rimcazole has been researched along with cocaine in 11 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 0 (0.00) | 18.7374 |
1990's | 2 (18.18) | 18.2507 |
2000's | 6 (54.55) | 29.6817 |
2010's | 3 (27.27) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
---|---|
Bowen, WD; Husbands, SM; Izenwasser, S; Katz, JL; Kopajtic, T; Newman, AH; Vilner, BJ | 1 |
Cao, J; Husbands, SM; Katz, JL; Kopajtic, T; Newman, AH | 1 |
Bowen, WD; Cao, J; George, C; Husbands, SM; Katz, JL; Kopajtic, T; Kulkarni, SS; Newman, AH; Williams, W | 1 |
Bowen, WD; Husbands, SM; Izenwasser, S; Katz, JL; Loeloff, RJ; Newman, AH; Vilner, BJ | 1 |
Bowen, WD; Cao, JJ; Hewett, KL; Husbands, SM; Matsumoto, RR; Newman, AH; Pouw, B | 1 |
Husbands, SM; Katz, JL; Kopajtic, T; Libby, TA; Newman, AH | 1 |
Blakely, RD; Henry, LK | 1 |
Cao, J; Katz, JL; Kopajtic, T; Newman, AH | 1 |
Bartlett, PJ; Berwick, ZC; Chakraborty, S; Kumar, S; Obukhov, AG; Sturek, M; Thomas, AP; Tune, JD | 1 |
Cao, J; Hiranita, T; Katz, JL; Kohut, SJ; Kopajtic, T; Newman, AH; Soto, PL; Tanda, G | 1 |
Atluri, VSR; Jayant, RD; Kaushik, A; Nair, M; Pilakka-Kanthikeel, S; Tiwari, S; Yndart, A | 1 |
11 other study(ies) available for rimcazole and cocaine
Article | Year |
---|---|
Structure-activity relationships at the monoamine transporters and sigma receptors for a novel series of 9-[3-(cis-3, 5-dimethyl-1-piperazinyl)propyl]carbazole (rimcazole) analogues.
Topics: Aniline Compounds; Animals; Brain; Carbazoles; Carrier Proteins; Dopamine; Dopamine Plasma Membrane Transport Proteins; Dopamine Uptake Inhibitors; Guinea Pigs; In Vitro Techniques; Male; Membrane Glycoproteins; Membrane Transport Proteins; Nerve Tissue Proteins; Norepinephrine Plasma Membrane Transport Proteins; Piperazines; Protein Binding; Rats; Rats, Sprague-Dawley; Receptors, sigma; Serotonin Plasma Membrane Transport Proteins; Structure-Activity Relationship; Symporters | 1999 |
[3-cis-3,5-Dimethyl-(1-piperazinyl)alkyl]-bis-(4'-fluorophenyl)amine analogues as novel probes for the dopamine transporter.
Topics: Animals; Carbazoles; Cocaine; Dopamine Plasma Membrane Transport Proteins; Dopamine Uptake Inhibitors; Membrane Glycoproteins; Membrane Transport Proteins; Molecular Probes; Nerve Tissue Proteins; Piperazines; Rats | 2001 |
Dual probes for the dopamine transporter and sigma1 receptors: novel piperazinyl alkyl-bis(4'-fluorophenyl)amine analogues as potential cocaine-abuse therapeutic agents.
Topics: Animals; Binding, Competitive; Brain; Cocaine-Related Disorders; Crystallography, X-Ray; Dopamine; Dopamine Plasma Membrane Transport Proteins; In Vitro Techniques; Membrane Glycoproteins; Membrane Transport Proteins; Models, Molecular; Nerve Tissue Proteins; Piperazines; Radioligand Assay; Rats; Receptors, sigma; Structure-Activity Relationship | 2003 |
Isothiocyanate derivatives of 9-[3-(cis-3,5-dimethyl-1-piperazinyl)propyl]carbazole (rimcazole): irreversible ligands for the dopamine transporter.
Topics: Animals; Binding Sites; Binding, Competitive; Brain; Carbazoles; Carrier Proteins; Cocaine; Cocaine-Related Disorders; Dopamine; Dopamine Plasma Membrane Transport Proteins; Guinea Pigs; Isothiocyanates; Ligands; Liver; Membrane Glycoproteins; Membrane Transport Proteins; Nerve Tissue Proteins; Protein Binding; Rats; Receptors, sigma | 1997 |
Rimcazole analogs attenuate the convulsive effects of cocaine: correlation with binding to sigma receptors rather than dopamine transporters.
Topics: Animals; Anticonvulsants; Binding Sites; Carbazoles; Cocaine; Dopamine; Dopamine Plasma Membrane Transport Proteins; Dose-Response Relationship, Drug; Ethylamines; Male; Membrane Glycoproteins; Membrane Transport Proteins; Mice; Nerve Tissue Proteins; Pyrrolidines; Radioligand Assay; Rats; Rats, Sprague-Dawley; Receptors, sigma; Seizures | 2001 |
Behavioral effects of rimcazole analogues alone and in combination with cocaine.
Topics: Animals; Behavior, Animal; Carbazoles; Cocaine; Conditioning, Operant; Dopamine Plasma Membrane Transport Proteins; Dopamine Uptake Inhibitors; Dose-Response Relationship, Drug; Male; Mice; Motor Activity; Rats; Rats, Sprague-Dawley; Receptors, sigma; Structure-Activity Relationship | 2003 |
Distinctions between dopamine transporter antagonists could be just around the bend.
Topics: Animals; Benztropine; Carbazoles; Cocaine; Discrimination Learning; Dopamine Plasma Membrane Transport Proteins; Dopamine Uptake Inhibitors; Dose-Response Relationship, Drug; Inhibitory Concentration 50; Mice; Models, Molecular; Motor Activity; Protein Conformation; Protein Structure, Secondary; Rats | 2008 |
Dual DAT/sigma1 receptor ligands based on 3-(4-(3-(bis(4-fluorophenyl)amino)propyl)piperazin-1-yl)-1-phenylpropan-1-ol.
Topics: Animals; Carbazoles; Cocaine; Combinatorial Chemistry Techniques; Dopamine Plasma Membrane Transport Proteins; Molecular Structure; Piperazines; Protein Binding; Rats; Receptors, sigma; Stereoisomerism; Structure-Activity Relationship | 2008 |
Bromoenol lactone inhibits voltage-gated Ca2+ and transient receptor potential canonical channels.
Topics: Animals; Behavior, Addictive; Calcium Channels; Carbazoles; Cocaine; Conditioning, Operant; Dopamine Plasma Membrane Transport Proteins; Dopamine Uptake Inhibitors; Dose-Response Relationship, Drug; Humans; Male; Naphthalenes; Phosphodiesterase Inhibitors; Phospholipases; Pyrones; Radioligand Assay; Rats; Rats, Sprague-Dawley; Receptors, sigma; Self Administration; Swine; Thapsigargin; Transient Receptor Potential Channels | 2011 |
Decreases in cocaine self-administration with dual inhibition of the dopamine transporter and σ receptors.
Topics: Animals; Anisoles; Antipsychotic Agents; Carbazoles; Cocaine; Cocaine-Related Disorders; Conditioning, Operant; Dopamine Plasma Membrane Transport Proteins; Dopamine Uptake Inhibitors; Male; Molecular Targeted Therapy; Oxalates; Piperidines; Propylamines; Radioligand Assay; Rats; Rats, Sprague-Dawley; Receptors, sigma; Reinforcement, Psychology; Self Administration | 2011 |
Novel nanoformulation to mitigate co-effects of drugs of abuse and HIV-1 infection: towards the treatment of NeuroAIDS.
Topics: AIDS Dementia Complex; Astrocytes; Blood-Brain Barrier; Carbazoles; Cocaine; Delayed-Action Preparations; Endothelial Cells; HIV Protease Inhibitors; HIV-1; Humans; Illicit Drugs; Magnets; Methamphetamine; Nanostructures; Nelfinavir; Neuroprotective Agents; Primary Cell Culture; Substance Abuse, Intravenous | 2017 |