Page last updated: 2024-08-23

rimcazole and pentazocine

rimcazole has been researched along with pentazocine in 14 studies

Research

Studies (14)

TimeframeStudies, this research(%)All Research%
pre-19903 (21.43)18.7374
1990's7 (50.00)18.2507
2000's4 (28.57)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
DeHaven-Hudkins, DL; Fleissner, LC1
DeHaven-Hudkins, DL; Fleissner, LC; Ford-Rice, FY1
della Puppa, A; London, ED1
Cook, L; Steinfels, GF; Tam, SW1
Su, TP; Vaupel, DB1
Appleyard, SM; Chavkin, C; Connor, M; Patterson, TA1
Matsunaga, KH; Matsuno, K; Mita, S1
Kobayashi, T; Matsuno, K; Mita, S1
Eaton, MJ; Lookingland, KJ; Moore, KE1
Kamei, J1
Devaud, LL1
Achison, M; Boylan, MT; Hupp, TR; Spruce, BA1
Dhir, A; Kulkarni, SK2

Reviews

1 review(s) available for rimcazole and pentazocine

ArticleYear
[Possible role of sigma-receptors in the regulation of cough reflex, gastrointestinal and retinal function].
    Nihon yakurigaku zasshi. Folia pharmacologica Japonica, 1999, Volume: 114, Issue:1

    Topics: Animals; Anti-Ulcer Agents; Antitussive Agents; Carbazoles; Guanidines; Haloperidol; Humans; Ligands; Pentazocine; Phenazocine; Receptors, N-Methyl-D-Aspartate; Receptors, sigma; Retinal Diseases

1999

Other Studies

13 other study(ies) available for rimcazole and pentazocine

ArticleYear
Competitive interactions at [3H]1,3-di(2-tolyl)guanidine (DTG)-defined sigma recognition sites in guinea pig brain.
    Life sciences, 1992, Volume: 50, Issue:9

    Topics: Animals; Antipsychotic Agents; Binding, Competitive; Carbazoles; Dopamine Agents; Guanidines; Guinea Pigs; Haloperidol; In Vitro Techniques; Kinetics; Male; Pentazocine; Piperidines; Radioligand Assay; Receptors, Opioid; Receptors, sigma

1992
Characterization of the binding of [3H](+)-pentazocine to sigma recognition sites in guinea pig brain.
    European journal of pharmacology, 1992, Dec-01, Volume: 227, Issue:4

    Topics: Animals; Antipsychotic Agents; Binding Sites; Binding, Competitive; Brain; Carbazoles; Dopamine Agents; Guinea Pigs; Haloperidol; Kinetics; Male; Pentazocine; Piperidines; Receptors, sigma

1992
Cerebral metabolic effects of sigma ligands in the rat.
    Brain research, 1989, Dec-29, Volume: 505, Issue:2

    Topics: Animals; Autoradiography; Blood Pressure; Brain; Carbazoles; Deoxyglucose; Heart Rate; Male; Pentazocine; Pyrimidines; Rats; Rats, Inbred F344; Receptors, Opioid; Receptors, sigma

1989
Electrophysiological effects of selective sigma-receptor agonists, antagonists, and the selective phencyclidine receptor agonist MK-801 on midbrain dopamine neurons.
    Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology, 1989, Volume: 2, Issue:3

    Topics: Animals; Anti-Anxiety Agents; Anticonvulsants; Antipsychotic Agents; Carbazoles; Cell Membrane; Dibenzocycloheptenes; Dizocilpine Maleate; Dopamine; Dopamine Agents; Male; Neurons; Pentazocine; Phencyclidine; Piperidines; Pyrimidines; Rats; Rats, Inbred Strains; Receptors, Neurotransmitter; Receptors, Opioid; Receptors, Phencyclidine; Receptors, sigma; Substantia Nigra

1989
Guinea-pig vas deferens preparation may contain both receptors and phencyclidine receptors.
    European journal of pharmacology, 1987, Jul-02, Volume: 139, Issue:1

    Topics: Animals; Antipsychotic Agents; Carbazoles; Electric Stimulation; Guinea Pigs; Haloperidol; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth; Pentazocine; Receptors, Neurotransmitter; Receptors, Phencyclidine; Vas Deferens

1987
Oocytes from Xenopus laevis contain an intrinsic sigma 2-like binding site.
    Neuroscience letters, 1994, Oct-24, Volume: 180, Issue:2

    Topics: Animals; Binding Sites; Binding, Competitive; Carbazoles; Dextromethorphan; Female; Guanidines; Haloperidol; Liver; Mazindol; Oocytes; Pentazocine; Phenazocine; Piperazines; Piperidines; Radioligand Assay; Rats; Receptors, sigma; Xenopus laevis; Zinc

1994
Acute effects of sigma ligands on the extracellular DOPAC level in rat frontal cortex and striatum.
    Neurochemical research, 1995, Volume: 20, Issue:2

    Topics: 3,4-Dihydroxyphenylacetic Acid; Animals; Anticonvulsants; Antipsychotic Agents; Carbazoles; Corpus Striatum; Extracellular Space; Frontal Lobe; Guanidines; Kinetics; Ligands; Male; Microdialysis; Pentazocine; Phenazocine; Piperidines; Rats; Rats, Wistar; Receptors, sigma; Time Factors

1995
Involvement of sigma-receptors in the increase in contraction of mouse vas deferens induced by exogenous ATP.
    The Journal of pharmacy and pharmacology, 1996, Volume: 48, Issue:1

    Topics: Adenosine Triphosphate; Analgesics, Opioid; Animals; Anticonvulsants; Antipsychotic Agents; Carbazoles; Dopamine Agonists; Dopamine Antagonists; Dose-Response Relationship, Drug; Drug Synergism; Guanidines; Haloperidol; Ligands; Male; Mice; Muscle Contraction; Muscle, Smooth; Pentazocine; Phenazocine; Piperidines; Receptors, sigma; Regression Analysis; Structure-Activity Relationship; Vas Deferens

1996
The sigma ligand rimcazole activates noradrenergic neurons projecting to the paraventricular nucleus and increases corticosterone secretion in rats.
    Brain research, 1996, Sep-16, Volume: 733, Issue:2

    Topics: 3,4-Dihydroxyphenylacetic Acid; Analysis of Variance; Animals; Antipsychotic Agents; Carbazoles; Corticosterone; Dopamine; Dose-Response Relationship, Drug; Kinetics; Male; Methoxyhydroxyphenylglycol; Neurons; Norepinephrine; Paraventricular Hypothalamic Nucleus; Pentazocine; Radioimmunoassay; Rats; Receptors, sigma; Sensitivity and Specificity

1996
Effects of ethanol or rimcazole on dizocilpine maleate-induced behaviors in male and female rats.
    Alcohol (Fayetteville, N.Y.), 2003, Volume: 29, Issue:2

    Topics: Animals; Antipsychotic Agents; Behavior, Animal; Binding, Competitive; Carbazoles; Central Nervous System Depressants; Dizocilpine Maleate; Drug Interactions; Ethanol; Female; Injections, Intraperitoneal; Male; Motor Activity; Narcotics; Neuroprotective Agents; Pentazocine; Rats; Rats, Sprague-Dawley; Receptors, sigma; Sex Characteristics; Stereotyped Behavior

2003
HIF-1alpha contributes to tumour-selective killing by the sigma receptor antagonist rimcazole.
    Oncogene, 2007, Feb-22, Volume: 26, Issue:8

    Topics: Apoptosis; Carbazoles; Cell Line, Tumor; Epithelial Cells; Fibroblasts; Humans; Hypoxia-Inducible Factor 1, alpha Subunit; Neoplasms; Pentazocine; Receptors, sigma; RNA Interference; Tumor Suppressor Protein p53; Up-Regulation

2007
Involvement of sigma-1 receptor modulation in the antidepressant action of venlafaxine.
    Neuroscience letters, 2007, Jun-15, Volume: 420, Issue:3

    Topics: Analgesics, Opioid; Animals; Antidepressive Agents, Second-Generation; Carbazoles; Cyclohexanols; Depression; Dose-Response Relationship, Drug; Ethylenediamines; Male; Mice; Motor Activity; Neuroprotective Agents; Pentazocine; Receptors, sigma; Sigma-1 Receptor; Swimming; Venlafaxine Hydrochloride

2007
Possible involvement of sigma-1 receptors in the anti-immobility action of bupropion, a dopamine reuptake inhibitor.
    Fundamental & clinical pharmacology, 2008, Volume: 22, Issue:4

    Topics: Analgesics, Opioid; Animals; Antidepressive Agents, Second-Generation; Behavior, Animal; Bupropion; Carbazoles; Dopamine Uptake Inhibitors; Dose-Response Relationship, Drug; Drug Synergism; Ethylenediamines; Male; Mice; Motor Activity; Neuroprotective Agents; Pentazocine; Progesterone; Receptors, sigma; Sigma-1 Receptor; Stress, Psychological

2008