Page last updated: 2024-08-16

ritanserin and mdl 100907

ritanserin has been researched along with mdl 100907 in 37 studies

Research

Studies (37)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's7 (18.92)18.2507
2000's17 (45.95)29.6817
2010's10 (27.03)24.3611
2020's3 (8.11)2.80

Authors

AuthorsStudies
Blackburn, TP; Holland, V; Kettle, A; Reavill, C; Riley, G1
Benwell, K; Bickerdike, M; Kennett, G; Knight, AR; Misra, A; Quirk, K; Revell, D1
Bonaventure, P; Carruthers, NI; Dvorak, CA; Dvorak, L; Lovenberg, TW; Miller, KL; Nepomuceno, D; Rudolph, DA; Shireman, BT1
Chen, Z; Collier, T; Fu, H; Liang, SH; Rong, J; Zhou, J1
Fadayel, GM; Schmidt, CJ1
Aghajanian, GK; Marek, GJ1
Dudley, MW; Kehne, JH; Ketteler, HJ; McCloskey, TC; Schmidt, CJ; Sullivan, CK1
Carlsson, A; Carlsson, ML; Martin, P; Waters, N1
Alsayegh, L; Backstrom, JR; Berry, SA; Friedman, L; Roth, BL; Sanders-Bush, E; Willins, DL1
Heron-Maxwell, CL; O'Neill, MF; Shaw, G1
Berndt, MC; Bobik, A; Jennings, G; Kannelakis, P; Taylor, AJ1
Abu-Amara, M; Aldairy, C; Hagan, JJ; Siddiqui, A; Wilson, C1
Calama, E; Martín, ML; Morán, A; Ortiz de Urbina, AV; San Román, L1
Harooni, HE; Naghdi, N1
Coimbra, NC; de Oliveira, R; de Oliveira, RC; Ferreira, CM1
Alexandropoulou, KN; Demonakou, MD; Hereti, RI; Kourentzi, KT; Manta, GA; Mykoniatis, MG; Panoutsopoulos, GI; Papadimas, GK; Skaltsas, SD; Tzirogiannis, KN1
Cheng, HY; Hsieh, CC; Hsieh, MT; Lin, YT; Lu, MC; Peng, WH; Wu, CR1
Beck, W; Deppisch, R; Hoenich, NA; Marshall, SM; Thompson, MG; Wang, Y1
Ago, Y; Baba, A; Matsuda, T; Nakamura, S1
Bray, JK; Goddard, WA1
Atwood, WJ; Lane, TE; O'Hara, BA; Schaumburg, C1
France, CP; Li, JX; Rice, KC1
Kłodzińska, A; Neuville, P; Palucha-Poniewiera, A; Pilc, A; Schann, S; Stachowicz, K1
France, CP; Javors, MA; Koek, W; Li, JX; Rice, KC; Unzeitig, A1
Nakamichi, K; Nukuzuma, C; Nukuzuma, S; Takegami, T1
Anwar, MA; Broadley, KJ; Ford, WR; Herbert, AA1
Choi, HS; Jun, DW; Kim, DC; Kim, EK; Kwon, YI; Lee, HL; Lee, KN; Lee, OY; Yoon, BC1
Regan, CM; Ring, RM1
Chaki, S; Fukumoto, K; Iijima, M1
Anisimova, VA; Mal'tsev, DV; Spasov, AA; Yakovlev, DS1
Dvorkin-Gheva, A; Johnson, E; Szechtman, H; Tucci, MC; Wong, M1
Guo, Y; Hu, L; Liu, C; Luo, B; Wang, H1
Braida, D; Ponzoni, L; Sala, M1
Barbosa Silva, RC; de Oliveira, RP; Nagaishi, KY1
Bjørn-Yoshimoto, WE; Che, T; Cheng, J; Ding, K; Gloriam, DE; Han, GW; Hanson, MA; Harpsøe, K; Huang, XP; Jensen, AA; Katritch, V; Lansu, K; Liu, ZJ; McCorvy, JD; Nikolajsen, LF; Peng, Y; Popov, P; Pu, M; Qu, L; Roth, BL; Shen, L; Stevens, RC; Wacker, D; Wu, Y; Yuan, S; Zhao, S1
Bova, S; Fusi, F; Saponara, S; Sgaragli, G; Spiga, O; Trezza, A1
Makiguchi, A; Okada, T; Shioda, K; Suda, S1

Reviews

2 review(s) available for ritanserin and mdl 100907

ArticleYear
Positron Emission Tomography (PET) Imaging Tracers for Serotonin Receptors.
    Journal of medicinal chemistry, 2022, 08-25, Volume: 65, Issue:16

    Topics: Brain; Humans; Ligands; Positron-Emission Tomography; Radiopharmaceuticals; Receptors, Serotonin

2022
Neuropsychotoxicity of abused drugs: effects of serotonin receptor ligands on methamphetamine- and cocaine-induced behavioral sensitization in mice.
    Journal of pharmacological sciences, 2008, Volume: 106, Issue:1

    Topics: Amphetamine-Related Disorders; Animals; Behavior, Animal; Brain; Bridged Bicyclo Compounds, Heterocyclic; Central Nervous System Stimulants; Cocaine; Cocaine-Related Disorders; Dioxanes; Dioxoles; Disease Models, Animal; Ligands; Methamphetamine; Mice; Motor Activity; Oxazines; Receptors, Serotonin; Ritanserin; Serotonin; Serotonin 5-HT1 Receptor Agonists; Serotonin 5-HT2 Receptor Antagonists; Serotonin 5-HT3 Receptor Antagonists; Serotonin Agents; Serotonin Antagonists; Serotonin Receptor Agonists

2008

Other Studies

35 other study(ies) available for ritanserin and mdl 100907

ArticleYear
Attenuation of haloperidol-induced catalepsy by a 5-HT2C receptor antagonist.
    British journal of pharmacology, 1999, Volume: 126, Issue:3

    Topics: Animals; Binding, Competitive; Catalepsy; Cell Line; Dopamine Antagonists; Fluorobenzenes; Haloperidol; Humans; Indoles; Male; Piperidines; Quinolines; Radioligand Assay; Rats; Rats, Sprague-Dawley; Receptor, Serotonin, 5-HT2A; Receptor, Serotonin, 5-HT2B; Receptor, Serotonin, 5-HT2C; Receptors, Serotonin; Serotonin Antagonists

1999
Pharmacological characterisation of the agonist radioligand binding site of 5-HT(2A), 5-HT(2B) and 5-HT(2C) receptors.
    Naunyn-Schmiedeberg's archives of pharmacology, 2004, Volume: 370, Issue:2

    Topics: Binding Sites; Binding, Competitive; Cell Line; Humans; Radioligand Assay; Receptor, Serotonin, 5-HT2A; Receptor, Serotonin, 5-HT2B; Receptor, Serotonin, 5-HT2C; Recombinant Proteins; Serotonin 5-HT2 Receptor Agonists; Serotonin 5-HT2 Receptor Antagonists; Serotonin Antagonists; Serotonin Receptor Agonists

2004
2-Alkyl-4-aryl-pyrimidine fused heterocycles as selective 5-HT2A antagonists.
    Bioorganic & medicinal chemistry letters, 2008, Mar-15, Volume: 18, Issue:6

    Topics: Animals; Azepines; Binding, Competitive; CHO Cells; Cricetinae; Cricetulus; Humans; Mice; Molecular Structure; NIH 3T3 Cells; Pyrimidines; Radioligand Assay; Receptor, Serotonin, 5-HT2A; Receptor, Serotonin, 5-HT2B; Receptor, Serotonin, 5-HT2C; Serotonin 5-HT2 Receptor Antagonists; Serotonin Antagonists; Structure-Activity Relationship

2008
The selective 5-HT2A receptor antagonist, MDL 100,907, increases dopamine efflux in the prefrontal cortex of the rat.
    European journal of pharmacology, 1995, Feb-06, Volume: 273, Issue:3

    Topics: 3,4-Dihydroxyphenylacetic Acid; Animals; Behavior, Animal; Dopamine; Electrophysiology; Fluorobenzenes; Homovanillic Acid; In Vitro Techniques; Male; Microdialysis; Piperidines; Prefrontal Cortex; Rats; Rats, Sprague-Dawley; Ritanserin; Serotonin Antagonists

1995
Excitation of interneurons in piriform cortex by 5-hydroxytryptamine: blockade by MDL 100,907, a highly selective 5-HT2A receptor antagonist.
    European journal of pharmacology, 1994, Jul-01, Volume: 259, Issue:2

    Topics: Animals; Dose-Response Relationship, Drug; Electrophysiology; Fluorobenzenes; In Vitro Techniques; Interneurons; Male; Olfactory Pathways; Piperidines; Rats; Rats, Sprague-Dawley; Receptors, Serotonin; Ritanserin; Serotonin; Serotonin Antagonists

1994
Effects of the selective 5-HT2A receptor antagonist MDL 100,907 on MDMA-induced locomotor stimulation in rats.
    Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology, 1996, Volume: 15, Issue:2

    Topics: 5,7-Dihydroxytryptamine; Animals; Brain Chemistry; Clozapine; Dopamine Antagonists; Fluorobenzenes; Male; Methiothepin; Motor Activity; N-Methyl-3,4-methylenedioxyamphetamine; Piperidines; Presynaptic Terminals; Rats; Receptors, Neurotransmitter; Ritanserin; Serotonin; Serotonin Agents; Serotonin Antagonists; Stimulation, Chemical

1996
The apparent antipsychotic action of the 5-HT2a receptor antagonist M100907 in a mouse model of schizophrenia is counteracted by ritanserin. (Rapid communication).
    Journal of neural transmission (Vienna, Austria : 1996), 1997, Volume: 104, Issue:4-5

    Topics: Animals; Antipsychotic Agents; Dizocilpine Maleate; Excitatory Amino Acid Antagonists; Fluorobenzenes; Male; Mice; Mice, Inbred Strains; Motor Activity; Piperidines; Ritanserin; Schizophrenia; Serotonin Antagonists

1997
Clozapine and other 5-hydroxytryptamine-2A receptor antagonists alter the subcellular distribution of 5-hydroxytryptamine-2A receptors in vitro and in vivo.
    Neuroscience, 1999, Volume: 91, Issue:2

    Topics: 3T3 Cells; Animals; Antipsychotic Agents; Benzodiazepines; Cell Line; Clozapine; Dendrites; Fluorobenzenes; Haloperidol; Mianserin; Mice; Olanzapine; Piperidines; Pirenzepine; Prefrontal Cortex; Pyramidal Cells; Rats; Receptor, Serotonin, 5-HT2A; Receptors, Serotonin; Recombinant Proteins; Risperidone; Ritanserin; Serotonin Antagonists; Transfection

1999
5-HT2 receptor antagonism reduces hyperactivity induced by amphetamine, cocaine, and MK-801 but not D1 agonist C-APB.
    Pharmacology, biochemistry, and behavior, 1999, Volume: 63, Issue:2

    Topics: Aminopyridines; Amphetamine; Animals; Benzazepines; Cocaine; Dizocilpine Maleate; Dopamine Agonists; Drug Interactions; Female; Fluorobenzenes; Indoles; Mice; Motor Activity; Piperidines; Ritanserin; Serotonin Antagonists

1999
Serotonin blockade protects against early microvascular constriction following atherosclerotic plaque rupture.
    European journal of pharmacology, 2004, Feb-13, Volume: 486, Issue:1

    Topics: Animals; Arteriosclerosis; Blood Flow Velocity; Disease Models, Animal; Iliac Artery; Indans; Microcirculation; Rabbits; Receptors, Serotonin, 5-HT2; Ritanserin; Rupture; Serotonin 5-HT2 Receptor Antagonists; Vasoconstriction

2004
5-HT7 receptor subtype as a mediator of the serotonergic regulation of luteinizing hormone release in the zona incerta.
    European journal of pharmacology, 2004, Apr-26, Volume: 491, Issue:1

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Female; Luteinizing Hormone; Male; Ovariectomy; Phenols; Piperazines; Rats; Rats, Wistar; Receptors, Serotonin; Ritanserin; Serotonin; Serotonin 5-HT1 Receptor Antagonists; Serotonin 5-HT2 Receptor Antagonists; Serotonin Antagonists; Serotonin Receptor Agonists; Subthalamus; Sulfonamides

2004
Vasoconstrictor responses to 5-hydroxytryptamine in the autoperfused hindquarters of spontaneously hypertensive rats.
    Pharmacology, 2004, Volume: 71, Issue:2

    Topics: Animals; Dose-Response Relationship, Drug; Hindlimb; Indoles; Injections, Intra-Arterial; Injections, Intravenous; Male; Perfusion; Piperazines; Prazosin; Pyridines; Rats; Rats, Inbred SHR; Rats, Wistar; Receptor, Serotonin, 5-HT1A; Receptor, Serotonin, 5-HT2A; Receptor, Serotonin, 5-HT2B; Receptor, Serotonin, 5-HT2C; Receptors, Serotonin, 5-HT2; Regional Blood Flow; Ritanserin; Serotonin; Serotonin 5-HT1 Receptor Antagonists; Serotonin 5-HT2 Receptor Agonists; Serotonin 5-HT2 Receptor Antagonists; Serotonin Receptor Agonists; Spiperone; Thiophenes; Vasoconstriction

2004
The effect of intrahippocampal injections of ritanserin (5HT2A/2C antagonist) and granisetron (5HT3 antagonist) on learning as assessed in the spatial version of the water maze.
    Behavioural brain research, 2005, Feb-28, Volume: 157, Issue:2

    Topics: Analysis of Variance; Animals; Escape Reaction; Granisetron; Hippocampus; Male; Maze Learning; Microinjections; Rats; Rats, Wistar; Reaction Time; Ritanserin; Serotonin 5-HT2 Receptor Antagonists; Serotonin 5-HT3 Receptor Antagonists; Serotonin Antagonists; Spatial Behavior; Swimming

2005
Involvement of 5-HT(2) serotonergic receptors of the nucleus raphe magnus and nucleus reticularis gigantocellularis/paragigantocellularis complex neural networks in the antinociceptive phenomenon that follows the post-ictal immobility syndrome.
    Experimental neurology, 2006, Volume: 201, Issue:1

    Topics: Analgesia; Analysis of Variance; Animals; Behavior, Animal; Brain; Male; Medulla Oblongata; Models, Neurological; Neural Pathways; Pain; Pain Measurement; Pain Threshold; Pentylenetetrazole; Raphe Nuclei; Rats; Rats, Wistar; Receptors, Serotonin, 5-HT2; Reticular Formation; Ritanserin; Seizures; Serotonin 5-HT2 Receptor Antagonists; Serotonin Antagonists; Syndrome; Time Factors

2006
Effect of 5-HT(2) receptor blockade on cadmium-induced acute toxicity.
    Digestive diseases and sciences, 2007, Volume: 52, Issue:9

    Topics: Animals; Apoptosis; Cadmium; Disease Models, Animal; In Situ Nick-End Labeling; Ketanserin; Liver Failure, Acute; Male; Rats; Rats, Wistar; Receptors, Serotonin, 5-HT2; Ritanserin; Serotonin 5-HT2 Receptor Antagonists; Serotonin Antagonists; Treatment Outcome

2007
Ameliorating effect of emodin, a constitute of Polygonatum multiflorum, on cycloheximide-induced impairment of memory consolidation in rats.
    Journal of ethnopharmacology, 2007, Jul-25, Volume: 112, Issue:3

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Administration, Oral; Animals; Baclofen; Bicuculline; Cycloheximide; Dose-Response Relationship, Drug; Emodin; GABA Agonists; GABA Antagonists; Injections, Subcutaneous; Learning; Male; Memory; Memory Disorders; Plant Roots; Polygonatum; Protein Synthesis Inhibitors; Rats; Rats, Sprague-Dawley; Ritanserin; Scopolamine; Serotonin 5-HT1 Receptor Agonists; Serotonin 5-HT2 Receptor Antagonists

2007
Differential effects of dialysis and ultrafiltrate from individuals with CKD, with or without diabetes, on platelet phosphatidylserine externalization.
    American journal of physiology. Renal physiology, 2008, Volume: 294, Issue:1

    Topics: Acetophenones; Adult; Aged; Aged, 80 and over; Benzopyrans; Blood Platelets; Case-Control Studies; Chronic Disease; Diabetes Mellitus, Type 2; Enzyme Inhibitors; Female; Hemodiafiltration; Humans; Kidney Diseases; Male; Middle Aged; Phosphatidylserines; Protein Kinase C-delta; Renal Dialysis; Ritanserin; Serotonin 5-HT2 Receptor Antagonists; Serotonin Antagonists

2008
The structure of human serotonin 2c G-protein-coupled receptor bound to agonists and antagonists.
    Journal of molecular graphics & modelling, 2008, Volume: 27, Issue:1

    Topics: Amino Acid Sequence; Binding Sites; Humans; Kinetics; Metergoline; Methiothepin; Molecular Sequence Data; Mutagenesis; Protein Structure, Secondary; Psilocybin; Receptor, Serotonin, 5-HT2B; Receptor, Serotonin, 5-HT2C; Ritanserin; Serotonin; Serotonin 5-HT2 Receptor Agonists; Serotonin 5-HT2 Receptor Antagonists; Structure-Activity Relationship; Thermodynamics

2008
Human embryonic stem cell-derived oligodendrocyte progenitor cells express the serotonin receptor and are susceptible to JC virus infection.
    Journal of virology, 2008, Volume: 82, Issue:17

    Topics: Antibodies, Monoclonal; Antigens; Biomarkers; Cell Line; Embryonic Stem Cells; Fetus; Humans; JC Virus; Ketanserin; Leukoencephalopathy, Progressive Multifocal; Oligodendroglia; Proteoglycans; Receptor, Serotonin, 5-HT2A; Ritanserin; Serotonin 5-HT2 Receptor Antagonists; Serotonin Antagonists

2008
Discriminative stimulus effects of 1-(2,5-dimethoxy-4-methylphenyl)-2-aminopropane in rhesus monkeys: antagonism and apparent pA2 analyses.
    The Journal of pharmacology and experimental therapeutics, 2009, Volume: 328, Issue:3

    Topics: Animals; DOM 2,5-Dimethoxy-4-Methylamphetamine; Dose-Response Relationship, Drug; Electroshock; Fluorobenzenes; Hallucinogens; Ketanserin; Macaca mulatta; Phenethylamines; Piperidines; Reaction Time; Receptor, Serotonin, 5-HT2A; Receptor, Serotonin, 5-HT2C; Receptors, Serotonin; Regression Analysis; Ritanserin; Serotonin Antagonists; Serotonin Receptor Agonists

2009
The group III mGlu receptor agonist ACPT-I exerts anxiolytic-like but not antidepressant-like effects, mediated by the serotonergic and GABA-ergic systems.
    Neuropharmacology, 2009, Volume: 57, Issue:3

    Topics: Animals; Anti-Anxiety Agents; Antidepressive Agents; Anxiety; Cyclopentanes; Depression; Flumazenil; GABA-A Receptor Antagonists; gamma-Aminobutyric Acid; Injections, Intraperitoneal; Male; Piperazines; Pyridines; Rats; Rats, Wistar; Receptors, Metabotropic Glutamate; Ritanserin; Serotonin; Serotonin 5-HT1 Receptor Antagonists; Serotonin 5-HT2 Receptor Antagonists; Serotonin Antagonists; Stress, Psychological; Tricarboxylic Acids

2009
Discriminative stimulus effects of 1-(2,5-dimethoxy-4-methylphenyl)-2-aminopropane (DOM), ketanserin, and (R)-(+)-{alpha}-(2,3-dimethoxyphenyl)-1-[2-(4-fluorophenyl)ethyl]-4-pipidinemethanol (MDL100907) in rats.
    The Journal of pharmacology and experimental therapeutics, 2009, Volume: 331, Issue:2

    Topics: Analgesics, Opioid; Anesthetics, Dissociative; Animals; Conditioning, Operant; Discrimination, Psychological; DOM 2,5-Dimethoxy-4-Methylamphetamine; Dose-Response Relationship, Drug; Excitatory Amino Acid Antagonists; Fluorobenzenes; Ketamine; Ketanserin; Male; Morphine; Phencyclidine; Piperidines; Rats; Rats, Sprague-Dawley; Receptor, Serotonin, 5-HT2A; Receptors, Adrenergic, alpha-1; Ritanserin; Serotonin Antagonists; Serotonin Receptor Agonists

2009
Inhibitory effect of serotonin antagonists on JC virus propagation in a carrier culture of human neuroblastoma cells.
    Microbiology and immunology, 2009, Volume: 53, Issue:9

    Topics: Cell Line, Tumor; Down-Regulation; Humans; JC Virus; Ketanserin; Neuroblastoma; Receptor, Serotonin, 5-HT2A; Ritanserin; Serotonin 5-HT2 Receptor Antagonists; Serotonin Antagonists; Virus Cultivation; Virus Replication

2009
Signal transduction and modulating pathways in tryptamine-evoked vasopressor responses of the rat isolated perfused mesenteric bed.
    Vascular pharmacology, 2013, Volume: 58, Issue:1-2

    Topics: Animals; Dinoprostone; Dose-Response Relationship, Drug; Male; Mesenteric Arteries; Nitric Oxide; Rats; Rats, Sprague-Dawley; Receptor, Serotonin, 5-HT2A; rho-Associated Kinases; Ritanserin; Serotonin 5-HT2 Receptor Antagonists; Signal Transduction; Tryptamines; Vasoconstriction; Vasodilation

2013
5-HT2A receptor antagonists inhibit hepatic stellate cell activation and facilitate apoptosis.
    Liver international : official journal of the International Association for the Study of the Liver, 2013, Volume: 33, Issue:4

    Topics: Actins; Animals; Apoptosis; Cell Line; Cell Survival; Collagen Type I; Dose-Response Relationship, Drug; Hepatic Stellate Cells; Humans; Ketanserin; Liver Cirrhosis, Experimental; Rats; Rats, Sprague-Dawley; Reactive Oxygen Species; Receptor, Serotonin, 5-HT2A; Ritanserin; RNA, Messenger; Serotonin 5-HT2 Receptor Antagonists; Smad2 Protein; Smad3 Protein; Succinates; Thioacetamide; Time Factors; Transforming Growth Factor beta; Wound Healing

2013
Captodiamine, a putative antidepressant, enhances hypothalamic BDNF expression in vivo by synergistic 5-HT2c receptor antagonism and sigma-1 receptor agonism.
    Journal of psychopharmacology (Oxford, England), 2013, Volume: 27, Issue:10

    Topics: Animals; Antidepressive Agents; Brain-Derived Neurotrophic Factor; Carbazoles; Corticotropin-Releasing Hormone; CREB-Binding Protein; Disks Large Homolog 4 Protein; Drug Interactions; Ethylamines; Gene Expression Regulation; Guanylate Kinases; Hypothalamus; Male; Membrane Proteins; Mice; Paraventricular Hypothalamic Nucleus; Phosphorylation; Receptor, Serotonin, 5-HT2C; Receptors, sigma; Ritanserin; Serotonin 5-HT2 Receptor Antagonists; Sigma-1 Receptor; Signal Transduction; Sulfides; Synapsins

2013
Serotonin-1A receptor stimulation mediates effects of a metabotropic glutamate 2/3 receptor antagonist, 2S-2-amino-2-(1S,2S-2-carboxycycloprop-1-yl)-3-(xanth-9-yl)propanoic acid (LY341495), and an N-methyl-D-aspartate receptor antagonist, ketamine, in the
    Psychopharmacology, 2014, Volume: 231, Issue:11

    Topics: Amino Acids; Animals; Antidepressive Agents; Dioxoles; Enzyme Inhibitors; Excitatory Amino Acid Antagonists; Feeding Behavior; Fenclonine; Ketamine; Male; Mice, Inbred C57BL; Neuropsychological Tests; Piperazines; Piperidines; Pyridines; Quinoxalines; Receptors, AMPA; Receptors, Metabotropic Glutamate; Receptors, N-Methyl-D-Aspartate; Ritanserin; Serotonin 5-HT1 Receptor Antagonists; Serotonin 5-HT2 Receptor Antagonists; Tryptophan Hydroxylase; Xanthenes

2014
Effect of 5-HT(2A) receptor antagonists on blood flow in the carotid vessels upon elevation of serotonin level.
    Bulletin of experimental biology and medicine, 2014, Volume: 157, Issue:3

    Topics: Animals; Animals, Outbred Strains; Carotid Arteries; Drug Evaluation, Preclinical; Ketanserin; Male; Rats; Regional Blood Flow; Ritanserin; Serotonin; Serotonin 5-HT2 Receptor Antagonists; Vasoconstriction

2014
5-HT2A/C receptors do not mediate the attenuation of compulsive checking by mCPP in the quinpirole sensitization rat model of obsessive-compulsive disorder (OCD).
    Behavioural brain research, 2015, Feb-15, Volume: 279

    Topics: Animals; Compulsive Behavior; Disease Models, Animal; Male; Obsessive-Compulsive Disorder; Piperazines; Quinpirole; Rats; Rats, Long-Evans; Receptor, Serotonin, 5-HT2A; Receptor, Serotonin, 5-HT2C; Ritanserin; Serotonin 5-HT2 Receptor Antagonists; Serotonin Receptor Agonists

2015
Activation of 5-HT2A/C receptor reduces glycine receptor-mediated currents in cultured auditory cortical neurons.
    Amino acids, 2016, Volume: 48, Issue:2

    Topics: Amphetamines; Animals; Auditory Cortex; Cells, Cultured; GTP-Binding Proteins; Guanosine Diphosphate; Ion Channels; Microtubules; Neurons; Nocodazole; Patch-Clamp Techniques; Rats; Rats, Sprague-Dawley; Receptor, Serotonin, 5-HT2A; Receptor, Serotonin, 5-HT2C; Receptors, Glycine; Risperidone; Ritanserin; Serotonin 5-HT2 Receptor Agonists; Serotonin 5-HT2 Receptor Antagonists; Strychnine; Thionucleotides; Tubulin Modulators

2016
Abuse potential of methylenedioxymethamphetamine (MDMA) and its derivatives in zebrafish: role of serotonin 5HT2-type receptors.
    Psychopharmacology, 2016, Volume: 233, Issue:15-16

    Topics: Amphetamines; Animals; Behavior, Animal; Conditioning, Psychological; DOM 2,5-Dimethoxy-4-Methylamphetamine; Female; Hallucinogens; Male; N-Methyl-3,4-methylenedioxyamphetamine; Receptors, Serotonin, 5-HT2; Reinforcement, Psychology; Reward; Ritanserin; Serotonin 5-HT2 Receptor Antagonists; Serotonin Receptor Agonists; Zebrafish

2016
Atypical antipsychotic clozapine reversed deficit on prepulse inhibition of the acoustic startle reflex produced by microinjection of DOI into the inferior colliculus in rats.
    Behavioural brain research, 2017, 05-15, Volume: 325, Issue:Pt A

    Topics: Amphetamines; Animals; Antipsychotic Agents; Clozapine; Inferior Colliculi; Male; Microinjections; Prepulse Inhibition; Rats, Wistar; Receptor, Serotonin, 5-HT2A; Ritanserin; Serotonin 5-HT2 Receptor Agonists; Serotonin 5-HT2 Receptor Antagonists

2017
5-HT
    Cell, 2018, 02-08, Volume: 172, Issue:4

    Topics: Ergotamine; HEK293 Cells; Humans; Obesity; Protein Domains; Receptor, Serotonin, 5-HT2C; Ritanserin; Schizophrenia; Serotonin 5-HT2 Receptor Agonists; Serotonin 5-HT2 Receptor Antagonists; Structure-Activity Relationship; Substance-Related Disorders

2018
Ritanserin blocks Ca
    Acta pharmacologica Sinica, 2020, Volume: 41, Issue:9

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Arteries; Binding Sites; Calcium Channels, L-Type; Electrophysiological Phenomena; Ketanserin; Male; Molecular Docking Simulation; Muscle, Smooth, Vascular; Myocytes, Smooth Muscle; Protein Binding; Rats, Wistar; Ritanserin; Serotonin 5-HT2 Receptor Antagonists; Vasoconstriction

2020
Risperidone and 5-HT2A Receptor Antagonists Attenuate and Reverse Cocaine-Induced Hyperthermia in Rats.
    The international journal of neuropsychopharmacology, 2020, 12-29, Volume: 23, Issue:12

    Topics: Animals; Benzazepines; Cocaine; Disease Models, Animal; Dopamine Antagonists; Dopamine Uptake Inhibitors; Haloperidol; Hyperthermia; Ketanserin; Male; Rats; Rats, Wistar; Risperidone; Ritanserin; Serotonin 5-HT2 Receptor Antagonists

2020