rimcazole has been researched along with pentazocine in 14 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 3 (21.43) | 18.7374 |
1990's | 7 (50.00) | 18.2507 |
2000's | 4 (28.57) | 29.6817 |
2010's | 0 (0.00) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
---|---|
DeHaven-Hudkins, DL; Fleissner, LC | 1 |
DeHaven-Hudkins, DL; Fleissner, LC; Ford-Rice, FY | 1 |
della Puppa, A; London, ED | 1 |
Cook, L; Steinfels, GF; Tam, SW | 1 |
Su, TP; Vaupel, DB | 1 |
Appleyard, SM; Chavkin, C; Connor, M; Patterson, TA | 1 |
Matsunaga, KH; Matsuno, K; Mita, S | 1 |
Kobayashi, T; Matsuno, K; Mita, S | 1 |
Eaton, MJ; Lookingland, KJ; Moore, KE | 1 |
Kamei, J | 1 |
Devaud, LL | 1 |
Achison, M; Boylan, MT; Hupp, TR; Spruce, BA | 1 |
Dhir, A; Kulkarni, SK | 2 |
1 review(s) available for rimcazole and pentazocine
Article | Year |
---|---|
[Possible role of sigma-receptors in the regulation of cough reflex, gastrointestinal and retinal function].
Topics: Animals; Anti-Ulcer Agents; Antitussive Agents; Carbazoles; Guanidines; Haloperidol; Humans; Ligands; Pentazocine; Phenazocine; Receptors, N-Methyl-D-Aspartate; Receptors, sigma; Retinal Diseases | 1999 |
13 other study(ies) available for rimcazole and pentazocine
Article | Year |
---|---|
Competitive interactions at [3H]1,3-di(2-tolyl)guanidine (DTG)-defined sigma recognition sites in guinea pig brain.
Topics: Animals; Antipsychotic Agents; Binding, Competitive; Carbazoles; Dopamine Agents; Guanidines; Guinea Pigs; Haloperidol; In Vitro Techniques; Kinetics; Male; Pentazocine; Piperidines; Radioligand Assay; Receptors, Opioid; Receptors, sigma | 1992 |
Characterization of the binding of [3H](+)-pentazocine to sigma recognition sites in guinea pig brain.
Topics: Animals; Antipsychotic Agents; Binding Sites; Binding, Competitive; Brain; Carbazoles; Dopamine Agents; Guinea Pigs; Haloperidol; Kinetics; Male; Pentazocine; Piperidines; Receptors, sigma | 1992 |
Cerebral metabolic effects of sigma ligands in the rat.
Topics: Animals; Autoradiography; Blood Pressure; Brain; Carbazoles; Deoxyglucose; Heart Rate; Male; Pentazocine; Pyrimidines; Rats; Rats, Inbred F344; Receptors, Opioid; Receptors, sigma | 1989 |
Electrophysiological effects of selective sigma-receptor agonists, antagonists, and the selective phencyclidine receptor agonist MK-801 on midbrain dopamine neurons.
Topics: Animals; Anti-Anxiety Agents; Anticonvulsants; Antipsychotic Agents; Carbazoles; Cell Membrane; Dibenzocycloheptenes; Dizocilpine Maleate; Dopamine; Dopamine Agents; Male; Neurons; Pentazocine; Phencyclidine; Piperidines; Pyrimidines; Rats; Rats, Inbred Strains; Receptors, Neurotransmitter; Receptors, Opioid; Receptors, Phencyclidine; Receptors, sigma; Substantia Nigra | 1989 |
Guinea-pig vas deferens preparation may contain both receptors and phencyclidine receptors.
Topics: Animals; Antipsychotic Agents; Carbazoles; Electric Stimulation; Guinea Pigs; Haloperidol; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth; Pentazocine; Receptors, Neurotransmitter; Receptors, Phencyclidine; Vas Deferens | 1987 |
Oocytes from Xenopus laevis contain an intrinsic sigma 2-like binding site.
Topics: Animals; Binding Sites; Binding, Competitive; Carbazoles; Dextromethorphan; Female; Guanidines; Haloperidol; Liver; Mazindol; Oocytes; Pentazocine; Phenazocine; Piperazines; Piperidines; Radioligand Assay; Rats; Receptors, sigma; Xenopus laevis; Zinc | 1994 |
Acute effects of sigma ligands on the extracellular DOPAC level in rat frontal cortex and striatum.
Topics: 3,4-Dihydroxyphenylacetic Acid; Animals; Anticonvulsants; Antipsychotic Agents; Carbazoles; Corpus Striatum; Extracellular Space; Frontal Lobe; Guanidines; Kinetics; Ligands; Male; Microdialysis; Pentazocine; Phenazocine; Piperidines; Rats; Rats, Wistar; Receptors, sigma; Time Factors | 1995 |
Involvement of sigma-receptors in the increase in contraction of mouse vas deferens induced by exogenous ATP.
Topics: Adenosine Triphosphate; Analgesics, Opioid; Animals; Anticonvulsants; Antipsychotic Agents; Carbazoles; Dopamine Agonists; Dopamine Antagonists; Dose-Response Relationship, Drug; Drug Synergism; Guanidines; Haloperidol; Ligands; Male; Mice; Muscle Contraction; Muscle, Smooth; Pentazocine; Phenazocine; Piperidines; Receptors, sigma; Regression Analysis; Structure-Activity Relationship; Vas Deferens | 1996 |
The sigma ligand rimcazole activates noradrenergic neurons projecting to the paraventricular nucleus and increases corticosterone secretion in rats.
Topics: 3,4-Dihydroxyphenylacetic Acid; Analysis of Variance; Animals; Antipsychotic Agents; Carbazoles; Corticosterone; Dopamine; Dose-Response Relationship, Drug; Kinetics; Male; Methoxyhydroxyphenylglycol; Neurons; Norepinephrine; Paraventricular Hypothalamic Nucleus; Pentazocine; Radioimmunoassay; Rats; Receptors, sigma; Sensitivity and Specificity | 1996 |
Effects of ethanol or rimcazole on dizocilpine maleate-induced behaviors in male and female rats.
Topics: Animals; Antipsychotic Agents; Behavior, Animal; Binding, Competitive; Carbazoles; Central Nervous System Depressants; Dizocilpine Maleate; Drug Interactions; Ethanol; Female; Injections, Intraperitoneal; Male; Motor Activity; Narcotics; Neuroprotective Agents; Pentazocine; Rats; Rats, Sprague-Dawley; Receptors, sigma; Sex Characteristics; Stereotyped Behavior | 2003 |
HIF-1alpha contributes to tumour-selective killing by the sigma receptor antagonist rimcazole.
Topics: Apoptosis; Carbazoles; Cell Line, Tumor; Epithelial Cells; Fibroblasts; Humans; Hypoxia-Inducible Factor 1, alpha Subunit; Neoplasms; Pentazocine; Receptors, sigma; RNA Interference; Tumor Suppressor Protein p53; Up-Regulation | 2007 |
Involvement of sigma-1 receptor modulation in the antidepressant action of venlafaxine.
Topics: Analgesics, Opioid; Animals; Antidepressive Agents, Second-Generation; Carbazoles; Cyclohexanols; Depression; Dose-Response Relationship, Drug; Ethylenediamines; Male; Mice; Motor Activity; Neuroprotective Agents; Pentazocine; Receptors, sigma; Sigma-1 Receptor; Swimming; Venlafaxine Hydrochloride | 2007 |
Possible involvement of sigma-1 receptors in the anti-immobility action of bupropion, a dopamine reuptake inhibitor.
Topics: Analgesics, Opioid; Animals; Antidepressive Agents, Second-Generation; Behavior, Animal; Bupropion; Carbazoles; Dopamine Uptake Inhibitors; Dose-Response Relationship, Drug; Drug Synergism; Ethylenediamines; Male; Mice; Motor Activity; Neuroprotective Agents; Pentazocine; Progesterone; Receptors, sigma; Sigma-1 Receptor; Stress, Psychological | 2008 |