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ritanserin and 1-(3-chlorophenyl)piperazine

ritanserin has been researched along with 1-(3-chlorophenyl)piperazine in 26 studies

Research

Studies (26)

TimeframeStudies, this research(%)All Research%
pre-19901 (3.85)18.7374
1990's14 (53.85)18.2507
2000's10 (38.46)29.6817
2010's1 (3.85)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Hamblin, MW; Monsma, FJ; Shen, Y; Sibley, DR; Ward, RP1
Hamblin, MW; Jose, PA; Metcalf, MA; Monsma, FJ; Shen, Y; Sibley, DR1
Audia, JE; Baez, M; Cohen, ML; Kursar, JD; Lucaites, VL; Nelson, DL; Nissen, JS; Schenck, KW; Wainscott, DB1
Baez, M; Kursar, JD; Lucaites, VL; Nelson, DL; Sasso, DA; Wainscott, DB1
Glennon, RA1
Benwell, K; Bickerdike, M; Kennett, G; Knight, AR; Misra, A; Quirk, K; Revell, D1
Cleves, AE; Jain, AN; Kirshner, D; Langham, JJ; Spitzer, R1
Aulakh, CS; Hill, JL; Murphy, DL1
Charney, DS; D'Amico, C; Heninger, GR; Krystal, JH; Price, LH; Seibyl, JP; Woods, SW1
Aghajanian, GK; Sheldon, PW1
Brownfield, MS; Rittenhouse, PA; Saydoff, JA; van de Kar, LD1
Borsini, F; D'Aranno, V; Lecci, A; Mancinelli, A; Meli, A; Stasi, MA; Volterra, G1
Broekkamp, CL; Jenck, F; Van Delft, AM1
Bagdy, G; Hill, J; Murphy, DL; Szemeredi, K; Zukowska-Grojec, Z1
Kennaway, DJ; Moyer, RW1
Bell, CJ; Malizia, AL; Nutt, DJ1
Aerts, N; Clincke, G; Meert, TF; Melis, W1
Bergqvist, PB; Blier, P; Dong, J1
Fernández, MM; Martín, ML; Morán, A; San Román, L1
Sugimoto, Y; Yamada, J1
Abi-Dargham, A; Abi-Saab, W; Charney, DS; D'Souza, DC; Erdos, JP; Gueorgueva, R; Heninger, GR; Karper, LP; Krystal, JH; Rajhans, S; Seibyl, JP; Wong, ML1
Calama, E; Martín, ML; Morán, A; Ortiz de Urbina, AV; San Román, L2
Kenis, G; Kim, YK; Kubera, M; Lasoń, W; Maes, M1
de Leeuw, AS; Westenberg, HG1
Dvorkin-Gheva, A; Johnson, E; Szechtman, H; Tucci, MC; Wong, M1

Reviews

2 review(s) available for ritanserin and 1-(3-chlorophenyl)piperazine

ArticleYear
Higher-end serotonin receptors: 5-HT(5), 5-HT(6), and 5-HT(7).
    Journal of medicinal chemistry, 2003, Jul-03, Volume: 46, Issue:14

    Topics: Animals; Humans; Ligands; Receptors, Serotonin; Serotonin Agents; Serotonin Antagonists; Serotonin Receptor Agonists

2003
Brain mechanisms of social anxiety disorder.
    The Journal of clinical psychiatry, 1998, Volume: 59 Suppl 17

    Topics: Animals; Brain; Caffeine; Carbon Dioxide; Cholecystokinin; Dopamine; Fear; Fenfluramine; Humans; Panic Disorder; Paroxetine; Phobic Disorders; Piperazines; Rats; Ritanserin; Selective Serotonin Reuptake Inhibitors; Serotonin; Tomography, Emission-Computed

1998

Trials

3 trial(s) available for ritanserin and 1-(3-chlorophenyl)piperazine

ArticleYear
Effects of ritanserin on the behavioral, neuroendocrine, and cardiovascular responses to meta-chlorophenylpiperazine in healthy human subjects.
    Psychiatry research, 1991, Volume: 38, Issue:3

    Topics: Adult; Anxiety; Data Interpretation, Statistical; Double-Blind Method; Growth Hormone; Humans; Hydrocortisone; Male; Personality Inventory; Piperazines; Placebos; Prolactin; Receptors, Serotonin; Ritanserin

1991
Ritanserin antagonism of m-chlorophenylpiperazine effects in neuroleptic-free schizophrenics patients: support for serotonin-2 receptor modulation of schizophrenia symptoms.
    Psychopharmacology, 2002, Volume: 162, Issue:1

    Topics: Adult; Antipsychotic Agents; Cross-Over Studies; Double-Blind Method; Humans; Male; Middle Aged; Piperazines; Psychiatric Status Rating Scales; Receptors, Serotonin; Regression Analysis; Ritanserin; Schizophrenia; Serotonin Antagonists; Serotonin Receptor Agonists

2002
Hypersensitivity of 5-HT2 receptors in OCD patients. An increased prolactin response after a challenge with meta-chlorophenylpiperazine and pre-treatment with ritanserin and placebo.
    Journal of psychiatric research, 2008, Volume: 42, Issue:11

    Topics: Adult; Dose-Response Relationship, Drug; Female; Humans; Hydrocortisone; Male; Middle Aged; Obsessive-Compulsive Disorder; Piperazines; Premedication; Prolactin; Receptor, Serotonin, 5-HT2C; Ritanserin; Serotonin Antagonists; Young Adult

2008

Other Studies

21 other study(ies) available for ritanserin and 1-(3-chlorophenyl)piperazine

ArticleYear
Cloning and expression of a novel serotonin receptor with high affinity for tricyclic psychotropic drugs.
    Molecular pharmacology, 1993, Volume: 43, Issue:3

    Topics: Amino Acid Sequence; Animals; Base Sequence; Binding, Competitive; Blotting, Northern; Brain Chemistry; Cell Line; Cloning, Molecular; DNA; GTP-Binding Proteins; Lysergic Acid Diethylamide; Molecular Sequence Data; Polymerase Chain Reaction; Psychotropic Drugs; Rats; Receptors, Serotonin; RNA; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Transfection

1993
Molecular cloning and expression of a 5-hydroxytryptamine7 serotonin receptor subtype.
    The Journal of biological chemistry, 1993, Aug-25, Volume: 268, Issue:24

    Topics: Amino Acid Sequence; Animals; Base Sequence; Binding, Competitive; Cell Line; Cell Membrane; Cloning, Molecular; Cyclic AMP; Gene Expression; Kidney Tubules, Proximal; Lysergic Acid Diethylamide; Molecular Sequence Data; Oligodeoxyribonucleotides; Polymerase Chain Reaction; Radioligand Assay; Rats; Receptors, Serotonin; Recombinant Proteins; Serotonin; Transfection

1993
Pharmacological characteristics of the newly cloned rat 5-hydroxytryptamine2F receptor.
    Molecular pharmacology, 1993, Volume: 43, Issue:3

    Topics: Animals; Binding Sites; Cell Line; Cloning, Molecular; Gastric Fundus; Inositol 1,4,5-Trisphosphate; Male; Muscle Contraction; Muscle, Smooth; Radioligand Assay; Rats; Rats, Wistar; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Temperature

1993
[3H]Rauwolscine: an antagonist radioligand for the cloned human 5-hydroxytryptamine2b (5-HT2B) receptor.
    Naunyn-Schmiedeberg's archives of pharmacology, 1998, Volume: 357, Issue:1

    Topics: Adrenergic alpha-Antagonists; Benzofurans; Binding, Competitive; Cell Line; Cloning, Molecular; Humans; Imidazoles; Radioligand Assay; Receptor, Serotonin, 5-HT2B; Receptors, Serotonin; Serotonin Antagonists; Transfection; Tritium; Yohimbine

1998
Pharmacological characterisation of the agonist radioligand binding site of 5-HT(2A), 5-HT(2B) and 5-HT(2C) receptors.
    Naunyn-Schmiedeberg's archives of pharmacology, 2004, Volume: 370, Issue:2

    Topics: Binding Sites; Binding, Competitive; Cell Line; Humans; Radioligand Assay; Receptor, Serotonin, 5-HT2A; Receptor, Serotonin, 5-HT2B; Receptor, Serotonin, 5-HT2C; Recombinant Proteins; Serotonin 5-HT2 Receptor Agonists; Serotonin 5-HT2 Receptor Antagonists; Serotonin Antagonists; Serotonin Receptor Agonists

2004
Physical binding pocket induction for affinity prediction.
    Journal of medicinal chemistry, 2009, Oct-08, Volume: 52, Issue:19

    Topics: Binding Sites; Ligands; Models, Molecular; Neural Networks, Computer; Peptide Fragments; Protein Binding; Receptor, Serotonin, 5-HT1A

2009
Effects of various serotonin receptor subtype-selective antagonists alone and on m-chlorophenylpiperazine-induced neuroendocrine changes in rats.
    The Journal of pharmacology and experimental therapeutics, 1992, Volume: 263, Issue:2

    Topics: Animals; Corticosterone; Ergolines; Male; Metergoline; Mianserin; Neurosecretory Systems; Piperazines; Prolactin; Rats; Rats, Wistar; Receptors, Serotonin; Ritanserin; Serotonin Antagonists; Spiperone

1992
Excitatory responses to serotonin (5-HT) in neurons of the rat piriform cortex: evidence for mediation by 5-HT1C receptors in pyramidal cells and 5-HT2 receptors in interneurons.
    Synapse (New York, N.Y.), 1991, Volume: 9, Issue:3

    Topics: Animals; Electrophysiology; Ergolines; Interneurons; Limbic System; Male; Neurons; Piperazines; Rats; Rats, Inbred Strains; Receptors, Serotonin; Ritanserin; Serotonin; Serotonin Antagonists; Spiperone

1991
Enhanced serotonergic transmission stimulates oxytocin secretion in conscious male rats.
    The Journal of pharmacology and experimental therapeutics, 1991, Volume: 257, Issue:1

    Topics: Animals; Male; Oxytocin; Piperazines; Piperidines; Rats; Rats, Inbred Strains; Receptors, Serotonin; Ritanserin; Serotonin; Synaptic Transmission

1991
Effect of serotoninergic drugs on stress-induced hyperthermia (SIH) in mice.
    Journal of neural transmission. General section, 1990, Volume: 82, Issue:3

    Topics: 5,7-Dihydroxytryptamine; 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Anti-Anxiety Agents; Body Temperature Regulation; Buspirone; Diazepam; Ergolines; Fenclonine; Fever; Flumazenil; Imidazoles; Male; Mice; Ondansetron; Piperazines; Piperidines; Ritanserin; Serotonin; Serotonin Antagonists; Stress, Psychological; Tetrahydronaphthalenes

1990
5-HT1C receptors in the serotonergic control of periaqueductal gray induced aversion in rats.
    Psychopharmacology, 1990, Volume: 100, Issue:3

    Topics: Amphetamines; Animals; Cyproheptadine; Indoles; Ketanserin; Male; Periaqueductal Gray; Piperazines; Piperidines; Rats; Rats, Inbred Strains; Receptors, Serotonin; Reinforcement, Psychology; Ritanserin; Serotonin; Serotonin Antagonists

1990
M-chlorophenylpiperazine increases blood pressure and heart rate in pithed and conscious rats.
    Life sciences, 1987, Aug-10, Volume: 41, Issue:6

    Topics: Adrenal Medulla; Animals; Blood Pressure; Brain; Heart Rate; Kinetics; Male; Metergoline; Piperazines; Piperidines; Rats; Rats, Inbred Strains; Receptors, Serotonin; Ritanserin; Serotonin Antagonists; Spinal Cord

1987
Serotonin 5-HT2c agonists mimic the effect of light pulses on circadian rhythms.
    Brain research, 1998, Sep-28, Volume: 806, Issue:2

    Topics: Amphetamines; Animals; Body Temperature; Circadian Rhythm; Ketanserin; Light; Male; Melatonin; Periodicity; Photic Stimulation; Piperazines; Proto-Oncogene Proteins c-fos; Rats; Rats, Wistar; Ritanserin; Serotonin Antagonists; Serotonin Receptor Agonists; Suprachiasmatic Nucleus

1998
Antagonism of meta-chlorophenylpiperazine-induced inhibition of exploratory activity in an emergence procedure, the open field test, in rats.
    Behavioural pharmacology, 1997, Volume: 8, Issue:4

    Topics: Adrenergic alpha-Antagonists; Animals; Behavior, Animal; Dose-Response Relationship, Drug; Injections, Intraperitoneal; Injections, Intravenous; Injections, Subcutaneous; Male; Methysergide; Mianserin; Mirtazapine; Piperazines; Pizotyline; Rats; Rats, Wistar; Ritanserin; Serotonin Antagonists; Serotonin Receptor Agonists

1997
Effect of atypical antipsychotic drugs on 5-HT2 receptors in the rat orbito-frontal cortex: an in vivo electrophysiological study.
    Psychopharmacology, 1999, Volume: 143, Issue:1

    Topics: Amphetamines; Animals; Antipsychotic Agents; Bicuculline; Clozapine; Electrophysiology; GABA Antagonists; Iontophoresis; Male; Neurons; Piperazines; Prefrontal Cortex; Rats; Rats, Sprague-Dawley; Receptor, Serotonin, 5-HT2A; Receptors, GABA-A; Receptors, Serotonin; Risperidone; Ritanserin; Serotonin Antagonists; Serotonin Receptor Agonists

1999
Mesenteric vasoconstrictor response to 5-hydroxytryptamine in the in situ blood autoperfused rat mesentery: involvement of 5-HT(2B) and/or 5-HT(2C) receptor activation.
    European journal of pharmacology, 2000, Aug-04, Volume: 401, Issue:2

    Topics: Amphetamines; Animals; Biguanides; Dose-Response Relationship, Drug; Enalapril; Indoles; Indomethacin; Male; Mesenteric Arteries; Mesentery; Perfusion; Piperazines; Prazosin; Propranolol; Pyridines; Rats; Rats, Wistar; Receptor, Serotonin, 5-HT2B; Receptor, Serotonin, 5-HT2C; Receptors, Serotonin; Ritanserin; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Splanchnic Circulation; Vasoconstriction

2000
The 5-HT(2C/2B) receptor agonist, m-chlorophenylpiperazine, increases plasma glucagon levels in rats.
    European journal of pharmacology, 2000, Oct-06, Volume: 406, Issue:1

    Topics: Adrenal Medulla; Animals; Blood Glucose; Dose-Response Relationship, Drug; Glucagon; Ketanserin; Male; Piperazines; Rats; Rats, Sprague-Dawley; Receptor, Serotonin, 5-HT2A; Receptor, Serotonin, 5-HT2B; Receptor, Serotonin, 5-HT2C; Receptors, Serotonin; Ritanserin; Serotonin Antagonists; Serotonin Receptor Agonists; Time Factors

2000
Vasoconstrictor responses to 5-hydroxytryptamine in the autoperfused hindquarters of spontaneously hypertensive rats.
    Pharmacology, 2004, Volume: 71, Issue:2

    Topics: Animals; Dose-Response Relationship, Drug; Hindlimb; Indoles; Injections, Intra-Arterial; Injections, Intravenous; Male; Perfusion; Piperazines; Prazosin; Pyridines; Rats; Rats, Inbred SHR; Rats, Wistar; Receptor, Serotonin, 5-HT1A; Receptor, Serotonin, 5-HT2A; Receptor, Serotonin, 5-HT2B; Receptor, Serotonin, 5-HT2C; Receptors, Serotonin, 5-HT2; Regional Blood Flow; Ritanserin; Serotonin; Serotonin 5-HT1 Receptor Antagonists; Serotonin 5-HT2 Receptor Agonists; Serotonin 5-HT2 Receptor Antagonists; Serotonin Receptor Agonists; Spiperone; Thiophenes; Vasoconstriction

2004
Effects of serotonin and serotonergic agonists and antagonists on the production of tumor necrosis factor alpha and interleukin-6.
    Psychiatry research, 2005, Apr-30, Volume: 134, Issue:3

    Topics: Adult; Depressive Disorder; Dose-Response Relationship, Drug; Female; Fenclonine; Humans; Immunocompetence; Interleukin-6; Male; Middle Aged; Piperazines; Receptor, Serotonin, 5-HT1A; Receptor, Serotonin, 5-HT2A; Receptor, Serotonin, 5-HT2B; Receptor, Serotonin, 5-HT2C; Ritanserin; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Tumor Necrosis Factor-alpha

2005
Effect of 5-hydroxytryptamine on neurogenic vasoconstriction in the isolated, autoperfused hindquarters of the rat.
    Clinical and experimental pharmacology & physiology, 2005, Volume: 32, Issue:10

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Biguanides; Biphenyl Compounds; Dose-Response Relationship, Drug; Electric Stimulation; Hindlimb; In Vitro Techniques; Infusions, Intravenous; Male; Methiothepin; Oxadiazoles; Perfusion; Piperazines; Pressure; Quinoxalines; Rats; Rats, Wistar; Ritanserin; Serotonin; Serotonin 5-HT1 Receptor Agonists; Serotonin 5-HT2 Receptor Agonists; Serotonin 5-HT3 Receptor Agonists; Serotonin Agents; Serotonin Antagonists; Serotonin Receptor Agonists; Tryptamines; Vasoconstriction

2005
5-HT2A/C receptors do not mediate the attenuation of compulsive checking by mCPP in the quinpirole sensitization rat model of obsessive-compulsive disorder (OCD).
    Behavioural brain research, 2015, Feb-15, Volume: 279

    Topics: Animals; Compulsive Behavior; Disease Models, Animal; Male; Obsessive-Compulsive Disorder; Piperazines; Quinpirole; Rats; Rats, Long-Evans; Receptor, Serotonin, 5-HT2A; Receptor, Serotonin, 5-HT2C; Ritanserin; Serotonin 5-HT2 Receptor Antagonists; Serotonin Receptor Agonists

2015