rilmenidine has been researched along with idazoxan in 38 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 3 (7.89) | 18.7374 |
1990's | 27 (71.05) | 18.2507 |
2000's | 7 (18.42) | 29.6817 |
2010's | 1 (2.63) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
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Arrault, A; Guillaumet, G; Mérour, JY; Pfeiffer, B; Renard, P; Rettori, MC; Scalbert, E; Touzeau, F | 1 |
Agbaba, D; Filipic, S; Nikolic, K | 1 |
Agbaba, D; Azzali, E; Costantino, G; Glisic, S; Laurila, JM; Nikolic, K; Perovic, V; Pieroni, M; Radi, M; Scheinin, M; Srdic-Rajic, T; Tassini, S; Veljkovic, N; Vucicevic, J | 1 |
Berger, SB; Maiese, K; Pek, L; Reis, DJ | 1 |
Bousquet, P; Feldman, J; Gonon, F; Mermet, C; Monassier, L; Tibiriça, E | 1 |
Bidet, M; Parini, A; Poujeol, P | 2 |
Belcourt, A; Bousquet, P; Bricca, G; Dontenwill, M; Feldman, J | 1 |
Belcourt, A; Bousquet, P; Bricca, G; Dontenwill, M; Feldman, J; Tibiriça, E | 1 |
Coupry, I; Koenig, E; Lachaud, V; Parini, A; Podevin, RA | 2 |
Bidet, M; Coupry, I; Lachaud, V; Parini, A; Podevin, RA; Poujeol, P | 1 |
Head, GA; Sannajust, F | 3 |
Advenier, C; Biyah, K | 1 |
Gundlach, AL; King, PR; Louis, WJ; Suzuki, S | 2 |
Szabo, B; Urban, R | 1 |
Chernobelski, M; Mayorov, D; Medvedev, O | 1 |
Hamilton, CA; Jardine, E; Reid, JL | 1 |
Starke, K; Szabo, B; Urban, R | 1 |
Godwin, SJ; Head, GA; Sannajust, F | 1 |
Feinstein, DL; Golanov, EV; Regunathan, S; Reis, DJ | 1 |
Anderson, WP; Evans, RG | 1 |
Gargalidis-Moudanos, C; Parini, A | 1 |
Hayashi, Y; Kamibayashi, T; Mammoto, T; Takada, K; Yamatodani, A; Yoshiya, I | 1 |
Chan, CK; Head, GA | 1 |
Boulanger, CM; Illiano, S; Marsault, R; Taddei, S; Vanhoutte, PM | 1 |
Bousquet, P; De Jong, W; Feldman, J; Monassier, L; Roegel, JC; Yannoulis, N | 1 |
Avellar, MC; Markus, RP | 1 |
Arrais, CA; Camargo, LA; Menani, JV; Renzi, A; Saad, R; Saad, WA; Silveira, JE | 1 |
Bousquet, P; De Jong, W; Feldman, J; Roegel, JC; Yannoulis, N | 1 |
Burke, SL; Head, GA | 1 |
Godwin, SJ; Head, GA; Parkin, ML | 1 |
Artigues-Varin, C; Mulder, P; Richard, V; Thuillez, C; Varin, R | 1 |
de Arruda Camargo, LA; Guarda, IF; Guarda, RS; Saad, WA; Simões, S | 1 |
Burke, SL; Chan, CK; Head, GA | 1 |
1 review(s) available for rilmenidine and idazoxan
Article | Year |
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Protection of focal ischemic infarction by rilmenidine in the animal: evidence that interactions with central imidazoline receptors may be neuroprotective.
Topics: Adrenergic alpha-Agonists; Animals; Brain Ischemia; Cerebral Infarction; Dioxanes; Idazoxan; Imidazoles; Imidazoline Receptors; Neurons; Neuroprotective Agents; Oxazoles; Receptors, Drug; Rilmenidine | 1994 |
37 other study(ies) available for rilmenidine and idazoxan
Article | Year |
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Synthesis and biological evaluation of new 2-(4,5-dihydro-1H-imidazol-2-yl)-3,4-dihydro-2H-1,4-benzoxazine derivatives.
Topics: Adrenal Medulla; Animals; Antihypertensive Agents; Binding Sites; Blood Pressure; Cattle; Frontal Lobe; Heart Rate; Imidazoles; Imidazoline Receptors; In Vitro Techniques; Kidney; Oxazines; Rabbits; Radioligand Assay; Rats; Rats, Inbred SHR; Rats, Wistar; Receptors, Adrenergic, alpha-1; Receptors, Adrenergic, alpha-2; Receptors, Drug; Stereoisomerism; Structure-Activity Relationship | 2003 |
QSAR study of imidazoline antihypertensive drugs.
Topics: Antihypertensive Agents; Binding Sites; Imidazoline Receptors; Imidazolines; Ligands; Models, Molecular; Molecular Structure; Quantitative Structure-Activity Relationship | 2008 |
A combined ligand- and structure-based approach for the identification of rilmenidine-derived compounds which synergize the antitumor effects of doxorubicin.
Topics: Adrenergic alpha-Agonists; Antibiotics, Antineoplastic; Apoptosis; Doxorubicin; Drug Synergism; Humans; K562 Cells; Ligands; Molecular Structure; Oxazoles; Receptors, Adrenergic, alpha-2; Rilmenidine | 2016 |
Reduction in focal cerebral ischemia by agents acting at imidazole receptors.
Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Benzazepines; Brain; Dioxanes; Dose-Response Relationship, Drug; Idazoxan; Imidazoles; Ischemic Attack, Transient; Male; Neurons; Oxazoles; Rats; Rats, Inbred SHR; Receptors, Drug; Rilmenidine | 1992 |
Selectivity of rilmenidine for the nucleus reticularis lateralis, a ventrolateral medullary structure containing imidazoline-preferring receptors.
Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Azepines; Blood Pressure; Catecholamines; Clonidine; Dioxanes; Electrochemistry; Hemodynamics; Idazoxan; Imidazoline Receptors; Male; Medulla Oblongata; Neurons; Oxazoles; Piperoxan; Rats; Rats, Inbred WKY; Receptors, Drug; Reticular Formation; Rilmenidine; Stereotaxic Techniques; Yohimbine | 1991 |
The imidazoline-guanidinium receptor site, a target for some alpha-2 adrenergic agonists, is involved in inhibition of Na(+)-H+ exchange in renal proximal tubule cells.
Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Brimonidine Tartrate; Carrier Proteins; Dioxanes; Hydrogen; Idazoxan; Imidazoles; Imidazoline Receptors; In Vitro Techniques; Ion Exchange; Kidney Tubules, Proximal; Oxazoles; Quinoxalines; Rabbits; Receptors, Drug; Rilmenidine; Sodium; Sodium-Hydrogen Exchangers | 1991 |
[Selectivity of a new antihypertensive agent, rilmenidine, for imidazoline receptors in the human brain].
Topics: Adrenergic alpha-Antagonists; Animals; Antihypertensive Agents; Blood Pressure; Brain; Dioxanes; Humans; Idazoxan; Imidazoline Receptors; Oxazoles; Rabbits; Receptors, Drug; Rilmenidine; Yohimbine | 1990 |
Effect of imidazolines on Na+ transport and intracellular pH in renal proximal tubule cells.
Topics: Amiloride; Animals; Biological Transport; Brimonidine Tartrate; Cimetidine; Dioxanes; Dioxins; Hydrogen-Ion Concentration; Idazoxan; Imidazoles; In Vitro Techniques; Kidney Tubules, Proximal; Oxazoles; Quinoxalines; Rabbits; Rilmenidine; Sodium | 1990 |
Evidence for the involvement of imidazoline receptors in the central hypotensive effect of rilmenidine in the rabbit.
Topics: Animals; Antihypertensive Agents; Blood Pressure; Brain; Cisterna Magna; Dioxanes; Heart Rate; Hemodynamics; Idazoxan; Imidazoline Receptors; Injections; Injections, Intraventricular; Male; Oxazoles; Rabbits; Receptors, Drug; Rilmenidine; Tissue Extracts; Yohimbine | 1990 |
Different affinities of alpha 2-agonists for imidazoline and alpha 2-adrenergic receptors.
Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Binding, Competitive; Dioxanes; Guanfacine; Guanidine; Guanidines; Idazoxan; Imidazoline Receptors; Male; Oxazoles; Phenylacetates; Rabbits; Receptors, Adrenergic, alpha; Receptors, Drug; Rilmenidine; Yohimbine | 1989 |
[Selectivity of alpha 2-adrenergic agonists for the imidazoline-guanidine and alpha 2-adrenergic receptors].
Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Clonidine; Dioxanes; Guanfacine; Guanidines; Idazoxan; Kidney Tubules, Proximal; Male; Oxazoles; Phenylacetates; Rabbits; Receptors, Adrenergic, alpha; Rilmenidine; Yohimbine | 1989 |
[Interaction of rilmenidine with renal imidazoline-guanidine sites].
Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Basement Membrane; Binding Sites; Dioxanes; Drug Interactions; Guanfacine; Guanidines; Idazoxan; Imidazoles; Imidazoline Receptors; Kidney; Male; Oxazoles; Phenylacetates; Rabbits; Receptors, Drug; Rilmenidine; Sodium Channels; Yohimbine | 1989 |
Rilmenidine-induced hypotension in conscious rabbits involves imidazoline-preferring receptors.
Topics: Adrenergic alpha-Antagonists; Analysis of Variance; Animals; Antihypertensive Agents; Blood Pressure; Dioxanes; Dose-Response Relationship, Drug; Female; Heart Rate; Hypotension; Idazoxan; Imidazoline Receptors; Male; Methyldopa; Oxazoles; Rabbits; Receptors, Drug; Rilmenidine | 1994 |
Effects of three alpha 2-adrenoceptor agonists, rilmenidine, UK 14304 and clonidine on bradykinin- and substance P-induced airway microvascular leakage in guinea-pigs.
Topics: Acetylcholine; Adrenergic alpha-1 Receptor Antagonists; Adrenergic alpha-2 Receptor Agonists; Adrenergic alpha-2 Receptor Antagonists; Adrenergic alpha-Agonists; Animals; Bradykinin; Brimonidine Tartrate; Capillaries; Capillary Permeability; Clonidine; Dioxanes; Extravascular Lung Water; Guinea Pigs; Idazoxan; Oxazoles; Prazosin; Quinoxalines; Rilmenidine; Substance P; Trachea | 1995 |
Distribution of nonadrenergic [3H]rilmenidine binding in rat brain and kidney.
Topics: Adrenergic alpha-2 Receptor Agonists; Adrenergic alpha-2 Receptor Antagonists; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Autoradiography; Binding Sites; Brain; Dioxanes; Idazoxan; Imidazoles; Imidazoline Receptors; In Vitro Techniques; Kidney; Male; Oxazoles; Radioligand Assay; Rats; Rats, Inbred WKY; Receptors, Adrenergic, alpha-2; Receptors, Drug; Rilmenidine; Tritium | 1995 |
Mechanism of sympathoinhibition by imidazolines.
Topics: Adrenergic alpha-2 Receptor Agonists; Adrenergic alpha-2 Receptor Antagonists; Animals; Antihypertensive Agents; Benzazepines; Brimonidine Tartrate; Dioxanes; Hemodynamics; Idazoxan; Imidazoles; Oxazoles; Quinoxalines; Rabbits; Rilmenidine; Sympathetic Nervous System; Yohimbine | 1995 |
Sympathoinhibitory action of rilmenidine in conscious sinoaortically denervated rats.
Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Blood Pressure; Cisterna Magna; Denervation; Dioxanes; Heart Rate; Idazoxan; Infusions, Intravenous; Injections; Injections, Intra-Arterial; Kidney; Male; Oxazoles; Phenylephrine; Rats; Rats, Wistar; Rilmenidine; Sinoatrial Node; Sympatholytics | 1993 |
Down-regulation of imidazoline sites in rabbit kidney.
Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Clonidine; Dioxanes; Down-Regulation; Guanabenz; Idazoxan; Imidazoline Receptors; Kidney; Male; Oxazoles; Rabbits; Receptors, Drug; Rilmenidine | 1993 |
Sympathoinhibition by rilmenidine in conscious rabbits: involvement of alpha 2-adrenoceptors.
Topics: Adrenergic alpha-2 Receptor Antagonists; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Blood Pressure; Catecholamines; Decerebrate State; Dioxanes; Dose-Response Relationship, Drug; Electric Stimulation; Electrodes, Implanted; Female; Heart Rate; Hemodynamics; Idazoxan; Kidney; Male; Oxazoles; Rabbits; Rilmenidine; Sympathetic Nervous System; Yohimbine | 1993 |
Differential receptors involved in the cardiovascular effects of clonidine and rilmenidine in conscious rabbits.
Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Blood Pressure; Cardiovascular Physiological Phenomena; Cardiovascular System; Clonidine; Dioxanes; Female; Idazoxan; Imidazoline Receptors; Male; Methyldopa; Oxazoles; Rabbits; Receptors, Adrenergic, alpha-2; Receptors, Drug; Rilmenidine | 1993 |
Effect of rilmenidine on baroreflex control of renal sympathetic nerve activity.
Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Baroreflex; Blood Pressure; Dioxanes; Female; Idazoxan; Imidazoline Receptors; Kidney; Male; Oxazoles; Rabbits; Receptors, Adrenergic, alpha-2; Receptors, Drug; Rilmenidine; Sympathetic Nervous System | 1993 |
Involvement of imidazoline-preferring receptors in regulation of sympathetic tone.
Topics: Adrenergic alpha-Antagonists; Animals; Antihypertensive Agents; Central Nervous System; Clonidine; Dioxanes; Dose-Response Relationship, Drug; Female; Hemodynamics; Hypertension; Idazoxan; Imidazoles; Imidazoline Receptors; Male; Oxazoles; Rabbits; Rats; Rats, Inbred SHR; Receptors, Drug; Rilmenidine | 1994 |
Differential characteristics and localisation of [3H]oxazoline and [3H]imidazoline binding sites in rat kidney.
Topics: Adrenergic alpha-Antagonists; Animals; Autoradiography; Binding Sites; Dioxanes; Idazoxan; Imidazoles; Kidney; Male; Oxazoles; Radioligand Assay; Rats; Rats, Inbred WKY; Rilmenidine | 1995 |
Renal effects of infusion of rilmenidine and guanabenz in conscious dogs: contribution of peripheral and central nervous system alpha 2-adrenoceptors.
Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Autonomic Nerve Block; Binding Sites; Blood Pressure; Central Nervous System; Consciousness; Dioxanes; Dogs; Dose-Response Relationship, Drug; Ganglia, Autonomic; Guanabenz; Heart Rate; Idazoxan; Imidazoles; Imidazoline Receptors; Kidney; Male; Oxazoles; Peripheral Nervous System; Receptors, Adrenergic, alpha-2; Receptors, Drug; Renal Circulation; Rilmenidine | 1995 |
Selectivity of rilmenidine for I1-imidazoline-binding sites in rabbit proximal tubule cells.
Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Antihypertensive Agents; Binding Sites; Binding, Competitive; Cells, Cultured; Clonidine; Dioxanes; Idazoxan; Imidazoles; Imidazoline Receptors; Kidney Tubules, Proximal; Kinetics; Male; Oxazoles; Rabbits; Radioligand Assay; Receptors, Adrenergic, alpha-2; Receptors, Drug; Rilmenidine; Tritium | 1995 |
Antiarrhythmic action of rilmenidine on adrenaline-induced arrhythmia via central imidazoline receptors in halothane-anaesthetized dogs.
Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Analysis of Variance; Anesthetics, Inhalation; Animals; Arrhythmias, Cardiac; Blood Pressure; Dogs; Epinephrine; Female; Halothane; Heart Rate; Idazoxan; Imidazoline Receptors; Male; Oxazoles; Receptors, Drug; Rilmenidine; Yohimbine | 1996 |
Relative importance of central imidazoline receptors for the antihypertensive effects of moxonidine and rilmenidine.
Topics: Adrenergic alpha-2 Receptor Antagonists; Animals; Antihypertensive Agents; Benzofurans; Blood Pressure; Cardiac Catheterization; Clonidine; Dose-Response Relationship, Drug; Female; Heart Rate; Idazoxan; Imidazoles; Imidazoline Receptors; Injections, Intravenous; Male; Oxazoles; Rabbits; Receptors, Drug; Rilmenidine; Time Factors | 1996 |
Rilmenidine activates postjunctional alpha 1- and alpha 2-adrenoceptors in the canine saphenous vein.
Topics: Adrenergic alpha-1 Receptor Agonists; Adrenergic alpha-2 Receptor Agonists; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Brimonidine Tartrate; Calcium Channel Blockers; Clonidine; Dihydropyridines; Dogs; Female; Idazoxan; Imidazoles; Imidazoline Receptors; In Vitro Techniques; Isotope Labeling; Male; Medetomidine; Muscle Contraction; Muscle, Smooth; Osmolar Concentration; Oxazoles; Phenoxybenzamine; Prazosin; Protein Binding; Quinoxalines; Radioligand Assay; Receptors, Adrenergic, alpha-1; Receptors, Adrenergic, alpha-2; Receptors, Drug; Rilmenidine; Saphenous Vein; Tritium; Yohimbine | 1996 |
Inhibition of centrally induced ventricular arrhythmias by rilmenidine and idazoxan in rabbits.
Topics: Adrenergic alpha-Antagonists; Analysis of Variance; Animals; Antihypertensive Agents; Arrhythmias, Cardiac; Bicuculline; Blood Pressure; Dose-Response Relationship, Drug; GABA Antagonists; Heart Rate; Idazoxan; Injections, Intravenous; Male; Oxazoles; Rabbits; Rilmenidine | 1996 |
Are imidazoline receptors involved in sympathetic neurotransmission in rat vas deferens?
Topics: Adrenergic alpha-2 Receptor Agonists; Adrenergic alpha-2 Receptor Antagonists; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Electric Stimulation; Idazoxan; Imidazoline Receptors; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth; Norepinephrine; Oxazoles; Rats; Rats, Wistar; Receptors, Adrenergic, alpha-2; Receptors, Drug; Rilmenidine; Sympathetic Nervous System; Synaptic Transmission; Vas Deferens; Yohimbine | 1996 |
Effect of rilmenidine injection into the paraventricular nucleus of the hypothalamus on the water intake induced by application of angiotensin II to the subfornical organ.
Topics: Angiotensin II; Animals; Drinking; Idazoxan; Imidazoles; Injections; Male; Oxazoles; Paraventricular Hypothalamic Nucleus; Rats; Rats, Sprague-Dawley; Rilmenidine; Subfornical Organ | 1997 |
Preventive effect of rilmenidine on the occurrence of neurogenic ventricular arrhythmias in rabbits.
Topics: Animals; Antihypertensive Agents; Bicuculline; Cardiac Complexes, Premature; GABA Antagonists; Hemodynamics; Idazoxan; Injections, Intravenous; Injections, Intraventricular; Male; Oxazoles; Rabbits; Rilmenidine; Sympathetic Nervous System; Tachycardia, Ventricular | 1998 |
Comparison of renal sympathetic baroreflex effects of rilmenidine and alpha-methylnoradrenaline in the ventrolateral medulla of the rabbit.
Topics: Adrenergic alpha-Antagonists; Animals; Antihypertensive Agents; Baroreflex; Blood Pressure; Dose-Response Relationship, Drug; Female; Idazoxan; Kidney; Male; Medulla Oblongata; Nordefrin; Oxazoles; Rabbits; Receptors, Adrenergic, alpha-2; Rilmenidine; Sympathetic Nervous System; Vasoconstrictor Agents | 2000 |
Importance of imidazoline-preferring receptors in the cardiovascular actions of chronically administered moxonidine, rilmenidine and clonidine in conscious rabbits.
Topics: Adrenergic alpha-2 Receptor Antagonists; Animals; Antihypertensive Agents; Benzofurans; Blood Pressure; Cardiovascular System; Clonidine; Dose-Response Relationship, Drug; Drug Administration Schedule; Female; Fourth Ventricle; Heart Rate; Idazoxan; Imidazoles; Imidazoline Receptors; Injections, Intraventricular; Male; Oxazoles; Rabbits; Receptors, Drug; Rilmenidine | 2003 |
Alpha2-adrenoceptor ligands inhibit alpha1-adrenoceptor-mediated contraction of isolated rat arteries.
Topics: Adrenergic alpha-1 Receptor Antagonists; Adrenergic alpha-2 Receptor Agonists; Adrenergic alpha-2 Receptor Antagonists; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Aorta, Thoracic; Arteries; Azepines; Brimonidine Tartrate; Clonidine; Idazoxan; In Vitro Techniques; Ligands; Male; Mesenteric Arteries; Muscle Contraction; Muscle, Smooth, Vascular; Nitric Oxide; Oxazoles; Prostaglandins; Quinoxalines; Rats; Rats, Wistar; Receptors, Adrenergic, alpha-2; Rilmenidine; Yohimbine | 2002 |
Moxonidine and rilmenidine injected into the medial septal area reduces the salivation induced by pilocarpine.
Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Analysis of Variance; Animals; Drug Interactions; Idazoxan; Imidazoles; Male; Muscarinic Agonists; Oxazoles; Pilocarpine; Rats; Rats, Sprague-Dawley; Rilmenidine; Salivation; Septum of Brain; Yohimbine | 2004 |
Contribution of imidazoline receptors and alpha2-adrenoceptors in the rostral ventrolateral medulla to sympathetic baroreflex inhibition by systemic rilmenidine.
Topics: Adrenergic alpha-2 Receptor Agonists; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Antihypertensive Agents; Baroreflex; Blood Pressure; Dose-Response Relationship, Drug; Idazoxan; Imidazoline Receptors; Injections, Intravenous; Kidney; Medulla Oblongata; Neural Inhibition; Oxazoles; Rabbits; Receptors, Adrenergic, alpha-2; Receptors, Drug; Rilmenidine; Sympathetic Nervous System | 2007 |