet aggregation by ketanserin, ritanserin, and the ergoline 5HT2 receptor antagonists-LY53857, sergolexole, and LY237733.
Topics: Adult; Ergolines; Female; Humans; Ketanserin; Lysergic Acid; Male; Piperidines; Platelet Aggregation; Platelet Aggregation Inhibitors; Receptors, Serotonin; Ritanserin; Serotonin; Serotonin Antagonists | 1990 |
Neurochemical effects of chronic co-administration of ritanserin and haloperidol: comparison with clozapine effects.
Topics: Animals; Clozapine; Dopamine; Drug Combinations; Haloperidol; Male; Nucleus Accumbens; Piperidines; Rats; Rats, Inbred Strains; Ritanserin; Serotonin; Substantia Nigra; Time Factors | 1990 |
Effects of the 5-HT1C/5-5-HT2 receptor agonists DOI and alpha-methyl-5-HT on plasma glucose and insulin levels in the rat.
Topics: Amphetamines; Animals; Blood Glucose; Catecholamines; Ergolines; Hyperglycemia; Insulin; Male; Piperazines; Piperidines; Rats; Rats, Inbred Strains; Receptors, Serotonin; Ritanserin; Serotonin | 1990 |
Studies on the role of 5-HT receptors in satiation and the effect of d-fenfluramine in the runway test.
Topics: Amidines; Animals; Feeding Behavior; Fenfluramine; Male; Metergoline; Piperidines; Rats; Receptors, Serotonin; Ritanserin; Satiation; Serotonin Antagonists | 1990 |
Renal vasodilatation induced by DOI, a 5-HT2 receptor agonist, in the canine kidney.
Topics: Amphetamines; Animals; Blood Pressure; Creatinine; Dogs; Female; Glomerular Filtration Rate; Male; Piperidines; Receptors, Serotonin; Renal Circulation; Ritanserin; Urodynamics; Vasodilation | 1990 |
Personality related differences in response to 5-HT uptake inhibition.
Topics: Adult; Analysis of Variance; Choice Behavior; Double-Blind Method; Emotions; Flicker Fusion; Fluoxetine; Humans; Male; Personality; Piperidines; Reaction Time; Reference Values; Ritanserin; Serotonin Antagonists | 1990 |
5HT-2 mediation of acute behavioral effects of hallucinogens in rats.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Amphetamines; Animals; Behavior, Animal; DOM 2,5-Dimethoxy-4-Methylamphetamine; Dose-Response Relationship, Drug; Hallucinogens; Ketanserin; Male; Mescaline; Piperidines; Quipazine; Rats; Rats, Inbred Strains; Ritanserin; Serotonin; Tetrahydronaphthalenes | 1990 |
Comparison of the cardiovascular effects of the 5-HT1A receptor agonist flesinoxan with that of 8-OH-DPAT in the rat.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Anesthesia; Animals; Antihypertensive Agents; Atropine; Blood Pressure; Decerebrate State; Heart Rate; Hemodynamics; Imidazoles; In Vitro Techniques; Male; Naphthalenes; Ondansetron; Piperazines; Piperidines; Rats; Rats, Inbred SHR; Rats, Inbred Strains; Receptors, Serotonin; Ritanserin; Serotonin Antagonists; Tetrahydronaphthalenes | 1990 |
Role of different serotonergic receptors in the long-lasting blood pressure depression following muscle stimulation in the spontaneously hypertensive rat.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Blood Pressure; Electric Stimulation; Heart Rate; Indoles; Male; Methiothepin; Muscles; Piperidines; Rats; Rats, Inbred SHR; Rats, Inbred Strains; Receptors, Serotonin; Ritanserin; Serotonin Antagonists; Tetrahydronaphthalenes; Time Factors; Tropisetron | 1990 |
Behavioural evidence for a functional interaction between central 5-HT2 and 5-HT1A receptors.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Apomorphine; Behavior, Animal; Central Nervous System; Dose-Response Relationship, Drug; Haloperidol; Ketanserin; Male; Methoxydimethyltryptamines; Piperidines; Prazosin; Pyrimidines; Quinolines; Rats; Rats, Inbred Strains; Receptors, Serotonin; Ritanserin; Serotonin; Stereotyped Behavior; Tetrahydronaphthalenes | 1990 |
Effect of serotonergic drugs on negative contrast in consummatory behavior.
Topics: Animals; Buspirone; Chlordiazepoxide; Cyproheptadine; Dose-Response Relationship, Drug; Ethanol; Feeding Behavior; Fenclonine; Injections, Intraperitoneal; Injections, Subcutaneous; Ketanserin; Male; Midazolam; Nucleus Accumbens; Piperidines; Pyrimidines; Rats; Rats, Inbred Strains; Ritanserin; Serotonin; Serotonin Antagonists | 1990 |
Effects of zimeldine, a selective 5-HT reuptake inhibitor, combined with ritanserin, a selective 5-HT2 antagonist, on waking and sleep stages in rats.
Topics: Animals; Arousal; Brain; Electroencephalography; Male; Piperidines; Rats; Rats, Inbred Strains; Reaction Time; Receptors, Serotonin; Ritanserin; Serotonin; Serotonin Antagonists; Sleep Stages; Sleep, REM; Wakefulness; Zimeldine | 1990 |
Receptor subtypes mediating facilitation by serotonin of excitability of spinal motoneurons.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Amphetamines; Animals; In Vitro Techniques; Injections, Intravenous; Iontophoresis; Ketanserin; Male; Methysergide; Microelectrodes; Motor Neurons; Piperidines; Prazosin; Quipazine; Rats; Rats, Inbred Strains; Receptors, Serotonin; Ritanserin; Serotonin; Serotonin Antagonists; Spinal Cord; Tetrahydronaphthalenes | 1990 |
Mediation of ACTH and prolactin responses to 5-HTP by 5-HT2 receptors.
Topics: 5-Hydroxytryptophan; Adrenocorticotropic Hormone; Animals; Dose-Response Relationship, Drug; Ketanserin; Male; Metergoline; Piperidines; Prolactin; Rats; Rats, Inbred Strains; Receptors, Serotonin; Ritanserin; Serotonin Antagonists; Spiperone | 1990 |
Ketanserin and ritanserin can reduce reperfusion-induced but not ischaemia-induced arrhythmias in anaesthetised rats.
Topics: Animals; Anti-Arrhythmia Agents; Arrhythmias, Cardiac; Coronary Vessels; Female; Guinea Pigs; Ketanserin; Male; Piperidines; Rats; Rats, Inbred Strains; Ritanserin; Serotonin Antagonists | 1987 |
Phencyclidine-induced head-weaving and head-twitch through interaction with 5-HT1 and 5-HT2 receptors in reserpinized rats.
Topics: Animals; Brain; Hydroxyindoleacetic Acid; Imipramine; In Vitro Techniques; Male; Methoxydimethyltryptamines; p-Chloroamphetamine; Phencyclidine; Pindolol; Piperidines; Rats; Rats, Inbred F344; Receptors, Serotonin; Reserpine; Ritanserin; Serotonin; Serotonin Antagonists; Stereotyped Behavior | 1987 |
Antihypertensive effects of ketanserin and ritanserin in the spontaneously hypertensive rat.
Topics: Animals; Antihypertensive Agents; Blood Pressure; Heart Rate; Hypertension; Ketanserin; Male; Phenylephrine; Piperidines; Prazosin; Rats; Rats, Inbred SHR; Receptors, Adrenergic, alpha; Receptors, Serotonin; Ritanserin; Serotonin; Sympathetic Nervous System | 1988 |
5-HT2-receptor antagonists: alpha 1- vs. 5-HT2-receptor blocking properties in blood vessels.
Topics: Adrenergic alpha-Antagonists; Animals; Blood Pressure; Ergolines; Ketanserin; Male; Muscle Contraction; Muscle, Smooth, Vascular; Phentolamine; Piperidines; Pyrimidinones; Rats; Rats, Inbred SHR; Rats, Inbred Strains; Receptors, Adrenergic, alpha; Receptors, Serotonin; Ritanserin; Serotonin Antagonists; Spiperone | 1988 |
Are drugs that act both on serotonin receptors and alpha 1-adrenoceptors more potent hypotensive agents than those that act only on alpha 1-adrenoceptors?
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Blood Pressure; Cats; Cinanserin; Ergolines; Ketanserin; Male; Metergoline; Piperidines; Prazosin; Receptors, Adrenergic, alpha; Receptors, Serotonin; Ritanserin; Serotonin Antagonists; Sympathetic Nervous System; Tetrahydronaphthalenes | 1988 |
Biochemical profile of risperidone, a new antipsychotic.
Topics: Animals; Antipsychotic Agents; Blood Platelets; Cerebral Cortex; Dopamine; Ergolines; Female; Haloperidol; Isoxazoles; Models, Molecular; Norepinephrine; Oxazoles; Phosphatidic Acids; Piperidines; Quinpirole; Radioligand Assay; Rats; Rats, Inbred Strains; Receptors, Adrenergic, alpha; Receptors, Dopamine; Receptors, Serotonin; Risperidone; Ritanserin; X-Ray Diffraction | 1988 |
Arterial and venous effects of serotonin in the forearm of healthy subjects are not age-related.
Topics: Adult; Aged; Aging; Blood Pressure; Forearm; Heart Rate; Humans; Ketanserin; Male; Methoxamine; Middle Aged; Piperidines; Regional Blood Flow; Ritanserin; Serotonin; Serotonin Antagonists | 1989 |
Arabinogalactan- and dextran-induced ear inflammation in mice: differential inhibition by H1-antihistamines, 5-HT-serotonin antagonists and lipoxygenase blockers.
Topics: 4,5-Dihydro-1-(3-(trifluoromethyl)phenyl)-1H-pyrazol-3-amine; Animals; Aprotinin; Astemizole; Benzimidazoles; Benzoquinones; Cinanserin; Cyproheptadine; Dextrans; Galactans; Histamine H1 Antagonists; Kinetics; Lipoxygenase Inhibitors; Male; Metergoline; Mice; Otitis; Piperidines; Pyrazoles; Quinones; Ritanserin; Serotonin Antagonists | 1989 |
Receptor occupancy by ritanserin and risperidone measured using ex vivo autoradiography.
Topics: Animals; Brain; Dopamine Antagonists; Isoxazoles; Male; Oxazoles; Piperidines; Rats; Rats, Inbred Strains; Receptors, Adrenergic, alpha; Receptors, Dopamine; Receptors, Serotonin; Risperidone; Ritanserin; Serotonin Antagonists | 1989 |
Serotonin blockade in conscious, unrestrained cirrhotic dogs with portal hypertension.
Topics: Animals; Blood Pressure; Cardiac Output; Common Bile Duct; Dogs; Female; Heart Rate; Hypertension, Portal; Ligation; Liver Cirrhosis, Biliary; Piperidines; Portal Vein; Ritanserin; Serotonin Antagonists; Vascular Resistance | 1989 |
Evidence that d-fenfluramine anorexia is mediated by 5-HT1 receptors.
Topics: Amidines; Animals; Appetite Depressants; Fenfluramine; Male; Metergoline; Pindolol; Piperidines; Rats; Receptors, Serotonin; Ritanserin; Serotonin Antagonists | 1989 |
Serotonin as a modulator of skeletal muscle oxygenation: effects of ketanserin and ritanserin on oxygen pressure distributions.
Topics: Animals; Ketanserin; Muscles; Oxygen; Oxygen Consumption; Piperidines; Pressure; Rabbits; Ritanserin; Serotonin; Serotonin Antagonists | 1989 |
The anti-conflict effect of cyproheptadine is not mediated by its 5-hydroxytryptamine antagonistic property.
Topics: Animals; Behavior Therapy; Conflict, Psychological; Cyproheptadine; Injections, Intraperitoneal; Male; Physostigmine; Piperidines; Rats; Rats, Inbred Strains; Ritanserin; Scopolamine; Serotonin Antagonists | 1989 |
Effects of 5-HT2 receptor antagonist on cycloheximide-induced amnesia in mice.
Topics: Amnesia; Animals; Cycloheximide; Male; Methysergide; Mice; Piperidines; Receptors, Serotonin; Ritanserin; Scopolamine | 1989 |
Involvement of serotonergic mechanisms in the disruption of ovine duodenal migrating myoelectric complex cycles by duodenal acidification.
Topics: Animals; Dose-Response Relationship, Drug; Duodenum; Ergolines; Gastrointestinal Motility; Humans; Hydrochloric Acid; Intestinal Secretions; Metergoline; Piperidines; Receptors, Serotonin; Ritanserin; Sheep | 1989 |
Effects of fenfluramine and ritanserin on prolactin response to insulin-induced hypoglycemia in obese patients: evidence for failure of the serotoninergic system.
Topics: Adolescent; Adult; Female; Fenfluramine; Humans; Hypoglycemia; Insulin; Middle Aged; Obesity; Piperidines; Prolactin; Ritanserin; Serotonin; Serotonin Antagonists | 1989 |
Antinociceptive effects of the 5-HT2 antagonist ritanserin in rats: evidence for an activation of descending monoaminergic pathways in the spinal cord.
Topics: Animals; Methysergide; Nociceptors; Pain; Piperidines; Rats; Receptors, Serotonin; Ritanserin; Spinal Cord; Yohimbine | 1989 |
Deuterated ritanserin analysis by gas chromatography/mass spectrometry: a sensitive technique to study human ritanserin pharmacokinetics.
Topics: Gas Chromatography-Mass Spectrometry; Humans; Isotope Labeling; Piperidines; Ritanserin; Serotonin Antagonists | 1989 |
Lack of a difference between ketanserin and ritanserin in central vs. peripheral serotonin receptor antagonism.
Topics: Animals; Blood Pressure; Corticosterone; Ketanserin; Male; Piperidines; Quipazine; Rats; Rats, Inbred Strains; Receptors, Serotonin; Ritanserin; Serotonin; Serotonin Antagonists | 1989 |
Effects of repeated ritanserin on middle-aged poor sleepers.
Topics: Attention; Electroencephalography; Female; Humans; Male; Middle Aged; Piperidines; Ritanserin; Serotonin Antagonists; Sleep; Sleep Stages; Sleep Wake Disorders; Substance Withdrawal Syndrome; Wakefulness | 1989 |
Ritanserin in schizophrenic patients.
Topics: Adult; Aged; Dose-Response Relationship, Drug; Humans; Middle Aged; Piperidines; Ritanserin; Schizophrenia; Serotonin Antagonists | 1989 |
Melatonin modulates the sensitivity of 5-hydroxytryptamine-2 receptor-mediated sleep-wakefulness regulation in the rat.
Topics: Animals; Male; Melatonin; Piperidines; Rats; Rats, Inbred Strains; Receptors, Serotonin; Ritanserin; Serotonin; Sleep; Wakefulness | 1989 |
1-5-Hydroxytryptophan-induced flat body posture in the rat: antagonism by ritanserin and potentiation after 5,7-dihydroxytryptamine.
Topics: 5-Hydroxytryptophan; 5,7-Dihydroxytryptamine; Animals; Behavior, Animal; Dihydroxytryptamines; Drug Synergism; Injections, Intraventricular; Male; Neurons; Piperidines; Posture; Rats; Rats, Inbred Strains; Ritanserin | 1989 |
Serotonergic mediation of the anxiolytic effect of intracerebrally injected propranolol measured in the elevated plus-maze.
Topics: Animal Testing Alternatives; Animals; Anxiety; Exploratory Behavior; Injections, Intraventricular; Male; Mesencephalon; Piperidines; Propranolol; Rats; Rats, Inbred Strains; Ritanserin; Serotonin Antagonists | 1989 |
The light-dark cycle modulates the effects of ritanserin on sleep-wakefulness patterns in the rat.
Topics: Animals; Circadian Rhythm; Male; Piperidines; Rats; Rats, Inbred Strains; Receptors, Serotonin; Ritanserin; Serotonin Antagonists; Sleep; Wakefulness | 1989 |
Facilitation of 8-OHDPAT-induced forepaw treading of rats by the 5-HT2 agonist DOI.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Alprenolol; Amphetamines; Animals; Behavior, Animal; Cerebral Cortex; Injections, Subcutaneous; Ketanserin; Male; Naphthalenes; Piperidines; Rats; Rats, Inbred Strains; Receptors, Serotonin; Ritanserin; Tetrahydronaphthalenes | 1989 |
Pharmacological characterization of serotonin receptors involved in the control of prolactin secretion.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Fenfluramine; Indoles; Male; Piperidines; Prolactin; Quipazine; Rats; Rats, Inbred Strains; Receptors, Serotonin; Ritanserin; Tetrahydronaphthalenes | 1989 |
Functional role of 5-HT2 receptors in the regulation of sleep and wakefulness in the rat.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Cinanserin; DOM 2,5-Dimethoxy-4-Methylamphetamine; Dose-Response Relationship, Drug; Indoles; Male; Piperidines; Rats; Rats, Inbred Strains; Receptors, Serotonin; Ritanserin; Sleep; Tetrahydronaphthalenes; Wakefulness | 1989 |
Ritanserin, a 5-HT2 receptor antagonist, activates midbrain dopamine neurons by blocking serotonergic inhibition.
Topics: Action Potentials; Animals; Apomorphine; Fenclonine; Male; Mesencephalon; Neurons; Piperidines; Rats; Rats, Inbred Strains; Receptors, Dopamine; Ritanserin; Serotonin Antagonists; Substantia Nigra | 1989 |
Effect of minaprine on cycloheximide-induced amnesia in mice.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Amnesia; Animals; Avoidance Learning; Cycloheximide; Drug Interactions; Male; Mice; p-Chloroamphetamine; Physostigmine; Piperidines; Pyridazines; Ritanserin; Scopolamine; Tetrahydronaphthalenes | 1989 |
Functional interactions between TRH and 5-hydroxytryptamine (5-HT) and proctolin in rat brain and spinal cord.
Topics: 5,7-Dihydroxytryptamine; Animals; Brain; Cerebral Ventricles; Male; Methoxydimethyltryptamines; Motor Activity; Neuropeptides; Neurotransmitter Agents; Oligopeptides; Pentobarbital; Piperidines; Pyrrolidonecarboxylic Acid; Rats; Rats, Inbred Strains; Receptors, Serotonin; Reference Values; Ritanserin; Sleep; Spinal Cord; Stereotyped Behavior; Thyrotropin-Releasing Hormone; Tryptamines | 1989 |
Evidence that central 5-HT2 receptors do not play an important role in the anorectic activity of D-fenfluramine in the rat.
Topics: Animals; Appetite Depressants; Brain Chemistry; Eating; Fenfluramine; Histamine H2 Antagonists; Male; Metergoline; Norfenfluramine; Piperidines; Rats; Rats, Inbred Strains; Receptors, Serotonin; Ritanserin; Spiperone | 1989 |
D2-dopamine receptor specific brain uptake of carbon-11-labeled YM-09151-2.
Topics: Animals; Antipsychotic Agents; Benzamides; Brain; Carbon Radioisotopes; Cerebellum; Corpus Striatum; Dogs; Male; Piperidines; Radionuclide Imaging; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Dopamine D2; Ritanserin; Serotonin Antagonists; Spiperone; Sulpiride | 1989 |
The 5-HT2 antagonist ritanserin blocks the effect of pre-frontal cortex inactivation on rat A10 dopamine neurons in vivo.
Topics: Animals; Cerebral Cortex; Histamine H2 Antagonists; Neurons; Piperidines; Rats; Rats, Inbred Strains; Receptors, Dopamine; Ritanserin | 1989 |
Behavioral analysis of zopiclone on the basis of their discriminative stimulus properties in the rat.
Topics: Animals; Anti-Anxiety Agents; Azabicyclo Compounds; Behavior, Animal; Benzodiazepines; Bicuculline; Discrimination Learning; Dose-Response Relationship, Drug; Flumazenil; Hypnotics and Sedatives; Male; Muscimol; Naphthyridines; Pentylenetetrazole; Piperazines; Piperidines; Rats; Rats, Inbred WKY; Ritanserin; Serotonin Antagonists; Sulfur Compounds | 1989 |
5-Hydroxytryptamine stimulates the formation of inositol phosphate in astrocytes from different regions of the brain.
Topics: Animals; Astrocytes; Brain; Cyclic AMP; Inositol Phosphates; Ketanserin; Piperidines; Rats; Rats, Inbred Strains; Ritanserin; Serotonin; Stimulation, Chemical; Sugar Phosphates; Tissue Distribution | 1987 |
Potentiation in phencyclidine-induced serotonin-mediated behaviors after intracerebroventricular administration of 5,7-dihydroxytryptamine in rats.
Topics: 5,7-Dihydroxytryptamine; Animals; Behavior, Animal; Biogenic Amines; Brain Chemistry; Dihydroxytryptamines; Drug Synergism; Injections, Intraventricular; Male; Methoxydimethyltryptamines; p-Chloroamphetamine; Phencyclidine; Piperidines; Rats; Rats, Inbred Strains; Receptors, N-Methyl-D-Aspartate; Receptors, Neurotransmitter; Receptors, Phencyclidine; Receptors, Serotonin; Ritanserin | 1987 |
Receptor-binding properties in vitro and in vivo of ritanserin: A very potent and long acting serotonin-S2 antagonist.
Topics: Animals; Binding, Competitive; Biogenic Amines; Brain; Cerebellum; Cerebral Cortex; Corpus Striatum; Female; Guinea Pigs; Haloperidol; Hippocampus; Histamine H2 Antagonists; In Vitro Techniques; Ketanserin; Kinetics; Male; Organ Specificity; Piperidines; Rats; Rats, Inbred Strains; Receptors, Serotonin; Ritanserin; Serotonin Antagonists | 1985 |
Behavioral and 5-HT antagonist effects of ritanserin: a pure and selective antagonist of LSD discrimination in rat.
Topics: 5-Hydroxytryptophan; Animals; Anti-Anxiety Agents; Anxiety; Chlordiazepoxide; Diazepam; Disease Models, Animal; Histamine H2 Antagonists; Humans; Lysergic Acid Diethylamide; Male; Motor Activity; Piperidines; Pyrimidines; Rats; Rats, Inbred Strains; Ritanserin; Serotonin Antagonists | 1985 |
Characterization of flufylline, fluprofylline, ritanserin, butanserin and R 56413 with respect to in-vivo alpha 1-,alpha 2- and 5-HT2-receptor antagonism and in-vitro affinity for alpha 1-,alpha 2- and 5-HT2-receptors: comparison with ketanserin.
Topics: Adrenergic alpha-Antagonists; Animals; Binding, Competitive; Blood Pressure; Brain; Decerebrate State; Histamine H2 Antagonists; Ketanserin; Male; Piperidines; Rats; Rats, Inbred Strains; Ritanserin; Serotonin Antagonists; Theophylline; Vasoconstriction | 1986 |
Recent developments in 5HT-related pharmacology of animal models of anxiety.
Topics: Animals; Anti-Anxiety Agents; Anxiety; Buspirone; Disease Models, Animal; Piperidines; Pyrimidines; Receptors, Serotonin; Ritanserin; Serotonin; Serotonin Antagonists; Social Behavior | 1986 |
Phencyclidine-induced head-weaving observed in mice after ritanserin treatment.
Topics: Animals; Fenclonine; Histamine H2 Antagonists; Male; Methoxydimethyltryptamines; Mice; Mice, Inbred Strains; Phencyclidine; Pindolol; Piperidines; Ritanserin; Stereotyped Behavior | 1987 |
Ritanserin assessments in plasma and CSF by means of HPLC technique with fluorescence detection.
Topics: Chromatography, High Pressure Liquid; Histamine H2 Antagonists; Humans; Piperidines; Ritanserin; Spectrometry, Fluorescence; Spectrophotometry, Ultraviolet | 1987 |
Quipazine reduces food intake in the rat by activation of 5-HT2-receptors.
Topics: Animals; Diet; Dose-Response Relationship, Drug; Eating; Histamine H2 Antagonists; Imidazoles; Ketanserin; Methysergide; Ondansetron; Pindolol; Piperidines; Quinolines; Quipazine; Rats; Receptors, Serotonin; Ritanserin; Serotonin Antagonists | 1988 |
Chronic 5-HT2 receptor blockade with ritanserin does not reduce blood pressure in the spontaneously hypertensive rat.
Topics: Animals; Blood Pressure; Decerebrate State; Dose-Response Relationship, Drug; Electric Stimulation; Heart Rate; Hypertension; Ketanserin; Male; Phenylephrine; Piperidines; Prazosin; Rats; Rats, Inbred SHR; Receptors, Serotonin; Ritanserin; Time Factors | 1985 |
Differential regulation of dopamine-D2 and serotonin-S2 receptors by chronic treatment with the serotonin-S2 antagonists, ritanserin, and setoperone.
Topics: Animals; Brain; Corpus Striatum; Frontal Lobe; Male; Piperidines; Pyrimidinones; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Dopamine D2; Receptors, Serotonin; Ritanserin; Serotonin Antagonists | 1987 |
5-HT2 receptors could be primarily involved in the regulation of slow-wave sleep in the rat.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; DOM 2,5-Dimethoxy-4-Methylamphetamine; Dose-Response Relationship, Drug; Indoles; Piperidines; Rats; Rats, Inbred Strains; Receptors, Serotonin; Ritanserin; Sleep; Tetrahydronaphthalenes | 1987 |
Ritanserin, a serotonin-S2 receptor antagonist, does not prevent 5-hydroxytryptophan-induced beta-EP, beta-LPH and cortisol secretion.
Topics: 5-Hydroxytryptophan; Adolescent; beta-Endorphin; beta-Lipotropin; Endorphins; Humans; Hydrocortisone; Male; Piperidines; Ritanserin; Secretory Rate; Serotonin; Time Factors | 1987 |
Antihypertensive mechanism of action of ketanserin and some ketanserin analogues in the spontaneously hypertensive rat.
Topics: Animals; Blood Pressure; Dose-Response Relationship, Drug; Electric Stimulation; Hypertension; Ketanserin; Phenylephrine; Piperidines; Prazosin; Pyrimidines; Rats; Rats, Inbred SHR; Receptors, Adrenergic, alpha; Ritanserin; Sympathetic Nervous System | 1985 |
Down regulation of serotonin-S2 receptor sites in rat brain by chronic treatment with the serotonin-S2 antagonists: ritanserin and setoperone.
Topics: Animals; Brain; Corpus Striatum; Frontal Lobe; Ketanserin; Male; Piperidines; Pyrimidinones; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Dopamine D2; Receptors, Neurotransmitter; Receptors, Serotonin; Ritanserin | 1986 |
Open pilot trial of ritanserin in parkinsonism.
Topics: Aged; Antiparkinson Agents; Dyskinesia, Drug-Induced; Humans; Levodopa; Parkinson Disease; Pilot Projects; Piperidines; Ritanserin | 1986 |
Evidence for separate receptors that mediate parallel effects of serotonin and small cardioactive peptideB (SCPB) on adenylate cyclase in Aplysia californica.
Topics: Adenylyl Cyclases; Animals; Aplysia; Enzyme Activation; Ketanserin; Neuropeptides; Piperidines; Receptors, Serotonin; Ritanserin; Serotonin; Serotonin Antagonists | 1986 |
Effect of hallucinogens on spontaneous and sensory-evoked locus coeruleus unit activity in the rat: reversal by selective 5-HT2 antagonists.
Topics: Animals; Dextroamphetamine; DOM 2,5-Dimethoxy-4-Methylamphetamine; Ergolines; Evoked Potentials, Somatosensory; Hallucinogens; Locus Coeruleus; Lysergic Acid Diethylamide; Male; Mescaline; Piperidines; Rats; Rats, Inbred Strains; Ritanserin | 1986 |
5-Hydroxytryptamine M-receptor antagonism in the hypothalamus facilitates gastric emptying in the guinea-pig.
Topics: Animals; Gastric Emptying; Guinea Pigs; Hypothalamus; Indoles; Male; Methysergide; Piperidines; Receptors, Serotonin; Ritanserin; Serotonin; Tropisetron | 1986 |
Antagonism by methysergide of neurogenic vasoconstriction in the dog forelimb.
Topics: Animals; Dogs; Electric Stimulation; Forelimb; Ketanserin; Median Nerve; Methysergide; Phentolamine; Piperidines; Receptors, Serotonin; Ritanserin; Serotonin; Serotonin Antagonists; Vascular Resistance; Vasoconstriction; Vasodilation | 1987 |
Serotonin receptors in the rat nucleus tractus solitarii and cardiovascular regulation.
Topics: Animals; Blood Pressure; Body Temperature; Cardiovascular Physiological Phenomena; Heart Rate; Indoles; Ketanserin; Male; Medulla Oblongata; Piperidines; Rats; Rats, Inbred Strains; Receptors, Serotonin; Ritanserin; Serotonin; Serotonin Antagonists | 1986 |
Vasoconstrictor expression of human platelet-vessel wall interactions: inhibition by the Ca2+ entry blocker flunarizine.
Topics: Animals; Arachidonic Acid; Arachidonic Acids; Basilar Artery; Blood Platelets; Dogs; Flunarizine; In Vitro Techniques; Piperidines; Ritanserin; Serotonin; Thromboxane A2; Vasodilator Agents | 1987 |
Effect of the 5HT2 antagonist ritanserin on food intake and on 5HT-induced anorexia in the rat.
Topics: Animals; Anorexia; Brain; Drinking Behavior; Feeding and Eating Disorders; Feeding Behavior; Food Deprivation; Male; Piperidines; Rats; Rats, Inbred Strains; Ritanserin; Satiation; Serotonin; Serotonin Antagonists | 1987 |
Phencyclidine-induced head-twitch responses as 5-HT2 receptor-mediated behavior in rats.
Topics: Animals; Male; Methoxydimethyltryptamines; Mice; Phencyclidine; Piperidines; Rats; Rats, Inbred F344; Receptors, Serotonin; Ritanserin; Serotonin Antagonists; Stereotyped Behavior | 1987 |
Allosteric properties of the 5-HT2 receptor system of the rat tail artery. Ritanserin and methysergide are not competitive 5-HT2 receptor antagonists but allosteric modulators.
Topics: Allosteric Regulation; Animals; Arteries; Binding, Competitive; In Vitro Techniques; Male; Methysergide; Muscle, Smooth, Vascular; Piperidines; Rats; Rats, Inbred Strains; Receptors, Serotonin; Regional Blood Flow; Ritanserin; Tail | 1987 |
M-chlorophenylpiperazine increases blood pressure and heart rate in pithed and conscious rats.
Topics: Adrenal Medulla; Animals; Blood Pressure; Brain; Heart Rate; Kinetics; Male; Metergoline; Piperazines; Piperidines; Rats; Rats, Inbred Strains; Receptors, Serotonin; Ritanserin; Serotonin Antagonists; Spinal Cord | 1987 |
Effects of 5-HT receptor subtype-selective drugs on locomotor activity and motor habituation in the DHT adult rat model.
Topics: 5-Hydroxytryptophan; 5,7-Dihydroxytryptamine; Animals; Habituation, Psychophysiologic; Male; Motor Activity; Piperidines; Rats; Rats, Inbred Strains; Receptors, Serotonin; Ritanserin; Serotonin; Serotonin Antagonists | 1987 |
Two distinct effects of 5-hydroxytryptamine on single cortical neurons.
Topics: Animals; Cinanserin; Electric Conductivity; Guinea Pigs; In Vitro Techniques; Membrane Potentials; Neurons; Piperidines; Potassium; Pyramidal Tracts; Ritanserin; Serotonin; Serotonin Antagonists; Somatosensory Cortex | 1987 |
The 5-hydroxytryptamine stimulated formation of inositol phosphate is inhibited in platelets from alcoholics.
Topics: Adult; Alcoholism; Blood Platelets; Humans; Inositol Phosphates; Male; Middle Aged; Piperidines; Receptors, Serotonin; Ritanserin; Serotonin; Sugar Phosphates | 1988 |
Mescaline: excitatory effects on acoustic startle are blocked by serotonin2 antagonists.
Topics: Animals; Dextroamphetamine; Dimethyl Sulfoxide; Dose-Response Relationship, Drug; Male; Mescaline; Piperidines; Rats; Rats, Inbred Strains; Reflex, Acoustic; Reflex, Startle; Ritanserin; Serotonin Antagonists | 1987 |
The effects of chronic ritanserin treatment on sleep and the neuroendocrine response to L-tryptophan.
Topics: Adult; Binding, Competitive; Growth Hormone; Humans; Lysergic Acid Diethylamide; Male; Neurosecretory Systems; Piperidines; Prolactin; Radioimmunoassay; Ritanserin; Sleep; Sleep Stages; Tryptophan | 1987 |
Ritanserin and serotonergic mechanisms in blood pressure and fluid regulation in sheep.
Topics: Animals; Blood Pressure; Cardiac Output; Heart Rate; Hypertension; Ketanserin; Phenylephrine; Piperidines; Ritanserin; Serotonin; Serotonin Antagonists; Sheep; Water-Electrolyte Balance | 1987 |
Protection with phencyclidine against inactivation of 5-HT2 receptors by sulfhydryl-modifying reagents.
Topics: Animals; Behavior, Animal; Ethylmaleimide; Ketanserin; Male; Phencyclidine; Piperidines; Rats; Rats, Inbred F344; Receptors, Serotonin; Ritanserin; Serotonin; Sulfhydryl Reagents | 1988 |
Putative selective 5-HT-2 antagonists block serotonin 5-HT-1c receptors in the choroid plexus.
Topics: Animals; Choroid Plexus; In Vitro Techniques; Lysergic Acid Diethylamide; Mianserin; Piperidines; Rats; Rats, Inbred Strains; Receptors, Serotonin; Ritanserin; Serotonin Antagonists | 1988 |
Effects of dopaminergic and serotonergic receptor blockade on neurochemical changes induced by acute administration of methamphetamine and 3,4-methylenedioxymethamphetamine.
Topics: 3,4-Methylenedioxyamphetamine; Amphetamines; Animals; Haloperidol; Male; Methamphetamine; Methiothepin; Piperidines; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Serotonin; Ritanserin; Serotonin Antagonists | 1988 |
Effects of ritanserin on the rewarding properties of d-amphetamine, morphine and diazepam revealed by conditioned place preference in rats.
Topics: Analgesia; Animals; Conditioning, Operant; Dextroamphetamine; Diazepam; Exploratory Behavior; Male; Morphine; Motor Activity; Piperidines; Rats; Rats, Inbred Strains; Reference Values; Reinforcement, Psychology; Reward; Ritanserin; Serotonin Antagonists | 1988 |
Increased food intake in satiated rats induced by the 5-HT antagonists methysergide, metergoline and ritanserin.
Topics: Animals; Chlordiazepoxide; Cyproheptadine; Diet; Eating; Ergolines; Male; Metergoline; Methysergide; Piperidines; Rats; Rats, Inbred Strains; Ritanserin; Satiation; Serotonin Antagonists | 1988 |
Interference of ketanserin with baroreflex control of the circulation in the conscious spontaneously hypertensive rat.
Topics: Animals; Blood Pressure; Heart Rate; Hypertension; Ketanserin; Male; Piperidines; Prazosin; Pressoreceptors; Rats; Rats, Inbred SHR; Ritanserin; Serotonin Antagonists | 1988 |
Effect of ritanserin on sleep stages and sleep EEG in the rat.
Topics: Animals; Dose-Response Relationship, Drug; Electroencephalography; Male; Piperidines; Rats; Rats, Inbred Strains; Ritanserin; Sleep Stages | 1988 |
Examination of the effects of some 5-HT2 receptor antagonists on central sympathetic outflow and blood pressure in anaesthetised cats.
Topics: Anesthesia; Animals; Blood Pressure; Cats; Cinanserin; Cyproheptadine; Male; Metergoline; Methiothepin; Piperidines; Quinolines; Ritanserin; Serotonin Antagonists; Sympathetic Nervous System | 1988 |
Study to establish the indication for the selective S2 antagonist ritanserin.
Topics: Adult; Depressive Disorder; Female; Humans; Male; Mental Disorders; Middle Aged; Piperidines; Psychiatric Status Rating Scales; Ritanserin; Serotonin Antagonists | 1988 |
Habituation of tactile startle is altered by drugs acting on serotonin-2 receptors.
Topics: Animals; Cinanserin; Cyproheptadine; Habituation, Psychophysiologic; Ketanserin; Male; Piperidines; Propranolol; Rats; Rats, Inbred Strains; Receptors, Serotonin; Reference Values; Reflex, Startle; Ritanserin; Serotonin; Serotonin Antagonists; Touch | 1988 |
Effects of prenatal administration of phencyclidine on the learning and memory processes of rat offspring.
Topics: Animals; Avoidance Learning; Body Weight; Brain; Female; Learning; Memory; Naloxone; Organ Size; Phencyclidine; Physostigmine; Piperidines; Pregnancy; Prenatal Exposure Delayed Effects; Rats; Rats, Inbred Strains; Ritanserin | 1988 |
Serotonin antagonism in panic disorder: an open trial with ritanserin.
Topics: Adult; Agoraphobia; Escape Reaction; Fear; Female; Humans; Male; Panic; Phobic Disorders; Piperidines; Ritanserin; Serotonin Antagonists | 1988 |
5-HT2 receptor antagonists do not reduce ethanol preference in Sardinian alcohol-preferring (sP) rats.
Topics: Alcohol Drinking; Animals; Antipsychotic Agents; Haloperidol; Isoxazoles; Male; Piperidines; Rats; Risperidone; Ritanserin; Serotonin Antagonists | 1993 |
The effect of risperidone and ritanserin on human IgG and IgM synthesis in vitro.
Topics: Antipsychotic Agents; B-Lymphocytes; Enzyme-Linked Immunosorbent Assay; Humans; Immunoglobulin G; Immunoglobulin M; In Vitro Techniques; Isoxazoles; Monocytes; Piperidines; Pokeweed Mitogens; Risperidone; Ritanserin; Schizophrenia | 1994 |
Effects of risperidone on phencyclidine-induced behaviors: comparison with haloperidol and ritanserin.
Topics: 3,4-Dihydroxyphenylacetic Acid; Animals; Antipsychotic Agents; Chromatography, High Pressure Liquid; Corpus Striatum; Dopamine; Dose-Response Relationship, Drug; Frontal Lobe; Haloperidol; Homovanillic Acid; Hydroxyindoleacetic Acid; Injections, Intraperitoneal; Isoxazoles; Locomotion; Male; Phencyclidine; Piperidines; Random Allocation; Rats; Rats, Wistar; Risperidone; Ritanserin; Schizophrenia; Serotonin; Stereotyped Behavior | 1994 |
Effects of MDL 28,133A, a 5-HT2 receptor antagonist, on platelet aggregation and coronary thrombosis in dogs.
Topics: Administration, Oral; Animals; Biological Availability; Blood Platelets; Blood Pressure; Coronary Thrombosis; Disease Models, Animal; Dogs; Drug Therapy, Combination; Electric Stimulation; Female; Heart Rate; Heparin; In Vitro Techniques; Male; Piperidines; Platelet Aggregation; Ritanserin; Serotonin; Serotonin Antagonists; Streptokinase | 1994 |
Risperidone prevents the development of supersensitivity, but not tolerance, to phencyclidine in rats treated with subacute phencyclidine.
Topics: Animals; Antipsychotic Agents; Dizocilpine Maleate; Drug Tolerance; Haloperidol; Isoxazoles; Male; Methamphetamine; Motor Activity; Phencyclidine; Piperidines; Rats; Rats, Wistar; Receptors, Phencyclidine; Receptors, Serotonin; Risperidone; Ritanserin | 1995 |
The selective 5-HT2A receptor antagonist, MDL 100,907, increases dopamine efflux in the prefrontal cortex of the rat.
Topics: 3,4-Dihydroxyphenylacetic Acid; Animals; Behavior, Animal; Dopamine; Electrophysiology; Fluorobenzenes; Homovanillic Acid; In Vitro Techniques; Male; Microdialysis; Piperidines; Prefrontal Cortex; Rats; Rats, Sprague-Dawley; Ritanserin; Serotonin Antagonists | 1995 |
Effect of NE-100, a novel sigma receptor ligand, on phencyclidine-induced cognitive dysfunction.
Topics: Animals; Anisoles; Anti-Anxiety Agents; Cognition Disorders; Drug Interactions; Ligands; Male; Phencyclidine; Physical Exertion; Piperidines; Propylamines; Pyrimidines; Rats; Rats, Wistar; Receptors, sigma; Ritanserin; Swimming | 1994 |
Excitation of interneurons in piriform cortex by 5-hydroxytryptamine: blockade by MDL 100,907, a highly selective 5-HT2A receptor antagonist.
Topics: Animals; Dose-Response Relationship, Drug; Electrophysiology; Fluorobenzenes; In Vitro Techniques; Interneurons; Male; Olfactory Pathways; Piperidines; Rats; Rats, Sprague-Dawley; Receptors, Serotonin; Ritanserin; Serotonin; Serotonin Antagonists | 1994 |
Effects of the selective 5-HT2A receptor antagonist MDL 100,907 on MDMA-induced locomotor stimulation in rats.
Topics: 5,7-Dihydroxytryptamine; Animals; Brain Chemistry; Clozapine; Dopamine Antagonists; Fluorobenzenes; Male; Methiothepin; Motor Activity; N-Methyl-3,4-methylenedioxyamphetamine; Piperidines; Presynaptic Terminals; Rats; Receptors, Neurotransmitter; Ritanserin; Serotonin; Serotonin Agents; Serotonin Antagonists; Stimulation, Chemical | 1996 |
5-HT3-like receptors in the rat medial prefrontal cortex: further pharmacological characterization.
Topics: Animals; Biguanides; Bridged Bicyclo Compounds, Heterocyclic; Dose-Response Relationship, Drug; Drug Interactions; Electrophysiology; Frontal Lobe; Glutamic Acid; Gyrus Cinguli; Hydrolysis; Indoles; Isomerism; Male; Neurons; Nicotinic Antagonists; Phosphatidylinositols; Piperidines; Prefrontal Cortex; Rats; Rats, Sprague-Dawley; Receptors, Serotonin; Ritanserin; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Tubocurarine | 1996 |
Pharmacological characterization of in vivo properties of putative mixed 5-HT1A agonist/5-HT(2A/2C) antagonist anxiolytics. II. Drug discrimination and behavioral observation studies in rats.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Amphetamines; Animals; Anti-Anxiety Agents; Behavior, Animal; Benzopyrans; Discrimination, Psychological; Ketanserin; Lysergic Acid Diethylamide; Male; Nicotinic Acids; Piperazines; Piperidines; Protein Binding; Rats; Rats, Sprague-Dawley; Receptors, Serotonin; Ritanserin; Serotonin Antagonists; Serotonin Receptor Agonists | 1997 |
The apparent antipsychotic action of the 5-HT2a receptor antagonist M100907 in a mouse model of schizophrenia is counteracted by ritanserin. (Rapid communication).
Topics: Animals; Antipsychotic Agents; Dizocilpine Maleate; Excitatory Amino Acid Antagonists; Fluorobenzenes; Male; Mice; Mice, Inbred Strains; Motor Activity; Piperidines; Ritanserin; Schizophrenia; Serotonin Antagonists | 1997 |
Evidence for a 5-HT3 receptor involvement in the facilitation of peristalsis on mucosal application of 5-HT in the guinea pig isolated ileum.
Topics: Animals; Dioxanes; Female; Granisetron; Guinea Pigs; Ileum; In Vitro Techniques; Male; Methiothepin; Mucous Membrane; Ondansetron; Peristalsis; Piperidines; Receptors, Serotonin; Receptors, Serotonin, 5-HT3; Ritanserin; Serotonin; Serotonin Antagonists | 1997 |
Characterization of 5-HT receptors on human pulmonary artery and vein: functional and binding studies.
Topics: Abortifacient Agents, Nonsteroidal; Adult; Aged; Benzamides; Binding Sites; Binding, Competitive; Bridged Bicyclo Compounds, Heterocyclic; Dinoprost; Dioxanes; Dose-Response Relationship, Drug; Endothelium, Vascular; Female; Humans; Male; Middle Aged; Oxadiazoles; Piperazines; Piperidines; Pulmonary Artery; Pulmonary Veins; Pyridines; Receptors, Serotonin; Ritanserin; Serotonin; Serotonin Antagonists; Sumatriptan; Vasoconstrictor Agents | 1997 |
Effects of serotonin 5-HT(2A/2C) antagonists on associative learning in the rabbit.
Topics: Animals; Conditioning, Classical; Female; Male; Nictitating Membrane; Piperidines; Rabbits; Receptor, Serotonin, 5-HT2A; Receptor, Serotonin, 5-HT2C; Receptors, Serotonin; Ritanserin; Serotonin Antagonists | 1998 |
Vascular and cardiac effects of DV-7028, a selective, 5-HT2-receptor antagonist in rats.
Topics: Animals; Baroreflex; Blood Pressure; Cardiovascular System; Coronary Circulation; Heart; Heart Rate; Hindlimb; Injections, Intravenous; Ketanserin; Male; Piperidines; Rats; Rats, Wistar; Receptor, Serotonin, 5-HT2A; Receptors, Serotonin; Ritanserin; Serotonin Antagonists; Triazines; Vagotomy | 1998 |
5-HT2A receptor antagonists block MK-801-induced stereotypy and hyperlocomotion.
Topics: Animals; Dizocilpine Maleate; Dose-Response Relationship, Drug; Histamine H2 Antagonists; Ketanserin; Locomotion; Male; Mice; Mice, Inbred BALB C; Neuroprotective Agents; Piperidines; Receptor, Serotonin, 5-HT2A; Receptors, Serotonin; Ritanserin; Serotonin Antagonists; Stereotypic Movement Disorder | 1998 |
Effect of 5-HT2 receptor antagonists on a cranial nerve reflex in the rabbit: evidence for inverse agonism.
Topics: Animals; Cranial Nerves; Ergolines; Female; Ketanserin; Lysergic Acid Diethylamide; Male; Mianserin; Piperidines; Rabbits; Receptors, Serotonin; Reflex; Ritanserin; Serotonin Antagonists; Serotonin Receptor Agonists | 1999 |
The motivation for beer in rats: effects of ritanserin, naloxone and SR 141716.
Topics: Alcohol Drinking; Animals; Beer; Ethanol; Male; Motivation; Motor Activity; Naloxone; Narcotic Antagonists; Piperidines; Pyrazoles; Rats; Rats, Wistar; Rimonabant; Ritanserin; Serotonin Antagonists | 1999 |
Clozapine and other 5-hydroxytryptamine-2A receptor antagonists alter the subcellular distribution of 5-hydroxytryptamine-2A receptors in vitro and in vivo.
Topics: 3T3 Cells; Animals; Antipsychotic Agents; Benzodiazepines; Cell Line; Clozapine; Dendrites; Fluorobenzenes; Haloperidol; Mianserin; Mice; Olanzapine; Piperidines; Pirenzepine; Prefrontal Cortex; Pyramidal Cells; Rats; Receptor, Serotonin, 5-HT2A; Receptors, Serotonin; Recombinant Proteins; Risperidone; Ritanserin; Serotonin Antagonists; Transfection | 1999 |
5-HT2 receptor antagonism reduces hyperactivity induced by amphetamine, cocaine, and MK-801 but not D1 agonist C-APB.
Topics: Aminopyridines; Amphetamine; Animals; Benzazepines; Cocaine; Dizocilpine Maleate; Dopamine Agonists; Drug Interactions; Female; Fluorobenzenes; Indoles; Mice; Motor Activity; Piperidines; Ritanserin; Serotonin Antagonists | 1999 |
Pharmacological characterization of the 5-HT receptor-mediated contraction in the mouse isolated ileum.
Topics: Animals; Atropine; Dioxanes; Dose-Response Relationship, Drug; Female; Granisetron; Ileum; In Vitro Techniques; Indoles; Ketanserin; Male; Mice; Muscle Contraction; Ondansetron; Piperidines; Receptors, Serotonin; Ritanserin; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Tetrodotoxin; Tropanes; Tropisetron | 2000 |
The pharmacology of the acute hyperthermic response that follows administration of 3,4-methylenedioxymethamphetamine (MDMA, 'ecstasy') to rats.
Topics: 3,4-Methylenedioxyamphetamine; Acute Disease; Animals; Benzazepines; Body Temperature; Corpus Striatum; Dopamine; Dopamine Antagonists; Dopamine Uptake Inhibitors; Fever; Hallucinogens; Hippocampus; Male; Methysergide; N-Methyl-3,4-methylenedioxyamphetamine; Neuroprotective Agents; Piperazines; Piperidines; Rats; Rats, Inbred Strains; Receptor, Serotonin, 5-HT2A; Receptor, Serotonin, 5-HT2C; Receptors, Serotonin; Remoxipride; Ritanserin; Selective Serotonin Reuptake Inhibitors; Serotonin Antagonists | 2002 |
Differential inverse agonist efficacies of SB-258719, SB-258741 and SB-269970 at human recombinant serotonin 5-HT7 receptors.
Topics: Animals; Binding, Competitive; CHO Cells; Clozapine; Cricetinae; Cricetulus; Cyclic AMP; Dose-Response Relationship, Drug; Ergolines; Humans; Loxapine; Methiothepin; Phenols; Pimozide; Pindolol; Piperidines; Plasmids; Pyrrolidines; Radioligand Assay; Receptors, Serotonin; Ritanserin; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Sulfonamides; Tosyl Compounds; Transfection | 2004 |
Discriminative stimulus effects of 1-(2,5-dimethoxy-4-methylphenyl)-2-aminopropane in rhesus monkeys: antagonism and apparent pA2 analyses.
Topics: Animals; DOM 2,5-Dimethoxy-4-Methylamphetamine; Dose-Response Relationship, Drug; Electroshock; Fluorobenzenes; Hallucinogens; Ketanserin; Macaca mulatta; Phenethylamines; Piperidines; Reaction Time; Receptor, Serotonin, 5-HT2A; Receptor, Serotonin, 5-HT2C; Receptors, Serotonin; Regression Analysis; Ritanserin; Serotonin Antagonists; Serotonin Receptor Agonists | 2009 |
Discriminative stimulus effects of 1-(2,5-dimethoxy-4-methylphenyl)-2-aminopropane (DOM), ketanserin, and (R)-(+)-{alpha}-(2,3-dimethoxyphenyl)-1-[2-(4-fluorophenyl)ethyl]-4-pipidinemethanol (MDL100907) in rats.
Topics: Analgesics, Opioid; Anesthetics, Dissociative; Animals; Conditioning, Operant; Discrimination, Psychological; DOM 2,5-Dimethoxy-4-Methylamphetamine; Dose-Response Relationship, Drug; Excitatory Amino Acid Antagonists; Fluorobenzenes; Ketamine; Ketanserin; Male; Morphine; Phencyclidine; Piperidines; Rats; Rats, Sprague-Dawley; Receptor, Serotonin, 5-HT2A; Receptors, Adrenergic, alpha-1; Ritanserin; Serotonin Antagonists; Serotonin Receptor Agonists | 2009 |
Serotonin-1A receptor stimulation mediates effects of a metabotropic glutamate 2/3 receptor antagonist, 2S-2-amino-2-(1S,2S-2-carboxycycloprop-1-yl)-3-(xanth-9-yl)propanoic acid (LY341495), and an N-methyl-D-aspartate receptor antagonist, ketamine, in the
Topics: Amino Acids; Animals; Antidepressive Agents; Dioxoles; Enzyme Inhibitors; Excitatory Amino Acid Antagonists; Feeding Behavior; Fenclonine; Ketamine; Male; Mice, Inbred C57BL; Neuropsychological Tests; Piperazines; Piperidines; Pyridines; Quinoxalines; Receptors, AMPA; Receptors, Metabotropic Glutamate; Receptors, N-Methyl-D-Aspartate; Ritanserin; Serotonin 5-HT1 Receptor Antagonists; Serotonin 5-HT2 Receptor Antagonists; Tryptophan Hydroxylase; Xanthenes | 2014 |
Neuropharmacology of light-induced locomotor activation.
Topics: Animals; Dopamine Agents; Dose-Response Relationship, Drug; Excitatory Amino Acid Agents; Haloperidol; Indoles; Ketamine; Light; Male; Motor Activity; Naphthyridines; Phencyclidine; Photic Stimulation; Piperazines; Piperidines; Pyridines; Quinpirole; Rats, Wistar; Receptors, N-Methyl-D-Aspartate; Ritanserin; Serotonin Antagonists | 2015 |
Ritanserin, a novel agent targeting the mesenchymal subtype of glioblastomas.
Topics: Adult; Diacylglycerol Kinase; Glioblastoma; Humans; Piperidines; Ritanserin | 2018 |
Identification of a novel DGKα inhibitor for XLP-1 therapy by virtual screening.
Topics: Cell Death; Computer Simulation; Diacylglycerol Kinase; Drug Evaluation, Preclinical; Humans; Lymphoproliferative Disorders; Piperidines; Protein Kinase Inhibitors; Pyrimidinones; Quinazolinones; Ritanserin; Thiazoles | 2019 |